chembl_id
stringlengths
7
13
canonical_smiles
stringlengths
1
2.03k
CHEMBL14510
CCc1ccc(OCCCN2CCC(c3noc4cc(F)ccc34)CC2)c(OC)c1
CHEMBL14597
CCN1CCCC1CNC(=O)c1cc(NS(=O)(=O)NC)ccc1OC
CHEMBL14598
COc1ccc(C(=O)/C(=N/O)SCCCN(C)C)cc1.O=C(O)C(=O)O
CHEMBL14599
C=CCCCCCCCC1CCC(CCCCC=C)N1
CHEMBL13899
CC(C)=CC(=O)c1cc(C(C)(C)C)c2c(c1)C(C)(C)CO2
CHEMBL13902
COC(Cn1c(=O)[nH]c2c(=O)n(CC(=O)NC(C(=O)C(F)(F)F)C(C)C)c(-c3ccccc3)cc2c1=O)OC
CHEMBL13994
c1ccc(-c2nnc3c4ccccc4c(N4CCCCC4)nn23)cc1
CHEMBL14296
O=C(Nc1ccncc1)c1c(O)c2cccnc2n(-c2ccccc2)c1=O
CHEMBL14298
COc1ccc(-c2cc(O)c(SCc3ccccc3)c(=O)o2)cc1C
CHEMBL14299
CCNC(=O)/C(C(=O)OCC)=C(C)/C=C/C=C(C)/C=C/C1=C(C)CCCC1(C)C
CHEMBL14574
C=CCOc1ccc2c(c1)CCc1ccccc1/C(CC)=C\2c1ccccc1
CHEMBL14575
C[C@]12CC[C@H]3[C@@H](CC[C@H]4CC(=O)CCN43)[C@@H]1CCC2=O
CHEMBL14576
O=C(CCCC1CC1)c1ccc2c(c1)CCO2
CHEMBL14314
CCN1CCCC1CNC(=O)c1cc(NS(=O)(=O)NC)c(C)cc1OC
CHEMBL14315
Nc1noc(C2CN3CCC2CC3)n1
CHEMBL14600
O=C1CC[C@H](/C=C/C(O)Cc2ccccc2)N1CCCCSc1nn[nH]n1
CHEMBL14601
COc1oc(=O)c2cc(NC(=O)C(c3ccccc3)c3ccccc3)ccc2c1Cl
CHEMBL14338
c1ccc(-c2[nH]ccc3c4ccccc4nc2-3)cc1
CHEMBL14339
Fc1ccc(-c2ncn(C3CCNCC3)c2-c2ccnc(Oc3cc(F)cc(F)c3)n2)cc1
CHEMBL14340
Cc1cc(C)c(NN=C2CCC(C)n3c2ncc(C(=O)O)c3=O)c(C)c1
CHEMBL13995
CCNCc1c(Cl)cccc1Cl.Cl
CHEMBL13996
CNC(=O)C1=CC(C)(C)Oc2ccc(C#N)cc21
CHEMBL13998
CC[C@@]1(O)C(=O)OCc2c1cc1n(c2=O)Cc2c-1nc1cnc(C#N)cc1c2C
CHEMBL14091
CC(C)CCN(C)CC(=O)N[C@@H](Cc1ccc(OC(=O)c2ccccc2)cc1)C(=O)NC(C)(C)C
CHEMBL14092
c1ccc(-c2ccccc2)cc1
CHEMBL14093
CCOC(=O)C1(CCCCCc2ccc(Cl)cc2)CO1
CHEMBL14383
Fc1ccccc1-c1[nH]ccc2c3ccccc3nc1-2
CHEMBL14384
CC1CCC(=NNc2ccccc2)c2ncc(C(=O)NO)c(=O)n21
CHEMBL14385
C#CCc1c(O)n(Cc2ccccc2)c2nc3c(n2c1=O)C(=O)N(C)CN3C
CHEMBL14386
O=C(Nc1cccnc1)c1c(O)c2cccnc2n(-c2ccccc2)c1=O
CHEMBL14387
N#Cc1nccc2c1ncn2CCOc1ccc(Cc2ccccc2)cc1
CHEMBL14316
Cc1ccc(-c2nnc3c4ccccc4c(N4CCCC4)nn23)cc1C
CHEMBL14317
CCN(CC)c1nc(NCCNC(=O)c2cc(O)c(O)c(O)c2)c2ccccc2n1.CS(=O)(=O)O
