| endpoint_id,split,assay_id,standard_type,assay_type,label_type,binary_semantics,n_pairs,n_unique_molecules,mean,std_population,std_sample,min,q25,median,q75,max,positive_fraction,label_counts,value_sources,value_types,units | |
| 135936|Inhibitory activity|binary|active_inactive,validation,135936,Inhibitory activity,F,binary,active_inactive,33,12,0.5833333333333334,0.4930066485916347,0.5149286505444373,0.0,0.0,1.0,1.0,1.0,0.5833333333333334,"{""0"": 5, ""1"": 7}","{""clean_label"": 12}","{""binary_label"": 12}","{""binary_label"": 12}" | |
| 335844|Activity|binary|active_inactive,validation,335844,Activity,F,binary,active_inactive,33,12,0.0,0.0,0.0,0.0,0.0,0.0,0.0,0.0,0.0,"{""0"": 12, ""1"": 0}","{""clean_label"": 12}","{""binary_label"": 12}","{""binary_label"": 12}" | |
| 424986|Activity|binary|active_inactive,validation,424986,Activity,F,binary,active_inactive,22,10,0.4,0.48989794855663565,0.5163977794943223,0.0,0.0,0.0,1.0,1.0,0.4,"{""0"": 6, ""1"": 4}","{""clean_label"": 10}","{""binary_label"": 10}","{""binary_label"": 10}" | |
| 432191|Activity|binary|active_inactive,validation,432191,Activity,F,binary,active_inactive,76,18,0.16666666666666666,0.372677996249965,0.3834824944236852,0.0,0.0,0.0,0.0,1.0,0.16666666666666666,"{""0"": 15, ""1"": 3}","{""clean_label"": 18}","{""binary_label"": 18}","{""binary_label"": 18}" | |
| 435149|Activity|binary|active_inactive,validation,435149,Activity,F,binary,active_inactive,60,16,0.25,0.4330127018922193,0.4472135954999579,0.0,0.0,0.0,0.25,1.0,0.25,"{""0"": 12, ""1"": 4}","{""clean_label"": 16}","{""binary_label"": 16}","{""binary_label"": 16}" | |
| 435161|Activity|binary|active_inactive,validation,435161,Activity,T,binary,active_inactive,100,23,0.21739130434782608,0.4124709991523973,0.42174116783664994,0.0,0.0,0.0,0.0,1.0,0.21739130434782608,"{""0"": 18, ""1"": 5}","{""clean_label"": 23}","{""binary_label"": 23}","{""binary_label"": 23}" | |
| 437563|Activity|binary|active_inactive,validation,437563,Activity,F,binary,active_inactive,27,11,0.2727272727272727,0.4453617714151233,0.4670993664969138,0.0,0.0,0.0,0.5,1.0,0.2727272727272727,"{""0"": 8, ""1"": 3}","{""clean_label"": 11}","{""binary_label"": 11}","{""binary_label"": 11}" | |
| 437564|Activity|binary|active_inactive,validation,437564,Activity,F,binary,active_inactive,27,11,0.36363636363636365,0.48104569292083466,0.504524979109513,0.0,0.0,0.0,1.0,1.0,0.36363636363636365,"{""0"": 7, ""1"": 4}","{""clean_label"": 11}","{""binary_label"": 11}","{""binary_label"": 11}" | |
| 457828|Activity|binary|active_inactive,validation,457828,Activity,B,binary,active_inactive,68,17,0.5882352941176471,0.49215295678475035,0.5072996561958923,0.0,0.0,1.0,1.0,1.0,0.5882352941176471,"{""0"": 7, ""1"": 10}","{""clean_label"": 17}","{""binary_label"": 17}","{""binary_label"": 17}" | |
| 466136|Activity|binary|active_inactive,validation,466136,Activity,B,binary,active_inactive,39,13,0.46153846153846156,0.4985185152621431,0.5188745216627708,0.0,0.0,0.0,1.0,1.0,0.46153846153846156,"{""0"": 7, ""1"": 6}","{""clean_label"": 13}","{""binary_label"": 13}","{""binary_label"": 13}" | |
| 466137|Activity|binary|active_inactive,validation,466137,Activity,B,binary,active_inactive,39,13,0.46153846153846156,0.4985185152621431,0.5188745216627708,0.0,0.0,0.0,1.0,1.0,0.46153846153846156,"{""0"": 7, ""1"": 6}","{""clean_label"": 13}","{""binary_label"": 13}","{""binary_label"": 13}" | |
| 470402|Activity|binary|active_inactive,validation,470402,Activity,F,binary,active_inactive,60,16,0.375,0.4841229182759271,0.5,0.0,0.0,0.0,1.0,1.0,0.375,"{""0"": 10, ""1"": 6}","{""clean_label"": 16}","{""binary_label"": 16}","{""binary_label"": 16}" | |
| 473194|Activity|binary|toxic_non_toxic,validation,473194,Activity,A,binary,toxic_non_toxic,85,19,0.6842105263157895,0.464829519280413,0.4775669329409193,0.0,0.0,1.0,1.0,1.0,0.6842105263157895,"{""0"": 6, ""1"": 13}","{""clean_label"": 19}","{""binary_label"": 19}","{""binary_label"": 19}" | |
| 475548|Activity|binary|active_inactive,validation,475548,Activity,B,binary,active_inactive,68,17,0.4117647058823529,0.49215295678475035,0.5072996561958923,0.0,0.0,0.0,1.0,1.0,0.4117647058823529,"{""0"": 10, ""1"": 7}","{""clean_label"": 17}","{""binary_label"": 17}","{""binary_label"": 17}" | |
| 475550|Activity|binary|active_inactive,validation,475550,Activity,B,binary,active_inactive,45,14,0.2857142857142857,0.45175395145262565,0.4688072309384954,0.0,0.0,0.0,0.75,1.0,0.2857142857142857,"{""0"": 10, ""1"": 4}","{""clean_label"": 14}","{""binary_label"": 14}","{""binary_label"": 14}" | |
| 490527|Activity|binary|active_inactive,validation,490527,Activity,F,binary,active_inactive,42,22,0.5909090909090909,0.4916660830178167,0.5032362797401965,0.0,0.0,1.0,1.0,1.0,0.5909090909090909,"{""0"": 9, ""1"": 13}","{""clean_label"": 22}","{""binary_label"": 22}","{""binary_label"": 22}" | |
