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Physical Examination X X X X X X X
Height
Weight X X X X X X X
12-Lead ECG X
Eastern Cooperative Oncology Group Performance Status X X X
HBV, HCV, and HIV
Serology
PK X X X X X X X
ADA X X
IV Administration CLBR0012
SWI0192 X X X X X X X
Adverse Events/Serious Adverse events(6) X X X X X X X X X X X X X X X X X X X X X X X X X X X X
Chemistry, Hematology, and Urinalysis X X X X X X
Prior and Concomitant Medications/ Nonpharmacologic therapies
CTC
Bone Marrow Biopsy(3) X
Archival Bone Marrow Sample X
Exploratory biomarkers4 X X X X X X X X
1Assessment Cycle 2 - Patients will be treated on an Outpatient basis 2Assessment Cycle 1 - Patients will be admitted on Day 28 for evaluation and scheduled procedures, i.e. bone marrow biopsy
CD19 Program timeline:
Schedule 1.94: Corporate Names
The Scripps Research Institute
Scripps Research
Calibr, a division of Scripps Research
Calibr
TSRI
Schedule 1.119: Existing Patents
[See attached.]
Matters 70 items
Client-Matter Cooley Docket Title Country Application Num Application Date Publication Num Publication Date Registration Num Registration Date Case Status Inventors Applicant TSRI Ref
SWITCHABLE CAR-T THERAPIES FOR TREATING HUMAN CANCERS World Intellectual Property Organization PCT US22/081010 12/6/2022 WO 2023 107910 6/15/2023 Published Travis YOUNG, Eduardo LABORDA 2120.1PC
SWITCHABLE CAR-T THERAPIES FOR TREATING HUMAN CANCERS United States 63/286,868 12/7/2021 Expired Travis YOUNG, Eduardo LABORDA 2120.0P
NOVEL THERAPIES WITH ENGINEERED EFFECTOR CELLS World Intellectual Property Organization PCT US22/023791 7/2022 WO 2022 216906 10/13/2022 Published Travis YOUNG, Nelson Bruno 2081.1PC
NOVEL CANCER THERAPIES WITH SWITCHABLE CAR-T PLATFORMS United States 63/172,212 8/2021 Abandoned Travis YOUNG, Nelson Bruno 2081.0P
CHIMERIC ANTIGEN RECEPTOR EFFECTOR CELL SWITCHES WITH HUMANI... United States 16/343,353 4/18/2019 20190359697 11/28/2019 11,174,306 11/16/2021 Issued Travis YOUNG, Leonard PRESTA, David RODGERS, Eric HAMPTON, Ti... 1924.1US
CHIMERIC ANTIGEN RECEPTOR EFFECTOR CELL SWITCHES WITH HUMANI... World Intellectual Property Organization PCT US17/057460 10/19/2017 WO 2018/075807 4/26/2018 Expired Travis YOUNG, Leonard PRESTA, David RODGERS, Eric HAMPTON, Ti... 1924.1PC
CHIMERIC ANTIGEN RECEPTOR EFFECTOR CELL SWITCHES WITH HUMANI... Republic of Korea 10-2019-0065433 5/17/2019 20200138985 12/11/2020 Published Travis YOUNG, Leonard PRESTA, David RODGERS, Eric HAMPTON, Ti... 1924.1KR
CHIMERIC ANTIGEN RECEPTOR EFFECTOR CELL SWITCHES WITH HUMANI... Japan 2022-153946 9/27/2022 2022-185016 12/13/2022 Published Travis YOUNG, Leonard PRESTA, David RODGERS, Eric HAMPTON, Ti... 1924.1JPD1
CHIMERIC ANTIGEN RECEPTOR EFFECTOR CELL SWITCHES WITH HUMANI... Japan 2019-520888 10/19/2017 2019-535241 12/12/2019 7149935 9/29/2022 Issued Travis YOUNG, Leonard PRESTA, David RODGERS, Eric HAMPTON, Ti... 1924.1JP
