SMILES
large_stringlengths
17
56
ID
large_stringlengths
1
7
SELFIES
stringlengths
63
275
SAFE
stringlengths
20
78
CCOc1ncc(NC(=O)c2ccccn2)c(OCC)n1
1498853
[C][C][O][C][=N][C][=C][Branch1][=C][N][C][=Branch1][C][=O][C][=C][C][=C][C][=N][Ring1][=Branch1][C][Branch1][Ring2][O][C][C][=N][Ring2][Ring1][C]
c16ncc8c7n1.c19ccccn1.C39=O.CC4.O46.N38.O57.C5C
CCCC(NC(=O)Cc1ccccc1)C(=O)N1CCN(C(C)C)CC1
1684711
[C][C][C][C][Branch1][#C][N][C][=Branch1][C][=O][C][C][=C][C][=C][C][=C][Ring1][=Branch1][C][=Branch1][C][=O][N][C][C][N][Branch1][=Branch1][C][Branch1][C][C][C][C][C][Ring1][=Branch2]
CCCC4C3=O.N13CCN5CC1.c16ccccc1.C2(=O)C6.C5(C)C.N24
O=C(CN1CCN(c2ccccc2F)C1=O)NCCc1ccncc1
1660700
[O][=C][Branch2][Ring1][Branch1][C][N][C][C][N][Branch1][#Branch2][C][=C][C][=C][C][=C][Ring1][=Branch1][F][C][Ring1][N][=O][N][C][C][C][=C][C][=N][C][=C][Ring1][=Branch1]
N15CCN7C1=O.c17ccccc1F.c16ccncc1.O=C3C5.C4C6.N34
COCCCN(C)C(=O)Nc1cc(C(F)(F)F)c[nH]c1=O
906234
[C][O][C][C][C][N][Branch1][C][C][C][=Branch1][C][=O][N][C][=C][C][Branch1][=Branch2][C][Branch1][C][F][Branch1][C][F][F][=C][NH1][C][Ring1][#Branch2][=O]
c16cc7c[nH]c1=O.C4CC5.C7(F)(F)F.N25C.C23=O.CO4.N36
CN(C)C(=O)C1CCCN1S(=O)(=O)c1cccc(Cl)c1
1800052
[C][N][Branch1][C][C][C][=Branch1][C][=O][C][C][C][C][N][Ring1][Branch1][S][=Branch1][C][=O][=Branch1][C][=O][C][=C][C][=C][C][Branch1][C][Cl][=C][Ring1][#Branch1]
S3(=O)(=O)c1cccc(Cl)c1.C14CCCN13.CN2C.C24=O
Brc1cccnc1SCCOCC1CCCO1
1215096
[Br][C][=C][C][=C][N][=C][Ring1][=Branch1][S][C][C][O][C][C][C][C][C][O][Ring1][Branch1]
Brc1cccnc16.C15CCCO1.C4C2.S46.O23.C35
NC(=O)c1cccc(CNC(=O)N2CCCC(O)C2)c1
999661
[N][C][=Branch1][C][=O][C][=C][C][=C][C][Branch2][Ring1][C][C][N][C][=Branch1][C][=O][N][C][C][C][C][Branch1][C][O][C][Ring1][#Branch1][=C][Ring1][P]
c16cccc7c1.N14CCCC(O)C1.NC6=O.C34=O.C57.N35
CCC(C)NC(=O)Nc1ccccc1C(=O)N1CC(C)CC(C)C1
590973
[C][C][C][Branch1][C][C][N][C][=Branch1][C][=O][N][C][=C][C][=C][C][=C][Ring1][=Branch1][C][=Branch1][C][=O][N][C][C][Branch1][C][C][C][C][Branch1][C][C][C][Ring1][Branch2]
N14CC(C)CC(C)C1.c16ccccc17.CCC5C.C23=O.C47=O.N25.N36
COc1ccc(C(NCC(F)(F)F)C(N)=O)cc1OC
497037
[C][O][C][=C][C][=C][Branch2][Ring1][Ring1][C][Branch1][O][N][C][C][Branch1][C][F][Branch1][C][F][F][C][Branch1][C][N][=O][C][=C][Ring1][S][O][C]
c12ccc6cc13.C46C(N)=O.C5C(F)(F)F.CO2.N45.O3C
CC(C)C(=O)N1CCCC(n2nc(-c3cccs3)ccc2=O)C1
1873141