| 493953|Activity|binary|active_inactive,validation,493953,Activity,B,binary,active_inactive,100,28,0.39285714285714285,0.48838551182776224,0.49734746139343805,0.0,0.0,0.0,1.0,1.0,0.39285714285714285,"{""0"": 17, ""1"": 11}","{""clean_label"": 28}","{""binary_label"": 28}","{""binary_label"": 28}" | |
| 495219|Activity|binary|active_inactive,validation,495219,Activity,F,binary,active_inactive,76,18,0.0,0.0,0.0,0.0,0.0,0.0,0.0,0.0,0.0,"{""0"": 18, ""1"": 0}","{""clean_label"": 18}","{""binary_label"": 18}","{""binary_label"": 18}" | |
| 1008|EC50|continuous,validation,1008,EC50,F,continuous,,100,39,7.9592307692307696,0.6280183919215392,0.6362281311116428,6.39,7.67,8.0,8.434999999999999,9.14,,,"{""pchembl"": 39}","{""pChEMBL"": 39}","{""pChEMBL"": 39}" | |
| 1011|IC50|continuous,validation,1011,IC50,B,continuous,,60,16,8.13125,0.6649424317187166,0.6867495904622004,6.9,7.65,8.25,8.7,9.4,,,"{""pchembl"": 16}","{""pChEMBL"": 16}","{""pChEMBL"": 16}" | |
| 1023|Ki|continuous,validation,1023,Ki,B,continuous,,100,28,8.487142857142858,0.8046954044093647,0.8194616893531145,6.5,7.887499999999999,8.850000000000001,9.115,9.54,,,"{""pchembl"": 28}","{""pChEMBL"": 28}","{""pChEMBL"": 28}" | |
| 1101|Ki|continuous,validation,1101,Ki,B,continuous,,22,10,7.787999999999999,1.1529163022526832,1.2152804888858648,5.85,7.154999999999999,7.865,8.759999999999998,9.23,,,"{""pchembl"": 10}","{""pChEMBL"": 10}","{""pChEMBL"": 10}" | |
| 1102|Ki|continuous,validation,1102,Ki,B,continuous,,60,16,7.3725000000000005,0.9270821161040699,0.9574862923300783,5.84,6.515,7.66,8.2025,8.47,,,"{""pchembl"": 16}","{""pChEMBL"": 16}","{""pChEMBL"": 16}" | |
| 1130|Ki|continuous,validation,1130,Ki,B,continuous,,52,15,8.101333333333333,0.8776777439483255,0.9084827749500552,6.1,7.705,8.31,8.785,9.49,,,"{""pchembl"": 15}","{""pChEMBL"": 15}","{""pChEMBL"": 15}" | |
| 1143|Ki|continuous,validation,1143,Ki,B,continuous,,100,42,8.02,0.861968953147662,0.8724174431554834,6.0,7.4399999999999995,7.98,8.577499999999999,10.15,,,"{""pchembl"": 42}","{""pChEMBL"": 42}","{""pChEMBL"": 42}" | |
| 1156|Ki|continuous,validation,1156,Ki,B,continuous,,33,12,7.054166666666667,0.6372526753354764,0.6655887118433824,6.06,6.48,7.005,7.7275,7.8,,,"{""pchembl"": 12}","{""pChEMBL"": 12}","{""pChEMBL"": 12}" | |
| 1159|Ki|continuous,validation,1159,Ki,B,continuous,,27,11,8.377272727272727,0.7088157974472239,0.7434122800854304,6.92,8.0,8.39,8.850000000000001,9.68,,,"{""pchembl"": 11}","{""pChEMBL"": 11}","{""pChEMBL"": 11}" | |
| 1160|Ki|continuous,validation,1160,Ki,B,continuous,,100,60,6.797166666666667,0.7250266470198795,0.7311451238231679,5.3,6.3,6.779999999999999,7.3,8.3,,,"{""pchembl"": 60}","{""pChEMBL"": 60}","{""pChEMBL"": 60}" | |
| 1164|Ki|continuous,validation,1164,Ki,B,continuous,,52,15,6.502,1.2379886913861533,1.2814400381713424,4.31,5.869999999999999,6.78,6.905,8.57,,,"{""pchembl"": 15}","{""pChEMBL"": 15}","{""pChEMBL"": 15}" | |
| 1167|Ki|continuous,validation,1167,Ki,B,continuous,,33,12,7.707916666666667,0.6713030188041431,0.701153135696454,6.71,7.3237499999999995,7.725,7.9025,9.22,,,"{""pchembl"": 12}","{""pChEMBL"": 12}","{""pChEMBL"": 12}" | |
| 118|IC50|continuous,validation,118,IC50,B,continuous,,39,13,7.356153846153846,0.630842397257441,0.656601584696261,6.09,6.94,7.42,7.64,8.64,,,"{""pchembl"": 13}","{""pChEMBL"": 13}","{""pChEMBL"": 13}" | |
| 1200|Ki|continuous,validation,1200,Ki,B,continuous,,68,17,7.534705882352942,0.6872461469051581,0.7083971136221796,6.36,7.08,7.38,7.96,9.0,,,"{""pchembl"": 17}","{""pChEMBL"": 17}","{""pChEMBL"": 17}" | |
| 1202|Ki|continuous,validation,1202,Ki,B,continuous,,27,11,6.6463636363636365,0.7540710447271317,0.7908763838587259,5.21,6.324999999999999,7.0,7.17,7.46,,,"{""pchembl"": 11}","{""pChEMBL"": 11}","{""pChEMBL"": 11}" | |
| 1206|Ki|continuous,validation,1206,Ki,B,continuous,,85,19,7.77421052631579,1.343543295639414,1.3803595175391152,5.37,6.705,7.85,8.969999999999999,9.52,,,"{""pchembl"": 19}","{""pChEMBL"": 19}","{""pChEMBL"": 19}" | |
| 1210|Ki|continuous,validation,1210,Ki,B,continuous,,27,11,8.671818181818182,0.8448648970189708,0.8861017795018604,7.29,8.04,8.73,9.245000000000001,10.35,,,"{""pchembl"": 11}","{""pChEMBL"": 11}","{""pChEMBL"": 11}" | |
| 1211|Ki|continuous,validation,1211,Ki,B,continuous,,22,10,6.399,0.9060513230496382,0.9550619526152915,4.69,5.91,6.545,7.18,7.54,,,"{""pchembl"": 10}","{""pChEMBL"": 10}","{""pChEMBL"": 10}" | |
| 1232|IC50|continuous,validation,1232,IC50,B,continuous,,100,26,7.691923076923077,0.771681576572424,0.7869638834445669,6.34,7.225,7.625,8.207500000000001,9.12,,,"{""pchembl"": 26}","{""pChEMBL"": 26}","{""pChEMBL"": 26}" | |
| 1261|Inhibition|continuous,validation,1261,Inhibition,B,continuous,,100,50,5.1626e-05,3.792188713658644e-05,3.830689078524454e-05,0.0,7.375e-06,6.539999999999999e-05,8.92e-05,9.6e-05,,,"{""standard_value"": 50}","{""raw standard value"": 50}","{""%"": 50}" | |
