smiles
stringlengths
1
1.34k
Hepatobiliary disorders
int64
0
1
Metabolism and nutrition disorders
int64
0
1
Product issues
int64
0
1
Eye disorders
int64
0
1
Investigations
int64
0
1
Musculoskeletal and connective tissue disorders
int64
0
1
Gastrointestinal disorders
int64
0
1
Social circumstances
int64
0
1
Immune system disorders
int64
0
1
Reproductive system and breast disorders
int64
0
1
Neoplasms benign, malignant and unspecified (incl cysts and polyps)
int64
0
1
General disorders and administration site conditions
int64
0
1
Endocrine disorders
int64
0
1
Surgical and medical procedures
int64
0
1
Vascular disorders
int64
0
1
Blood and lymphatic system disorders
int64
0
1
Skin and subcutaneous tissue disorders
int64
0
1
Congenital, familial and genetic disorders
int64
0
1
Infections and infestations
int64
0
1
Respiratory, thoracic and mediastinal disorders
int64
0
1
Psychiatric disorders
int64
0
1
Renal and urinary disorders
int64
0
1
Pregnancy, puerperium and perinatal conditions
int64
0
1
Ear and labyrinth disorders
int64
0
1
Cardiac disorders
int64
0
1
Nervous system disorders
int64
0
1
Injury, poisoning and procedural complications
int64
0
1
CC1C(C(CC(O1)OC2CC(CC3=C(C4=C(C(=C23)O)C(=O)C5=C(C4=O)C=CC=C5OC)O)(C(=O)C)O)N)O
1
0
1
1
1
1
1
1
1
1
1
0
0
1
1
1
0
1
1
1
1
0
1
1
1
1
1
CC1C(C(CC(O1)OC2CC(CC3=C(C4=C(C(=C23)O)C(=O)C5=CC=CC=C5C4=O)O)(C(=O)C)O)N)O
1
0
0
1
0
1
0
1
1
1
1
0
0
1
1
1
1
1
0
0
1
0
0
1
1
1
1
C1=CC=C(C=C1)C(=C(C2=CC=CC=C2)C3=CC=C(C=C3)OCCO)CCCl
0
0
0
0
1
0
0
0
1
1
0
0
0
1
0
1
0
0
0
0
0
0
0
1
1
0
0
CCN(CC)CCOC1=CC=C(C=C1)C(=C(C2=CC=CC=C2)Cl)C3=CC=CC=C3
1
0
1
1
1
1
1
1
1
1
1
1
0
1
1
1
1
1
1
1
1
1
1
1
1
1
1
CCC(=C(C1=CC=CC=C1)C2=CC=C(C=C2)OCCN(C)C)C3=CC=CC=C3
1
0
1
1
1
1
1
1
1
1
1
1
0
1
1
1
1
1
1
1
1
0
0
1
1
1
1
CN(C)CCOC1=CC=C(C=C1)C(=C(CCCl)C2=CC=CC=C2)C3=CC=CC=C3
1
0
1
1
1
1
0
0
1
1
1
1
0
1
1
1
0
0
1
1
0
0
1
1
1
0
1
C1=CN(C(=O)N=C1N)C2C(C(C(O2)CO)O)O
1
0
1
1
1
1
0
1
0
1
1
0
0
1
1
1
0
1
1
1