CHEMBL14318
COc1nccc(-c2c(-c3ccc(F)cc3)ncn2CCCN2CCOCC2)n1
CHEMBL14400
COc1oc(=O)c2cc(NC(=O)C(Cc3ccccc3)NS(=O)(=O)c3ccc(C)cc3)ccc2c1Cl
CHEMBL4543262
CC(CO)NC(=O)CCC1CCCCC1
CHEMBL4543263
COc1ccc2[nH]cc(C3=CCN(Cc4ccco4)CC3)c2c1
CHEMBL4543264
CCOc1cc2c(cc1OC)CCN(C=O)[C@H]2CCc1c[nH]c2ccccc12
CHEMBL4543265
Cc1ccc(-c2cnc(N)c(C(=O)Nc3c(C)cccc3Cl)c2)c(F)c1
CHEMBL14341
O=C([O-])C1(CCCCCc2ccc(Cl)cc2)CO1.[Na+]
CHEMBL14342
O=c1cc(-c2ccccc2)oc(O)c1SCc1ccc2c(c1)OCCO2
CHEMBL14343
OC1COC(O)C(O)C1O
CHEMBL14423
COc1oc(=O)c2cc(NC(=O)OCc3ccccc3)ccc2c1Cl
CHEMBL14424
Nc1nsc(-c2ccc(N3CCN(c4cccc(C(F)(F)F)c4)CC3)nn2)n1
CHEMBL14094
CC(C)CC(C)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1
CHEMBL14095
CC(C)NCC(O)COc1ccccc1/C=C\CO
CHEMBL546
C=CCOc1ccccc1OCC(O)CNC(C)C
CHEMBL14189
c1ccc(-c2ncc[nH]2)cc1
CHEMBL14190
Cc1cccc(C)c1NN=C1CCC(C)n2c1ncc(C(=O)O)c2=O
CHEMBL14191
COc1cc(OC)c(-c2nnc3c4ccccc4c(N4CCCC4)nn23)cc1OC
CHEMBL14192
c1ccc(Cn2ccnc2)cc1
CHEMBL14470
COc1ccc(NC(C)=O)cc1OCCCN1CCC(c2noc3cc(F)ccc23)CC1
CHEMBL14471
Nc1ccc(Cn2cnc3ncnc-3c2O)cc1
CHEMBL14472
CCC(c1ccc(O)c([N+](=O)[O-])c1)C(CC)c1ccc(O)c([N+](=O)[O-])c1
CHEMBL14473
CCC(c1ccc(O)c(CO)c1)C(CC)c1ccc(O)c(CO)c1
CHEMBL14474
c1ccc2ncccc2c1
CHEMBL4543288
CC(=O)c1c(C)cccc1NC(=O)CN1CCCC1=O
CHEMBL4543289
COc1ccccc1NCc1ccc(CNc2ccccc2OC)o1
CHEMBL14475
CCOc1ccc2c(c1)[nH]c1c(C)nccc12
CHEMBL14401
COc1cc2c(cc1C(F)(F)F)N(C(=O)Nc1cncc(-c3ccc(F)cc3)c1)CC2
CHEMBL14402
CC(C)(C)c1[nH]ccc2c3ccccc3nc1-2
CHEMBL14403
CCCC(=O)NCCc1c(-c2ccccc2)[nH]c2ccc(OC)cc12
CHEMBL14404
Cc1nsc(-c2nccc(N3CCN(c4cccc(C(F)(F)F)c4)CC3)n2)n1
CHEMBL14490
OC(c1ccccc1)(c1ccccc1)c1noc(C2CN3CCC2CC3)n1
CHEMBL14425
Cc1nccc2c1[nH]c1cc(OCCC3(C)OCC(C)(C)CO3)ccc12
CHEMBL14427
Cc1sc2c(c1C(C)C)C(N1CCN(C)CC1)=Nc1cc(F)ccc1N2
CHEMBL14512
CC(C)(C)c1cc(C(=O)CCCC2CC2)cc2c1SCC2(C)C
CHEMBL14513
O=C(NCCCCNCCCNC(=O)c1cccc(O)c1O)c1cccc(O)c1O
CHEMBL4543311
Cn1nc(N2CCCC2)c(=O)n(C)c1=O
