PDBID
stringlengths
4
4
Resolution
stringlengths
1
13
Year
int64
1.98k
2.02k
Ligand Name
stringlengths
1
7
Ligand Chain
stringclasses
53 values
Ligand Residue Number
stringlengths
1
9
Binding Affinity Measurement
stringclasses
4 values
Binding Affinity Sign
stringclasses
6 values
Binding Affinity Value
float64
0
500M
Binding Affinity Unit
stringclasses
6 values
Log Binding Affinity
float64
-14
2.97
Binding Affinity Source
stringclasses
3 values
Binding Affinity Annotation
stringlengths
6
72
Protein UniProtID
stringlengths
6
55
Protein UniProtName
stringlengths
2
575
Ligand SMILES
stringlengths
4
352
Ligand MW
float64
44
1.82k
Ligand LogP
float64
-23.01
13.7
Ligand TPSA
float64
0
786
Ligand NumRotBond
int64
0
59
Ligand NumHeavyAtoms
int64
3
120
Ligand NumHDon
int64
0
30
Ligand NumHAcc
int64
0
56
Ligand QED
float64
0.01
0.95
7rlj
NMR
2,021
JDP
F
803
ki
=
26
nM
-7.585027
BindingDB
IC50=1030nM,Ki=26nM
P55072,P55072
Transitional endoplasmic reticulum ATPase,Transitional endoplasmic reticulum ATPase
Cc1cc2c(C(N)=O)cccc2n1-c1nc2c(c(NCc3ccccc3)n1)COCC2
413.481
3.51262
95.06
5
31
2
6
0.522051
7rlj
NMR
2,021
JDP
G
803
ki
=
26
nM
-7.585027
BindingDB
IC50=1030nM,Ki=26nM
P55072,P55072
Transitional endoplasmic reticulum ATPase,Transitional endoplasmic reticulum ATPase
Cc1cc2c(C(N)=O)cccc2n1-c1nc2c(c(NCc3ccccc3)n1)COCC2
413.481
3.51262
95.06
5
31
2
6
0.522051
7rlj
NMR
2,021
JDP
H
803
ki
=
26
nM
-7.585027
BindingDB
IC50=1030nM,Ki=26nM
P55072,P55072
Transitional endoplasmic reticulum ATPase,Transitional endoplasmic reticulum ATPase
Cc1cc2c(C(N)=O)cccc2n1-c1nc2c(c(NCc3ccccc3)n1)COCC2
413.481
3.51262
95.06
5
31
2
6
0.522051
7rlj
NMR
2,021
JDP
I
803
ki
=
26
nM
-7.585027
BindingDB
IC50=1030nM,Ki=26nM
P55072,P55072
Transitional endoplasmic reticulum ATPase,Transitional endoplasmic reticulum ATPase
Cc1cc2c(C(N)=O)cccc2n1-c1nc2c(c(NCc3ccccc3)n1)COCC2
413.481
3.51262
95.06
5
31
2
6
0.522051
7rlj
NMR
2,021
JDP
J
803
ki
=
26
nM
-7.585027
BindingDB
IC50=1030nM,Ki=26nM
P55072,P55072
Transitional endoplasmic reticulum ATPase,Transitional endoplasmic reticulum ATPase
Cc1cc2c(C(N)=O)cccc2n1-c1nc2c(c(NCc3ccccc3)n1)COCC2
413.481
3.51262
95.06
5
31
2
6
0.522051
7rlj
NMR
2,021
JDP
K
803
ki
=
26
nM
-7.585027
BindingDB
IC50=1030nM,Ki=26nM
P55072,P55072