CHIMERIC ANTIGEN RECEPTOR EFFECTOR CELL SWITCHES WITH HUMANI... Hong Kong 62020002300.5 10/19/2017 HK1291004 7/31/2020 Published Travis YOUNG, Leonard PRESTA, David RODGERS, Eric HAMPTON, Ti... 1924.1HK
CHIMERIC ANTIGEN RECEPTOR EFFECTOR CELL SWITCHES WITH HUMANI... European Patent Office 17794509.4 5/14/2019 3529268 8/28/2019 Published Travis YOUNG, Leonard PRESTA, David RODGERS, Eric HAMPTON, Ti... 1924.1EP
CHIMERIC ANTIGEN RECEPTOR EFFECTOR CELL SWITCHES WITH HUMANI... China 201780076966.5 6/12/2019 110267982 9/20/2019 Published Travis YOUNG, Leonard PRESTA, David RODGERS, Eric HAMPTON, Ti... 1924.1CN
CHIMERIC ANTIGEN RECEPTOR EFFECTOR CELL SWITCHES WITH HUMANI... Canada 3,040,343 10/19/2017 3040343 4/26/2018 Published Travis YOUNG, Leonard PRESTA, David RODGERS, Eric HAMPTON, Ti... 1924.1CA
CHIMERIC ANTIGEN RECEPTOR EFFECTOR CELL SWITCHES WITH HUMANI... United States 17/461,365 8/30/2021 20220073597 3/10/2022 Published Travis YOUNG, Leonard PRESTA, David RODGERS, Eric HAMPTON, Ti... 1924.1C1
CHIMERIC ANTIGEN RECEPTOR EFFECTOR CELL SWITCHES WITH HUMANI... Australia 2017345479 10/19/2017 2017345479 5/9/2019 Published Travis YOUNG, Leonard PRESTA, David RODGERS, Eric HAMPTON, Ti... 1924.1AU
CHIMERIC ANTIGEN RECEPTOR EFFECTOR CELL SWITCHES WITH HUMANI... United States 62/410,315 10/19/2016 Expired Travis YOUNG, Leonard PRESTA, David RODGERS, Eric HAMPTON, Ti... 1924.0P
OPTIMIZED PNE-BASED CHIMERIC RECEPTOR T CELL SWITCHES AND USES... United States 15/566,680 10/13/2017 20190169289 6/6/2019 11,091,546 8/17/2021 Issued Travis YOUNG, David RODGERS, Ian Hardy, Chanhyuk KIM, Peter G. S... 1923.2US
OPTIMIZED PNE-BASED CHIMERIC RECEPTOR T CELL SWITCHES AND USES... World Intellectual Property Organization PCT US2016/027997 4/15/2016 WO 16/168773 10/20/2016 Expired Eric HAMPTON, Travis YOUNG, David RODGERS, Ian Hardy, Peter G... 1923.2PC
OPTIMIZED PNE-BASED CHIMERIC RECEPTOR T CELL SWITCHES AND USES... Hong Kong 18110231.8 8/19/2018 HK1250661 1/11/2019 Published Eric HAMPTON, Travis YOUNG, David RODGERS, Ian Hardy, Chanhyu... 1923.2HK
OPTIMIZED PNE-BASED CHIMERIC RECEPTOR T CELL SWITCHES AND USES... European Patent Office 16780958.1 4/15/2016 3283113 2/21/2018 Published Travis YOUNG, David RODGERS, Ian Hardy, Chanhyuk KIM, Peter G. S... 1923.2EP
CHIMERIC RECEPTOR T CELL SWITCHES AND USES THEREOF United States 62/253,467 11/10/2015 Expired Travis YOUNG, David RODGERS, Ian Hardy, Chanhyuk KIM, Peter G. S... 1923.1P
OPTIMIZED CHIMERIC RECEPTOR CELL SWITCHES AND USES THEREOF United States 62/148,063 4/15/2015 Expired Travis YOUNG, David RODGERS, Ian Hardy, Chanhyuk KIM, Peter G. S... 1923.0P
CHIMERIC RECEPTOR T CELLS AND USES THEREOF United States 15/561,274 9/25/2017 20180118808 5/3/2018 10,800,828 10/13/2020 Issued Travis YOUNG, Chanhyuk KIM, Peter G. SCHULTZ 1922.1US
SWITCHABLE NON-scFv CHIMERIC RECEPTOR T CELLS AND USES THEREOF World Intellectual Property Organization PCT US2016/024252 3/28/2016 WO 16/154621 9/29/2016 Expired Travis YOUNG, Chanhyuk KIM, Peter G. SCHULTZ 1922.1PC
