chembl_id
stringlengths
7
13
canonical_smiles
stringlengths
1
2.03k
CHEMBL13414
CCN(C)C(=O)c1ccc(N(c2ccccc2)[C@H]2C[C@@H]3CC[C@H](C2)N3CCc2ccccc2)cc1
CHEMBL13339
CCCCC1C(=O)N(Cc2ccccc2)c2nc3ncncc3n2C1=O
CHEMBL13340
Cc1c(C(=O)c2cccc(N)c2)c2ccccc2n1CCN1CCOCC1
CHEMBL13341
CN1C(=O)CN=C(c2ccccc2)c2cc([N+](=O)[O-])ccc21
CHEMBL13455
CNCc1cccc(F)c1.Cl
CHEMBL13456
O=C(O)c1cc2c(O)nc3ccccc3n2n1
CHEMBL13458
O=C1CN=C(c2ccccc2)c2ccccc2N1
CHEMBL13183
CC(C)c1c(O)n(Cc2ccccc2)c2nc3c(c(=O)n(C)c(=O)n3C)n2c1=O
CHEMBL13184
CC(C)=CCc1c(O)n(Cc2ccccc2)c2nc3c(c(=O)n(C)c(=O)n3C)n2c1=O
CHEMBL13389
COC(=O)Nc1ccc(S(=O)(=O)Nc2ccc(CCNC[C@H](O)COc3ccc(O)cc3)cc2)cc1
CHEMBL13473
COc1ccc2c(=O)cc(-c3ccc(OC)c(OC)c3)oc2c1
CHEMBL13474
CC(C)N1C(=O)NC(c2ccc3c(c2)OCO3)c2cc3c(cc21)OCO3
CHEMBL13475
Cl.NCc1cccc(C(F)(F)F)c1
CHEMBL13476
O=C(Nc1cccc(NC(=O)c2cccnc2)c1)c1cccnc1
CHEMBL13136
CC(C)c1ccccc1Sc1c(O)cc(-c2ccc(Cl)c(Cl)c2)oc1=O
CHEMBL13137
CC1(C)CCC(C)(C)c2cc(CCc3ccc(C(=O)O)cc3)ccc21
CHEMBL13139
O=C(O)CCN1CCC(C(=O)N2CCC3(CC2)CCN(c2ccncc2)C3)CC1
CHEMBL13140
CN1C(=O)CN=C(c2ccccc2C(F)(F)F)c2cc([N+](=O)[O-])ccc21
CHEMBL13430
COC[C@H]1OC(=O)c2coc3c2[C@@]1(C)C1=C(C3=O)[C@@H]2C[C@@H](O)C(=O)[C@@]2(C)C[C@H]1OC(C)=O
CHEMBL13431
CC(C)=CCc1c(O)n(Cc2ccc([S+](C)[O-])cc2)c2nc3c(c(=O)n(C)c(=O)n3C)n2c1=O
CHEMBL13432
O=C(Nc1ccc(S(=O)(=O)Nc2ccc(CCNC[C@H](O)COc3ccc(O)cc3)cc2)cc1)NC1CCCCC1
CHEMBL13160
O=C(O)c1cn2c(ccc3cc([N+](=O)[O-])ccc32)n1
CHEMBL13161
CSc1ccc2c(c1)C(c1ccccc1)=NCC(=O)N2
CHEMBL13185
[O-][N+]1=Cc2ccccc2CC12CCCC2
CHEMBL13186
CCn1c(=O)c2nc(C(=O)Nc3nn[nH]n3)cn2c2ccccc21
CHEMBL13187
CCOC(=O)c1cc2c(=O)n(C)c3ccccc3n2c1
CHEMBL13188
COC(=O)/C=C/C(N)Cc1ccccc1
CHEMBL13280
CN1C(=O)CN=C(c2ccccc2F)c2cc([N+](=O)[O-])ccc21
CHEMBL521
CC(C)Cc1ccc(C(C)C(=O)O)cc1
CHEMBL13281
Cc1ccc(C2NC(=O)N(C(C)C)c3cc4c(cc32)OCO4)cc1
CHEMBL13393
CCN(CC)C(=O)c1ccc(N(c2ccccc2)[C@@H]2C[C@@H]3CC[C@H](C2)N3)cc1
CHEMBL13394
CC(C)NC(=O)C1=CC(C)(C)Oc2ccc([N+](=O)[O-])cc21
CHEMBL13117
CS(=O)(=O)c1ccc2ccc3nc(C(=O)O)cn3c2c1
