smiles
stringlengths
4
580
activity
stringclasses
3 values
HIV_active
int64
0
1
CC1=C(C(=O)Nc2ccc([N+](=O)[O-])cc2)C(c2ccccc2O)C(C(=O)Nc2ccc([N+](=O)[O-])cc2)=C(C)N1
CI
0
CC1=C(C(=O)Nc2ccc([N+](=O)[O-])cc2)C(c2ccccc2F)C(C(=O)Nc2ccc([N+](=O)[O-])cc2)=C(C)N1
CI
0
CCc1ccccc1NC(=O)C1=C(C)NC(C)=C(C(=O)Nc2ccccc2CC)C1c1ccccc1Cl
CI
0
CCc1ccccc1NC(=O)C1=C(C)NC(C)=C(C(=O)Nc2ccccc2CC)C1c1ccc(NC(C)=O)cc1
CI
0
CC1=C(C(=O)Nc2cccc(Cl)c2)C(c2ccc([N+](=O)[O-])cc2)C(C(=O)Nc2cccc(Cl)c2)=C(C)N1
CI
0
CCOc1ccc(NC(=O)C2=C(C)NC(C)=C(C(=O)Nc3ccc(OCC)cc3)C2c2ccc(O)c(OC)c2)cc1
CI
0
CC1=C(C(=O)Nc2ccc([N+](=O)[O-])cc2)C(c2cccc([N+](=O)[O-])c2)C(C(=O)Nc2ccc([N+](=O)[O-])cc2)=C(C)N1
CI
0
CC1=C(C(=O)Nc2ccccc2C)C(c2ccccc2)C(C(=O)Nc2ccccc2C)=C(C)N1
CI
0
CC1=C(C(=O)Nc2ccc([N+](=O)[O-])cc2)C(c2ccc(N(C)C)cc2)C(C(=O)Nc2ccc([N+](=O)[O-])cc2)=C(C)N1
CI
0
CCOc1ccc(NC(=O)C2=C(C)NC(C)=C(C(=O)Nc3ccc(OCC)cc3)C2c2ccc([N+](=O)[O-])cc2)cc1
CI
0
CCc1ccccc1NC(=O)C1=C(C)NC(C)=C(C(=O)Nc2ccccc2CC)C1c1cccc([N+](=O)[O-])c1
CI
0
CCOc1ccccc1NC(=O)C1=C(C)NC(C)=C(C(=O)Nc2ccccc2OCC)C1c1ccc(NC(C)=O)cc1
CI
0
COc1cc(C2C(C(=O)Nc3ccc(Cl)c(Cl)c3)=C(C)NC(C)=C2C(=O)Nc2ccc(Cl)c(Cl)c2)ccc1O
CI
0
COc1cc(C2C(C(=O)Nc3cc(F)c(F)cc3F)=C(C)NC(C)=C2C(=O)Nc2cc(F)c(F)cc2F)ccc1O
CI
0
CC1=C(C(=O)Nc2ccc(C)cc2)C(c2cccc([N+](=O)[O-])c2)C(C(=O)Nc2ccc(C)cc2)=C(C)N1
CI
0
Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1
CI
0
Nc1ccc(S(=O)(=O)Nc2ccc(S(=O)(=O)O)cc2)cc1
CI
0
CC(=O)Nc1ccc(S(=O)(=O)Nc2ccc([N+](=O)[O-])cc2)cc1
CI
0
Cc1ccc(S(=O)(=O)N(CCC(=O)O)c2ccccc2)cc1
CI
0
O=S(=O)(Nc1cccc(F)c1)c1ccc(F)cc1
CI
0
COc1ccc(S(=O)(=O)O)cc1NS(=O)(=O)c1ccc(C)cc1.[NaH]
CI
0
COc1cc([N+](=O)[O-])c(S(=O)(=O)O)cc1NS(=O)(=O)c1ccc(C)cc1.[NaH]
CI
0
Cc1ccc(S(=O)(=O)Nc2cccc(C)c2C)cc1
CI
0
O=C(O)c1ccccc1NS(=O)(=O)c1ccc(Cl)cc1
CI
0
O=C(O)c1ccccc1NS(=O)(=O)c1ccc([N+](=O)[O-])cc1
