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Tetracyclines: Concomitant treatment with Accutane and tetracyclines should be avoided because Accutane use has been associated with a number of cases of pseudotumor cerebri (benign intracranial hypertension), some of which involved concomitant use of tetracyclines
Accutane
tetracyclines
ADVISE
Isotretinoin_ddi.xml
DDI-DrugBank.d163.s2
DDI-DrugBank.d163.s2.p4
In order to maintain phenytoin levels, limit adverse experiences, and achieve the felbamate dose of 3600 mg/day, a phenytoin dose reduction of approximately 40% was necessary for eight of these 10 subjects.
felbamate
phenytoin
ADVISE
Felbamate_ddi.xml
DDI-DrugBank.d434.s15
DDI-DrugBank.d434.s15.p2
Acellular, live and live-attenuated vaccines should not be administered during RAPTIVA treatment.
live vaccines
RAPTIVA
ADVISE
Efalizumab_ddi.xml
DDI-DrugBank.d44.s2
DDI-DrugBank.d44.s2.p4
ketoconazole), macrolide antibiotics (e.g. erythromycin), and HIV protease inhibitors (e.g. ritonavir, indinavir and saquinavir) should have their dose of SUBUTEX or SUBOXONE adjusted.
ketoconazole
indinavir
NONE
Buprenorphine_ddi.xml
DDI-DrugBank.d380.s2
DDI-DrugBank.d380.s2.p4
Etonogestrel may interact with the following medications: acetaminophen (Tylenol), antibiotics such as ampicillin and tetracycline, anticonvulsants (Dilantin, Phenobarbital, Tegretol, Trileptal, Topamax, Felbatol), antifungals (Gris-PEG, Nizoral, Sporanox), atorvastatin (Lipitor), clofibrate (Atromid-S), cyclosporine (Neoral, Sandimmune), HIV drugs classified as protease inhibitors (Agenerase, Crixivan, Fortovase, Invirase, Kaletra, Norvir, Viracept), morphine (Astramorph, Kadian, MS Contin), phenylbutazone, prednisolone (Prelone), rifadin (rifampin), St. Johns wort, temazepam, theophylline (Theo-Dur), and vitamin C.
anticonvulsants
Sporanox
NONE
Etonogestrel_ddi.xml
DDI-DrugBank.d484.s0
DDI-DrugBank.d484.s0.p258
FLEXERIL may enhance the effects of alcohol, barbiturates, and other CNS depressants.
alcohol
CNS depressants
NONE
Cyclobenzaprine_ddi.xml
DDI-DrugBank.d150.s1
DDI-DrugBank.d150.s1.p4
Drugs that reportedly may increase oral anticoagulant response, ie, increased prothrombin response, in man include:alcohol*;allopurinol;aminosalicylic acid;amiodarone;anabolic steroids;antibiotics;bromelains;chloral hydrate*;chlorpropamide;chymotrypsin;cimetidine;cinchophen;clofibrate;dextran;dextrothyroxine;diazoxide;dietary deficiencies;diflunisal;disulfiram;drugs affecting blood elements;ethacrynic acid;fenoprofen;glucagon;hepatotoxic drugs;ibuprofen;indomethacin;influenza virus vaccine;inhalation anesthetics;mefenamic acid;methyldopa;methylphenidate;metronidazole;miconazole;monoamine oxidase inhibitors;nalidixic acid;naproxen;oxolinic acid;oxyphenbutazone;pentoxifylline;phenylbutazone;phenyramidol;phenytoin;prolonged hot weather;prolonged narcotics;pyrazolones;quinidine;quinine;ranitidine*;salicylates;sulfinpyrazone;sulfonamides, long acting;sulindac;thyroid drugs;tolbutamide;triclofos sodium;trimethoprim/sulfamethoxazole;unreliable prothrombin time determinations;warfarin sodium overdosage.
quinine
warfarin sodium
NONE
Anisindione_ddi.xml
DDI-DrugBank.d64.s87
DDI-DrugBank.d64.s87.p1429
When digoxin and BREVIBLOC were concomitantly administered intravenously to normal volunteers, there was a 10-20% increase in digoxin blood levels at some time points.
digoxin
BREVIBLOC
MECHANISM
Esmolol_ddi.xml
DDI-DrugBank.d422.s4
DDI-DrugBank.d422.s4.p0
DOSTINEX should not be administered concurrently with D2-antagonists, such as phenothiazines, butyrophenones, thioxanthines, or metoclopramide.
DOSTINEX
thioxanthines
ADVISE
Cabergoline_ddi.xml
DDI-DrugBank.d282.s0
DDI-DrugBank.d282.s0.p2
Nonetheless, the range of individual Simulect clearance values in the presence of azathioprine (12-57 mL/h) or mycophenolate mofetil (7-54 mL/h) did not extend outside the range observed with dual therapy (10-78 mL/h).