CHIMERIC RECEPTOR T CELLS AND USES THEREOF United States 62/138,901 3/26/2015 Expired Travis YOUNG, Chanhyuk KIM, Peter G. SCHULTZ 1922.0P
OPTIMIZED CHIMERIC RECEPTOR T CELL SWITCHES AND USES THEREOF United States 15/566,685 4/15/2016 Abandoned Chanhyuk KIM, Travis YOUNG, Jennifer MA, Ji Young KIM, Hui WANG... 1771.3US
OPTIMIZED CHIMERIC RECEPTOR T CELL SWITCHES AND USES THEREOF World Intellectual Property Organization PCT US2016/027990 4/15/2016 WO 16/168766 10/20/2016 Expired Chanhyuk KIM, Travis YOUNG, Jennifer MA, Ji Young KIM, Hui WANG... 1771.3PC
CHIMERIC RECEPTOR T CELL SWITCHES FOR HER2 World Intellectual Property Organization PCT US2016/027993 4/15/2016 WO 16/168769 10/20/2016 Expired Yu J. CAO, Travis YOUNG, Peter G. SCHULTZ 1771.2PC
CHIMERIC RECEPTOR T CELL SWITCHES FOR HER2 United States 62/253,465 11/10/2015 Expired Yu J. CAO, Travis YOUNG, Peter G. SCHULTZ 1771.1P
CHIMERIC RECEPTOR T CELL SWITCHES FOR HER2 United States 62/148,070 4/15/2015 Expired Yu J. CAO, Travis YOUNG, Peter G. SCHULTZ 1771.0P
PEPTIDIC CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THE... United States 18/056,554 11/17/2022 Pending Travis YOUNG, Chanhyuk KIM, Peter G. SCHULTZ 1666.6C
PEPTIDIC CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THE... United States 17/713,489 5/2022 Abandoned Travis YOUNG, Chanhyuk KIM, Peter G. SCHULTZ 1666.6C3
PEPTIDIC CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THE... United States 16/532,860 8/6/2019 20200197497 6/25/2020 Abandoned Travis YOUNG, Chanhyuk KIM, Peter G. SCHULTZ 1666.6C2
PEPTIDIC CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THE... United States 15/484,477 4/2/2017 20170246270 8/31/2017 10,391,155 8/27/2019 Issued Travis YOUNG, Chanhyuk KIM, Peter G. SCHULTZ 1666.6C1
PEPTIDIC CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THE... United States 14/688,899 4/16/2015 20150307564 10/29/2015 9,624,276 4/18/2017 Issued Travis YOUNG, Chanhyuk KIM, Peter G. SCHULTZ 1666.6
PEPTIDIC CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THE... World Intellectual Property Organization PCT US14/060684 10/15/2014 WO 15/057834 4/23/2015 Expired Travis YOUNG, Chanhyuk KIM, Peter G. SCHULTZ 1666.5PC
PEPTIDIC CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THE... Republic of Korea 10-2016-7012414 10/15/2014 20160062760 6/2/2016 10-2339240 12/9/2021 Issued Travis YOUNG, Chanhyuk KIM, Peter G. SCHULTZ 1666.5KR
PEPTIDIC CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THE... Japan 2020-037808 3/5/2020 20200196604 6/25/2020 Abandoned Travis YOUNG, Chanhyuk KIM, Peter G. SCHULTZ 1666.5JPD1
PEPTIDIC CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THE... Japan 2016-522782 10/15/2014 2016533174 10/27/2016 6734477 7/14/2020 Issued Travis YOUNG, Chanhyuk KIM, Peter G. SCHULTZ 1666.5JP
PEPTIDIC CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THE... Italy 14854285.5 10/15/2014 502020000012146 9/23/2020 Issued Travis YOUNG, Chanhyuk KIM, Peter G. SCHULTZ 1666.5IT