1
0
1
1
1
1
1
C1=CN(C(=O)N=C1N)C2C(C(C(O2)CO)O)(F)F
1
0
0
1
1
1
0
1
1
1
1
0
0
1
1
1
0
1
1
1
1
0
1
1
1
1
1
CCCCCOC(=O)NC1=NC(=O)N(C=C1F)[C@H]2[C@@H]([C@@H]([C@H](O2)C)O)O
1
0
1
1
1
1
1
1
1
1
1
1
0
1
1
1
1
1
1
1
1
0
1
1
1
1
1
C1CC(OC1CO)N2C=CC(=NC2=O)N
1
0
1
1
1
1
1
1
1
0
1
0
0
1
1
1
1
1
1
1
1
0
1
1
1
1
1
CCCCCC(C=CC1C(CC(=O)C1CC=CCCCC(=O)O)O)O
1
0
1
1
1
1
0
1
1
0
1
0
0
1
1
1
0
1
1
1
1
1
1
1
1
1
0
CCCCCC(C=CC1C(CC(=O)C1CCCCCCC(=O)O)O)O
1
1
1
1
1
1
1
0
1
1
1
0
1
1
1
1
1
1
1
1
1
0
0
1
1
1
1
CCCCC(C)(CC=C[C@H]1[C@@H](CC(=O)[C@@H]1CCCCCCC(=O)OC)O)O
1
0
1
1
1
1
0
1
1
0
1
0
0
1
1
1
1
1
1
1
1
1
1
1
1
1
0
CCCCC(C)(C)C(C=CC1C(CC(=O)C1CCCCC=CC(=O)OC)O)O
0
0
0
1
1
1
0
1
1
0
1
0
1
1
0
0
0
0
1
0
0
0
0
1
1
0
0
C[C@H](C1=CC(=CC(=C1)C(F)(F)F)C(F)(F)F)O[C@H]2[C@H](N(CCO2)CC3=NC(=O)NN3)C4=CC=C(C=C4)F
1
0
1
1
1
1
1
1
1
1
1
1
0
1
1
1
0
1
1
1
1
0
1
1
1
1
0
C[C@H](C1=CC(=CC(=C1)C(F)(F)F)C(F)(F)F)O[C@@H]2[C@@H](N(CCO2)CC3=NC(=O)N(N3)P(=O)([O-])[O-])C4=CC=C(C=C4)F.C[NH2+]C[C@@H]([C@H]([C@@H]([C@@H](CO)O)O)O)O.C[NH2+]C[C@@H]([C@H]([C@@H]([C@@H](CO)O)O)O)O
1
0
1
1
1
1
0
1
1
1
1
0
0
1
1
1
0
1
1
1
1
0
1
1
1
1
0
C[C@H](C1=CC(=CC(=C1)C(F)(F)F)C(F)(F)F)O[C@@H]2[C@@H](N(CCO2)CC3=NC(=O)N(N3)P(=O)(O)O)C4=CC=C(C=C4)F
1
0
1
1
1
1
0
1
1
0
1
0
0
1
1
1
0
1
1
1
1
0
1
1
1
1
0
CNCCC(C1=CC=CC=C1)OC2=CC=C(C=C2)C(F)(F)F
1
0
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
CC1=CC=CC=C1O[C@H](CCNC)C2=CC=CC=C2.Cl
1
0
1
1
1
1
0
0
1
0
1
0
0
1
0
1
0
1
1
1
1
0
1
1
1
1
1
C1=CC=C(C=C1)COC2=CC=C(C=C2)O
0
0
0
0
0
0
0
1
0
0
0
0
0
0
0
1
0
0
0
0
0
0
0
0
1
0
0
C1[C@@H]([C@@H]2[C@H](O1)[C@@H](CO2)O[N+](=O)[O-])O
1
0
1
1
1
1
1
1
1
0
1
0
0
1
1
1
0
1
1
1
1
0
1
1
1
0
1
C1C(C2C(O1)C(CO2)O[N+](=O)[O-])O[N+](=O)[O-]
0
0
0
0
0
1
0
0
0
0
1
0
0
1
1
1
0
0
0
0
0
0
0
1
1
0
0
C1[C@H]([C@@H]2[C@H](O1)[C@H](CO2)O)O
1
0
1
1
1
1
1
1
1
0
1
0
0
1
1
1
0
1
1
1
1
0
1
1
1
0
0
CC[C@H](C)[C@H]1C(=O)NC(C(=O)N[C@H](C(=O)N[C@@H](CSSCCC(=O)N[C@@H](C(=O)N1)CC2=CC=C(C=C2)OCC)C(=O)N3CCC[C@H]3C(=O)N[C@@H](CCCN)C(=O)NCC(=O)N)CC(=O)N)[C@@H](C)O