CI
0
Nc1ccccc1S(=O)(=O)N(CC(=O)O)c1ccccc1
CI
0
Nc1cccc(S(=O)(=O)N(CC(=O)O)c2ccccc2)c1
CI
0
COc1ccc(S(=O)(=O)N(CC(=O)O)c2ccccc2)cc1
CI
0
Cc1ccc(S(=O)(=O)N(CC(=O)O)c2ccccc2)cc1
CI
0
O=C(O)CN(c1ccccc1)S(=O)(=O)c1ccccc1[N+](=O)[O-]
CI
0
O=C(O)CN(c1ccccc1)S(=O)(=O)c1cccc([N+](=O)[O-])c1
CI
0
O=C(O)CN(c1ccccc1)S(=O)(=O)c1ccc([N+](=O)[O-])cc1
CI
0
COc1ccc(N(CC(=O)O)S(=O)(=O)c2ccccc2)cc1
CI
0
Cc1ccccc1N(CC(=O)O)S(=O)(=O)c1ccccc1
CI
0
Cc1cccc(N(CC(=O)O)S(=O)(=O)c2ccccc2)c1
CI
0
Cc1ccc(N(CC(=O)O)S(=O)(=O)c2ccccc2)cc1
CI
0
O=C(O)CN(c1ccccc1Cl)S(=O)(=O)c1ccccc1
CI
0
O=C(O)CN(c1cccc(Cl)c1)S(=O)(=O)c1ccccc1
CI
0
O=C(O)CN(c1ccc(Cl)cc1)S(=O)(=O)c1ccccc1
CI
0
O=C(O)CN(c1ccc(F)cc1)S(=O)(=O)c1ccccc1
CI
0
O=C(O)CN(c1ccccc1)S(=O)(=O)c1ccc(Cl)cc1
CI
0
COc1ccc(S(=O)(=O)Nc2ccccc2C(=O)O)cc1
CI
0
CCc1cccc(C)c1NS(=O)(=O)c1ccccc1
CI
0
Cc1ccc(S(=O)(=O)Nc2ccccc2C(C)(C)C)cc1
CI
0
CC(C)(C)c1ccccc1NS(=O)(=O)c1ccccc1
CI
0
O=[N+]([O-])c1ccccc1S(=O)(=O)Nc1ccccc1
CI
0
Cc1cc(N(CCC#N)S(=O)(=O)c2ccccc2)ccc1C=O
CI
0
N#CCCN(c1ccc(C=O)cc1)S(=O)(=O)c1ccccc1
CI
0
CN(c1ccccc1)S(=O)(=O)c1ccccc1[N+](=O)[O-]
CI
0
CN(c1ccccc1)S(=O)(=O)c1ccc([N+](=O)[O-])cc1
CI
0
Cc1ccc(N(C)S(=O)(=O)c2ccccc2[N+](=O)[O-])cc1
CM
1
Cc1ccc(N(C)S(=O)(=O)c2ccc([N+](=O)[O-])cc2)cc1
CI
0
CN(c1ccc(Cl)cc1)S(=O)(=O)c1ccccc1[N+](=O)[O-]
CI
0
CN(c1ccc(Cl)cc1)S(=O)(=O)c1cccc([N+](=O)[O-])c1
CI
0
CN(c1ccc(Cl)cc1)S(=O)(=O)c1ccc([N+](=O)[O-])cc1
CI
0
CN(c1c(Cl)cccc1Cl)S(=O)(=O)c1ccccc1[N+](=O)[O-]
CI
0
CN(c1ccccc1Cl)S(=O)(=O)c1ccccc1[N+](=O)[O-]
CM
1
CN(c1ccccc1Cl)S(=O)(=O)c1ccc([N+](=O)[O-])cc1
CI
0
Cc1ccccc1N(C)S(=O)(=O)c1ccccc1[N+](=O)[O-]
CI
0
COc1ccc(N(C)S(=O)(=O)c2ccccc2)cc1
CI
0
CN(c1ccc(Cl)cc1)S(=O)(=O)c1ccccc1
CI
0
Cc1ccc(N(C)S(=O)(=O)c2ccccc2)cc1
CI
0
CN(c1ccccc1Cl)S(=O)(=O)c1ccccc1
CI
0