Simulect
mycophenolate mofetil
NONE
Basiliximab_ddi.xml
DDI-DrugBank.d544.s4
DDI-DrugBank.d544.s4.p1
Amphotericin B injection and potassium-depleting agents: When corticosteroids are administered concomitantly with potassium-depleting agents (e.g., amphotericin B, diuretics), patients should be observed closely for development of hypokalemia.
corticosteroids
diuretics
ADVISE
Dexamethasone_ddi.xml
DDI-DrugBank.d314.s1
DDI-DrugBank.d314.s1.p4
Agents that have been found, or are expected to have decreased plasma levels in the presence of EQUETROTM due to induction of CYP enzymes are the following: Acetaminophen, alprazolam, amitriptyline, bupropion, buspirone, citalopram, clobazam, clonazepam, clozapine, cyclosporin, delavirdine, desipramine, diazepam, dicumarol, doxycycline, ethosuximide, felbamate, felodipine, glucocorticoids, haloperidol, itraconazole, lamotrigine, levothyroxine, lorazepam, methadone, midazolam, mirtazapine, nortriptyline, olanzapine, oral contraceptives(3), oxcarbazepine, Phenytoin(4), praziquantel, protease inhibitors, quetiapine, risperidone, theophylline, topiramate, tiagabine, tramadol, triazolam, valproate, warfarin(5) , ziprasidone, and zonisamide.
felodipine
mirtazapine
NONE
Carbamazepine_ddi.xml
DDI-DrugBank.d94.s11
DDI-DrugBank.d94.s11.p665
Before taking glimepiride, tell your doctor if you are taking any of the following medicines: - aspirin or another salicylate such as magnesium/choline salicylate (Trilisate), salsalate (Disalcid, others), choline salicylate (Arthropan), magnesium salicylate (Magan), or bismuth subsalicylate (Pepto-Bismol);
magnesium salicylate
bismuth subsalicylate
NONE
Glimepiride_ddi.xml
DDI-DrugBank.d521.s1
DDI-DrugBank.d521.s1.p73
Quinidine at 648 mg bid decreased the bioavailability (AUC) of nisoldipine by 26%, but not the peak concentration.
Quinidine
nisoldipine
MECHANISM
Nisoldipine_ddi.xml
DDI-DrugBank.d106.s8
DDI-DrugBank.d106.s8.p0
Antibiotics (e.g., erythromycin, trimethoprim and sulfamethoxazole, amoxicillin).
Antibiotics
amoxicillin
NONE
Doxazosin_ddi.xml
DDI-DrugBank.d367.s11
DDI-DrugBank.d367.s11.p3
Bacteriostatic Antibiotics: Chloramphenicol, erythromycins, sulfonamides, or tetracyclines may interfere with the bactericidal effect of penicillins.
erythromycins
penicillins
EFFECT
Ampicillin_ddi.xml
DDI-DrugBank.d211.s2
DDI-DrugBank.d211.s2.p11
Phenobarbital toxicity has been reported to have occurred in a patient on chronic phenobarbital treatment following the initiation of diclofenac therapy.
phenobarbital
diclofenac
EFFECT
Diclofenac_ddi.xml
DDI-DrugBank.d249.s17
DDI-DrugBank.d249.s17.p2
Based on total ertapenem concentrations, probenecid increased the AUC by 25% and reduced the plasma and renal clearances by 20% and 35%, respectively.
ertapenem
probenecid
MECHANISM
Ertapenem_ddi.xml
DDI-DrugBank.d329.s1
DDI-DrugBank.d329.s1.p0
Antihypertensives: Amphetamines may antagonize the hypotensive effects of antihypertensives.
Amphetamines
antihypertensives
EFFECT
Dextroamphetamine_ddi.xml
DDI-DrugBank.d236.s15
DDI-DrugBank.d236.s15.p2
Agents that have been found, or are expected to have decreased plasma levels in the presence of EQUETROTM due to induction of CYP enzymes are the following: Acetaminophen, alprazolam, amitriptyline, bupropion, buspirone, citalopram, clobazam, clonazepam, clozapine, cyclosporin, delavirdine, desipramine, diazepam, dicumarol, doxycycline, ethosuximide, felbamate, felodipine, glucocorticoids, haloperidol, itraconazole, lamotrigine, levothyroxine, lorazepam, methadone, midazolam, mirtazapine, nortriptyline, olanzapine, oral contraceptives(3), oxcarbazepine, Phenytoin(4), praziquantel, protease inhibitors, quetiapine, risperidone, theophylline, topiramate, tiagabine, tramadol, triazolam, valproate, warfarin(5) , ziprasidone, and zonisamide.
felbamate
haloperidol
NONE
Carbamazepine_ddi.xml
DDI-DrugBank.d94.s11
DDI-DrugBank.d94.s11.p631
Meperidine: Amphetamines potentiate the analgesic effect of meperidine.
Amphetamines
meperidine
EFFECT
Dextroamphetamine_ddi.xml
DDI-DrugBank.d236.s20
DDI-DrugBank.d236.s20.p2
Caution is advised in patients receiving concomitant high-dose aspirin and carbonic anhydrase inhibitors, as anorexia, tachypnea, lethargy and coma have been rarely reported due to a possible drug interaction.
aspirin
carbonic anhydrase inhibitors
ADVISE
Dichlorphenamide_ddi.xml
DDI-DrugBank.d36.s0
DDI-DrugBank.d36.s0.p0
Furosemide: Clinical studies, as well as post-marketing observations, have shown that NSAIDs can reduce the natriuretic effect of furosemide and thiazides in some patients.