CHEMBL13118
CCCCC1C(=O)N(Cc2ccccc2)c2nc3ccccc3n2C1=O
CHEMBL13235
Cn1cc(C(=O)c2ccccc2)cc1CCC(=O)NO
CHEMBL13236
NC(Cc1ccccc1)C(=O)Nc1ccc([N+](=O)[O-])cc1
CHEMBL13237
CCCNCc1cccc(Br)c1.Cl
CHEMBL13238
CC(C)S(=O)(=O)Nc1ccc(CCNC[C@H](O)COc2ccc(O)cc2)cc1
CHEMBL13239
CC(C)(S)C(N)C(=O)O
CHEMBL13240
Cn1c(=O)c2c(nc3n(Cc4ccccc4)c(O)c(CC=C4CCCCC4)c(=O)n23)n(C)c1=O
CHEMBL13162
CC(C)N(CCC(CCCN1CCCCC1)(C(N)=O)c1ccccc1F)C(C)C
CHEMBL13164
CC(C)Cc1c(O)n(Cc2ccccc2)c2nc3c(c(=O)n(C)c(=O)n3C)n2c1=O
CHEMBL13165
NCc1cccc(Cl)c1Cl
CHEMBL13260
O=c1[nH]c2cc(-n3ccnc3)c([N+](=O)[O-])cc2[nH]c1=O
CHEMBL13261
Cc1ccc(S(=O)(=O)O)cc1.N/C(=N\O)N/N=C/C1CC2C=CC1C2
CHEMBL13262
OCc1cn2c(cnc3ccccc32)n1
CHEMBL13282
COC(=O)c1cn2c(n1)COc1ccc(NC(C)=O)cc1-2
CHEMBL13283
Cc1c(O)n(Cc2ccc(F)cc2)c2nc3c(c(=O)n(C)c(=O)n3C)n2c1=O
CHEMBL13284
COC(=O)c1ccccc1OCC(O)CNC(C)C
CHEMBL13364
C#CCc1c(O)n(Cc2ccccc2)c2nc3c(c(=O)n(C)c(=O)n3C)n2c1=O
CHEMBL13365
COC(=O)c1ccccc1OCC(O)CNC(C)(C)C
CHEMBL3309339
C=CCn1c(=O)c2cccnc2n(C2CCCCC2)c1=O
CHEMBL13214
CN(C)Cc1ccc(CSCCNC(=O)NCCSCc2ccc(CN(C)C)o2)o1
CHEMBL13299
COC(=O)c1ccccc1OCC(O)CNCCNC(=O)Nc1ccccc1
CHEMBL13300
CC(C)c1ccc(C(CCN2CCCCC2)(CCN(C(C)C)C(C)C)C(N)=O)cc1
CHEMBL13301
CCN(CC)C(=O)c1ccc(N(c2ccccc2)[C@@H]2C[C@@H]3CC[C@H](C2)N3CC2CCCCC2)cc1
CHEMBL13321
CCC[C@H](NC(=O)[C@H](Cc1ccc(OP(=O)(O)O)cc1)NC(C)=O)C(=O)NCCCc1ccccc1
CHEMBL13322
OCc1cn2c(n1)COc1ccccc1-2
CHEMBL13324
O=C(O)c1cn2c(cnc3ccccc32)n1
CHEMBL13325
CN1CCc2cc(Cl)c(O)cc2C(c2ccccc2Br)C1
CHEMBL13326
CCc1ccccc1CCNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](Cc1ccc(OP(=O)(O)O)cc1)NC(C)=O
CHEMBL13263
NCc1cc(Cl)cc(Cl)c1
CHEMBL13264
CNn1cc(C(=O)O)c(=O)c2cc(F)c(N3CCCC(O)C3)cc21
CHEMBL13265
O=C([C@@H](NS(=O)(=O)c1cnccc1N[C@H](CO)Cc1ccccc1)c1ccc(O)c(O)c1)N1CCC(CCF)CC1
CHEMBL13342
O=C(Nc1cc(Cl)cc(Cl)c1)Nc1cccc(NC(=O)Nc2cc(Cl)cc(Cl)c2)c1
CHEMBL3309316
COc1cc2c(Oc3ccc(NC(=O)c4nn(-c5ccccc5F)c(=O)c5ccccc45)cc3F)ccnc2cc1OCCCN1CCOCC1
CHEMBL13366
CC(C)(N)C(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC2(CC1)Cc1ccccc1C2=O