[C][C][Branch1][C][C][C][=Branch1][C][=O][N][C][C][C][C][Branch2][Ring1][Ring1][N][N][=C][Branch1][Branch2][C][=C][C][=C][S][Ring1][Branch1][C][=C][C][Ring1][O][=O][C][Ring2][Ring1][C]
n15nc6ccc1=O.N14CCCC5C1.CC(C)C4=O.c16cccs1
Cc1nnc(C(C)NC(C)c2cnn(Cc3ccccc3)c2)o1
1562321
[C][C][=N][N][=C][Branch2][Ring1][N][C][Branch1][C][C][N][C][Branch1][C][C][C][C][=N][N][Branch1][#Branch2][C][C][=C][C][=C][C][=C][Ring1][=Branch1][C][=Ring1][N][O][Ring2][Ring1][=Branch1]
Cc1nnc7o1.c18cnn6c1.c19ccccc1.C47C.C58C.N45.C69
O=C(NCc1cccnc1)c1cn(Cc2ccc(F)cc2)nn1
1859683
[O][=C][Branch1][O][N][C][C][=C][C][=C][N][=C][Ring1][=Branch1][C][=C][N][Branch1][=N][C][C][=C][C][=C][Branch1][C][F][C][=C][Ring1][#Branch1][N][=N][Ring1][=N]
c18ccc(F)cc1.c17cccnc1.c15cn6nn1.O=C35.N34.C47.C68
Cn1cc(Cl)cc1CNC(=O)N1CCCC(C2(C)OCCO2)C1
1926181
[C][N][C][=C][Branch1][C][Cl][C][=C][Ring1][=Branch1][C][N][C][=Branch1][C][=O][N][C][C][C][C][Branch1][O][C][Branch1][C][C][O][C][C][O][Ring1][=Branch1][C][Ring1][N]
Cn1cc(Cl)cc16.N14CCCC7C1.C17(C)OCCO1.C34=O.C56.N35
O=C(Nc1ccc2[nH]c(=O)[nH]c2c1)c1ccccc1F
1612913
[O][=C][Branch2][Ring1][C][N][C][=C][C][=C][NH1][C][=Branch1][C][=O][NH1][C][Ring1][=Branch1][=C][Ring1][#Branch2][C][=C][C][=C][C][=C][Ring1][=Branch1][F]
c14ccc2[nH]c(=O)[nH]c2c1.c15ccccc1F.O=C35.N34
COc1ccccc1N1CC(C(=O)N2CCCCC2)CC1=O
515088
[C][O][C][=C][C][=C][C][=C][Ring1][=Branch1][N][C][C][Branch1][=N][C][=Branch1][C][=O][N][C][C][C][C][C][Ring1][=Branch1][C][C][Ring1][=N][=O]
c14ccccc16.N16CC5CC1=O.N13CCCCC1.C35=O.CO4
O=C(NCC1CCCC1)c1ccc(-c2cnco2)cc1
1536018
[O][=C][Branch1][#Branch2][N][C][C][C][C][C][C][Ring1][Branch1][C][=C][C][=C][Branch1][Branch2][C][=C][N][=C][O][Ring1][Branch1][C][=C][Ring1][O]
c15ccc7cc1.C16CCCC1.c17cnco1.O=C35.N34.C46
Cc1nn(C)c2ncc(NC(=O)N3CCOCC3)cc12
1831417
[C][C][=N][N][Branch1][C][C][C][=N][C][=C][Branch1][=C][N][C][=Branch1][C][=O][N][C][C][O][C][C][Ring1][=Branch1][C][=C][Ring2][Ring1][Ring1][Ring1][#C]
Cc1nn(C)c2ncc6cc12.N15CCOCC1.C45=O.N46
Nc1cccc(OCCC(=O)Nc2ccccc2)c1
1816614
[N][C][=C][C][=C][C][Branch1][P][O][C][C][C][=Branch1][C][=O][N][C][=C][C][=C][C][=C][Ring1][=Branch1][=C][Ring2][Ring1][C]
Nc1cccc5c1.c16ccccc1.C4CC3=O.O45.N36
CCCCNC(=O)C1CCN(C(=O)c2c[nH]c3cccc(F)c23)CC1
1382381
[C][C][C][C][N][C][=Branch1][C][=O][C][C][C][N][Branch2][Ring1][Branch1][C][=Branch1][C][=O][C][=C][NH1][C][=C][C][=C][C][Branch1][C][F][=C][Ring1][#Branch2][Ring1][#Branch1][C][C][Ring2][Ring1][C]
c18c[nH]c2cccc(F)c12.C17CCN5CC1.CCCC6.C47=O.C58=O.N46
Cc1ccc(C(=O)N2CCCC2C(=O)NC2CCCC2)cc1
1679873