NSAIDs
furosemide
EFFECT
Rofecoxib_ddi.xml
DDI-DrugBank.d210.s13
DDI-DrugBank.d210.s13.p3
Etonogestrel may interact with the following medications: acetaminophen (Tylenol), antibiotics such as ampicillin and tetracycline, anticonvulsants (Dilantin, Phenobarbital, Tegretol, Trileptal, Topamax, Felbatol), antifungals (Gris-PEG, Nizoral, Sporanox), atorvastatin (Lipitor), clofibrate (Atromid-S), cyclosporine (Neoral, Sandimmune), HIV drugs classified as protease inhibitors (Agenerase, Crixivan, Fortovase, Invirase, Kaletra, Norvir, Viracept), morphine (Astramorph, Kadian, MS Contin), phenylbutazone, prednisolone (Prelone), rifadin (rifampin), St. Johns wort, temazepam, theophylline (Theo-Dur), and vitamin C.
clofibrate
Atromid-S
NONE
Etonogestrel_ddi.xml
DDI-DrugBank.d484.s0
DDI-DrugBank.d484.s0.p665
Certain drugs, including nonsteroidal anti-inflammatory agents (NSAIDs), salicylates, monoamine oxidase inhibitors, and non-selective beta-adrenergic-blocking agents may potentiate the hypoglycemic action of Starlix and other oral antidiabetic drugs.
salicylates
Starlix
EFFECT
Nateglinide_ddi.xml
DDI-DrugBank.d460.s14
DDI-DrugBank.d460.s14.p13
Corticosteroids may increase the clearance of chronic high dose aspirin.
Corticosteroids
aspirin
EFFECT
Cortisone acetate_ddi.xml
DDI-DrugBank.d487.s4
DDI-DrugBank.d487.s4.p0
Other drugs Drug interactions have been reported with concomitant administration of erythromycin and other medications, including cyclosporine, hexobarbital, carbamazepine, alfentanil, disopyramide, phenytoin, bromocriptine, valproate, astemizole, and lovastatin.
bromocriptine
lovastatin
NONE
Dirithromycin_ddi.xml
DDI-DrugBank.d522.s24
DDI-DrugBank.d522.s24.p51
Agents that are CYP3A4 inhibitors that have been found, or are expected, to increase plasma levels of EQUETROTM are the following: Acetazolamide, azole antifungals, cimetidine, clarithromycin(1), dalfopristin, danazol, delavirdine, diltiazem, erythromycin(1), fluoxetine, fluvoxamine, grapefruit juice, isoniazid, itraconazole, ketoconazole, loratadine, nefazodone, niacinamide, nicotinamide, protease inhibitors, propoxyphene, quinine, quinupristin, troleandomycin, valproate(1), verapamil, zileuton.
nicotinamide
quinupristin
NONE
Carbamazepine_ddi.xml
DDI-DrugBank.d94.s4
DDI-DrugBank.d94.s4.p318
Both ibogaine and 18-MC block morphine-induced and nicotine-induced dopamine release in the nucleus accumbens;
18-MC
nicotine
EFFECT
11085336.xml
DDI-MedLine.d110.s6
DDI-MedLine.d110.s6.p4
Two different types of therapy with magnesium are used: physiological oral magnesium supplementation which is totally atoxic since it palliates magnesium deficiencies by simply normalizing the magnesium intake and pharmacological magnesium therapy which may induce toxicity since it creates iatrogenic magnesium overload.
magnesium
magnesium
NONE
7786695.xml
DDI-MedLine.d103.s1
DDI-MedLine.d103.s1.p10
Antagonism between lincomycin and erythromycin in vitro has been demonstrated.
lincomycin
erythromycin
EFFECT
Lincomycin_ddi.xml
DDI-DrugBank.d130.s2
DDI-DrugBank.d130.s2.p0
Certain drugs, including nonsteroidal anti-inflammatory agents (NSAIDs), salicylates, monoamine oxidase inhibitors, and non-selective beta-adrenergic-blocking agents may potentiate the hypoglycemic action of Starlix and other oral antidiabetic drugs.
monoamine oxidase inhibitors
antidiabetic drugs
EFFECT
Nateglinide_ddi.xml
DDI-DrugBank.d460.s14
DDI-DrugBank.d460.s14.p17
Patients taking REVIA may not benefit from opioid containing medicines, such as cough and cold preparations, antidiarrheal preparations, and opioid analgesics.
REVIA
opioid analgesics
EFFECT
Naltrexone_ddi.xml
DDI-DrugBank.d346.s4
DDI-DrugBank.d346.s4.p1
Hydrocodone increases gabapentin AUC values by 14%.