1
0
0
1
0
1
0
1
1
0
1
0
0
1
0
1
0
0
1
1
0
1
0
1
1
0
0
CCC(C)C1C(=O)NC(C(=O)NC(C(=O)NC(CSSCC(C(=O)NC(C(=O)N1)CC2=CC=C(C=C2)O)N)C(=O)N3CCCC3C(=O)NC(CC(C)C)C(=O)NCC(=O)N)CC(=O)N)C(C)O
1
0
1
1
1
1
0
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
0
1
1
1
0
CCC(C)C1C(=O)NC(C(=O)NC(C(=O)NC(CSSCC(C(=O)NC(C(=O)N1)CC2=CC=C(C=C2)O)N)C(=O)N3CCCC3C(=O)NC(CC(C)C)C(=O)NCC(=O)N)CC(=O)N)CCC(=O)N
1
0
1
1
1
1
0
1
1
0
1
0
0
1
1
1
1
0
1
0
0
1
0
1
1
1
0
CC1=C(C(=NO1)C2=C(C=CC=C2Cl)Cl)C(=O)NC3C4N(C3=O)C(C(S4)(C)C)C(=O)[O-]
0
0
0
1
1
1
0
1
0
0
1
0
0
1
1
1
0
1
1
1
1
0
0
0
1
1
1
CC1=C(C(=NO1)C2=C(C=CC=C2Cl)F)C(=O)NC3C4N(C3=O)C(C(S4)(C)C)C(=O)O
1
0
0
1
1
1
0
1
1
0
1
0
0
0
1
1
0
1
1
0
1
0
0
0
1
1
1
CC1=C(C(=NO1)C2=CC=CC=C2)C(=O)NC3C4N(C3=O)C(C(S4)(C)C)C(=O)[O-]
0
0
0
1
1
1
0
1
0
0
1
0
0
1
1
1
0
1
1
0
1
0
0
0
0
0
1
C1=CC=C(C(=C1)CC(=O)[O-])NC2=C(C=CC=C2Cl)Cl
1
0
1
1
1
1
1
1
1
1
1
0
1
1
1
1
1
1
1
1
1
0
1
1
1
1
1
CC1=C(C(=C(C=C1)Cl)NC2=CC=CC=C2C(=O)[O-])Cl
1
0
1
1
1
1
0
1
0
0
1
0
0
1
1
1
0
1
0
1
1
0
1
1
1
0
1
CC1=C(C(=CC=C1)NC2=CC=CC=C2C(=O)O)C
1
0
1
1
0
1
0
1
0
0
1
0
0
1
1
1
0
1
1
1
1
0
1
1
1
1
1
CCC[C@@H](C(=O)OCC)N[C@H](C)C(=O)N1[C@H]2CCCC[C@H]2C[C@H]1C(=O)O.CC(C)(C)N
1
0
1
1
1
1
0
1
1
0
1
0
1
1
1
1
0
1
1
1
1
0
1
1
1
1
1
CCC[C@@H](C(=O)OCC)N[C@H](C)C(=O)N1[C@H]2CCCC[C@H]2C[C@H]1C(=O)O
1
0
1
1
1
1
0
1
1
0
1
0
1
1
1
1
0
1
1
1
1
0
1
1
1
1
1
CCC[C@@H](C(=O)O)N[C@@H](C)C(=O)N1[C@H]2CCCC[C@H]2C[C@H]1C(=O)O
1
0
0
1
1
1
0
1
0
0
1
0
0
1
1
1
0
0
1
0
1
0
0
1
1
1
1
CCCC1CC(N(C1)C)C(=O)NC(C2C(C(C(C(O2)SC)O)O)O)C(C)Cl
0
0
0
1
1
1
0
1
1
0
1
1
0
1
1
1
0
1
1
0
1
1
1
1
1
1
1
CCCC1CC(N(C1)C)C(=O)NC(C2C(C(C(C(O2)SC)O)O)O)C(C)O
0
0
0
1
0
1
0
1
1
0
1
0
0
1
1
1
0
1
0
0
1
0
1
1
0
0
1
CCCC1CC(N(C1)C)C(=O)NC(C2C(C(C(C(O2)SC)OP(=O)(O)O)O)O)C(C)Cl
0
0
1
1
1
1
0
1
1
0
1
1
0
1
1
1
0
1
1
1
1
1
1
1
1
1
1
C1CC1N2C=C(C(=O)C3=CC(=C(C=C32)N4CCNCC4)F)C(=O)O
1
0
1
1
1
1
1
1
1
1
1
0
1
1
1
1
1
1
1
1
1
0
1
1
1
1
1