COc1ccc(S(=O)(=O)N(C)c2ccccc2)cc1
CI
0
CN(c1ccccc1)S(=O)(=O)c1ccc(Cl)cc1
CI
0
Cc1ccc(S(=O)(=O)N(C)c2ccccc2)cc1
CI
0
CN(c1ccccc1)S(=O)(=O)c1cccc([N+](=O)[O-])c1
CM
1
Cc1cccc(N(CCC#N)S(=O)(=O)c2ccccc2)c1
CI
0
O=S(=O)(Nc1ccccc1Cl)c1ccccc1
CI
0
CSC(=NN=C(C)c1ccc(S(=O)(=O)N(C)c2ccccc2)cc1)SC
CI
0
CSC(=S)NN=C(C)c1ccc(S(=O)(=O)N(C)c2ccccc2)cc1
CI
0
CCCNC(=S)NN=C(C)c1ccc(S(=O)(=O)N(C)c2ccccc2)cc1
CI
0
OCC12C3C4C5C3C1C5C42
CI
0
COC(=O)C12C3C4C1C1C2C3C41C(=O)O
CI
0
COC(=O)C12C3C4C1C1C2C3C41I
CI
0
CC(C)N(C(=O)C12C3C4C1C1C4(C#N)C3C12C#N)C(C)C
CI
0
OCC12C3C4C1C1C2C3C41CO
CI
0
O=C(O)CC12C3C4C5C3C1C5C42
CI
0
CC(C)N(C(=O)C12C3C4C5C3C1(C(=O)O)C5C42)C(C)C
CI
0
O=C(O)C12C3C4C1C1C2C3C41I
CI
0
CC(C)N(C(=O)C12C3C4C1C1C2C3C41I)C(C)C
CI
0
CN(C(=O)C12C3C4C1C1C4(C#N)C3C12C(=O)O)C(C)(C)C
CI
0
CN(C(=O)C12C3C4C1(C(=O)O)C1C2C3(C(=O)O)C41C(=O)N(C)C(C)(C)C)C(C)(C)C
CI
0
CN(C(=O)C12C3C4C1C1C2C3C41C(N)=O)C(C)(C)C
CI
0
CC(C)N(C(=O)C12C3C4C1C1C2C3C41C(=O)N(C(C)C)C(C)C)C(C)C
CI
0
CC(C)N(C(=O)C12C3C4C1(I)C1C2C3(I)C41C(=O)N(C(C)C)C(C)C)C(C)C
CI
0
CN(C(=O)C12C3C4C1C1C2C3C41C(=O)N(C)C(C)(C)C)C(C)(C)C
CI
0
CN(C(=O)C12C3(C(=O)C(C)(C)C)C4C5(C#N)C3C1(C(=O)C(C)(C)C)C5C42C(=O)C(C)(C)C)C(C)(C)C
CI
0
CN(C(=O)C12C3C4C1C1C2C3C41C#N)C(C)(C)C
CI
0
CN(C(=O)C12C3C4C1C1C2C3C41C(O)C(C)(C)C)C(C)(C)C
CI
0
CC(C)N(C(=O)C12C3C4C1C1C2C3C41C(O)C(C)(C)C)C(C)C
CI
0
CN(C(=O)C12C3C4C1C1C2C3C41C(=O)C(C)(C)C)C(C)(C)C
CI
0
CC(C)N(C(=O)C12C3C4C1C1C2C3C41C(=O)C(C)(C)C)C(C)C
CI
0
CC(C)N(C(=O)C12C3C4C1C1C2C3C41C(=O)O)C(C)C
CI
0
CC(C)N(C(=O)C12C3C4C1C1C2C3C41C(N)=O)C(C)C
CI
0
COC(=O)C12C3C4C1C1C2C3C41C(=O)N(C(C)C)C(C)C
CI
0
CC(C)N(C(=O)C12C3C4C5(C#N)C3C1(I)C5C42I)C(C)C
CI
0
CC(C)N(C(=O)C12C3C4C5(C#N)C3C1(C#N)C5C42C#N)C(C)C
CI
0
CC(C)N(C(=O)C12C3C4C5(C(=O)O)C(C1C35I)C42C(=O)O)C(C)C
CI
0
CC(C)N(C(=O)C12C3C4C5(C#N)C3C1(C#N)C5C42I)C(C)C
CI
0