Hydrocodone
gabapentin
MECHANISM
Gabapentin_ddi.xml
DDI-DrugBank.d438.s24
DDI-DrugBank.d438.s24.p0
Analgesic/anti-inflammatory (e.g., acetaminophen, aspirin, codeine and codeine combinations, ibuprofen, indomethacin).
anti-inflammatory
ibuprofen
NONE
Doxazosin_ddi.xml
DDI-DrugBank.d367.s9
DDI-DrugBank.d367.s9.p11
The most commonly occurring drug interactions are listed below: - Drugs that may increase plasma phenytoin concentrations include: acute alcohol intake, amiodarone, chboramphenicol, chlordiazepoxide, cimetidine, diazepam, dicumarol, disulfiram, estrogens, ethosuximide, fluoxetine, H2-antagonists, halothane, isoniazid, methylphenidate, phenothiazines, phenylbutazone, salicylates, succinimides, sulfonamides, tolbutamide, trazodone
ethosuximide
fluoxetine
NONE
Fosphenytoin_ddi.xml
DDI-DrugBank.d40.s10
DDI-DrugBank.d40.s10.p153
Dexamethasone: Steady-state trough concentrations of albendazole sulfoxide were about 56% higher when 8 mg dexamethasone was coadministered with each dose of albendazole (15 mg/kg/day) in eight neurocysticercosis patients.
dexamethasone
albendazole
MECHANISM
Albendazole_ddi.xml
DDI-DrugBank.d321.s0
DDI-DrugBank.d321.s0.p5
Tricyclic antidepressants have been reported to blunt the hypotensive effect of systemic clonidine.
Tricyclic antidepressants
clonidine
EFFECT
Apraclonidine_ddi.xml
DDI-DrugBank.d224.s2
DDI-DrugBank.d224.s2.p0
Other depressasnts such as alcohol, barbiturates, and MAOIs may enhance CNS depression when administered with ethchlorvynol.
barbiturates
ethchlorvynol
EFFECT
Ethchlorvynol_ddi.xml
DDI-DrugBank.d405.s1
DDI-DrugBank.d405.s1.p4
Nelfinavir steady-state Cmax, A.C. and Cmin were increased by 12%, 15%, and 14%, respectively, by concomitant amprenavir.
Nelfinavir
amprenavir
MECHANISM
Amprenavir_ddi.xml
DDI-DrugBank.d437.s8
DDI-DrugBank.d437.s8.p0
Coadministration of NIZORAL Tablets with midazolam or triazolam has resulted in elevated plasma concentrations of the latter two drugs.
NIZORAL
triazolam
MECHANISM
Ketoconazole_ddi.xml
DDI-DrugBank.d458.s12
DDI-DrugBank.d458.s12.p1
Diazepam at doses of 0.25 mg/kg and 2.5 mg/kg injected with morphine was found to decrease the antinociceptive effect of morphine.
Diazepam
morphine
EFFECT
11210678.xml
DDI-MedLine.d67.s5
DDI-MedLine.d67.s5.p0
- Phenothiazines (acetophenazine [e.g., Tindal], chlorpromazine [e.g., Thorazine], fluphenazine [e.g., Prolixin], mesoridazine [e.g., Serentil], perphenazine [e.g., Trilafon], prochlorperazine [e.g., Compazine], promazine [e.g., Sparine], promethazine [e.g., Phenergan], thioridazine [e.g., Mellaril], trifluoperazine [e.g., Stelazine], triflupromazine [e.g., Vesprin], trimeprazine [e.g., Temaril]) or
Prolixin
trimeprazine
NONE
Sulfapyridine_ddi.xml
DDI-DrugBank.d179.s21
DDI-DrugBank.d179.s21.p145
Other drugs which may enhance the neuromuscular blocking action of nondepolarizing agents such as NIMBEX include certain antibiotics (e. g., aminoglycosides, tetracyclines, bacitracin, polymyxins, lincomycin, clindamycin, colistin, and sodium colistemethate), magnesium salts, lithium, local anesthetics, procainamide, and quinidine.
procainamide
quinidine
NONE
Cisatracurium Besylate_ddi.xml
DDI-DrugBank.d60.s12
DDI-DrugBank.d60.s12.p119
When used in therapeutic doses, azithromycin had a modest effect on the pharmacokinetics of atorvastatin, carbamazepine, cetirizine, didanosine, efavirenz, fluconazole, indinavir, midazolam, rifabutin, sildenafil, theophylline (intravenous and oral), triazolam, trimethoprim/sulfamethoxazole or zidovudine.
azithromycin
indinavir
MECHANISM
Azithromycin_ddi.xml
DDI-DrugBank.d53.s7
DDI-DrugBank.d53.s7.p6
or with multivitamins containing zinc may substantially interfere with drug absorption and result in insufficient plasma and tissue quinolone concentrations.
zinc
quinolone
MECHANISM
Enoxacin_ddi.xml
DDI-DrugBank.d395.s16
DDI-DrugBank.d395.s16.p2
Quinolones, including norfloxacin, may enhance the effects of oral anticoagulants, including warfarin or its derivatives or similar agents.