CHEMBL13367
CCCCN(C)C(=O)CCCCCCCSC(Cc1ccc(OCc2ccccc2)cc1)c1ccc(OC)cc1
CHEMBL13368
COc1cccc2c1C=[N+]([O-])C1(CCCCC1)C2
CHEMBL1163481
O=C(CC(Nc1ccc([N+](=O)[O-])cc1)C1CCCCC1)c1ccc(F)cc1
CHEMBL3309356
COc1nonc1S(N)(=O)=O
CHEMBL3309357
CCOc1nonc1S(N)(=O)=O
CHEMBL3309358
CCCCOc1nonc1S(N)(=O)=O
CHEMBL13302
CCCCCCCc1cc(O)cc(O)n1
CHEMBL13303
CC(=O)O.CCN(CCc1ccccn1)C(=O)CNC(=O)[C@@H](CCCN=C(N)N)NC(=O)[C@@H](N)Cc1ccc(O)cc1
CHEMBL13304
Cc1ccccc1C(=O)c1c(C)n(CCN2CCOCC2)c2ccccc12
CHEMBL13390
Cc1c(O)n(-c2ccccc2)c2nc3c(c(=O)n(C)c(=O)n3C)n2c1=O
CHEMBL4543366
CNC(=O)CN(C)C(=O)C(C)OCc1ccccc1
CHEMBL13391
COc1ccc2c(ccc3nc(C(=O)O)cn32)c1
CHEMBL13392
CCOC(=O)c1cn2c(cc(Cl)c3ccc(Cl)cc32)n1
CHEMBL13416
O=C(O)c1cn2c(cc(Cl)c3ccc(Cl)cc32)n1
CHEMBL13417
CCN(CCCCCC(C)F)CCCC(O)c1ccc(NS(C)(=O)=O)cc1
CHEMBL13419
O=C(O)c1cn2ccc3ccccc3c2n1
CHEMBL4543209
O=C(N/N=C/c1cc(Cl)cc(Cl)c1O)c1cccc(Br)c1Br
CHEMBL4543210
C/C=C1\CN2CCc3c([nH]c4ccccc34)[C@H]2C[C@@H]1/C(=C\OC)C(=O)OC
CHEMBL13420
CCCN(CCC)C(=O)c1ccc(N(c2ccccc2)[C@@H]2C[C@@H]3CC[C@H](C2)N3)cc1
CHEMBL13421
O=C(Nc1ccc(Br)cc1Br)NC1CCCC(NC(=O)Nc2ccc(Br)cc2Br)C1
CHEMBL13344
CCSCCc1c(O)n(Cc2ccccc2)c2nc3c(c(=O)n(C)c(=O)n3C)n2c1=O
CHEMBL13345
O=C(Nc1nn[nH]n1)c1cn2c(n1)COc1ccccc1-2
CHEMBL13346
CC(C)(C)NC(=O)NC1CCCC(NC(=O)NC(C)(C)C)C1
CHEMBL13347
O=C(NCC(c1ccccc1)c1ccccc1)Nc1cccc(NC(=O)NCC(c2ccccc2)c2ccccc2)c1
CHEMBL13348
O=C(O)c1nc2n(c1C(=O)N1CCOCC1)-c1ccccc1OC2
CHEMBL13433
Cn1nnnc1SCC1=C(C(=O)OC(C)(C)C)N2C(=O)[C@@H](NC3=NCCN3)C2SC1
CHEMBL13459
CCCCCNC(=O)Nc1ccc(S(=O)(=O)Nc2ccc(CCNC[C@H](O)COc3ccc(O)cc3)cc2)cc1
CHEMBL13460
Clc1ccc2c(Cl)cc3nc(-c4nn[nH]n4)cn3c2c1
CHEMBL13461
O=C(O)c1cn2c(ccc3c(Cl)cccc32)n1
CHEMBL13189
CC(C)N(CCC(CCN(C(C)C)C(C)C)(C(N)=O)c1ccccc1F)C(C)C
CHEMBL13477
COc1ccc2c(c1)C=CC21CCN(S(=O)(=O)C[C@]23CCC(CC2=O)C3(C)C)CC1
CHEMBL13208
CN(C)[C@@H]1C(=O)C(C(N)=O)=C(O)[C@@]2(O)C(O)=C3C(=O)c4c(O)cccc4[C@](C)(O)C3C(=O)[C@@H]12
CHEMBL13209
O=C1CN=C(c2ccccc2)c2cc([N+](=O)[O-])ccc2N1