| 128|IC50|continuous,validation,128,IC50,B,continuous,,33,12,6.689166666666666,0.6394197673585709,0.6678521656411059,5.8,6.12,6.76,7.075,7.75,,,"{""pchembl"": 12}","{""pChEMBL"": 12}","{""pChEMBL"": 12}" | |
| 1291|Inhibition|continuous,validation,1291,Inhibition,B,continuous,,100,27,39.25925925925926,31.671452962954454,32.27477294514973,0.0,6.5,35.0,70.5,86.0,,,"{""standard_value"": 27}","{""raw standard value"": 27}","{""%"": 27}" | |
| 12|CC50|continuous,validation,12,CC50,F,continuous,,22,10,5.866868855504382,0.4142860421783107,0.43669583203334894,5.200659450546418,5.5779440026597875,5.970786987771497,6.130486416945223,6.494850021680094,,,"{""standard_value_p_transform"": 10}","{""pChEMBL"": 10}","{""pChEMBL"": 10}" | |
| 1315|Ki|continuous,validation,1315,Ki,B,continuous,,22,10,6.981,0.3326695056659087,0.35066444866218704,6.35,6.7875,7.0,7.157500000000001,7.47,,,"{""pchembl"": 10}","{""pChEMBL"": 10}","{""pChEMBL"": 10}" | |
| 1343|Ki|continuous,validation,1343,Ki,B,continuous,,33,12,7.744166666666666,3.3971494382136855,3.5482068668127242,6.41,6.68,6.715,6.8275,19.0,,,"{""pchembl"": 11, ""standard_value"": 1}","{""pChEMBL"": 11, ""raw standard value"": 1}","{""%"": 1, ""pChEMBL"": 11}" | |
| 1349|Ki|continuous,validation,1349,Ki,B,continuous,,76,18,8.090555555555556,0.6028955338127477,0.620374386225743,6.21,7.85,8.280000000000001,8.4725,8.82,,,"{""pchembl"": 18}","{""pChEMBL"": 18}","{""pChEMBL"": 18}" | |
| 1355|Ki|continuous,validation,1355,Ki,B,continuous,,100,24,6.496666666666666,0.7472821124284694,0.7633545342287136,5.22,6.0225,6.32,6.855,8.49,,,"{""pchembl"": 24}","{""pChEMBL"": 24}","{""pChEMBL"": 24}" | |
| 1361|Ki|continuous,validation,1361,Ki,B,continuous,,27,11,7.078181818181818,0.5755600937240204,0.6036525189513944,6.15,6.699999999999999,6.97,7.57,8.0,,,"{""pchembl"": 11}","{""pChEMBL"": 11}","{""pChEMBL"": 11}" | |
| 1371|IC50|continuous,validation,1371,IC50,B,continuous,,52,15,6.343999999999999,0.8117947195360823,0.8402873658117542,5.2,5.845000000000001,6.08,6.77,8.02,,,"{""pchembl"": 15}","{""pChEMBL"": 15}","{""pChEMBL"": 15}" | |
| 1400|IC50|continuous,validation,1400,IC50,B,continuous,,100,24,4.8741666661122505,0.8096908708535788,0.827105570051817,2.860000001448153,4.45,4.835,5.34,6.24,,,"{""pchembl"": 21, ""standard_value_p_transform"": 3}","{""pChEMBL"": 24}","{""pChEMBL"": 24}" | |
| 1419|Ki|continuous,validation,1419,Ki,B,continuous,,100,33,7.306363636363637,0.8747564792967386,0.8883194040638558,5.34,6.71,7.34,7.82,9.22,,,"{""pchembl"": 33}","{""pChEMBL"": 33}","{""pChEMBL"": 33}" | |
| 1422|Ki|continuous,validation,1422,Ki,B,continuous,,100,26,7.524230769230769,0.6592605010798263,0.6723164319093983,6.47,6.967499999999999,7.54,8.015,8.92,,,"{""pchembl"": 26}","{""pChEMBL"": 26}","{""pChEMBL"": 26}" | |
| 1423|Ki|continuous,validation,1423,Ki,B,continuous,,95,20,7.4915,0.5550790484246367,0.5694990873797042,6.72,6.955,7.505,7.789999999999999,8.89,,,"{""pchembl"": 20}","{""pChEMBL"": 20}","{""pChEMBL"": 20}" | |
| 1432|Ki|continuous,validation,1432,Ki,F,continuous,,100,38,7.971578947368421,0.8037495234206313,0.8145385903813789,6.88,7.25,7.744999999999999,8.635,9.66,,,"{""pchembl"": 38}","{""pChEMBL"": 38}","{""pChEMBL"": 38}" | |
| 1445|Ki|continuous,validation,1445,Ki,B,continuous,,100,34,8.651470588235293,0.7849021383471998,0.7967058403692239,7.19,8.0925,9.0,9.2925,9.82,,,"{""pchembl"": 34}","{""pChEMBL"": 34}","{""pChEMBL"": 34}" | |
| 1446|Ki|continuous,validation,1446,Ki,B,continuous,,100,28,7.049642857142857,0.602971701200794,0.6140363250375408,5.63,6.6850000000000005,6.93,7.307499999999999,8.42,,,"{""pchembl"": 28}","{""pChEMBL"": 28}","{""pChEMBL"": 28}" | |
| 1449|Ki|continuous,validation,1449,Ki,B,continuous,,95,20,6.511500010122271,1.4581572908930835,1.4960378143914383,3.3000002024454176,5.58,6.9,7.382499999999999,8.42,,,"{""pchembl"": 19, ""standard_value_p_transform"": 1}","{""pChEMBL"": 20}","{""pChEMBL"": 20}" | |
| 1451|Ki|continuous,validation,1451,Ki,B,continuous,,85,19,7.477631578947368,0.8026016387858409,0.8245947968228811,5.28,7.125,7.54,8.01,8.72,,,"{""pchembl"": 19}","{""pChEMBL"": 19}","{""pChEMBL"": 19}" | |
| 1468|Ki|continuous,validation,1468,Ki,B,continuous,,100,30,8.889666666666667,0.7067224034623182,0.7188040034684691,7.38,8.5025,8.940000000000001,9.22,10.4,,,"{""pchembl"": 30}","{""pChEMBL"": 30}","{""pChEMBL"": 30}" | |
| 1472|Ki|continuous,validation,1472,Ki,B,continuous,,45,14,7.947857142857143,0.31688615737310744,0.3288483066570493,7.54,7.647500000000001,7.885,8.2775,8.42,,,"{""pchembl"": 14}","{""pChEMBL"": 14}","{""pChEMBL"": 14}" | |
| 1475|KiAH|continuous,validation,1475,KiAH,B,continuous,,27,11,54.84909090909091,55.7757858792351,58.49813774378556,0.032,1.671,38.9,91.6,166.0,,,"{""standard_value"": 11}","{""raw standard value"": 11}","{""nM"": 11}" | |
| 1513|Ki|continuous,validation,1513,Ki,B,continuous,,100,42,6.915238095238095,0.6847287891853452,0.6930288351275397,5.0,6.475,6.93,7.4375,8.28,,,"{""pchembl"": 42}","{""pChEMBL"": 42}","{""pChEMBL"": 42}" | |