Quinolones
warfarin
EFFECT
Norfloxacin_ddi.xml
DDI-DrugBank.d217.s5
DDI-DrugBank.d217.s5.p2
Combination hormonal contraceptives may also decrease the plasma concentration of acetaminophen.
hormonal contraceptives
acetaminophen
MECHANISM
Ethynodiol Diacetate_ddi.xml
DDI-DrugBank.d485.s3
DDI-DrugBank.d485.s3.p0
Sympathomimetic amines may reduce the antihypertensive effects of reserpine, veratrum alkaloids, methyldopa and mecamylamine.
Sympathomimetic amines
methyldopa
EFFECT
Carbinoxamine_ddi.xml
DDI-DrugBank.d389.s2
DDI-DrugBank.d389.s2.p2
Oxytocin or other oxytocics (concurrent use with dinoprost may result in uterine hypertonus, possibly causing uterine rupture or cervical laceration, especially in the absence of adequate cervical dilatation;
Oxytocin
dinoprost
EFFECT
Dinoprost Tromethamine_ddi.xml
DDI-DrugBank.d181.s0
DDI-DrugBank.d181.s0.p1
Based on the chemical resemblance of itraconazole and ketoconazole, coadministration of astemizole with itraconazole is contraindicated.
astemizole
itraconazole
ADVISE
Itraconazole_ddi.xml
DDI-DrugBank.d165.s6
DDI-DrugBank.d165.s6.p5
Drugs that have been reported to diminish oral anticoagulant response, ie, decreased prothrom-bin time response, in man significantly include: adrenocortical steroids;
anticoagulant
adrenocortical steroids
EFFECT
Anisindione_ddi.xml
DDI-DrugBank.d64.s6
DDI-DrugBank.d64.s6.p0
Praziquantel: In the fed state, praziquantel (40 mg/kg) increased mean maximum plasma concentration and area under the curve of albendazole sulfoxide by about 50% in healthy subjects (n=10) compared with a separate group of subjects (n=6) given albendazole alone.
praziquantel
albendazole sulfoxide
MECHANISM
Albendazole_ddi.xml
DDI-DrugBank.d321.s1
DDI-DrugBank.d321.s1.p3
Aspirin: Concomitant administration of diclofenac and aspirin is not recommended because diclofenac is displaced from its binding sites during the concomitant administration of aspirin, resulting in lower plasma concentrations, peak plasma levels, and AUC values.
diclofenac
aspirin
MECHANISM
Diclofenac_ddi.xml
DDI-DrugBank.d249.s0
DDI-DrugBank.d249.s0.p9
Nafazodone, fluvoxamine, cimetidine (consider Xanax dose reduction).
fluvoxamine
Xanax
ADVISE
Adinazolam_ddi.xml
DDI-DrugBank.d449.s1
DDI-DrugBank.d449.s1.p4
These results suggest that both dexamethasone and retinyl acetate, and possibly other glucocorticoids and retinoids, may regulate the proliferation of prostate epithelium by a dose-dependent modification of the activity of insulin and EGF.
dexamethasone
insulin
EFFECT
3881461.xml
DDI-MedLine.d12.s7
DDI-MedLine.d12.s7.p3
Methamphetamine, like MPTP, produced depletions of striatal dopamine but these actions were potentiated by pargyline pretreatment.
Methamphetamine
pargyline
EFFECT
3871245.xml
DDI-MedLine.d73.s4
DDI-MedLine.d73.s4.p1
Propantheline and diphenoxylate, by decreasing gut motility, may increase digoxin absorption.
diphenoxylate
digoxin
MECHANISM
Digoxin_ddi.xml
DDI-DrugBank.d450.s5
DDI-DrugBank.d450.s5.p2
Drugs that have been reported to diminish oral anticoagulant response, ie, decreased prothrom-bin time response, in man significantly include: adrenocortical steroids;alcohol*;antacids;antihistamines;barbiturates;carbamazepine;chloral hydrate*;chlordiazepoxide;cholestyramine;diet high in vitamin K;diuretics*;ethchlorvynol;glutethimide;griseofulvin;haloperidol;meprobamate;oral contraceptives;paraldehyde;primidone;ranitidine*;rifampin;unreliable prothrombin time determinations;vitamin C;warfarin sodium under-dosage.
anticoagulant
griseofulvin
EFFECT
Anisindione_ddi.xml
DDI-DrugBank.d64.s29
DDI-DrugBank.d64.s29.p13
Concomitant administration of Targretin capsules and gemfibrozil resulted in substantial increases in plasma concentrations of bexarotene, probably at least partially related to cytochrome P450 3A4 inhibition by gemfibrozil.
Targretin
gemfibrozil
MECHANISM
Bexarotene_ddi.xml
DDI-DrugBank.d467.s4
DDI-DrugBank.d467.s4.p0
However, appropriate monitoring of blood glucose should be performed when initiating EXTRANEAL in diabetic patients and insulin dosage should be adjusted if needed.