CHEMBL4543312
Cc1cc2c(cc1S(=O)(=O)Nc1cc(C(F)(F)F)ccc1Cl)OCC(=O)N2
CHEMBL14193
O=Cc1ccc(O)cc1
CHEMBL14194
CCOC(=O)C1(CCCc2cc(Cl)ccc2OC)CO1
CHEMBL14538
Nc1ccccc1OCCCN1CCC(c2noc3cc(F)ccc23)CC1
CHEMBL14539
COc1ccccc1OCCCN1CCC(c2noc3cc(F)ccc23)CC1
CHEMBL14540
Oc1cc(-c2cccs2)nc2cc3c(cc12)OCO3
CHEMBL14541
COc1ccc(NC(=O)c2c(O)c3cccnc3n(-c3ccccc3)c2=O)cn1
CHEMBL14553
CCC(=O)c1ccc2c(c1)sc(=O)n2C(=O)CC
CHEMBL14554
Cc1cc([C@@H]2C[C@H](CF)CN2C)on1
CHEMBL14555
FC(F)(F)c1cccc(N2CCN(C3CCN(c4ccc(-c5ncns5)nn4)CC3)CC2)c1
CHEMBL14556
CC(=O)c1ccc(OCCCN2CCC(c3noc4cc(F)ccc34)CC2)c(C)c1
CHEMBL14557
O=C(O)c1cc(NC(=O)[C@H](Cc2ccccc2)NC(=O)c2cc3cc[nH]c3cc2C(=O)NCC23CC4CC(CC(C4)C2)C3)cc(C(=O)O)c1
CHEMBL14558
CCC(=Cc1ccccc1OCC(O)CNC(C)C)CO
CHEMBL14491
C[C@H]1CN(C(=O)N2Cc3c(C(=O)OC(C)(C)C)ncn3-c3ccc(C(F)(F)F)cc32)C[C@@H](C)N1C
CHEMBL14492
CC1CCn2c(ncc(C(=O)O)c2=O)/C1=N/Nc1ccccc1
CHEMBL14493
NCCn1cnc2ncnc-2c1O
CHEMBL14494
CC(=O)c1cc(C)ccc1OCCCN1CCC(c2noc3cc(F)ccc23)CC1
CHEMBL14578
O=c1cc(-c2ccc3c(c2)OCCO3)oc(O)c1SCc1ccccc1
CHEMBL14765
CCCc1c(OCCCOc2cccc(NC(=O)C(=O)OCC)c2C#N)ccc(C(C)=O)c1O
CHEMBL14766
CN1CCN(C2=Nc3cc(F)ccc3Nc3sc4c(c32)CCCC4)CC1
CHEMBL14854
CNc1nsc(-c2ccc(N3CCN(c4cccc(C(F)(F)F)c4)CC3)nn2)n1
CHEMBL14855
O=C(O)c1cccc(CSc2c(O)cc(-c3ccccc3)oc2=O)c1
CHEMBL3309988
Nc1nc2c3ccc(F)cc3nc(Cc3ccc4c(c3)OCO4)n2n1
CHEMBL14699
COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCN1CCOCC1
CHEMBL14785
CC(C)CCn1c(Cn2c(=O)n(C(=O)NCc3ccccc3)c3ccccc32)nc2ccccc21
CHEMBL3310021
COc1ccc(/C=C/C(=N\NC(=O)c2ccc(OC)cc2)c2ccc(Br)cc2)cc1
CHEMBL3310022
COc1ccc(/C=C/C(=N\NC(=O)c2ccco2)c2ccc(Br)cc2)cc1
CHEMBL14532
COC(=O)c1c(CS(=O)(=O)CCO)nc2ccccc2[n+]1[O-]
CHEMBL4543320
CC(C)(C)C(=O)N1CCc2cnccc21
CHEMBL4543321
COC(=O)N[C@H](C(=O)N1CCC[C@H]1c1ncc(-c2cc3c4c(c2)OCc2cc(-c5cnc([C@@H]6CCCN6C(=O)[C@H](NC(=O)OC)c6ccccc6)[nH]5)cc(c2-4)OC3)[nH]1)C(C)C
CHEMBL4543322
COc1ccc(-c2c(C)[nH]c3c(C4=CCOCC4)c(-c4ccccc4)nn3c2=O)cc1