[C][C][=C][C][=C][Branch2][Ring1][Branch2][C][=Branch1][C][=O][N][C][C][C][C][Ring1][Branch1][C][=Branch1][C][=O][N][C][C][C][C][C][Ring1][Branch1][C][=C][Ring2][Ring1][Branch1]
Cc1ccc7cc1.N13CCCC16.C15CCCC1.C37=O.C46=O.N45
CN(C(=O)c1ccccc1-n1cccn1)c1ccc(F)cc1
762897
[C][N][Branch2][Ring1][Ring2][C][=Branch1][C][=O][C][=C][C][=C][C][=C][Ring1][=Branch1][N][C][=C][C][=N][Ring1][Branch1][C][=C][C][=C][Branch1][C][F][C][=C][Ring1][#Branch1]
c14ccccc15.c13ccc(F)cc1.n15cccn1.CN23.C24=O
CC(=O)Nc1ccc(F)c(NC(=O)NCC(=O)N2CCCC2)c1
1825687
[C][C][=Branch1][C][=O][N][C][=C][C][=C][Branch1][C][F][C][Branch2][Ring1][Ring1][N][C][=Branch1][C][=O][N][C][C][=Branch1][C][=O][N][C][C][C][C][Ring1][Branch1][=C][Ring2][Ring1][Ring1]
c18ccc(F)c9c1.N16CCCC1.C7C6=O.CC3=O.C45=O.N38.N49.N57
CCN(CC(=O)NCc1cccs1)S(=O)(=O)c1cccs1
152227
[C][C][N][Branch1][#C][C][C][=Branch1][C][=O][N][C][C][=C][C][=C][S][Ring1][Branch1][S][=Branch1][C][=O][=Branch1][C][=O][C][=C][C][=C][S][Ring1][Branch1]
S6(=O)(=O)c1cccs1.c17cccs1.C4C2=O.N346.CC3.N25.C57
NC(=O)NC(Cc1ccccc1)C(=O)Nc1ccc(C(N)=O)cc1
359018
[N][C][=Branch1][C][=O][N][C][Branch1][#Branch2][C][C][=C][C][=C][C][=C][Ring1][=Branch1][C][=Branch1][C][=O][N][C][=C][C][=C][Branch1][=Branch1][C][Branch1][C][N][=O][C][=C][Ring1][=Branch2]
c15ccc6cc1.C4(C7)C3=O.c17ccccc1.NC2=O.C6(N)=O.N24.N35
O=C(Oc1cc(Cl)cc(Cl)c1)C1CCCN1
704944
[O][=C][Branch1][S][O][C][=C][C][Branch1][C][Cl][=C][C][Branch1][C][Cl][=C][Ring1][Branch2][C][C][C][C][N][Ring1][Branch1]
c13cc(Cl)cc(Cl)c1.C14CCCN1.O=C24.O23
Cc1cccc(Nc2nc(C(=O)NCC(F)(F)F)cs2)n1
837342
[C][C][=C][C][=C][C][Branch2][Ring1][=Branch2][N][C][=N][C][Branch1][#C][C][=Branch1][C][=O][N][C][C][Branch1][C][F][Branch1][C][F][F][=C][S][Ring1][=N][=N][Ring2][Ring1][Ring2]
Cc1cccc5n1.c16nc7cs1.C4C(F)(F)F.C37=O.N56.N34
CSc1ncccc1C(=O)Nc1cc(-c2nnc(C)o2)sc1C
867465
[C][S][C][=N][C][=C][C][=C][Ring1][=Branch1][C][=Branch1][C][=O][N][C][C][=C][Branch1][O][C][=N][N][=C][Branch1][C][C][O][Ring1][=Branch1][S][C][=Ring1][O][C]
c16ncccc15.c14cc7sc1C.c17nnc(C)o1.C35=O.CS6.N34
CCOC(=O)CS(=O)(=O)Nc1c(C)cccc1O
572095
[C][C][O][C][=Branch1][C][=O][C][S][=Branch1][C][=O][=Branch1][C][=O][N][C][=C][Branch1][C][C][C][=C][C][=C][Ring1][#Branch1][O]
c15c(C)cccc1O.C2(=O)CS4(=O)=O.CC3.O23.N45
CCn1c(-c2ccc(OC)c(C)c2)ccc(C(C)=O)c1=O
1250418
[C][C][N][C][Branch1][S][C][=C][C][=C][Branch1][Ring1][O][C][C][Branch1][C][C][=C][Ring1][=Branch2][=C][C][=C][Branch1][=Branch1][C][Branch1][C][C][=O][C][Ring2][Ring1][C][=O]
