File size: 1,927 Bytes
a7834dc
 
 
 
 
975d2c6
 
 
 
 
 
 
 
11fad9c
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
 
a7834dc
 
11fad9c
975d2c6
a7834dc
11fad9c
975d2c6
a7834dc
11fad9c
975d2c6
11fad9c
 
a7834dc
 
 
 
 
 
 
 
 
 
1
2
3
4
5
6
7
8
9
10
11
12
13
14
15
16
17
18
19
20
21
22
23
24
25
26
27
28
29
30
31
32
33
34
35
36
37
38
39
40
41
42
43
44
45
46
47
48
49
50
51
52
53
54
55
56
57
58
59
60
61
62
63
64
65
66
67
68
69
70
71
72
73
74
75
76
77
78
79
80
81
82
83
84
85
86
87
88
89
90
91
92
93
94
95
96
97
98
99
100
101
102
---
dataset_info:
  features:
  - name: SMILES
    dtype: string
  - name: Deep SMILES
    dtype: string
  - name: SELFIES
    dtype: string
  - name: SAFE
    dtype: string
  - name: Group SELFIES
    dtype: string
  - name: DBPP
    dtype: float64
  - name: RA
    dtype: float64
  - name: SYBA
    dtype: float64
  - name: QED
    dtype: float64
  - name: SA
    dtype: float64
  - name: NP
    dtype: float64
  - name: logP
    dtype: float64
  - name: Weight
    dtype: float64
  - name: Rings
    dtype: float64
  - name: gsk3b_current
    dtype: float64
  - name: jnk3_current
    dtype: float64
  - name: drd2_current
    dtype: float64
  - name: Celecoxib
    dtype: float64
  - name: Troglitazone
    dtype: float64
  - name: Thiothixene
    dtype: float64
  - name: Aripiprazole
    dtype: float64
  - name: Albuterol
    dtype: float64
  - name: Mestranol
    dtype: float64
  - name: Median 1
    dtype: float64
  - name: Median 2
    dtype: float64
  - name: c7h8n2o2
    dtype: float64
  - name: c9h10n2o2pf2cl
    dtype: float64
  - name: Osimertinib
    dtype: float64
  - name: Fexofenadine
    dtype: float64
  - name: Ranolazine
    dtype: float64
  - name: Perindopril
    dtype: float64
  - name: Amlodipine
    dtype: float64
  - name: Sitagliptin
    dtype: float64
  - name: Zaleplon
    dtype: float64
  - name: valsartan_smarts
    dtype: float64
  - name: Deco Hop
    dtype: float64
  - name: Scaffold Hop
    dtype: float64
  - name: Penalized logP
    dtype: float64
  splits:
  - name: train
    num_bytes: 1098896649
    num_examples: 1228690
  - name: valid
    num_bytes: 68629127
    num_examples: 76842
  - name: test
    num_bytes: 205923041
    num_examples: 230304
  download_size: 730840130
  dataset_size: 1373448817
configs:
- config_name: default
  data_files:
  - split: train
    path: data/train-*
  - split: valid
    path: data/valid-*
  - split: test
    path: data/test-*
---