CC1CN(CC(N1)C)C2=C(C3=C(C(=C2F)N)C(=O)C(=CN3C4CC4)C(=O)O)F
1
0
1
1
1
1
1
1
1
1
1
0
0
1
1
1
0
1
1
1
1
0
1
1
1
1
1
CC1CN(CCN1)C2=C(C=C3C(=C2OC)N(C=C(C3=O)C(=O)O)C4CC4)F
1
0
1
1
1
1
1
1
1
0
1
0
0
1
1
1
0
1
1
1
1
0
1
1
1
1
1
CCN(CC)CCCC(C)NC1=C2C=CC(=CC2=NC=C1)Cl
1
0
1
1
1
1
0
1
0
0
1
0
0
1
1
1
0
0
0
1
0
0
1
1
1
1
1
CCN(CCCC(C)NC1=C2C=CC(=CC2=NC=C1)Cl)CCO
1
0
1
1
1
1
0
1
0
0
1
0
0
1
1
1
1
0
1
1
0
0
1
1
1
1
1
CC(CCCN)NC1=C2C(=CC(=C1)OC)C=CC=N2
0
0
0
0
0
1
0
0
0
0
0
0
0
0
1
0
0
0
0
0
0
0
0
0
0
0
0
C1CN(CCN1CCOCC(=O)O)C(C2=CC=CC=C2)C3=CC=C(C=C3)Cl
1
0
1
1
1
1
1
1
1
0
1
1
0
1
1
1
1
1
1
1
1
1
1
1
1
1
1
C1CN(CCN1CCOCCO)C(C2=CC=CC=C2)C3=CC=C(C=C3)Cl
0
0
0
0
0
1
0
1
0
0
0
0
0
1
0
1
0
0
0
1
0
0
0
0
1
1
0
CN1CCN(CC1)C(C2=CC=CC=C2)C3=CC=CC=C3
0
0
1
0
1
1
0
1
0
0
1
0
0
1
1
1
0
0
1
1
1
0
0
1
1
1
1
CN(C)CCOC(C1=CC=C(C=C1)Cl)C2=CC=CC=N2
1
0
1
0
0
1
0
0
0
0
1
0
0
1
1
1
0
1
1
1
1
0
1
1
1
1
0
CN(C)CCC(C1=CC=C(C=C1)Cl)C2=CC=CC=N2
1
0
1
0
0
1
1
0
0
0
1
0
0
1
1
1
0
1
1
1
1
0
1
1
1
1
0
CC(C)N(CCC(C1=CC=CC=C1)(C2=CC=CC=N2)C(=O)N)C(C)C
1
0
1
1
1
1
0
0
1
0
1
0
0
1
1
1
0
0
1
1
1
0
1
1
1
1
1
CC(CCCC(C)(C)O)C1CCC2C1(CCCC2=CC=C3CC(CC(C3=C)O)O)C
1
0
1
1
1
1
0
1
0
1
1
0
0
1
1
1
0
1
1
1
1
0
0
1
1
1
0
CC(C)C(C)C=CC(C)C1CCC2C1(CCCC2=CC=C3CC(CCC3=C)O)C
1
0
0
1
1
1
1
0
0
0
1
0
0
1
1
0
0
0
0
0
1
0
0
0
1
1
0
CC(C)C(C)C=CC(C)C1CCC2C1(CCCC2=CC=C3CC(CC(C3=C)O)O)C
1
0
1
1
1
1
0
0
0
0
1
0
0
1
1
1
0
1
1
1
1
0
0
1
1
1
0
CCCCN1CCCCC1C(=O)NC2=C(C=CC=C2C)C
1
0
1
1
1
1
0
1
1
0
1
0
1
1
1
1
0
1
1
1
1
1
1
1
1
1
0
CC1=C(C(=CC=C1)C)NC(=O)C2CCCCN2C
1
0
1
1
1
1
0
1
0
0
1
0
1
1
0
1
0
1
1
1
1
0
1
1
1
1
0
CCCN1CCCCC1C(=O)NC2=C(C=CC=C2C)C
1
0
1
1
1
1
1
1
1
0
1
0
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
CN(C)CC(C1=CC=C(C=C1)O)C2(CCCCC2)O
1
0
1
1
1
1
1
1
1
0
1
0
0
1
1
1
0
0
1
1
1
0
1
1
1
1
0
CCN(CC)CC#CCOC(=O)C(C1CCCCC1)(C2=CC=CC=C2)O
1
0
1
1
1
1
1
1
1
0
1
0
1
1
0
1
0
1
1
1
1
0
1
1
1
1
0
CN(C)CC(C1=CC=C(C=C1)OC)C2(CCCCC2)O
1
0
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