n15c6ccc4c1=O.c16ccc3c(C)c1.C4(C)=O.CC5.O3C
CN(Cc1ccco1)C(=O)Nc1nnc(Cc2ccccc2)s1
583645
[C][N][Branch1][=Branch2][C][C][=C][C][=C][O][Ring1][Branch1][C][=Branch1][C][=O][N][C][=N][N][=C][Branch1][#Branch2][C][C][=C][C][=C][C][=C][Ring1][=Branch1][S][Ring1][N]
c16nnc8s1.c19ccccc1.c17ccco1.CN35.C34=O.C57.N46.C89
COc1cccc(OC(C)C(=O)Nc2nc3c(s2)CCCC3)c1
547066
[C][O][C][=C][C][=C][C][Branch2][Ring1][#Branch2][O][C][Branch1][C][C][C][=Branch1][C][=O][N][C][=N][C][=C][Branch1][Ring2][S][Ring1][Branch1][C][C][C][C][Ring1][#Branch1][=C][Ring2][Ring1][Branch1]
c18nc2c(s1)CCCC2.c16cccc7c1.C5(C)C4=O.CO6.O57.N48
Cc1nnnn1-c1cccc(NC(=O)c2scnc2C2CC2)c1
1909963
[C][C][=N][N][=N][N][Ring1][Branch1][C][=C][C][=C][C][Branch2][Ring1][C][N][C][=Branch1][C][=O][C][S][C][=N][C][=Ring1][Branch1][C][C][C][Ring1][Ring1][=C][Ring1][P]
c16cccc4c1.Cc1nnnn16.c15scnc17.C35=O.C17CC1.N34
Cc1ccc(C(O)CNC(=O)c2ccc3ccccc3c2)o1
687545
[C][C][=C][C][=C][Branch2][Ring1][=Branch2][C][Branch1][C][O][C][N][C][=Branch1][C][=O][C][=C][C][=C][C][=C][C][=C][C][Ring1][=Branch1][=C][Ring1][#Branch2][O][Ring2][Ring1][Branch1]
c16ccc2ccccc2c1.Cc1ccc7o1.C7(O)C5.C46=O.N45
COCn1nc(C#N)cc1-c1ccc(OC)cc1C
1129176
[C][O][C][N][N][=C][Branch1][Ring1][C][#N][C][=C][Ring1][#Branch1][C][=C][C][=C][Branch1][Ring1][O][C][C][=C][Ring1][Branch2][C]
n13nc(C#N)cc14.c14ccc2cc1C.COC3.O2C
CC(=O)c1ccc(S(=O)(=O)Nc2ccc(Cl)cc2F)cc1
128318
[C][C][=Branch1][C][=O][C][=C][C][=C][Branch2][Ring1][Branch1][S][=Branch1][C][=O][=Branch1][C][=O][N][C][=C][C][=C][Branch1][C][Cl][C][=C][Ring1][#Branch1][F][C][=C][Ring2][Ring1][C]
c15ccc(S3(=O)=O)cc1.c14ccc(Cl)cc1F.CC5=O.N34
CN(CCc1ccccn1)C(=O)Nc1ccnn1CC1CC=CCC1
1506021
[C][N][Branch1][O][C][C][C][=C][C][=C][C][=N][Ring1][=Branch1][C][=Branch1][C][=O][N][C][=C][C][=N][N][Ring1][Branch1][C][C][C][C][=C][C][C][Ring1][=Branch1]
c17ccccn1.c15ccnn16.C18CC=CCC1.CN24.C4C7.C23=O.N35.C68
Cc1c(C(=O)NC2CC3C(=O)NCC(=O)N3C2)sc2ccccc12
915821
[C][C][=C][Branch2][Ring1][=Branch2][C][=Branch1][C][=O][N][C][C][C][C][=Branch1][C][=O][N][C][C][=Branch1][C][=O][N][Ring1][Branch2][C][Ring1][O][S][C][=C][C][=C][C][=C][Ring2][Ring1][#Branch1][Ring1][=Branch1]
C15CC2C(=O)NCC(=O)N2C1.Cc1c6sc2ccccc12.C46=O.N45
COC(=O)CC(C)NC(=O)c1ccccc1OC(F)F
983745
[C][O][C][=Branch1][C][=O][C][C][Branch1][C][C][N][C][=Branch1][C][=O][C][=C][C][=C][C][=C][Ring1][=Branch1][O][C][Branch1][C][F][F]
c16ccccc14.C2(=O)CC5C.O4C(F)F.C36=O.CO2.N35
OCc1c(-c2cccnc2)nc2sc(C3CCC3)nn12