EXTRANEAL
insulin
ADVISE
Icodextrin_ddi.xml
DDI-DrugBank.d501.s6
DDI-DrugBank.d501.s6.p0
Therefore, co-administration of tricyclic antidepressants with other drugs that are metabolized by this isoenzyme, including other antidepressants, phenothiazines, carbamazepine, and Type 1C antiarrhythmics (eg, propafenone, flecainide, and encainide), or that inhibit this enzyme (eg, quinidine), should be approached with caution.
tricyclic antidepressants
carbamazepine
ADVISE
Nortriptyline_ddi.xml
DDI-DrugBank.d202.s16
DDI-DrugBank.d202.s16.p2
SINCE CHOLESTYRAMINE RESIN MAY BIND OTHER DRUGS GIVEN CONCURRENTLY, IT IS RECOMMENDED THAT PATIENTS TAKE OTHER DRUGS AT LEAST 1 HOUR BEFORE OR 4 TO 6 HOURS AFTER CHOLESTYRAMINE RESIN (OR AT AS GREAT AN INTERVAL AS POSSIBLE) TO AVOID IMPEDING THEIR ABSORPTION.
RESIN
RESIN
NONE
Cholestyramine_ddi.xml
DDI-DrugBank.d566.s5
DDI-DrugBank.d566.s5.p4
fluoxetine, fluvoxamine, paroxetine, sertraline).
paroxetine
sertraline
NONE
Dihydroergotamine_ddi.xml
DDI-DrugBank.d410.s8
DDI-DrugBank.d410.s8.p5
Since Zarontin (ethosuximide) may interact with concurrently administered antiepileptic drugs, periodic serum level determinations of these drugs may be necessary (eg, ethosuximide may elevate phenytoin serum levels and valproic acid has been reported to both increase and decrease ethosuximide levels).
ethosuximide
phenytoin
MECHANISM
Ethosuximide_ddi.xml
DDI-DrugBank.d205.s0
DDI-DrugBank.d205.s0.p15
Beta Blockers: Although the results of a clinical study did not indicate a safe problem associated with the administration of D.H.E. 45 (dihydroergotamine mesylate) Injection, USP to subjects already receiving propranolol, there have been reports that propranolol may potentiate the vasoconstrictive action of ergotamine by blocking the vasodilating property of epinephrine.
propranolol
ergotamine
EFFECT
Dihydroergotamine_ddi.xml
DDI-DrugBank.d410.s3
DDI-DrugBank.d410.s3.p14
No interactions have been observed between nizatidine and theophylline, chlordiazepoxide, lorazepam, lidocaine, phenytoin, and warfarin.
chlordiazepoxide
warfarin
NONE
Nizatidine_ddi.xml
DDI-DrugBank.d475.s0
DDI-DrugBank.d475.s0.p14
WelChol decreased the Cmax and AUC of sustained-release verapamil (Calan SR ) by approximately 31% and 11%, respectively.
WelChol
Calan SR
MECHANISM
Colesevelam_ddi.xml
DDI-DrugBank.d551.s2
DDI-DrugBank.d551.s2.p1
Although specific studies have not been performed, coadministration with drugs that are mainly metabolized by CYP3A4 (eg, calcium channel blockers, dapsone, disopyramide, quinine, amiodarone, quinidine, warfarin, tacrolimus, cyclosporine, ergot derivatives, pimozide, carbamazepine, fentanyl, alfentanyl, alprazolam, and triazolam) may have elevated plasma concentrations when coadministered with saquinavir;
cyclosporine
saquinavir
MECHANISM
Saquinavir_ddi.xml
DDI-DrugBank.d124.s26
DDI-DrugBank.d124.s26.p107
Antiepileptic Drugs: Sporadic cases of seizures have been reported during concomitant use of TORADOL and antiepileptic drugs (phenytoin, carbamazepine).
TORADOL
carbamazepine
EFFECT
Ketorolac_ddi.xml
DDI-DrugBank.d3.s18
DDI-DrugBank.d3.s18.p6
Echistatin alone had no effect on tyrosine phosphorylation in T24 cells, but dose-dependently inhibits the effects of contortrostatin when both are added simultaneously.
Echistatin
contortrostatin
EFFECT
10978746.xml
DDI-MedLine.d69.s3
DDI-MedLine.d69.s3.p0
Co-administration of lovastatin, atenolol, warfarin, furosemide, digoxin, celecoxib, hydrochlorothiazide, ramipril, valsartan, metformin and amlodipine did not result in clinically significant increases in aliskiren exposure.
valsartan
amlodipine
NONE
Aliskiren_ddi.xml
DDI-DrugBank.d533.s1
DDI-DrugBank.d533.s1.p61
Serious anticholinergic symptoms (i.e., severe dry mouth, urinary retention and blurred vision) have been associated with elevations in the serum levels of tricyclic antidepressant when cimetidine therapy is initiated.
tricyclic antidepressant
cimetidine
EFFECT
Doxepin_ddi.xml
DDI-DrugBank.d223.s23
DDI-DrugBank.d223.s23.p0
Bentiromide may interact with acetaminophen (e.g., Tylenol), chloramphenicol (e.g., Chloromycetin), local anesthetics (e.g., benzocaine and lidocaine), para-aminobenzoic acid (PABA)-containing preparations (e.g., sunscreens and some multivitamins), procainamide (e.g., Pronestyl), sulfonamides (sulfa medicines), thiazide diuretics (use of these medicines during the test period will affect the test results), and pancreatic supplements (use of pancreatic supplements may give false test results).