| 1514|Ki|continuous,validation,1514,Ki,B,continuous,,100,45,9.003777777777778,0.7125674670245116,0.7206193323955598,7.43,8.76,9.24,9.52,10.12,,,"{""pchembl"": 45}","{""pChEMBL"": 45}","{""pChEMBL"": 45}" | |
| 1526|Ki|continuous,validation,1526,Ki,B,continuous,,33,12,8.091666666666667,0.9349316671405576,0.976504278567486,6.1,7.7,8.05,8.825000000000001,9.5,,,"{""pchembl"": 12}","{""pChEMBL"": 12}","{""pChEMBL"": 12}" | |
| 1530|Ki|continuous,validation,1530,Ki,B,continuous,,45,14,6.822857142857143,0.8024732178123595,0.8327658140791451,6.0,6.3175,6.465,7.1125,8.59,,,"{""pchembl"": 14}","{""pChEMBL"": 14}","{""pChEMBL"": 14}" | |
| 157|Ki|continuous,validation,157,Ki,B,continuous,,100,44,7.872045454545455,1.4540860602664334,1.470896862217465,4.21,6.859999999999999,8.01,8.8725,10.55,,,"{""pchembl"": 44}","{""pChEMBL"": 44}","{""pChEMBL"": 44}" | |
| 1596|EC50|continuous,validation,1596,EC50,F,continuous,,45,14,9.358571428571429,0.4646635824959378,0.48220418820337835,8.4,9.1075,9.46,9.6425,10.05,,,"{""pchembl"": 14}","{""pChEMBL"": 14}","{""pChEMBL"": 14}" | |
| 1616|IC50|continuous,validation,1616,IC50,B,continuous,,100,30,7.185333333333333,0.559188300624714,0.5687477674580409,6.24,6.795,7.1,7.4625,8.57,,,"{""pchembl"": 30}","{""pChEMBL"": 30}","{""pChEMBL"": 30}" | |
| 1618|IC50|continuous,validation,1618,IC50,B,continuous,,100,26,6.68076923076923,0.9366220938807508,0.9551708667120163,5.14,6.0075,6.475,7.5874999999999995,8.51,,,"{""pchembl"": 26}","{""pChEMBL"": 26}","{""pChEMBL"": 26}" | |
| 165|IC50|continuous,validation,165,IC50,B,continuous,,100,25,6.7272,0.5912462769438807,0.6034382045136575,5.4,6.35,6.92,7.16,7.52,,,"{""pchembl"": 25}","{""pChEMBL"": 25}","{""pChEMBL"": 25}" | |
| 166|IC50|continuous,validation,166,IC50,B,continuous,,39,13,7.691538461538461,0.5585950253688838,0.5814041358906636,6.52,7.3,7.7,8.0,8.52,,,"{""pchembl"": 13}","{""pChEMBL"": 13}","{""pChEMBL"": 13}" | |
| 1671|Activity|continuous,validation,1671,Activity,F,continuous,,33,12,81.5,13.363507523600731,13.957728390328485,60.0,68.5,82.5,92.0,102.0,,,"{""standard_value"": 12}","{""raw standard value"": 12}","{""%"": 12}" | |
| 1676|EC50|continuous,validation,1676,EC50,B,continuous,,100,40,8.290000000000001,0.4512704289004545,0.457019328548221,7.5,7.9125,8.235,8.56,9.3,,,"{""pchembl"": 40}","{""pChEMBL"": 40}","{""pChEMBL"": 40}" | |
| 1678|EC50|continuous,validation,1678,EC50,F,continuous,,68,17,8.454117647058823,0.49936499469213436,0.5147336547129181,7.51,8.06,8.52,8.74,9.52,,,"{""pchembl"": 17}","{""pChEMBL"": 17}","{""pChEMBL"": 17}" | |
| 1680|EC50|continuous,validation,1680,EC50,F,continuous,,100,25,8.984,0.45971295391798556,0.4691925688527756,8.11,8.74,8.96,9.52,9.7,,,"{""pchembl"": 25}","{""pChEMBL"": 25}","{""pChEMBL"": 25}" | |
| 1685|ED50|continuous,validation,1685,ED50,F,continuous,,33,12,8.6575,0.448276793213003,0.4682098402911398,7.85,8.4275,8.715,8.8775,9.6,,,"{""pchembl"": 12}","{""pChEMBL"": 12}","{""pChEMBL"": 12}" | |
| 1687|Efficacy|continuous,validation,1687,Efficacy,F,continuous,,100,40,80.725,12.55186739095024,12.71177023722906,59.0,72.75,77.5,90.75,115.0,,,"{""standard_value"": 40}","{""raw standard value"": 40}","{""%"": 40}" | |
| 1699|IC50|continuous,validation,1699,IC50,B,continuous,,76,18,8.253888888888888,0.3290919980945702,0.33863287232964,7.54,8.0275,8.27,8.4375,8.89,,,"{""pchembl"": 18}","{""pChEMBL"": 18}","{""pChEMBL"": 18}" | |
| 1704|IC50|continuous,validation,1704,IC50,B,continuous,,100,33,8.746060606060606,0.7552440480298281,0.7669539563833812,6.68,8.31,9.0,9.22,10.0,,,"{""pchembl"": 33}","{""pChEMBL"": 33}","{""pChEMBL"": 33}" | |
| 1712|Ki|continuous,validation,1712,Ki,B,continuous,,100,23,7.34608695652174,0.3365133130053961,0.34407635424336724,6.78,7.140000000000001,7.4,7.58,8.08,,,"{""pchembl"": 23}","{""pChEMBL"": 23}","{""pChEMBL"": 23}" | |
| 1716|Ki|continuous,validation,1716,Ki,B,continuous,,100,21,7.884285714285714,0.2756562978744059,0.28246365126457307,7.13,7.68,7.96,8.07,8.21,,,"{""pchembl"": 21}","{""pChEMBL"": 21}","{""pChEMBL"": 21}" | |
| 1726|Ki|continuous,validation,1726,Ki,B,continuous,,100,27,6.773333333333333,0.7139509268331584,0.7275512141634904,5.72,6.25,6.47,7.34,8.42,,,"{""pchembl"": 27}","{""pChEMBL"": 27}","{""pChEMBL"": 27}" | |
| 1739|Selectivity|continuous,validation,1739,Selectivity,B,continuous,,100,25,133.62,139.30163530985556,142.17413618517259,6.0,26.0,98.0,200.0,556.0,,,"{""standard_value"": 25}","{""raw standard value"": 25}","{"""": 25}" | |
| 1743|IC50|continuous,validation,1743,IC50,B,continuous,,52,15,6.54,0.7965174197718465,0.8244738582011821,5.51,5.93,6.3,7.02,8.14,,,"{""pchembl"": 15}","{""pChEMBL"": 15}","{""pChEMBL"": 15}" | |
| 192|IC50|continuous,validation,192,IC50,F,continuous,,39,13,5.218480370980502,0.6328977765799154,0.6587408913220614,3.8002448227465253,5.14,5.27,5.58,6.18,,,"{""pchembl"": 12, ""standard_value_p_transform"": 1}","{""pChEMBL"": 13}","{""pChEMBL"": 13}" | |