844573
[O][C][C][=C][Branch1][=Branch2][C][=C][C][=C][N][=C][Ring1][=Branch1][N][=C][S][C][Branch1][#Branch1][C][C][C][C][Ring1][Ring2][=N][N][Ring2][Ring1][C][Ring1][=Branch2]
c14c6nc2sc5nn12.c16cccnc1.C15CCC1.OC4
O=C(CNC(=O)c1ccco1)Nc1cccc2c1CCCC2
377081
[O][=C][Branch1][=C][C][N][C][=Branch1][C][=O][C][=C][C][=C][O][Ring1][Branch1][N][C][=C][C][=C][C][=C][Ring1][=Branch1][C][C][C][C][Ring1][=Branch1]
c16cccc2c1CCCC2.c17ccco1.O=C3C5.C47=O.N45.N36
COc1ccccc1NC(=O)c1cccnc1NCc1ccccc1
352007
[C][O][C][=C][C][=C][C][=C][Ring1][=Branch1][N][C][=Branch1][C][=O][C][=C][C][=C][N][=C][Ring1][=Branch1][N][C][C][=C][C][=C][C][=C][Ring1][=Branch1]
c13ccccc16.c17cccnc15.c18ccccc1.C27=O.CO3.N26.N45.C48
COCCn1cc(CC(=O)Nc2cccc(C)c2)c2cccnc21
868075
[C][O][C][C][N][C][=C][Branch2][Ring1][C][C][C][=Branch1][C][=O][N][C][=C][C][=C][C][Branch1][C][C][=C][Ring1][#Branch1][C][=C][C][=C][N][=C][Ring1][=Branch1][Ring2][Ring1][Ring2]
n16cc7c2cccnc21.c15cccc(C)c1.C7C3=O.C4C6.CO4.N35
COc1cc(C(=O)NCC=Cc2ccccc2)cc(OC)c1OC
1217899
[C][O][C][=C][C][Branch1][P][C][=Branch1][C][=O][N][C][C][=C][C][=C][C][=C][C][=C][Ring1][=Branch1][=C][C][Branch1][Ring1][O][C][=C][Ring2][Ring1][Ring2][O][C]
c14cc8cc5c16.C=9c1ccccc1.C38=O.C7C=9.CO4.N37.O5C.O6C
CC(=O)Nc1cc(NS(=O)(=O)c2ccc(C)cc2)ccc1Cl
852405
[C][C][=Branch1][C][=O][N][C][=C][C][Branch2][Ring1][Ring2][N][S][=Branch1][C][=O][=Branch1][C][=O][C][=C][C][=C][Branch1][C][C][C][=C][Ring1][#Branch1][=C][C][=C][Ring1][P][Cl]
S4(=O)(=O)c1ccc(C)cc1.c15cc6ccc1Cl.CC3=O.N35.N46
Cc1nc2c(SCC(N)=O)nnc(-c3ccccc3)c2s1
1609602
[C][C][=N][C][=C][Branch1][Branch2][S][C][C][Branch1][C][N][=O][N][=N][C][Branch1][=Branch2][C][=C][C][=C][C][=C][Ring1][=Branch1][=C][Ring1][P][S][Ring2][Ring1][Ring2]
Cc1nc2c5nnc6c2s1.c16ccccc1.C4C(N)=O.S45
N#CC(NC(=O)c1scnc1C1CC1)c1cccc(Cl)c1
1376275
[N][#C][C][Branch2][Ring1][C][N][C][=Branch1][C][=O][C][S][C][=N][C][=Ring1][Branch1][C][C][C][Ring1][Ring1][C][=C][C][=C][C][Branch1][C][Cl][=C][Ring1][#Branch1]
c15cccc(Cl)c1.c14scnc16.N#CC35.C24=O.C16CC1.N23
COC(=O)c1sc(COc2cccc(C)c2)nc1C
707866
[C][O][C][=Branch1][C][=O][C][S][C][Branch1][=C][C][O][C][=C][C][=C][C][Branch1][C][C][=C][Ring1][#Branch1][=N][C][=Ring1][=C][C]
c16sc7nc1C.c15cccc(C)c1.C36=O.CO3.C47.O45
CC(C)CNC(=O)c1nc(-c2c[nH]c3ccccc23)no1
226838
[C][C][Branch1][C][C][C][N][C][=Branch1][C][=O][C][=N][C][Branch1][=C][C][=C][NH1][C][=C][C][=C][C][=C][Ring1][=Branch2][Ring1][=Branch1][=N][O][Ring1][=C]
c17c[nH]c2ccccc12.c16nc7no1.CC(C)C5.C46=O.N45