lidocaine
multivitamins
NONE
Bentiromide_ddi.xml
DDI-DrugBank.d537.s0
DDI-DrugBank.d537.s0.p79
Because fluvoxamine reduces the clearance of both diazepam and its active metabolite, N-desmethyldiazepam, there is a strong likelihood of substantial accumulation of both species during chronic co-administration.
fluvoxamine
diazepam
MECHANISM
Fluvoxamine_ddi.xml
DDI-DrugBank.d76.s20
DDI-DrugBank.d76.s20.p0
The concurrent use of two or more drugs with anticholinergic activity--such as an antipsychotic drug (eg, chlorpromazine), an antiparkinsonian drug (eg, trihexyphenidyl), and/or a tricyclic antidepressant (eg, amitriptyline)--commonly results in excessive anticholinergic effects, including dry mouth and associated dental complications, blurred vision, and, in patients exposed to high temperature and humidity, hyperpyrexia.
chlorpromazine
tricyclic antidepressant
EFFECT
Chlorpromazine_ddi.xml
DDI-DrugBank.d86.s0
DDI-DrugBank.d86.s0.p7
Cyclosporine, hexobarbital and phenytoin concentrations.
Cyclosporine
phenytoin
NONE
Azithromycin_ddi.xml
DDI-DrugBank.d53.s15
DDI-DrugBank.d53.s15.p1
Laboratory Tests: The combination of Amprenavir and low-dose ritonavir has been associated with elevations of cholesterol and triglycerides, SGOT (AST), and SGPT (ALT) in some patients.
Amprenavir
ritonavir
EFFECT
Amprenavir_ddi.xml
DDI-DrugBank.d437.s13
DDI-DrugBank.d437.s13.p0
If nifedipine therapy is initiated in a patient currently receiving cimetidine, cautious titration is advised.
nifedipine
cimetidine
ADVISE
Nifedipine_ddi.xml
DDI-DrugBank.d373.s14
DDI-DrugBank.d373.s14.p0
Warfarin, Digoxin, Salicylate, and Heparin The in vitro binding of warfarin to plasma proteins is only slightly reduced by ketorolac tromethamine (99.5% control vs 99.3%) when ketorolac plasma concentrations reach 5 to10 m g/mL.
warfarin
ketorolac tromethamine
MECHANISM
Ketorolac_ddi.xml
DDI-DrugBank.d3.s1
DDI-DrugBank.d3.s1.p18
Cytochrome P-450 inducers, such as phenytoin, carbamazepine and phenobarbital, induce clonazepam metabolism, causing an approximately 30% decrease in plasma clonazepam levels.
phenobarbital
clonazepam
MECHANISM
Clonazepam_ddi.xml
DDI-DrugBank.d333.s5
DDI-DrugBank.d333.s5.p7
Because of foscarnets tendency to cause renal impairment, the use of FOSCAVIR should be avoided in combination with potentially nephrotoxic drugs such as aminoglycosides, amphotericin B and intravenous pentamidine unless the potential benefits outweigh the risks to the patient.
FOSCAVIR
amphotericin B
ADVISE
Foscarnet_ddi.xml
DDI-DrugBank.d511.s4
DDI-DrugBank.d511.s4.p5
Lithium: Diclofenac decreases lithium renal clearance and increases lithium plasma levels.
Diclofenac
lithium
MECHANISM
Diclofenac_ddi.xml
DDI-DrugBank.d249.s8
DDI-DrugBank.d249.s8.p3
Plasma TCA concentrations may need to be monitored and the dose of the TCA may need to be reduced if a TCA is co-administered with Duloxetine.
TCA
Duloxetine
ADVISE
Duloxetine_ddi.xml
DDI-DrugBank.d548.s10
DDI-DrugBank.d548.s10.p5
Macrolide Antibiotics (e. g. erythromycin and troleandomycin): Agents of the ergot alkaloid class, of which D.H.E. 45 (dihydroergotamine mesylate) Injection, USP is a member, have been shown to interact with antibiotics of the macrolide class, resulting in increased plasma levels of unchanged alkaloids and peripheral vasoconstriction.
dihydroergotamine mesylate
macrolide class
MECHANISM
Dihydroergotamine_ddi.xml
DDI-DrugBank.d410.s5
DDI-DrugBank.d410.s5.p26
In general, these are drugs that have one or more pharmacologic activities similar to bepridil hydrochloride, including anti-arrhythmic agents such as quinidine and procainamide, cardiac glycosides and tricyclic anti-depressants.
quinidine
tricyclic anti-depressants
NONE
Bepridil_ddi.xml
DDI-DrugBank.d137.s9
DDI-DrugBank.d137.s9.p11
Products containing calcium and other multivalent cations (such as aluminum, magnesium, iron) are likely to interfere with absorption of Ibandronate.
calcium
iron
NONE
Ibandronate_ddi.xml
DDI-DrugBank.d440.s1
DDI-DrugBank.d440.s1.p2
Other drugs which may enhance the neuromuscular blocking action of nondepolarizing agents such as NIMBEX include certain antibiotics (e. g., aminoglycosides, tetracyclines, bacitracin, polymyxins, lincomycin, clindamycin, colistin, and sodium colistemethate), magnesium salts, lithium, local anesthetics, procainamide, and quinidine.