C1C2CC3CC1CC(C2)(C3)N
1
0
1
1
1
1
1
1
0
0
1
0
0
1
1
1
0
0
1
1
1
0
0
1
1
1
0
CC12CC3CC(C1)(CC(C3)(C2)N)C
1
0
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
CC(C12CC3CC(C1)CC(C3)C2)N
1
0
1
0
0
1
1
0
1
0
1
0
0
1
0
1
0
0
1
1
1
0
1
1
1
1
0
CC1=NN=C2N1C3=C(C=C(C=C3)Cl)C(=NC2)C4=CC=CC=C4
1
0
1
1
1
1
1
1
1
0
1
1
1
1
0
1
0
1
1
1
1
0
1
1
1
1
1
C1C2=NN=CN2C3=C(C=C(C=C3)Cl)C(=N1)C4=CC=CC=C4
1
0
1
1
1
1
1
1
1
1
1
0
0
1
1
1
0
1
1
1
1
0
1
1
1
1
0
CC1=NN=C2N1C3=C(C=C(C=C3)Cl)C(=NC2)C4=CC=CC=C4Cl
1
0
1
0
1
1
1
1
1
0
1
0
0
1
0
1
0
1
1
1
1
0
1
1
1
1
1
CO[C@@H]1[C@H]([C@@H]([C@@H](O[C@@H]1C(=O)[O-])O[C@H]2[C@@H](O[C@H]([C@H]([C@@H]2[O-])NOS(=O)(=O)O)OC)COS(=O)(=O)O)OS(=O)(=O)O)O
1
0
1
1
1
1
0
1
1
0
1
1
0
1
1
1
0
1
1
0
1
0
0
1
1
0
0
C1[C@H]([C@@H]([C@H]([C@@H](O1)O[C@@H]2CO[C@H]([C@@H]([C@H]2OS(=O)(=O)O)OS(=O)(=O)O)O)OS(=O)(=O)O)OS(=O)(=O)O)O
1
0
1
1
1
1
0
1
1
1
1
0
0
0
1
1
0
1
1
1
1
0
1
1
1
0
1
C([C@@H]1[C@H]([C@@H]([C@H]([C@H](O1)O)NS(=O)(=O)O)O)O[C@H]2[C@@H]([C@H]([C@@H]([C@@H](O2)C(=O)O)O)O)OS(=O)(=O)O)OS(=O)(=O)O
1
0
1
1
1
1
0
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
0
1
1
1
1
C[C@@H](C(=O)N1CC2=CC=CC=C2C[C@H]1C(=O)O)N[C@@H](CCC3=CC=CC=C3)C(=O)O
1
0
1
1
1
1
0
1
1
0
1
0
1
1
1
1
0
1
1
1
1
0
1
1
1
1
1
CCOC(=O)C(CCC1=CC=CC=C1)NC(C)C(=O)N2CC3=CC=CC=C3CC2C(=O)O
1
0
1
1
1
1
0
1
1
0
1
0
1
1
1
1
0
1
1
1
1
1
1
1
1
1
1
C[C@@H](C(=O)N1CC2=CC(=C(C=C2C[C@H]1C(=O)O)OC)OC)N[C@@H](CCC3=CC=CC=C3)C(=O)O
1
0
0
1
1
1
0
1
0
0
1
0
0
1
1
1
0
1
1
1
1
0
1
1
1
0
1
CC1=C(C(CCC1)(C)C)C=CC(=CC=CC(=CCO)C)C
0
0
0
0
0
0
0
1
0
0
0
0
0
0
0
0
0
0
0
0
0
0
0
0
0
0
0
CCC(CC)OC1C=C(CC(C1NC(=O)C)N)C(=O)OCC
1
0
1
1
1
1
0
1
1
0
1
0
0
0
1
1
0
1
1
1
0
0
1
1
1
1
1
CC1=C(C(CCC1)(C)C)C=CC(=CC=CC(=CC(=O)O)C)C
1
0
1
1
1
1
0
1
1
1
1
1
0
1
1
1
1
1
1
1
1
1
1
1
1
1
1
C[C@H](C(=O)N1CCC[C@H]1C(=O)O)N[C@@H](CCC2=CC=CC=C2)C(=O)O
1
0
1
1
1
1
0
1
1
0
1
0
0
1
1
1
0
1
1
1
1
0
1
1
1
0
1
CCOC(=O)C(CCC1=CC=CC=C1)NC(C)C(=O)N2CCCC2C(=O)O