| 207|IC50|continuous,validation,207,IC50,B,continuous,,33,12,4.632499999999999,0.2799739571222057,0.29242326110684774,4.52,4.52,4.52,4.5325,5.52,,,"{""pchembl"": 12}","{""pChEMBL"": 12}","{""pChEMBL"": 12}" | |
| 208|IC50|continuous,validation,208,IC50,B,continuous,,45,14,6.2821428571428575,0.8740887383149263,0.9070847519679445,5.0,5.375,6.475,7.165,7.46,,,"{""pchembl"": 14}","{""pChEMBL"": 14}","{""pChEMBL"": 14}" | |
| 234|IC50|continuous,validation,234,IC50,B,continuous,,22,10,6.6,0.2897240065993843,0.30539591789456966,6.22,6.335,6.59,6.78,7.19,,,"{""pchembl"": 10}","{""pChEMBL"": 10}","{""pChEMBL"": 10}" | |
| 235|IC50|continuous,validation,235,IC50,B,continuous,,45,14,6.453571428571428,0.7971521376827921,0.827243868265228,5.42,5.9624999999999995,6.195,6.7675,8.3,,,"{""pchembl"": 14}","{""pChEMBL"": 14}","{""pChEMBL"": 14}" | |
| 236|Ki|continuous,validation,236,Ki,B,continuous,,22,10,9.045,0.5577320145015884,0.5879011632730266,7.85,8.774999999999999,9.094999999999999,9.4775,9.78,,,"{""pchembl"": 10}","{""pChEMBL"": 10}","{""pChEMBL"": 10}" | |
| 238|Ki|continuous,validation,238,Ki,B,continuous,,60,16,7.828125,0.7671148769089281,0.7922728381056616,6.14,7.3325000000000005,7.869999999999999,8.37,9.24,,,"{""pchembl"": 16}","{""pChEMBL"": 16}","{""pChEMBL"": 16}" | |
| 260|IC50|continuous,validation,260,IC50,B,continuous,,33,12,3.9849864975122125,0.14475048925891557,0.15118695521179465,3.826813731587726,3.8786618011656224,3.9469385629966727,4.039999999999999,4.33,,,"{""pchembl"": 4, ""standard_value_p_transform"": 8}","{""pChEMBL"": 12}","{""pChEMBL"": 12}" | |
| 271|Ki|continuous,validation,271,Ki,B,continuous,,33,12,8.793333333333333,0.5952217140603062,0.6216888045453044,7.78,8.305,8.945,9.3025,9.52,,,"{""pchembl"": 12}","{""pChEMBL"": 12}","{""pChEMBL"": 12}" | |
| 296|Kd|continuous,validation,296,Kd,F,continuous,,100,22,7.838181818181818,0.5044586329885675,0.5163298720745652,7.05,7.34,7.93,8.1125,8.84,,,"{""pchembl"": 22}","{""pChEMBL"": 22}","{""pChEMBL"": 22}" | |
| 330|Ratio|continuous,validation,330,Ratio,B,continuous,,22,10,34.047000000000004,64.0233607443408,67.48654780357671,1.0,2.09,4.41,11.582500000000001,208.0,,,"{""standard_value"": 10}","{""raw standard value"": 10}","{"""": 10}" | |
| 337|Relative IC50|continuous,validation,337,Relative IC50,B,continuous,,33,12,7.767500000000001,9.241623346757503,9.652560776573983,0.25,0.8875,3.95,10.075,31.0,,,"{""standard_value"": 12}","{""raw standard value"": 12}","{"""": 12}" | |
| 339|Relative IC50|continuous,validation,339,Relative IC50,B,continuous,,33,12,10.033333333333333,8.902371718942218,9.298224007678547,0.4,3.1,7.05,15.0,31.0,,,"{""standard_value"": 12}","{""raw standard value"": 12}","{"""": 12}" | |
| 343|Relative ID50|continuous,validation,343,Relative ID50,B,continuous,,22,10,0.5726,0.784059334489425,0.8264711059007985,0.013,0.07750000000000001,0.24,0.505,2.5,,,"{""standard_value"": 10}","{""raw standard value"": 10}","{"""": 10}" | |
| 346|Relative ID50|continuous,validation,346,Relative ID50,B,continuous,,22,10,8.244,13.371455567738314,14.09475174193099,0.07,0.245,1.5,5.925,38.0,,,"{""standard_value"": 10}","{""raw standard value"": 10}","{"""": 10}" | |
| 349|IC50|continuous,validation,349,IC50,B,continuous,,27,11,8.673636363636364,0.6791474967295759,0.7122959037825883,7.5,8.16,8.72,9.114999999999998,9.77,,,"{""pchembl"": 11}","{""pChEMBL"": 11}","{""pChEMBL"": 11}" | |
| 371|IC50|continuous,validation,371,IC50,B,continuous,,100,29,4.973158060190569,0.8806204346943591,0.8962078471863939,3.714442690992226,4.05,5.03,5.94,6.08,,,"{""pchembl"": 23, ""standard_value_p_transform"": 6}","{""pChEMBL"": 29}","{""pChEMBL"": 29}" | |
| 37|Kd|continuous,validation,37,Kd,B,continuous,,100,25,4.312971534347746,0.48689209116683113,0.49693215964808535,2.799423073245152,4.24,4.41,4.6,4.96,,,"{""pchembl"": 20, ""standard_value_p_transform"": 5}","{""pChEMBL"": 25}","{""pChEMBL"": 25}" | |
| 381|k obs / 1|continuous,validation,381,k obs / 1,F,continuous,,27,11,105920.0,165235.14704257634,173300.0842469501,100.0,19910.0,59300.0,101900.0,610000.0,,,"{""standard_value"": 11}","{""raw standard value"": 11}","{""M-1 s-1"": 11}" | |
| 393|Ki|continuous,validation,393,Ki,B,continuous,,52,15,6.3566666666666665,1.6661919323882093,1.7246725016927817,4.23,4.9399999999999995,5.92,8.11,8.52,,,"{""pchembl"": 15}","{""pChEMBL"": 15}","{""pChEMBL"": 15}" | |
| 42|Kd|continuous,validation,42,Kd,B,continuous,,100,35,3.5901982009740583,0.2894005829622138,0.29362563247924384,3.0390538042661683,3.360022875122684,3.614393726401688,3.7790268136984744,4.22,,,"{""pchembl"": 2, ""standard_value_p_transform"": 33}","{""pChEMBL"": 35}","{""pChEMBL"": 35}" | |
| 437|Activity|continuous,validation,437,Activity,F,continuous,,100,28,6.570857142857142e-08,1.1670462656743689e-07,1.1884617448818532e-07,1.6e-10,7.825e-10,1.15e-08,4.5500000000000004e-08,4.3e-07,,,"{""standard_value"": 28}","{""raw standard value"": 28}","{"""": 28}" | |