PEPTIDIC CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THE... Hong Kong 17100359.6 7/17/2023 1226751A 10/6/2017 Published Travis YOUNG, Chanhyuk KIM, Peter G. SCHULTZ 1666.5HK
PEPTIDIC CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THE... United Kingdom 14854285.5 10/15/2014 3057990 9/23/2020 Issued Travis YOUNG, Chanhyuk KIM, Peter G. SCHULTZ 1666.5GB
PEPTIDIC CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THE... France 14854285.5 10/15/2014 3057990 9/23/2020 Issued Travis YOUNG, Chanhyuk KIM, Peter G. SCHULTZ 1666.5FR
PEPTIDIC CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THE... Spain 14854285.5 10/15/2014 3057990 9/23/2020 Issued Travis YOUNG, Chanhyuk KIM, Peter G. SCHULTZ 1666.5ES
PEPTIDIC CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THE... European Patent Office 14854285.5 10/15/2014 3057990 8/24/2016 3057990 9/23/2020 Issued Travis YOUNG, Chanhyuk KIM, Peter G. SCHULTZ 1666.5EP
PEPTIDIC CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THE... Germany 14854285.5 10/15/2014 602014070576.6 9/23/2020 Issued Travis YOUNG, Chanhyuk KIM, Peter G. SCHULTZ 1666.5DE
PEPTIDIC CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THE... China 201480066872.6 10/15/2014 105829349 8/3/2016 ZL 201480066872.6 2/3/2023 Issued Travis YOUNG, Chanhyuk KIM, Peter G. SCHULTZ 1666.5CN
PEPTIDIC CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THE... Canada 2,927,543 10/15/2014 2927543 4/23/2015 2,927,543 7/20/2021 Issued Travis YOUNG, Chanhyuk KIM, Peter G. SCHULTZ 1666.5CA
PEPTIDIC CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THE... Australia 2020207804 10/15/2014 2020207804 8/6/2020 Abandoned Travis YOUNG, Chanhyuk KIM, Peter G. SCHULTZ 1666.5AUD1
PEPTIDIC CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THE... Australia 2014337367 10/15/2014 2014337367 4/7/2016 2014337367 8/13/2020 Issued Travis YOUNG, Chanhyuk KIM, Peter G. SCHULTZ 1666.5AU
CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THEREOF United States 14/432,065 3/27/2015 2015-0238631 8/27/2015 Abandoned Chanhyuk KIM, Travis YOUNG, Yu J. CAO, Jennifer MA, Minsoo KIM, St... 1666.4US
CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THEREOF World Intellectual Property Organization PCT US14/060713 10/15/2014 WO 15/057852 4/23/2015 Expired Chanhyuk KIM, Travis YOUNG, Yu J. CAO, Jennifer MA, Minsoo KIM, St... 1666.4PC
CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THEREOF Republic of Korea 10-2016-7012417 10/15/2014 20160062761 6/2/2016 10-2357968 1/26/2022 Issued Chanhyuk KIM, Travis YOUNG, Yu J. CAO, Jennifer MA, Minsoo KIM, St... 1666.4KR
CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THEREOF Japan 2019-186117 10/9/2019 2020015760 1/30/2020 Abandoned Chanhyuk KIM, Travis YOUNG, Yu J. CAO, Jennifer MA, Minsoo KIM, St... 1666.4JPD1
CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THEREOF Japan 2016-522791 10/15/2014 2016534995 11/10/2016 6637415 12/27/2019 Issued Chanhyuk KIM, Travis YOUNG, Yu J. CAO, Jennifer MA, Minsoo KIM, St... 1666.4JP
CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THEREOF Italy 14853242.7 10/15/2014 502019000006215 5/8/2019 Issued Chanhyuk KIM, Travis YOUNG, Yu J. CAO, Jennifer MA, Minsoo KIM, St... 1666.4IT
CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THEREOF Hong Kong 17100358.7 10/15/2014 HK1226750A 10/6/2017 Abandoned Chanhyuk KIM, Travis YOUNG, Yu J. CAO, Jennifer MA, Minsoo KIM, St... 1666.4HK
CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THEREOF United Kingdom 14853242.7 10/15/2014 3057991 5/8/2019 Issued Chanhyuk KIM, Travis YOUNG, Yu J. CAO, Jennifer MA, Minsoo KIM, St... 1666.4GB
CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THEREOF France 14853242.7 10/15/2014 3057991 5/8/2019 Issued Chanhyuk KIM, Travis YOUNG, Yu J. CAO, Jennifer MA, Minsoo KIM, St... 1666.4FR
CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THEREOF Spain 14853242.7 10/15/2014 3057991 5/8/2019 Issued Chanhyuk KIM, Travis YOUNG, Yu J. CAO, Jennifer MA, Minsoo KIM, St... 1666.4ES
CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THEREOF European Patent Office 14853242.7 10/15/2014 3057991 8/24/2016 3057991 5/8/2019 Issued Chanhyuk KIM, Travis YOUNG, Yu J. CAO, Jennifer MA, Minsoo KIM, St... 1666.4EP
CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THEREOF Germany 14853242.7 10/15/2014 602014046575.7 5/8/2019 Issued Chanhyuk KIM, Travis YOUNG, Yu J. CAO, Jennifer MA, Minsoo KIM, St... 1666.4DE
CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THEREOF China 201480064779.1 10/15/2014 105814083 7/27/2016 Abandoned Chanhyuk KIM, Travis YOUNG, Yu J. CAO, Jennifer MA, Minsoo KIM, St... 1666.4CN
CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THEREOF Canada 2,926,698 10/15/2014 2,926,698 4/23/2015 2,926,698 6/22/2021 Issued Chanhyuk KIM, Travis YOUNG, Yu J. CAO, Jennifer MA, Minsoo KIM, St... 1666.4CA
CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THEREOF United States 15/644,657 7/7/2017 201801044535 4/19/2018 Abandoned Chanhyuk KIM, Travis YOUNG, Yu J. CAO, Jennifer MA, Minsoo KIM, St... 1666.4C2
CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THEREOF United States 15/363,350 11/29/2016 201801044535 Abandoned Chanhyuk KIM, Travis YOUNG, Yu J. CAO, Jennifer MA, Minsoo KIM, St... 1666.4C1
CHIMERIC ANTIGEN RECEPTOR T CELL SWITCHES AND USES THEREOF Australia 2014337385 10/15/2014 2014337385 4/7/2016 2014337385 8/13/2020 Issued Chanhyuk KIM, Travis YOUNG, Yu J. CAO, Jennifer MA, Minsoo KIM, St... 1666.4AU
CHIMERIC ANTIGEN RECEPTOR T CELLS AND USES THEREOF United States 62/009,056 6/6/2014 Abandoned Yu J. CAO, Chanhyuk KIM, Peter G. SCHULTZ, Travis YOUNG, Jennifer... 1666.2P
METHODS OF PRODUCING SWITCHABLE CHIMERIC ANTIGEN RECEPTOR T C... United States 61/895,704 10/25/2013 Abandoned Yu J. CAO, Chanhyuk KIM, Peter G. SCHULTZ, Travis YOUNG 1666.1P
METHODS OF PRODUCING SWITCHABLE CHIMERIC ANTIGEN RECEPTOR T C... United States 61/891,347 10/15/2013 Abandoned Yu J. CAO, Chanhyuk KIM, Peter G. SCHULTZ, Travis YOUNG 1666.0P