Drug_ID
stringlengths
6
9
Drug
stringlengths
4
325
Y
float64
0
1
Drug 1062
O=C(Oc1ccccc1)c1ccccc1O
0
Drug 1063
CC1CC(OC(=O)c2ccccc2O)CC(C)(C)C1
1
Drug 1065
O=C(OCc1ccccc1)c1ccccc1O
1
Drug 1074
Cc1occc(=O)c1O
0
Drug 1079
CC(C)(C)c1cc(Cc2cc(C(C)(C)C)c(O)c(C(C)(C)C)c2)cc(C(C)(C)C)c1O
0
Drug 1089
CC(=O)c1ccccc1O
0
Drug 1091
CCCCCCCCCCOC(=O)c1ccccc1C(=O)OCCCCCCCC
0
Drug 1096
CCCCCCCCCCCCCCOS(=O)(=O)[O-].[Na+]
1
Drug 1104
O=c1ssc(Cl)c1Cl
0
Drug 1114
COC(=O)c1ccccc1O
0
Drug 1121
CC1COC(Cn2cncn2)(c2ccc(Oc3ccc(Cl)cc3)cc2Cl)O1
1
Drug 1125
CCC(C)OC(=O)N1CCCCC1CCO
0
Drug 1131
O=C(c1ccccc1)c1ccccc1
0
Drug 1132
c1ccc2c(c1)CCCC2
0
Drug 1141
Cc1cc(-c2ccc(N)c(C)c2)ccc1N
0
Drug 1144
N#Cc1nn(-c2c(Cl)cc(C(F)(F)F)cc2Cl)c(N)c1S(=O)C(F)(F)F
1
Drug 1147
Cc1ccc(-c2c(Cl)nc(C#N)n2S(=O)(=O)N(C)C)cc1
1
Drug 1148
c1ccc2cc3ccccc3cc2c1
0
Drug 1149
COc1ccc(C=O)cc1OC
0
Drug 1155
Oc1ccc(Cl)cc1Cc1ccccc1
1
Drug 1156
CC(Oc1ccc(Cl)cc1Cl)C(=O)O
0
Drug 1162
O=C(CC(=O)c1ccccc1)c1ccccc1
0
Drug 1163
CCOC(=O)c1ccc(O)cc1
0
Drug 1165
CC(C)(C#N)c1cc(Cn2cncn2)cc(C(C)(C)C#N)c1
0
Drug 1166
O=C(OCc1ccccc1)c1ccccc1
1
Drug 1173
COC(=O)c1ccc(C(=O)OC)cc1
0
Drug 1176
CN(C)Cc1ccccc1O
0
Drug 1185
Clc1ccc(Cl)c(Cl)c1
0
Drug 1189
O=C1CCCC1
0
Drug 1193
CCC(C)(C)c1ccc(O)c(C(C)(C)CC)c1
1
Drug 1197
COc1ccc(O)c(C(C)(C)C)c1
1
Drug 1204
CC1C=[C-]C=C1.[C-]#[O+].[C-]#[O+].[C-]#[O+].[Mn+]
0
Drug 1206
Cc1ccc([N+](=O)[O-])cc1[N+](=O)[O-]
0
Drug 1214
CCOc1cc(C=O)ccc1O
0
Drug 1230
CN(C)c1ccccc1
0
Drug 1236
CCCOC(=O)c1cc(O)c(O)c(O)c1
1
Drug 1245
O=C(O)c1cccc(C(=O)O)c1
0
Drug 1251
CCCCOC(=O)[C@@H](C)Oc1ccc(Oc2ccc(C#N)cc2F)cc1
1
Drug 1259
COP(=S)(OC)Oc1ccc([N+](=O)[O-])c(C)c1
0
Drug 1270
CCNc1nc(Cl)nc(NCC)n1
0
Drug 1273
CCCCCC(C=O)=Cc1ccccc1
1
Drug 1274
CC(C)OC(=O)Nc1ccccc1
0
Drug 1275
CCOCn1c(-c2ccc(Cl)cc2)c(C#N)c(Br)c1C(F)(F)F
1
Drug 1280
CCOC(OCC)OCC
0
Drug 1285
CC(=O)C=Cc1ccccc1
0
Drug 1314
OCCOc1ccccc1
0
Drug 1315
NCCCN1CCOCC1
0
Drug 1322
CCc1ccc(O)cc1
0
Drug 1324
COc1ccc(C=O)cc1
0
Drug 1325
COCCOC[C@H](CC1(C(=O)N[C@H]2CC[C@@H](C(=O)O)CC2)CCCC1)C(=O)Oc1ccc2c(c1)CCC2
0
Drug 1327
CC(C)CC(C)CC(O)CC(C)C
0
Drug 1330
CCOC(=O)CCC(=O)OCC
0
Drug 1334
CC1=NNC(=O)N(/N=C/c2cccnc2)C1