| 447|IC50|continuous,validation,447,IC50,F,continuous,,33,12,4.963333333333334,0.36533850361304954,0.3815836220359315,4.48,4.71,4.795,5.25,5.62,,,"{""pchembl"": 12}","{""pChEMBL"": 12}","{""pChEMBL"": 12}" | |
| 450|IC50|continuous,validation,450,IC50,F,continuous,,33,12,5.004166666666666,0.30820605481109914,0.3219107254372168,4.5,4.797499999999999,4.92,5.26,5.55,,,"{""pchembl"": 12}","{""pChEMBL"": 12}","{""pChEMBL"": 12}" | |
| 458|IC50|continuous,validation,458,IC50,F,continuous,,100,28,8.954285714285714,0.9016232526925637,0.9181681786213267,6.85,8.2225,8.969999999999999,9.665,10.42,,,"{""pchembl"": 28}","{""pChEMBL"": 28}","{""pChEMBL"": 28}" | |
| 461|IC50|continuous,validation,461,IC50,F,continuous,,76,18,9.511271041404463,1.3886314558539845,1.4288899797800434,7.22,8.64,9.26,10.225000000000001,12.0,,,"{""pchembl"": 15, ""standard_value_p_transform"": 3}","{""pChEMBL"": 18}","{""pChEMBL"": 18}" | |
| 502|Basal uptake|continuous,validation,502,Basal uptake,F,continuous,,76,18,113.02777777777777,36.951346473069684,38.02262183545251,82.0,95.0,102.5,113.0,251.0,,,"{""standard_value"": 18}","{""raw standard value"": 18}","{""%"": 18}" | |
| 506|Basal uptake|continuous,validation,506,Basal uptake,F,continuous,,76,18,132.91666666666666,44.08900404610857,45.3672108854998,80.0,102.25,120.0,157.0,255.0,,,"{""standard_value"": 18}","{""raw standard value"": 18}","{""%"": 18}" | |
| 508|Basal uptake|continuous,validation,508,Basal uptake,F,continuous,,39,13,117.46153846153847,46.506600664050296,48.40560467655129,66.0,89.0,108.0,120.0,214.0,,,"{""standard_value"": 13}","{""raw standard value"": 13}","{""%"": 13}" | |
| 517|IC50|continuous,validation,517,IC50,F,continuous,,100,60,7.240666666666667,0.7315892897581873,0.7377631484947159,5.9,6.7275,7.1899999999999995,7.67,9.7,,,"{""pchembl"": 60}","{""pChEMBL"": 60}","{""pChEMBL"": 60}" | |
| 520|Activity|continuous,validation,520,Activity,F,continuous,,22,10,57.5,44.075503400415066,46.459659921269335,4.0,10.5,66.0,93.0,121.0,,,"{""standard_value"": 10}","{""raw standard value"": 10}","{""%"": 10}" | |
| 522|EC|continuous,validation,522,EC,F,continuous,,95,20,1.22005,1.9843530047599898,2.035903225778878,0.067,0.08025,0.365,1.1400000000000001,8.18,,,"{""standard_value"": 20}","{""raw standard value"": 20}","{""uM"": 20}" | |
| 524|EC50|continuous,validation,524,EC50,F,continuous,,39,13,7.594615384615385,1.148052634712802,1.194931067639576,6.4,6.64,7.09,8.85,9.68,,,"{""pchembl"": 13}","{""pChEMBL"": 13}","{""pChEMBL"": 13}" | |
| 526|Glucose transport|continuous,validation,526,Glucose transport,F,continuous,,100,26,246.0,191.88097272087114,195.68096483817735,100.0,129.75,198.5,243.0,868.0,,,"{""standard_value"": 26}","{""raw standard value"": 26}","{""%"": 26}" | |
| 527|Glucose transport|continuous,validation,527,Glucose transport,F,continuous,,100,26,178.03846153846155,130.88441194405402,133.47643410556958,63.0,109.75,126.5,164.75,611.0,,,"{""standard_value"": 26}","{""raw standard value"": 26}","{""%"": 26}" | |
| 528|Glucose transport|continuous,validation,528,Glucose transport,F,continuous,,100,26,156.1323076923077,167.61552299390624,170.9349645053976,0.1,3.9749999999999996,113.0,287.75,543.0,,,"{""standard_value"": 26}","{""raw standard value"": 26}","{""%"": 26}" | |
| 534|IC50|continuous,validation,534,IC50,F,continuous,,52,15,6.516666666666667,0.5029998895515673,0.520654350198817,5.55,6.1899999999999995,6.41,6.875,7.39,,,"{""pchembl"": 15}","{""pChEMBL"": 15}","{""pChEMBL"": 15}" | |
| 535|Ki|continuous,validation,535,Ki,B,continuous,,100,54,7.093703703703704,1.0245799433702834,1.0342006233898653,4.47,6.3475,7.215,7.9425,8.92,,,"{""pchembl"": 54}","{""pChEMBL"": 54}","{""pChEMBL"": 54}" | |
| 536|Ki|continuous,validation,536,Ki,B,continuous,,60,16,6.2584375,0.6672043323403632,0.6890856713791108,5.05,5.82,6.105,6.6362499999999995,8.11,,,"{""pchembl"": 16}","{""pChEMBL"": 16}","{""pChEMBL"": 16}" | |
| 541|IC50|continuous,validation,541,IC50,B,continuous,,39,13,6.102307692307692,0.8401662275650149,0.8744727349109086,4.52,5.43,6.3,6.6,7.3,,,"{""pchembl"": 13}","{""pChEMBL"": 13}","{""pChEMBL"": 13}" | |
| 542|IC50|continuous,validation,542,IC50,B,continuous,,39,13,6.106153846153846,0.8457362605949961,0.880270209098116,4.52,5.43,6.3,6.6,7.35,,,"{""pchembl"": 13}","{""pChEMBL"": 13}","{""pChEMBL"": 13}" | |
| 547|IC50|continuous,validation,547,IC50,B,continuous,,27,11,5.274391133395091,0.9497226269023497,0.996077494402584,3.4383024673460065,4.84,5.22,6.1850000000000005,6.6,,,"{""pchembl"": 10, ""standard_value_p_transform"": 1}","{""pChEMBL"": 11}","{""pChEMBL"": 11}" | |
| 559|IC50|continuous,validation,559,IC50,B,continuous,,100,21,4.9695238095238095,0.8859456942965694,0.907824191077084,4.01,4.26,4.89,5.27,7.19,,,"{""pchembl"": 21}","{""pChEMBL"": 21}","{""pChEMBL"": 21}" | |