CC(C)CCNC(=O)CNc1cccc(F)c1F
677877
[C][C][Branch1][C][C][C][C][N][C][=Branch1][C][=O][C][N][C][=C][C][=C][C][Branch1][C][F][=C][Ring1][#Branch1][F]
c15cccc(F)c1F.CC(C)CC3.C2(=O)C4.N23.N45
CCCCNC(=O)c1csc(Nc2ncccn2)n1
776857
[C][C][C][C][N][C][=Branch1][C][=O][C][=C][S][C][Branch1][#Branch2][N][C][=N][C][=C][C][=N][Ring1][=Branch1][=N][Ring1][N]
c17csc5n1.c16ncccn1.CCCC4.C37=O.N34.N56
Cc1cc(C)c(OC(=O)CN(C)C(=O)c2cccs2)c(C)c1
1088223
[C][C][=C][C][Branch1][C][C][=C][Branch2][Ring1][=Branch1][O][C][=Branch1][C][=O][C][N][Branch1][C][C][C][=Branch1][C][=O][C][=C][C][=C][S][Ring1][Branch1][C][Branch1][C][C][=C][Ring2][Ring1][Branch1]
Cc1cc(C)c5c(C)c1.c17cccs1.C3(=O)C6.N46C.C47=O.O35
Cc1cc(Cl)ccc1N(CC(=O)N(C)C)S(C)(=O)=O
23369
[C][C][=C][C][Branch1][C][Cl][=C][C][=C][Ring1][#Branch1][N][Branch1][O][C][C][=Branch1][C][=O][N][Branch1][C][C][C][S][Branch1][C][C][=Branch1][C][=O][=O]
Cc1cc(Cl)ccc15.C3C2=O.S4(C)(=O)=O.N345.N2(C)C
CNc1ccc(Oc2ccc(F)cc2C(N)=O)cc1
959244
[C][N][C][=C][C][=C][Branch2][Ring1][C][O][C][=C][C][=C][Branch1][C][F][C][=C][Ring1][#Branch1][C][Branch1][C][N][=O][C][=C][Ring1][P]
c14ccc(F)cc16.c15ccc3cc1.C6(N)=O.CN5.O34
CN(C(=O)CSc1nc2c(c(=O)[nH]1)CCC2)c1ccccc1
297702
[C][N][Branch2][Ring1][=Branch2][C][=Branch1][C][=O][C][S][C][=N][C][=C][Branch1][Branch2][C][=Branch1][C][=O][NH1][Ring1][#Branch1][C][C][C][Ring1][Branch2][C][=C][C][=C][C][=C][Ring1][=Branch1]
c16nc2c(c(=O)[nH]1)CCC2.c15ccccc1.C3(=O)C4.CN35.S46
Cc1nonc1CN(C)S(=O)(=O)NCc1ccccc1
978846
[C][C][=N][O][N][=C][Ring1][Branch1][C][N][Branch1][C][C][S][=Branch1][C][=O][=Branch1][C][=O][N][C][C][=C][C][=C][C][=C][Ring1][=Branch1]
N2(C)S(=O)(=O)N3.Cc1nonc14.c15ccccc1.C24.C35
CC1CC1CNC(=O)NCc1cccc(Cl)c1
634138
[C][C][C][C][Ring1][Ring1][C][N][C][=Branch1][C][=O][N][C][C][=C][C][=C][C][Branch1][C][Cl][=C][Ring1][#Branch1]
c17cccc(Cl)c1.CC1CC16.C23=O.C46.N24.N35.C57
CC(C)N1CC(C(=O)NCc2ncc3c(n2)CCC3)CC1=O
1155597
[C][C][Branch1][C][C][N][C][C][Branch2][Ring1][=Branch1][C][=Branch1][C][=O][N][C][C][=N][C][=C][C][=Branch1][Ring2][=N][Ring1][=Branch1][C][C][C][Ring1][=Branch1][C][C][Ring2][Ring1][C][=O]
c18ncc2c(n1)CCC2.N17CC6CC1=O.CC7C.C46=O.N45.C58
CCOCCCNC(=O)c1sccc1Br
534806
[C][C][O][C][C][C][N][C][=Branch1][C][=O][C][S][C][=C][C][=Ring1][Branch1][Br]
c16sccc1Br.C4CC5.C26=O.CC3.O34.N25
COc1ccc(F)cc1NC(=O)CCc1nc(C2CCCC2)no1
1445065
[C][O][C][=C][C][=C][Branch1][C][F][C][=C][Ring1][#Branch1][N][C][=Branch1][C][=O][C][C][C][=N][C][Branch1][Branch2][C][C][C][C][C][Ring1][Branch1][=N][O][Ring1][#Branch2]