Transitional endoplasmic reticulum ATPase,Transitional endoplasmic reticulum ATPase
Cc1cc2c(C(N)=O)cccc2n1-c1nc2c(c(NCc3ccccc3)n1)COCC2
413.481
3.51262
95.06
5
31
2
6
0.522051
7rlj
NMR
2,021
JDP
L
803
ki
=
26
nM
-7.585027
BindingDB
IC50=1030nM,Ki=26nM
P55072,P55072
Transitional endoplasmic reticulum ATPase,Transitional endoplasmic reticulum ATPase
Cc1cc2c(C(N)=O)cccc2n1-c1nc2c(c(NCc3ccccc3)n1)COCC2
413.481
3.51262
95.06
5
31
2
6
0.522051
7s3k
1.9
2,021
Z26
A
401
ic50
=
1,350
nM
-5.869666
BindingDB
IC50=1350nM
P0DTD1
3C-like proteinase
COc1ccc(Cl)cc1CC(=O)Nc1cncc2ccccc12
326.783
4.078
51.22
4
23
1
3
0.785675
7s3s
2.0
2,021
860
A
401
ic50
=
728
nM
-6.137869
BindingDB
IC50=728nM
P0DTD1
3C-like proteinase
O=C(Cc1cccc(Cl)c1)Nc1cncc2ccccc12
296.757
4.0694
41.99
3
21
1
2
0.791409
7slv
2.13
2,022
9TC
A
502
ic50
=
7.66
nM
-8.115771
BindingDB
IC50=7.66nM
O95497
Pantetheinase
O=C(c1cnc(NCc2cnccn2)nc1)N1CCC2(CCOCC2)C1
354.414
1.5214
93.13
4
26
1
7
0.889571
7slx
2.35
2,022
9SS
A
502
ic50
=
1,177
nM
-5.929224
BindingDB
IC50=1177nM
O95497
Pantetheinase
N#C[C@@H]1CCCN(C(=O)c2cnc(NC3(c4cncnc4)CC3)nc2)C1
349.398
1.74358
107.69
4
26
1
7
0.895443
7sly
2.17
2,022
9S5
A
502
ic50
=
0.242
nM
-9.616185
BindingDB
IC50=0.242nM
O95497
Pantetheinase
C[C@H](Nc1ncc(C(=O)N2CCC3(CCOCC3)C2)cn1)c1cnccn1
368.441
2.0824
93.13
4
27
1
7
0.882945
7std
1.8
1,999
CRP
A
600
ki
=
19
pM
-10.721246
MOAD
Ki=19.0pM
P56221,P56221
Scytalone dehydratase,Scytalone dehydratase
CC[C@@]1(C(=O)N[C@H](C)c2ccc(Cl)cc2)[C@@H](C)C1(Cl)Cl
334.674
4.7372
29.1
4
20
1
1
0.791879
7std
1.8
1,999
CRP
B
601
ki
=
19
pM
-10.721246
MOAD
Ki=19.0pM
P56221,P56221
Scytalone dehydratase,Scytalone dehydratase
CC[C@@]1(C(=O)N[C@H](C)c2ccc(Cl)cc2)[C@@H](C)C1(Cl)Cl
334.674
4.7372
29.1
4
20
1
1
0.791879
7std
1.8
1,999
CRP
C
602
ki
=
19
pM
-10.721246
MOAD
Ki=19.0pM
P56221,P56221
Scytalone dehydratase,Scytalone dehydratase
CC[C@@]1(C(=O)N[C@H](C)c2ccc(Cl)cc2)[C@@H](C)C1(Cl)Cl
334.674
4.7372
29.1
4
20
1
1
0.791879
7svd
NMR
2,022
VX8
A
1511
ec50
=
2,600
nM
-5.585027
BindingDB
EC50=2600nM
P13569
Cystic fibrosis transmembrane conductance regulator
Cc1ccc(NC(=O)C2(c3ccc4c(c3)OC(F)(F)O4)CC2)nc1-c1cccc(C(=O)[O-])c1
451.405
3.41232
100.58
5
33
1
6
0.638217
7svr
NMR
2,022
VX8
A
1501
ec50
=
2,600
nM
-5.585027