| 560|IC50|continuous,validation,560,IC50,B,continuous,,100,34,5.450000000455981,1.2094359397755412,1.2276239669834914,3.33999999963408,4.4925,5.16,6.57,7.28,,,"{""pchembl"": 29, ""standard_value_p_transform"": 5}","{""pChEMBL"": 34}","{""pChEMBL"": 34}" | |
| 561|IC50|continuous,validation,561,IC50,B,continuous,,39,13,8.611538461538462,1.1669081181537033,1.2145564770307866,5.52,8.52,9.0,9.52,9.7,,,"{""pchembl"": 13}","{""pChEMBL"": 13}","{""pChEMBL"": 13}" | |
| 575|Ki|continuous,validation,575,Ki,B,continuous,,85,19,7.05157894736842,0.7288149224156528,0.748786152218633,5.35,6.765,7.02,7.4350000000000005,8.62,,,"{""pchembl"": 19}","{""pChEMBL"": 19}","{""pChEMBL"": 19}" | |
| 581|Ki|continuous,validation,581,Ki,B,continuous,,100,24,7.7175,0.827749207187781,0.8455523021387701,6.42,6.98,7.765000000000001,8.3125,9.52,,,"{""pchembl"": 24}","{""pChEMBL"": 24}","{""pChEMBL"": 24}" | |
| 588|Ki|continuous,validation,588,Ki,B,continuous,,52,15,7.542666666666666,0.7098682193822236,0.7347834148010327,6.19,6.895,7.96,8.094999999999999,8.39,,,"{""pchembl"": 15}","{""pChEMBL"": 15}","{""pChEMBL"": 15}" | |
| 589|Ki|continuous,validation,589,Ki,B,continuous,,100,25,7.2104,1.2487801407773909,1.27453089409398,6.0,6.33,6.84,7.8,10.0,,,"{""pchembl"": 25}","{""pChEMBL"": 25}","{""pChEMBL"": 25}" | |
| 654|Emax|continuous,validation,654,Emax,F,continuous,,33,12,9.5,2.9011491975882016,3.0301515113634467,4.0,8.0,9.0,12.0,15.0,,,"{""standard_value"": 12}","{""raw standard value"": 12}","{""%"": 12}" | |
| 659|Emax|continuous,validation,659,Emax,F,continuous,,45,14,12.090714285714286,2.129119416518462,2.2094916376178695,7.47,11.282499999999999,12.175,13.075,16.99,,,"{""standard_value"": 14}","{""raw standard value"": 14}","{""%"": 14}" | |
| 662|Emax|continuous,validation,662,Emax,F,continuous,,76,18,6.399444444444445,2.9303725061314916,3.0153284324523515,1.8,3.4299999999999997,6.85,7.845,12.75,,,"{""standard_value"": 18}","{""raw standard value"": 18}","{""%"": 18}" | |
| 666|Emin|continuous,validation,666,Emin,F,continuous,,33,12,6.734999999999999,2.9468896031805016,3.07792580689127,1.43,4.6049999999999995,7.565,8.3425,10.83,,,"{""standard_value"": 12}","{""raw standard value"": 12}","{""%"": 12}" | |
| 669|FSC recovery|continuous,validation,669,FSC recovery,F,continuous,,100,25,35.32,28.817661251392348,29.411902352619084,-15.0,12.0,33.0,52.0,111.0,,,"{""standard_value"": 25}","{""raw standard value"": 25}","{""%"": 25}" | |
| 690|IC50|continuous,validation,690,IC50,B,continuous,,68,17,6.89764705882353,0.7038008526127318,0.7254613136805151,5.84,6.34,7.0,7.2,8.4,,,"{""pchembl"": 17}","{""pChEMBL"": 17}","{""pChEMBL"": 17}" | |
| 72|ED50|continuous,validation,72,ED50,F,continuous,,22,10,1.612,2.43608620537123,2.5678603284966,0.07,0.7,0.79,0.915,8.8,,,"{""standard_value"": 10}","{""raw standard value"": 10}","{""ug ml-1"": 10}" | |
| 732|Inhibition|continuous,validation,732,Inhibition,F,continuous,,27,11,33.06363636363636,9.041648354071159,9.482960795792918,18.9,27.1,32.9,41.75,46.2,,,"{""standard_value"": 11}","{""raw standard value"": 11}","{""%"": 11}" | |
| 733|IC50|continuous,validation,733,IC50,B,continuous,,100,32,6.575,0.4333661846521946,0.4403004839073338,5.82,6.2524999999999995,6.62,6.94,7.24,,,"{""pchembl"": 32}","{""pChEMBL"": 32}","{""pChEMBL"": 32}" | |
| 734|IC50|continuous,validation,734,IC50,B,continuous,,76,18,6.414444444444444,0.39877900064825966,0.4103402063743209,5.29,6.285,6.525,6.705,6.92,,,"{""pchembl"": 18}","{""pChEMBL"": 18}","{""pChEMBL"": 18}" | |
| 736|IC50|continuous,validation,736,IC50,B,continuous,,45,14,5.5042857142857144,0.41692264246010724,0.4326610733537331,4.68,5.362499999999999,5.605,5.842499999999999,6.0,,,"{""pchembl"": 14}","{""pChEMBL"": 14}","{""pChEMBL"": 14}" | |
| 757|IC50|continuous,validation,757,IC50,B,continuous,,76,18,6.309444444444444,0.981373596446567,1.00982509972081,5.18,5.494999999999999,5.92,6.822500000000001,8.64,,,"{""pchembl"": 18}","{""pChEMBL"": 18}","{""pChEMBL"": 18}" | |
| 801|Ki|continuous,validation,801,Ki,B,continuous,,45,14,6.807857142857143,0.4143700653044428,0.4300121388524277,6.0,6.59,6.84,7.1125,7.38,,,"{""pchembl"": 14}","{""pChEMBL"": 14}","{""pChEMBL"": 14}" | |
| 802|IC50|continuous,validation,802,IC50,B,continuous,,100,57,5.887719298245615,0.45501886424692345,0.45906355591674597,5.0,5.6,6.0,6.2,6.7,,,"{""pchembl"": 57}","{""pChEMBL"": 57}","{""pChEMBL"": 57}" | |
| 80|IC50|continuous,validation,80,IC50,B,continuous,,27,11,8.110909090909091,0.19080949783176393,0.20012268964085736,7.71,8.0,8.11,8.23,8.39,,,"{""pchembl"": 11}","{""pChEMBL"": 11}","{""pChEMBL"": 11}" | |
| 815|Efficacy|continuous,validation,815,Efficacy,F,continuous,,68,17,83.23529411764706,29.336845758041914,30.239728445715055,20.0,62.0,82.0,103.0,128.0,,,"{""standard_value"": 17}","{""raw standard value"": 17}","{""%"": 17}" | |
| 826|IC50|continuous,validation,826,IC50,B,continuous,,45,14,7.685714285714285,0.5794543527654059,0.601328200233121,6.72,7.255,7.78,8.127500000000001,8.44,,,"{""pchembl"": 14}","{""pChEMBL"": 14}","{""pChEMBL"": 14}" | |
