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Off target assessment using Retrogenix cell microarray technology
PK and ADA methods
Development of the PK and ADA methods in rat and mouse (4 week study), with validation of methods to support the 13-week GLP tox study (rat only).
Extension of validation for PK and ADA methods up to 300 mg/kg in monkey
Development and validation of the PK and ADA methods in human
Proposed PD biomarkers for clinical phase 1
On skin biopsies (after LPS challenge in Healthy Volunteers): - IHC (3 panels: neutrophils, macrophages and NETosis (eg CITH3)). Validation needed. - RNA seq (3 gene expression signatures product-related available in human on whole blood, neutrophils and macrophages; 3 gene expression signatures linked to the mechanism...
On whole blood: - PBMC subsets - ex vivo LPS challenge (multiplex cytokines). No validation needed for the multiplex cytokines portion on the ex vivo LPS challenge.
On skin exudates from blister suctions: -NETosis (Validation needed). - Multiplex cytokines (No validation needed).
CMC¹
New OSE230 GMP Drug Substance (DS) batch Manufacturing & release
Stability studies for new GMP DS batch
Analytical method transfer and partial validation of methods for Drug Product (DP) release
OSE230 clinical GMP DP batch manufacturing & release
Stability studies for clinical DP batch
Compatibility & in-use stability study (design to be discussed with AbbVie depending on clinical trial use)
Placebo batch manufacturing & release
TBC= To be confirmed ¹ See Appendix A for CMC documentations to be provided by OSE. In the event that a replacement GMP batch is needed due to nonconformity, OSE would not be responsible for the cost of more than one replacement batch.
Transition Development Plan Timeline²
[Timeline chart image]
*PD biomarkers requiring validation before Phase 1 start ²Timelines based on vendor projections summarized in the Workplan Table
Transition Development Budget
Study
TOXICOLOGY PACKAGE
4-w preli study in mice
Revised 65 965€ signed -ERBC + TK and ADA- planned at Nantes
4-w preli study in rat
Revised 77 565 signed- ERBC
SD GLP Resp Study in Rats
13-w additional GLP study in monkey
1 186 860€ signed ERBC
QPS Bioanalysis (ADA and PK)
77 900€ +11 550€ validation of new dose, signed QPS
10 000 € Cytokines Kit- Nantes
PK modeling Calvagone (PK analysis) 6 600
Total 1 292 910€ revised
Off target assessment
13-w GLP rat study
+ 250 k€ bioanalysis at QPS
378 530€ revised (number of animals reduced 148 vs 250 confirmed) + 6K€ QPS validation PK ADA 102 930€ (60 370+ 42 560) + bioanalysis 78090 €
Total revised 565,590€
PHASE 1 HUMAN PK/BIOMARKERS
Total 1,200 k€ still estimated
PK and ADA methods
Cytokine and biomarkers assessment
CMC
Additional GMP 250L DS batch
Catalent Madison 1 576 000$ 1 321 000$ already paid Additional stability cost updated
DP-related activities (production, analytical method validation, stability, Placebo)
TOTAL
Appendix A: CMC Documentations
Item #
1
2
3
4
5
6
³ Work may be performed at AbbVie or a CMO(s) selected by AbbVie.
Schedule 10.2.1 Existing Patents
List of Patents
[Table with patent information including IP family references, filing numbers, dates, etc.]