BindingDB
EC50=2600nM
P13569
Cystic fibrosis transmembrane conductance regulator
Cc1ccc(NC(=O)C2(c3ccc4c(c3)OC(F)(F)O4)CC2)nc1-c1cccc(C(=O)[O-])c1
451.405
3.41232
100.58
5
33
1
6
0.638217
7upj
2.0
1,997
INU
A
100
ki
=
3.2
nM
-8.49485
MOAD
Ki=3.2nM
P03367,P03367
HIV-1 PROTEASE,HIV-1 PROTEASE
O=c1oc2c(c(O)c1[C@H](c1cccc(NS(=O)(=O)c3ccccc3)c1)C1CC1)CCCCCC2
479.598
5.3471
96.61
6
34
2
5
0.496968
7vfw
NMR
2,021
6I7
A
2420
ic50
=
16
nM
-7.79588
BindingDB
IC50=16nM
Q00975
Voltage-dependent N-type calcium channel subunit alpha-1B
COc1ccccc1-n1nc(C2CC(C)(C)OC(C)(C)C2)cc1-c1ccc(Cl)cc1
424.972
6.6525
36.28
4
30
0
4
0.469822
7vkn
2.7
2,021
7GI
A
801
ic50
=
0.4
nM
-9.39794
BindingDB
IC50=0.400000nM
P04629
Tyrosine-protein kinase receptor
C[C@H]1CNC(=O)c2cnn3ccc(nc23)N[C@H](C)c2cc(F)ccc2O1
355.373
2.5522
80.55
0
26
2
6
0.647765
7vko
2.9
2,021
7GI
A
801
ic50
=
0.4
nM
-9.39794
BindingDB
IC50=0.400000nM
P04629
Tyrosine-protein kinase receptor
C[C@H]1CNC(=O)c2cnn3ccc(nc23)N[C@H](C)c2cc(F)ccc2O1
355.373
2.5522
80.55
0
26
2
6
0.647765
7vnp
NMR
2,021
7YV
A
1108
ec50
=
1,600
nM
-5.79588
BindingDB
EC50=1600nM
P56696,P56696
Potassium voltage-gated channel subfamily KQT member 4,Maltodextrin-binding protein,Potassium voltage-gated channel subfamily KQT member 4,Maltodextrin-binding protein
Cc1cc(C)c(NC(=O)[C@H]2C[C@@H]3CC[C@H]2C3)c(C)c1
257.377
3.98656
29.1
2
19
1
1
0.85254
7vnp
NMR
2,021
7YV
A
1107
ec50
=
1,600
nM
-5.79588
BindingDB
EC50=1600nM
P56696,P56696,P56696
Potassium voltage-gated channel subfamily KQT member 4,Maltodextrin-binding protein,Potassium voltage-gated channel subfamily KQT member 4,Maltodextrin-binding protein,Potassium voltage-gated channel subfamily KQT member 4,Maltodextrin-binding protein
Cc1cc(C)c(NC(=O)[C@H]2C[C@@H]3CC[C@H]2C3)c(C)c1
257.377
3.98656
29.1
2
19
1
1
0.85254
7vnp
NMR
2,021
7YV
C
1103
ec50
=
1,600
nM
-5.79588
BindingDB
EC50=1600nM
P56696,P56696
Potassium voltage-gated channel subfamily KQT member 4,Maltodextrin-binding protein,Potassium voltage-gated channel subfamily KQT member 4,Maltodextrin-binding protein
Cc1cc(C)c(NC(=O)[C@H]2C[C@@H]3CC[C@H]2C3)c(C)c1
257.377
3.98656
29.1
2
19
1
1
0.85254
7vnp
NMR
2,021
7YV
E
1103
ec50
=
1,600
nM
-5.79588
BindingDB
EC50=1600nM
P56696,P56696