1
0
1
1
1
1
0
1
1
0
1
1
0
1
1
1
0
1
1
1
1
0
1
1
1
1
1
C1CC(N(C1)C(=O)C(CCCCN)NC(CCC2=CC=CC=C2)C(=O)O)C(=O)O
1
0
1
1
1
1
0
1
1
1
1
1
0
1
1
1
1
1
1
1
1
0
1
1
1
1
1
C1=CC(=C(C=C1C[C@@H](C(=O)O)N)O)O.C1=CC(=C(C(=C1CNNC(=O)C(CO)N)O)O)O
1
0
1
1
1
1
0
0
0
0
1
0
1
1
1
1
0
0
1
1
1
0
0
1
1
0
0
CCCCCCCN(CC)CCCC(C1=CC=C(C=C1)NS(=O)(=O)C)O.CCCCCCCN(CC)CCCC(C1=CC=C(C=C1)NS(=O)(=O)C)O.C(=CC(=O)O)C(=O)O
0
0
0
0
0
1
0
0
0
0
0
0
0
1
0
0
0
0
0
0
1
0
0
1
1
0
0
C[C@](CC1=CC(=C(C=C1)O)O)(C(=O)O)NN.C1=CC(=C(C=C1C[C@@H](C(=O)O)N)O)O
1
0
1
1
1
1
0
1
1
1
1
0
0
1
1
1
0
1
1
1
1
0
0
1
1
1
0
CCNC(=NCCCC[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCCN=C(NCC)NCC)C(=O)N1CCC[C@H]1C(=O)N[C@H](C)C(=O)N)NC(=O)[C@H](CC2=CC=C(C=C2)O)NC(=O)[C@H](CO)NC(=O)[C@@H](CC3=CN=CC=C3)NC(=O)[C@@H](CC4=CC=C(C=C4)Cl)NC(=O)[C@@H](CC5=CC6=CC=CC=C6C=C5)NC(=O)C)NCC
0
0
0
0
1
1
0
1
1
1
1
0
0
0
0
1
1
0
1
0
1
1
0
0
1
1
0
C[C@H](C(=O)N)NC(=O)[C@@H]1CCCN1C(=O)[C@H](CCCCNC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](CC(=O)N)NC(=O)[C@H](CC2=CC=C(C=C2)O)N(C)C(=O)[C@H](CO)NC(=O)[C@@H](CC3=CN=CC=C3)NC(=O)[C@@H](CC4=CC=C(C=C4)Cl)NC(=O)[C@@H](CC5=CC6=CC=CC=C6C=C5)NC(=O)C
0
0
0
1
1
1
0
1
1
0
1
0
0
1
0
0
0
1
0
1
1
0
0
0
1
0
0
C[C@H](C(=O)N)NC(=O)[C@@H]1CCCN1C(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](CCCNC(=O)N)NC(=O)[C@H](CC2=CC=C(C=C2)O)NC(=O)[C@H](CO)NC(=O)[C@@H](CC3=CN=CC=C3)NC(=O)[C@@H](CC4=CC=C(C=C4)Cl)NC(=O)[C@@H](CC5=CC6=CC=CC=C6C=C5)NC(=O)C.C(=O)(C(F)(F)F)O
0
0
1
0
0
1
0
1
1
1
1
0
1
1
0
1
1
0
1
0
0
1
0
0
1
1
0
CC(=O)NCCC1=CNC2=C1C=C(C=C2)OC
1
0
1
1
1
1
0
1
1
0
1
0
0
1
1
1
0
1
0
1
1
0
1
1
1
0
1
CC(C)NCC(COC1=CC=CC2=C1C=CN2)O
0
0
1
1
1
1
0
0
1
0
1
0
0
1
0
1
0
1
1
1
1
0
1
1
1
0
0
CNS(=O)(=O)CC1=CC2=C(C=C1)NC=C2CCN(C)C
1
0
1
1
1
1
1
1
1
1
1
1
1
1
1
1
0
1
1
1
1
1
1
1
1
1
0
CC1CCC2CC(C(=CC=CC=CC(CC(C(=O)C(C(C(=CC(C(=O)CC(OC(=O)C3CCCCN3C(=O)C(=O)C1(O2)O)C(C)CC4CCC(C(C4)OC)OC(=O)C(C)(CO)CO)C)C)O)OC)C)C)C)OC
1
0
1
1
1
1
0
1
1
0
1
0
0
1
1
1
0