NIMBEX
aminoglycosides
EFFECT
Cisatracurium Besylate_ddi.xml
DDI-DrugBank.d60.s12
DDI-DrugBank.d60.s12.p16
In both species, (-)-NANM, but not (+)-NANM, antagonized the rate-decreasing effects of morphine on FI and FR responding.
(-)-NANM
morphine
EFFECT
3968644.xml
DDI-MedLine.d30.s7
DDI-MedLine.d30.s7.p1
The incidence of akathisia in clinical trials of the weekly dosage schedule was greater (8.5%, 4/47 patients) when prochlorperazine was administered on the same day as CAMPTOSAR than when these drugs were given on separate days (1.3%, 1/80 patients).
prochlorperazine
CAMPTOSAR
EFFECT
Irinotecan_ddi.xml
DDI-DrugBank.d279.s8
DDI-DrugBank.d279.s8.p0
When used in therapeutic doses, azithromycin had a modest effect on the pharmacokinetics of atorvastatin, carbamazepine, cetirizine, didanosine, efavirenz, fluconazole, indinavir, midazolam, rifabutin, sildenafil, theophylline (intravenous and oral), triazolam, trimethoprim/sulfamethoxazole or zidovudine.
azithromycin
theophylline
MECHANISM
Azithromycin_ddi.xml
DDI-DrugBank.d53.s7
DDI-DrugBank.d53.s7.p10
Fluvoxamine has also been shown to inhibit P450 1A2, an isoform also involved in TCAmetabolism.
Fluvoxamine
TCA
MECHANISM
Clomipramine_ddi.xml
DDI-DrugBank.d238.s17
DDI-DrugBank.d238.s17.p0
The IV methylprednisolone dose should be reduced by approximately 25%, and the oral methylprednisolone dose should be reduced by approximately 50% when coadministered with Aprepitant to achieve exposures of methylprednisolone similar to those obtained when it is given without Aprepitant.
methylprednisolone
Aprepitant
ADVISE
Aprepitant_ddi.xml
DDI-DrugBank.d382.s14
DDI-DrugBank.d382.s14.p4
High-dose cyclosporin A resulting in concentrations above 2000 ng/mL administered with oral etoposide has led to an 80% increase in etoposide exposure with a 38% decrease in total body clearance of etoposide compared to etoposide alone.
etoposide
etoposide
NONE
Etoposide_ddi.xml
DDI-DrugBank.d194.s1
DDI-DrugBank.d194.s1.p7
Caution should be observed when anileridine is coadministered with other opioids, sedatives, phenothiazines, or anesthetics, as these agents may increase respiratory and circulatory depression.
anileridine
phenothiazines
ADVISE
Anileridine_ddi.xml
DDI-DrugBank.d215.s0
DDI-DrugBank.d215.s0.p2
Clindamycin has been shown to have neuromuscular blocking properties that may enhance the action of other neuromuscular blocking agents.
Clindamycin
neuromuscular blocking agents
EFFECT
Clindamycin_ddi.xml
DDI-DrugBank.d256.s0
DDI-DrugBank.d256.s0.p0
Appropriate laboratory testing should be considered prior to initiating combination therapy with Amprenavir and ritonavir and at periodic intervals or if any clinical signs or symptoms of hyperlipidemia or elevated liver function tests occur during therapy.
Amprenavir
ritonavir
ADVISE
Amprenavir_ddi.xml
DDI-DrugBank.d437.s14
DDI-DrugBank.d437.s14.p0
Antacids, kaolin-pectin, sulfasalazine, neomycin, cholestyramine, certain anticancer drugs, and metoclopramide may interfere with intestinal digoxin absorption, resulting in unexpectedly low serum concentrations.
cholestyramine
digoxin
MECHANISM
Digoxin_ddi.xml
DDI-DrugBank.d450.s6
DDI-DrugBank.d450.s6.p19
[The GABA-ergic system and brain edema] It has been shown in rats with experimental toxic and traumatic edemas that picrotoxin (1 mg/kg) removes the antiedematous action of diazepam, phenazepam, phenibut and amizyl and reduces the action of phentolamine.
picrotoxin
phentolamine
EFFECT
2857099.xml
DDI-MedLine.d27.s0
DDI-MedLine.d27.s0.p4
Anticoagulants: Flurbiprofen like other nonsteroidal anti-inflammatory drugs, has been shown to affect bleeding parameters in patients receiving anti-coagulants, and serious clinical bleeding has been reported.
nonsteroidal anti-inflammatory drugs
anti-coagulants
EFFECT
Flurbiprofen_ddi.xml
DDI-DrugBank.d529.s2
DDI-DrugBank.d529.s2.p5