Potassium voltage-gated channel subfamily KQT member 4,Maltodextrin-binding protein,Potassium voltage-gated channel subfamily KQT member 4,Maltodextrin-binding protein
Cc1cc(C)c(NC(=O)[C@H]2C[C@@H]3CC[C@H]2C3)c(C)c1
257.377
3.98656
29.1
2
19
1
1
0.85254
7vnq
NMR
2,021
7YV
A
1101
ec50
=
1,600
nM
-5.79588
BindingDB
EC50=1600nM
P56696,P56696,P56696
Potassium voltage-gated channel subfamily KQT member 4,Maltodextrin-binding protein,Potassium voltage-gated channel subfamily KQT member 4,Maltodextrin-binding protein,Potassium voltage-gated channel subfamily KQT member 4,Maltodextrin-binding protein
Cc1cc(C)c(NC(=O)[C@H]2C[C@@H]3CC[C@H]2C3)c(C)c1
257.377
3.98656
29.1
2
19
1
1
0.85254
7vnq
NMR
2,021
7YV
C
1101
ec50
=
1,600
nM
-5.79588
BindingDB
EC50=1600nM
P56696,P56696,P56696
Potassium voltage-gated channel subfamily KQT member 4,Maltodextrin-binding protein,Potassium voltage-gated channel subfamily KQT member 4,Maltodextrin-binding protein,Potassium voltage-gated channel subfamily KQT member 4,Maltodextrin-binding protein
Cc1cc(C)c(NC(=O)[C@H]2C[C@@H]3CC[C@H]2C3)c(C)c1
257.377
3.98656
29.1
2
19
1
1
0.85254
7vnq
NMR
2,021
7YV
E
1101
ec50
=
1,600
nM
-5.79588
BindingDB
EC50=1600nM
P56696,P56696,P56696
Potassium voltage-gated channel subfamily KQT member 4,Maltodextrin-binding protein,Potassium voltage-gated channel subfamily KQT member 4,Maltodextrin-binding protein,Potassium voltage-gated channel subfamily KQT member 4,Maltodextrin-binding protein
Cc1cc(C)c(NC(=O)[C@H]2C[C@@H]3CC[C@H]2C3)c(C)c1
257.377
3.98656
29.1
2
19
1
1
0.85254
7vnq
NMR
2,021
7YV
G
1101
ec50
=
1,600
nM
-5.79588
BindingDB
EC50=1600nM
P56696,P56696,P56696
Potassium voltage-gated channel subfamily KQT member 4,Maltodextrin-binding protein,Potassium voltage-gated channel subfamily KQT member 4,Maltodextrin-binding protein,Potassium voltage-gated channel subfamily KQT member 4,Maltodextrin-binding protein
Cc1cc(C)c(NC(=O)[C@H]2C[C@@H]3CC[C@H]2C3)c(C)c1
257.377
3.98656
29.1
2
19
1
1
0.85254
7vnr
NMR
2,021
7YV
A
1101
ec50
=
1,600
nM
-5.79588
BindingDB
EC50=1600nM
P56696,P56696
Potassium voltage-gated channel subfamily KQT member 4,Maltodextrin-binding protein,Potassium voltage-gated channel subfamily KQT member 4,Maltodextrin-binding protein
Cc1cc(C)c(NC(=O)[C@H]2C[C@@H]3CC[C@H]2C3)c(C)c1