c14ccc(F)cc15.c16nc7no1.C3(=O)CC6.C17CCCC1.CO4.N35
Cc1noc(C)c1NC(=O)N(C)Cc1cccc(Cl)c1
1850410
[C][C][=N][O][C][Branch1][C][C][=C][Ring1][=Branch1][N][C][=Branch1][C][=O][N][Branch1][C][C][C][C][=C][C][=C][C][Branch1][C][Cl][=C][Ring1][#Branch1]
Cc1noc(C)c15.c16cccc(Cl)c1.C23=O.N34C.N25.C46
O=C(NCCn1nnn(-c2cccs2)c1=O)C1CCCCC1
1794763
[O][=C][Branch2][Ring1][Branch1][N][C][C][N][N][=N][N][Branch1][Branch2][C][=C][C][=C][S][Ring1][Branch1][C][Ring1][#Branch2][=O][C][C][C][C][C][C][Ring1][=Branch1]
n16nnn7c1=O.C15CCCCC1.c17cccs1.O=C35.C4C6.N34
CCC(NC(=O)Nc1cc(C)cc2cccnc12)c1c(C)noc1C
1919166
[C][C][C][Branch2][Ring1][Branch2][N][C][=Branch1][C][=O][N][C][=C][C][Branch1][C][C][=C][C][=C][C][=C][N][=C][Ring1][O][Ring1][=Branch1][C][C][Branch1][C][C][=N][O][C][=Ring1][=Branch1][C]
c16cc(C)cc2cccnc12.c17c(C)noc1C.CCC57.C34=O.N35.N46
CCOC(CC)C(=O)N(Cc1cccc(C)c1)C1CC1
1579004
[C][C][O][C][Branch1][Ring1][C][C][C][=Branch1][C][=O][N][Branch1][=N][C][C][=C][C][=C][C][Branch1][C][C][=C][Ring1][#Branch1][C][C][C][Ring1][Ring1]
c17cccc(C)c1.C4(CC)C2=O.N256.C16CC1.CC3.O34.C57
COc1ccc(-c2cc(CO)ccn2)c(-n2nc(C)cc2C)c1
1935460
[C][O][C][=C][C][=C][Branch1][=N][C][=C][C][Branch1][Ring1][C][O][=C][C][=N][Ring1][Branch2][C][Branch1][N][N][N][=C][Branch1][C][C][C][=C][Ring1][=Branch1][C][=C][Ring2][Ring1][Branch1]
c13ccc6c5c1.c16cc4ccn1.n15nc(C)cc1C.CO3.C4O
CC1(C)C2CCC1(CS(=O)(=O)NCCCO)C(=O)C2
1275499
[C][C][Branch1][C][C][C][C][C][C][Ring1][=Branch1][Branch1][=C][C][S][=Branch1][C][=O][=Branch1][C][=O][N][C][C][C][O][C][=Branch1][C][=O][C][Ring1][S]
CC1(C)C2CCC15C(=O)C2.C5S4(=O)=O.C3CCO.N34
O=C(CNc1cc(F)cc(F)c1)Nc1cccc(F)c1
1620438
[O][=C][Branch1][P][C][N][C][=C][C][Branch1][C][F][=C][C][Branch1][C][F][=C][Ring1][Branch2][N][C][=C][C][=C][C][Branch1][C][F][=C][Ring1][#Branch1]
c14cc(F)cc(F)c1.c15cccc(F)c1.O=C2C3.N34.N25
Cc1nnc(SCCCOc2ccccc2)n1N
1190471
[C][C][=N][N][=C][Branch1][=C][S][C][C][C][O][C][=C][C][=C][C][=C][Ring1][=Branch1][N][Ring1][S][N]
Cc1nnc6n1N.c14ccccc1.C5CC3.S56.O34
COC(=O)C(C)CNC(=O)Nc1cc(F)ccc1-n1cccn1
1290746
[C][O][C][=Branch1][C][=O][C][Branch1][C][C][C][N][C][=Branch1][C][=O][N][C][=C][C][Branch1][C][F][=C][C][=C][Ring1][#Branch1][N][C][=C][C][=N][Ring1][Branch1]
c16cc(F)ccc17.C2(=O)C(C)C5.n17cccn1.C34=O.CO2.N35.N46
CCN(C)C(=O)c1cccc(OCC(=O)Nc2ccccc2Cl)c1
1124304