| 827|IC50|continuous,validation,827,IC50,B,continuous,,45,14,7.026428571428572,0.7163060712817545,0.7433459402009179,5.28,6.6450000000000005,6.98,7.3025,8.11,,,"{""pchembl"": 14}","{""pChEMBL"": 14}","{""pChEMBL"": 14}" | |
| 829|IC50|continuous,validation,829,IC50,B,continuous,,100,21,7.176666666666667,0.3285369202030541,0.33665016461206926,6.57,6.92,7.21,7.49,7.7,,,"{""pchembl"": 21}","{""pChEMBL"": 21}","{""pChEMBL"": 21}" | |
| 831|IC50|continuous,validation,831,IC50,B,continuous,,100,35,7.118571428571428,0.899965532219803,0.9131044101665188,5.04,6.485,7.21,7.9399999999999995,8.7,,,"{""pchembl"": 35}","{""pChEMBL"": 35}","{""pChEMBL"": 35}" | |
| 835|IC50|continuous,validation,835,IC50,B,continuous,,100,30,8.086,1.0974929005085485,1.1162548219766877,4.7,7.430000000000001,8.4,9.0,9.52,,,"{""pchembl"": 30}","{""pChEMBL"": 30}","{""pChEMBL"": 30}" | |
| 842|IC50|continuous,validation,842,IC50,B,continuous,,100,21,6.796190476190477,0.5724922639566838,0.5866300042656887,6.03,6.24,6.68,7.11,7.85,,,"{""pchembl"": 21}","{""pChEMBL"": 21}","{""pChEMBL"": 21}" | |
| 843|IC50|continuous,validation,843,IC50,B,continuous,,39,13,6.817692307692307,0.49926336269091864,0.5196497834464068,6.16,6.43,6.63,7.24,7.77,,,"{""pchembl"": 13}","{""pChEMBL"": 13}","{""pChEMBL"": 13}" | |
| 844|IC50|continuous,validation,844,IC50,B,continuous,,45,14,6.491428571428571,0.7997129587086422,0.8299013578349319,5.16,5.7475000000000005,6.545,7.205,7.52,,,"{""pchembl"": 14}","{""pChEMBL"": 14}","{""pChEMBL"": 14}" | |
| 845|IC50|continuous,validation,845,IC50,B,continuous,,68,17,7.481764705882353,0.8430702663766779,0.8690169395221651,6.0,6.85,7.4,7.89,9.12,,,"{""pchembl"": 17}","{""pChEMBL"": 17}","{""pChEMBL"": 17}" | |
| 846|IC50|continuous,validation,846,IC50,B,continuous,,45,14,8.078571428571427,0.6486013208970421,0.6730854002605882,6.5,8.0,8.15,8.5575,8.89,,,"{""pchembl"": 14}","{""pChEMBL"": 14}","{""pChEMBL"": 14}" | |
| 857|IC50|continuous,validation,857,IC50,B,continuous,,68,17,6.446470588235294,0.5860831217545309,0.6041206540964167,5.07,6.09,6.59,6.77,7.29,,,"{""pchembl"": 17}","{""pChEMBL"": 17}","{""pChEMBL"": 17}" | |
| 858|IC50|continuous,validation,858,IC50,B,continuous,,100,23,8.075652173913044,0.7971134122949454,0.8150283100880971,6.83,7.32,8.06,8.77,9.41,,,"{""pchembl"": 23}","{""pChEMBL"": 23}","{""pChEMBL"": 23}" | |
| 862|IC50|continuous,validation,862,IC50,B,continuous,,100,38,7.871315789473685,0.6569433647488454,0.66576179106844,6.27,7.4425,8.015,8.355,9.15,,,"{""pchembl"": 38}","{""pChEMBL"": 38}","{""pChEMBL"": 38}" | |
| 863|IC50|continuous,validation,863,IC50,B,continuous,,100,24,7.11625,1.0553862345921834,1.078085309603377,5.7,6.3,6.83,7.7524999999999995,9.3,,,"{""pchembl"": 24}","{""pChEMBL"": 24}","{""pChEMBL"": 24}" | |
| 894|Ki|continuous,validation,894,Ki,B,continuous,,60,16,7.44125,0.57130196700169,0.5900381343608226,6.54,7.1675,7.43,7.897499999999999,8.48,,,"{""pchembl"": 16}","{""pChEMBL"": 16}","{""pChEMBL"": 16}" | |
| 8|CC50|continuous,validation,8,CC50,F,continuous,,22,10,6.115853543937424,0.5151278172025855,0.5429923961570122,5.443697499232712,5.625569708000178,6.197239738281265,6.279899052318158,7.154901959985743,,,"{""standard_value_p_transform"": 10}","{""pChEMBL"": 10}","{""pChEMBL"": 10}" | |
| 922|Ki|continuous,validation,922,Ki,B,continuous,,39,13,8.596923076923076,0.33349857837050517,0.34711632573208606,7.96,8.35,8.73,8.86,9.04,,,"{""pchembl"": 13}","{""pChEMBL"": 13}","{""pChEMBL"": 13}" | |
| 924|Ki|continuous,validation,924,Ki,B,continuous,,100,55,7.436909090909092,0.9092991761436592,0.9176799908773023,5.63,6.654999999999999,7.28,8.059999999999999,9.47,,,"{""pchembl"": 55}","{""pChEMBL"": 55}","{""pChEMBL"": 55}" | |
| 929|Ki|continuous,validation,929,Ki,B,continuous,,45,14,7.541428571428571,0.763187461925847,0.7919970584915959,6.0,6.955000000000001,7.734999999999999,7.947500000000001,8.86,,,"{""pchembl"": 14}","{""pChEMBL"": 14}","{""pChEMBL"": 14}" | |
| 949|Ki|continuous,validation,949,Ki,B,continuous,,100,24,7.047916666666667,0.6929765458192328,0.7078809723495133,5.7,6.640000000000001,7.005,7.405000000000001,8.7,,,"{""pchembl"": 24}","{""pChEMBL"": 24}","{""pChEMBL"": 24}" | |
| 94|Concentration|continuous,validation,94,Concentration,B,continuous,,22,10,3.3174000000000006e-06,5.742876826121209e-06,6.053523697447261e-06,1e-09,2.95e-07,9.5e-07,3.3e-06,2e-05,,,"{""standard_value"": 10}","{""raw standard value"": 10}","{"""": 10}" | |
| 961|Ki|continuous,validation,961,Ki,B,continuous,,26,17,7.473529411764706,0.5136139678381785,0.5294211600473505,6.22,7.16,7.39,7.82,8.29,,,"{""pchembl"": 17}","{""pChEMBL"": 17}","{""pChEMBL"": 17}" | |
| 987|Inhibition|continuous,validation,987,Inhibition,B,continuous,,95,20,32.845,53.37252546957095,54.75905572789332,0.0,0.0,14.5,42.25,242.9,,,"{""standard_value"": 20}","{""raw standard value"": 20}","{""%"": 20}" | |