257.377
3.98656
29.1
2
19
1
1
0.85254
7vnr
NMR
2,021
7YV
C
1101
ec50
=
1,600
nM
-5.79588
BindingDB
EC50=1600nM
P56696,P56696
Potassium voltage-gated channel subfamily KQT member 4,Maltodextrin-binding protein,Potassium voltage-gated channel subfamily KQT member 4,Maltodextrin-binding protein
Cc1cc(C)c(NC(=O)[C@H]2C[C@@H]3CC[C@H]2C3)c(C)c1
257.377
3.98656
29.1
2
19
1
1
0.85254
7vnr
NMR
2,021
7YV
E
1101
ec50
=
1,600
nM
-5.79588
BindingDB
EC50=1600nM
P56696,P56696
Potassium voltage-gated channel subfamily KQT member 4,Maltodextrin-binding protein,Potassium voltage-gated channel subfamily KQT member 4,Maltodextrin-binding protein
Cc1cc(C)c(NC(=O)[C@H]2C[C@@H]3CC[C@H]2C3)c(C)c1
257.377
3.98656
29.1
2
19
1
1
0.85254
7vnr
NMR
2,021
7YV
G
1101
ec50
=
1,600
nM
-5.79588
BindingDB
EC50=1600nM
P56696,P56696
Potassium voltage-gated channel subfamily KQT member 4,Maltodextrin-binding protein,Potassium voltage-gated channel subfamily KQT member 4,Maltodextrin-binding protein
Cc1cc(C)c(NC(=O)[C@H]2C[C@@H]3CC[C@H]2C3)c(C)c1
257.377
3.98656
29.1
2
19
1
1
0.85254
7vsi
NMR
2,021
7R3
A
703
ic50
=
3.1
nM
-8.508638
BindingDB
IC50=3.1nM,EC50=3.0nM
P31639
Sodium/glucose cotransporter 2
OC[C@H]1O[C@@H](c2ccc(Cl)c(Cc3ccc(O[C@H]4CCOC4)cc3)c2)[C@H](O)[C@@H](O)[C@@H]1O
450.915
1.6134
108.61
6
31
4
7
0.529157
7wf7
NMR
2,022
S1P
A
401
ic50
=
1.4
nM
-8.853872
BindingDB
IC50=1.40nM,EC50=4.3nM
P21453
Sphingosine 1-phosphate receptor 1
CCCCCCCCCCCCCC=C[C@@H](O)[C@@H]([NH3+])COP(=O)([O-])[O-]
378.47
2.0604
120.29
17
25
2
5
0.227956
830c
1.6
1,999
RS1
A
1
ki
=
0.52
nM
-9.283997
MOAD
Ki=0.52nM
P45452,P45452
MMP-13,MMP-13
O=C(NO)C1(CS(=O)(=O)c2ccc(Oc3ccc(Cl)cc3)cc2)CCOCC1
425.89
3.2082
101.93
6
28
2
6
0.543924
830c
1.6
1,999
RS1
B
1
ki
=
0.52
nM
-9.283997
MOAD
Ki=0.52nM
P45452,P45452
MMP-13,MMP-13
O=C(NO)C1(CS(=O)(=O)c2ccc(Oc3ccc(Cl)cc3)cc2)CCOCC1
425.89
3.2082
101.93
6
28
2
6
0.543924
8a3h
0.97
2,000
IDC
A
500
ki
=
88
uM
-4.055517
MOAD
Ki=88.0uM
O85465
PROTEIN (ENDOGLUCANASE)
OC[C@@H]1[C@@H](O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)[C@H](O)[C@@H](O)c2nccn21
362.335
-3.9905
177.89
4
25
7
11
0.27917
8abp
1.49
1,991
GAL
A
308
kd
=
0.01
uM
-8
MOAD
Kd=0.01uM
P02924
L-ARABINOSE-BINDING PROTEIN
OC[C@H]1O[C@@H](O)[C@H](O)[C@@H](O)[C@H]1O