Schedule 10.2.10 Third Party Agreements
ACTIVE BIOMARKER
1. Amendment 1 to the Project Order 1 between OSE Immunotherapeutics and Active Biomarkers, effective as from June 15th, 2022 (executed)
2. Amendment 2 to the Project Order 1 between OSE Immunotherapeutics and Active Biomarkers, effective as from July 18th, 2022 (executed)
3. Project Order 1 between OSE Immunotherapeutics and Active Biomarkers, as from May 3rd, 2022 (executed)
AGRO-BIO
4. Contract for the provision of services (Contrat de prestation de services) between OSE Immunotherapeutics and Agro-Bio, effective as from August 11, 2023 (French language) (executed)
5. Contract for the provision of services (Contrat de prestation de services) between OSE Immunotherapeutics and Agro-Bio, effective as from June 9, 2022 (French language) (executed)
6. Contract for the provision of services between OSE Immunotherapeutics and Agro-Bio, effective as from June 9, 2022 (translation from French)
7. Contract for the provision of services between OSE Immunotherapeutics and Agro-Bio, effective as from August 11, 2023 (translation from French)
Ambiotis
8. Patent Assignment Agreement (Contrat de Cession de Droits sur les brevets) between OSE Immunotherapeutics and Ambiotis, effective as from April 3, 2018 - in French
9. Patent Assignment Agreement between OSE Immunotherapeutics and Ambiotis, effective as from April 3, 2018 - Translation from French
ANAPATH
10. Services Agreement between OSE Immunotherapeutics and AnaPath Research S.A.U, effective as from April 5th, 2022 (executed)
B&S
11. Engagement letter (Lettre de mission) OSE Immunotherapeutics - Accompagnement dans la définition et la mise en œuvre opérationnelle de la stratégie PI - January 1st, 2023 (French language) (executed)
12. Engagement letter OSE Immunotherapeutics - Support in the definition and operational implementation of the IP strategy - January 1st, 2023 (translation from French)
BIOTEM
13. Contract for the provision of services (Contrat de prestation de services) between OSE Immunotherapeutics and Biotem, effective as from July 31, 2020 (French language) (executed)
14. Contract for the provision of services between OSE Immunotherapeutics and Biotem, effective as from July 31, 2020 (translation from French)
CALVAGONE
15. Consulting Agreement between OSE Immunotherapeutics and Calvagone Sarl, effective as from April 27th, 2021 (executed)
16. Amendment 2 to the Consulting Agreement between OSE Immunotherapeutics and Calvagone Sarl, effective as from June 13th, 2022 (executed)
17. Services Agreement between OSE Immunotherapeutics and Calvagone SAS, effective as from December 23rd, 2022 (executed)
18. Services Agreement between OSE Immunotherapeutics and Calvagone SAS, effective as from September 26, 2023 (executed)
19. Services Agreement between OSE Immunotherapeutics and Calvagone SAS, effective as from January 10, 2024 (executed)
CATALENT FRANCE LIMOGES
20. Customized Solution for OSE Immunotherapeutics - Clinical Program Phase 1 for OSE 230 Product - 9 March 2022 (executed)
21. Solution for OSE Immunotherapeutics - Cancellation and Postponement fees for OSE 230 Product - 23 March 2023 (executed)
CATALENT MADISON US
22. Statement of Work (SOW) - QTE-9193180 - OSE Immunotherapeutics SA - Catalent Pharma Solutions LLC - OSE 230 - April 28, 2021
23. Statement of Work (SOW) - QTE -9194626- OSE Immunotherapeutics SA - Catalent Pharma Solutions LLC - OSE 230 - June 4, 2021
24. Statement of Work (SOW) - QTE 9188753- OSE Immunotherapeutics SA - Catalent Pharma Solutions LLC - OSE 230 - September 29, 2021
25. Statement of Work (SOW) - QTE-9201531 - OSE Immunotherapeutics SA - Catalent Pharma Solutions LLC - OSE 230 - November 10, 2021
26. Statement of Work (SOW) - QTE-9209608 - OSE Immunotherapeutics SA - Catalent Pharma Solutions LLC - OSE 230 - July 21, 2022
27. Statement of Work (SOW) - QTE-9188753 - OSE Immunotherapeutics SA - Catalent Pharma Solutions LLC - OSE 230 - September 26, 2022
28. Statement of Work (SOW) - QTE-9209608 - OSE Immunotherapeutics SA - Catalent Pharma Solutions LLC - OSE 230 - October 28, 2022