0
Drug 1336
Oc1ccc(O)cc1
1
Drug 1337
O=c1ccc(=O)[nH][nH]1
0
Drug 1355
CCCCCC(=O)OCC
0
Drug 1359
NC(=O)N=NC(N)=O
0
Drug 1363
CC(=O)OCCC(C)C
0
Drug 1368
O=C(O)CCCCCCCC(=O)O
0
Drug 1371
O=C(O)CCCCC(=O)O
0
Drug 1375
NCCCCCCN
0
Drug 1378
CCCCCCCC=O
0
Drug 1380
CCCCCCCCCC
0
Drug 1381
CCCCC(CC)COP(=O)(Oc1ccccc1)Oc1ccccc1
1
Drug 1382
CCCCCCCCC=O
0
Drug 1392
Fc1ccc(Oc2ccnc3cc(Cl)cc(Cl)c23)cc1
1
Drug 1399
CC1(C)[C@@H]2CC[C@@]1(C)[C@H](O)C2
0
Drug 1406
C[C@]12C[C@H](O)[C@@]3(F)[C@@H](CCC4=CC(=O)C=C[C@@]43C)[C@@H]1C[C@@H](O)[C@]2(O)C(=O)CO
0
Drug 1408
CC1(C)CCC(Cc2ccc(Cl)cc2)C1(O)Cn1cncn1
1
Drug 1409
CC(=O)O[C@@H]1C[C@H]2CC[C@]1(C)C2(C)C
0
Drug 1427
CC(CCC(=O)O)(c1ccc(O)cc1)c1ccc(O)cc1
0
Drug 1429
CC1(C)C(=O)N(Br)C(=O)N1Cl
0
Drug 1431
O=[N+]([O-])C(CO)(CO)CO
0
Drug 1432
CC(=O)OC[C@H]1O[C@H](O[C@]2(COC(C)=O)O[C@H](COC(C)=O)[C@@H](OC(C)=O)[C@@H]2OC(C)=O)[C@H](OC(C)=O)[C@@H](OC(C)=O)[C@@H]1OC(C)=O
0
Drug 1445
O=P(OCC(Br)CBr)(OCC(Br)CBr)OCC(Br)CBr
0
Drug 1446
CCCCOP(=O)(OCCCC)OCCCC
0
Drug 1449
CC1(C(=O)Nc2ccc(O)c(Cl)c2Cl)CCCCC1
0
Drug 1451
CC(C)CC(C)(O)C#CC(C)(O)CC(C)C
0
Drug 1452
CCCCC(CC)COS(=O)(=O)[O-].[Na+]
0
Drug 1453
C=C(C)C#N
0
Drug 1463
CC(=O)N(C)C
0
Drug 1465
COC(=O)[C@]1(C)CCC[C@]2(C)[C@H]3CCC(C(C)C)=CC3=CC[C@@H]12
1
Drug 1472
CC(C)COC(=O)CC(C(=O)OCC(C)C)S(=O)(=O)[O-].[Na+]
0
Drug 1477
CC(=O)/C(C)=C/C1C(C)=CCCC1(C)C
0
Drug 1502
Nc1ccc(N)c2c1C(=O)c1ccccc1C2=O
1
Drug 1503
c1cc2ccc3cccc4ccc(c1)c2c34
0
Drug 1505
CC(=O)CC(c1ccccc1)c1c([O-])c2ccccc2oc1=O.[Na+]
0
Drug 1516
C[C@]12CC[C@@H]3c4ccc(O)cc4C[C@@H](CCCCCCCCCS(=O)CCCC(F)(F)C(F)(F)F)[C@H]3[C@@H]1CC[C@@H]2O
0
Drug 1532
O=S(=O)([O-])c1cccc2ccccc12.[Na+]
0
Drug 1541
[As]#[In]
0
Drug 1567
C=CCOC(=O)c1ccccc1C(=O)OCC=C
0
Drug 1568
CCCCCOC(=O)c1ccccc1C(=O)OCCCCC
1
Drug 1570
N#Cc1c[nH]cc1-c1cccc2c1OC(F)(F)O2
0
Drug 1577
O=C(c1ccccc1)c1ccc(O)cc1O
0
Drug 1582
CC(=O)c1cc(C(C)(C)C)cc2c1CCC2(C)C
0
Drug 1586
CC1(c2ccc(Oc3ccccc3)cc2)OC(=O)N(Nc2ccccc2)C1=O
1
Drug 1589
CO/C=C(/C(=O)OC)c1ccccc1Oc1cc(Oc2ccccc2C#N)ncn1
0
Drug 1596
Cc1ccc(N=Nc2c(O)ccc(N=Nc3ccc(S(=O)(=O)[O-])cc3)c2O)c(C)c1.[Na+]
0
Drug 1607
CC(C)CCCC(C)(C)O
0
Drug 1611
c1ccc2c(c1)oc1ccccc12
0