1
1
1
1
0
0
1
1
1
0
C[C@@H]1CC[C@H]2C[C@@H](/C(=C/C=C/C=C/[C@H](C[C@H](C(=O)[C@@H]([C@@H](/C(=C/[C@H](C(=O)C[C@H](OC(=O)[C@@H]3CCCCN3C(=O)C(=O)[C@@]1(O2)O)[C@H](C)C[C@@H]4CC[C@H]([C@@H](C4)OC)OCCO)C)/C)O)OC)C)C)/C)OC
1
0
1
1
1
1
0
1
1
1
1
1
0
1
1
1
1
1
1
1
1
0
0
1
1
1
1
CC1CCC2CC(C(=CC=CC=CC(CC(C(=O)C(C(C(=CC(C(=O)CC(OC(=O)C3CCCCN3C(=O)C(=O)C1(O2)O)C(C)CC4CCC(C(C4)OC)O)C)C)O)OC)C)C)C)OC
1
0
1
1
1
1
0
1
1
1
1
1
1
1
1
1
1
1
1
1
1
0
1
1
1
1
1
CCOC1=CC=CC=C1OCCN[C@@H](C)CC2=CC(=C(C=C2)OC)S(=O)(=O)N.Cl
1
0
1
1
1
1
0
1
1
0
1
0
0
1
0
1
1
1
1
1
1
0
1
1
1
1
0
CC(COC1=CC=CC=C1)NC(C)C(C2=CC=C(C=C2)O)O
1
0
0
0
0
1
0
0
0
0
1
0
0
1
0
1
0
0
1
0
0
0
0
1
1
0
0
CN(CCC1=CC=C(C=C1)NS(=O)(=O)C)CCOC2=CC=C(C=C2)NS(=O)(=O)C
0
0
0
0
1
1
0
0
0
0
1
0
0
1
0
1
0
1
1
1
0
0
0
1
1
1
1
C1CC(N(C1)C(=O)C2CSSCC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)N2)CC(=O)N)CCC(=O)N)CC3=CC=CC=C3)CC4=CC=C(C=C4)O)N)C(=O)NC(CCCN=C(N)N)C(=O)NCC(=O)N
0
0
0
1
0
1
0
1
0
0
0
0
0
1
0
1
0
1
1
0
0
0
1
1
1
0
0
C1C[C@H](N(C1)C(=O)[C@@H]2CSSC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N2)CC(=O)N)CCC(=O)N)CC3=CC=CC=C3)CC4=CC=C(C=C4)O)NC(=O)CNC(=O)CNC(=O)CN)C(=O)N[C@@H](CCCCN)C(=O)NCC(=O)N
1
0
0
1
0
1
0
0
1
0
1
0
0
1
0
1
0
0
1
0
0
1
0
1
1
0
0
C1CC(N(C1)C(=O)C2CSSCCC(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)N2)CC(=O)N)CCC(=O)N)CC3=CC=CC=C3)CC4=CC=C(C=C4)O)C(=O)NC(CCCN=C(N)N)C(=O)NCC(=O)N
1
0
1
1
1
1
1
1
1
0
1
1
1
1
0
1
0
1
1
1
1
0
1
1
1
1
0
C1CN2C(=CC=C2C(=O)C3=CC=CC=C3)C1C(=O)O
1
0
1
1
1
1
1
1
1
0
1
0
0
1
1
1
0
1
1
1
1
0
1
1
1
1
1
C1CN2C(=CC=C2C(=O)C3=CC=CC=C3)C1C(=O)O.C(C(CO)(CO)N)O
1
0
1
1
1
1
1
1
1
0
1
0
1
1
1
1
0
1
1
1
1
0
1
1
1
1
1
CN1C=CNC1=S
0
0
0
1
1
1
0
1
0
0
1
0
0
0
1
1
0
0
0
0
1
0
1
0
1
0
1
CCOC(=O)N1C=CN(C1=S)C
0
0
0
1
1
1
0
1
0
0
1
0
0
1
1
1
0
1
1
1
0
0
0
0
1
1
1
C[C@@]1(C2C[C@H]3[C@@H](C(=O)C(=C([C@]3(C(=O)C2=C(C4=C1C=CC=C4O)O)O)O)C(=O)NCNCCCC[C@@H](C(=O)O)N)N(C)C)O
0
0
1
1
0
1
0
1
1
0
0
0
0
0
1
1
1
1
0
0
0
0
0
0
1
1
1