180.156
-3.2214
110.38
1
12
5
6
0.290153
8abp
1.49
1,991
GLA
A
307
kd
=
0.01
uM
-8
MOAD
Kd=0.01uM
P02924
L-ARABINOSE-BINDING PROTEIN
OC[C@H]1O[C@H](O)[C@H](O)[C@@H](O)[C@H]1O
180.156
-3.2214
110.38
1
12
5
6
0.290153
8cat
2.5
1,985
NDP
A
508
kd
<
10
nM
-8
MOAD
Kd<10.0nM
P00432
CATALASE
NC(=O)C1=CN([C@@H]2O[C@H](CO[P@@](=O)([O-])O[P@@](=O)([O-])OC[C@H]3O[C@@H](n4cnc5c(N)ncnc54)[C@H](OP(=O)([O-])[O-])[C@H]3O)[C@@H](O)[C@H]2O)C=CC1
741.393
-5.0974
375.47
13
48
5
23
0.119838
8cat
2.5
1,985
NDP
B
508
kd
<
10
nM
-8
MOAD
Kd<10.0nM
P00432
CATALASE
NC(=O)C1=CN([C@@H]2O[C@H](CO[P@@](=O)([O-])O[P@@](=O)([O-])OC[C@H]3O[C@@H](n4cnc5c(N)ncnc54)[C@H](OP(=O)([O-])[O-])[C@H]3O)[C@@H](O)[C@H]2O)C=CC1
741.393
-5.0974
375.47
13
48
5
23
0.119838
8cpa
2.0
1,994
AGF
A
309
ki
=
710
pM
-9.148742
MOAD
Ki=710.0pM
P00730
CARBOXYPEPTIDASE A
C[C@H](NC(=O)OCc1ccccc1)C(=O)NC[P@@](=O)([O-])O[C@@H](Cc1ccccc1)C(=O)[O-]
462.395
0.3062
156.92
11
32
2
8
0.451797
8gpb
2.2
1,992
AMP
A
930
kd
=
250
uM
-3.60206
MOAD
Kd=250.0uM
P00489
GLYCOGEN PHOSPHORYLASE B
Nc1ncnc2c1ncn2[C@@H]1O[C@H](COP(=O)([O-])[O-])[C@@H](O)[C@H]1O
345.208
-3.127
191.73
4
23
3
12
0.474435
8gpb
2.2
1,992
AMP
A
940
kd
=
250
uM
-3.60206
MOAD
Kd=250.0uM
P00489
GLYCOGEN PHOSPHORYLASE B
Nc1ncnc2c1ncn2[C@@H]1O[C@H](COP(=O)([O-])[O-])[C@@H](O)[C@H]1O
345.208
-3.127
191.73
4
23
3
12
0.474435
8nse
2.25
2,001
NRG
A
705
ki
=
750
nM
-6.124939
BindingDB
IC50=1200nM,Ki=750nM
P29473
PROTEIN (NITRIC OXIDE SYNTHASE)
[NH2+]=C(NCCC[C@H]([NH3+])C(=O)[O-])N[N+](=O)[O-]
220.209
-5.387
160.56
6
15
4
4
0.114766
8nse
2.25
2,001
NRG
B
706
ki
=
750
nM
-6.124939
BindingDB
IC50=1200nM,Ki=750nM
P29473
PROTEIN (NITRIC OXIDE SYNTHASE)
[NH2+]=C(NCCC[C@H]([NH3+])C(=O)[O-])N[N+](=O)[O-]
220.209
-5.387
160.56
6
15
4
4
0.114766
966c
1.9
1,999
RS2
A
1
ki
=
23
nM
-7.638272
MOAD
Ki=23.0nM
P03956
MMP-1
O=C(CC1(S(=O)(=O)c2ccc(Oc3ccccc3)cc2)CCOCC1)NO
391.445
2.6973
101.93
6
27
2
6
0.579855
9abp
1.97
1,992
GLA
A
307
kd
=
0.01
uM
-8
MOAD
Kd=0.01uM
P02924
L-ARABINOSE-BINDING PROTEIN
OC[C@H]1O[C@H](O)[C@H](O)[C@@H](O)[C@H]1O
180.156
-3.2214
110.38
1
12
5
6
0.290153
9abp
1.97
1,992
GAL
A
308
kd
=
0.01
uM
-8
MOAD
Kd=0.01uM
P02924
L-ARABINOSE-BINDING PROTEIN
OC[C@H]1O[C@@H](O)[C@H](O)[C@@H](O)[C@H]1O
180.156
-3.2214
110.38
1
12
5
6
0.290153