[C][C][N][Branch1][C][C][C][=Branch1][C][=O][C][=C][C][=C][C][Branch1][P][O][C][C][=Branch1][C][=O][N][C][=C][C][=C][C][=C][Ring1][=Branch1][Cl][=C][Ring2][Ring1][C]
c19cccc6c1.c18ccccc1Cl.C5C4=O.N37C.C39=O.CC7.O56.N48
CNC(=O)c1ccc(S(=O)(=O)NC(C(=O)OC)C(C)(C)C)cc1
997832
[C][N][C][=Branch1][C][=O][C][=C][C][=C][Branch2][Ring1][#Branch2][S][=Branch1][C][=O][=Branch1][C][=O][N][C][Branch1][#Branch1][C][=Branch1][C][=O][O][C][C][Branch1][C][C][Branch1][C][C][C][C][=C][Ring2][Ring1][Ring1]
c16ccc(S5(=O)=O)cc1.C4(C2=O)C(C)(C)C.C36=O.CN3.N45.O2C
CC(NC(N)=O)C(=O)NCCCC1CCCCC1
621613
[C][C][Branch1][#Branch1][N][C][Branch1][C][N][=O][C][=Branch1][C][=O][N][C][C][C][C][C][C][C][C][C][Ring1][=Branch1]
C16CCCCC1.CC4C3=O.C5CC6.C2(N)=O.N24.N35
COCCN1CCN(C(=O)c2ccccc2-n2cccn2)CC1=O
1418667
[C][O][C][C][N][C][C][N][Branch2][Ring1][Ring2][C][=Branch1][C][=O][C][=C][C][=C][C][=C][Ring1][=Branch1][N][C][=C][C][=N][Ring1][Branch1][C][C][Ring2][Ring1][Ring1][=O]
N16CCN3CC1=O.c15ccccc17.n17cccn1.C4C6.C35=O.CO4
COc1ccc(C2CCCN2C(=O)COc2ccc(C)nc2)cc1
1457449
[C][O][C][=C][C][=C][Branch2][Ring1][=Branch2][C][C][C][C][N][Ring1][Branch1][C][=Branch1][C][=O][C][O][C][=C][C][=C][Branch1][C][C][N][=C][Ring1][#Branch1][C][=C][Ring2][Ring1][=Branch1]
c15ccc7cc1.c16ccc(C)nc1.C17CCCN13.C3(=O)C4.CO5.O46
CC(=O)NC(C(=O)NC(C)c1ccc(CC(C)C)cc1)C(C)C
401177
[C][C][=Branch1][C][=O][N][C][Branch2][Ring1][#Branch2][C][=Branch1][C][=O][N][C][Branch1][C][C][C][=C][C][=C][Branch1][#Branch1][C][C][Branch1][C][C][C][C][=C][Ring1][#Branch2][C][Branch1][C][C][C]
C4(C3=O)C(C)C.c16ccc7cc1.C7C(C)C.CC2=O.C56C.N24.N35
Cc1cc(NC(=O)CN2CCOC(CNc3cccnn3)C2)no1
1211562
[C][C][=C][C][Branch2][Ring1][O][N][C][=Branch1][C][=O][C][N][C][C][O][C][Branch1][O][C][N][C][=C][C][=C][N][=N][Ring1][=Branch1][C][Ring1][=C][=N][O][Ring2][Ring1][#Branch1]
N15CCOC9C1.Cc1cc7no1.c18cccnn1.C4(=O)C5.N47.C69.N68
Cc1cc(=O)oc(C)c1C(=O)Nc1ccccc1C(=O)N1CCCC1
1761430
[C][C][=C][C][=Branch1][C][=O][O][C][Branch1][C][C][=C][Ring1][Branch2][C][=Branch1][C][=O][N][C][=C][C][=C][C][=C][Ring1][=Branch1][C][=Branch1][C][=O][N][C][C][C][C][Ring1][Branch1]
Cc1cc(=O)oc(C)c15.c14ccccc16.N13CCCC1.C25=O.C36=O.N24
Cc1nn(-c2ccccc2)c(C)c1C(=O)Nc1cccc(O)c1
1577704
[C][C][=N][N][Branch1][=Branch2][C][=C][C][=C][C][=C][Ring1][=Branch1][C][Branch1][C][C][=C][Ring1][N][C][=Branch1][C][=O][N][C][=C][C][=C][C][Branch1][C][O][=C][Ring1][#Branch1]
Cc1nn6c(C)c15.c14cccc(O)c1.c16ccccc1.C35=O.N34
Cn1ccc(NC(=O)c2cc3c(nc4sccn43)s2)n1
372370
[C][N][C][=C][C][Branch2][Ring1][=Branch2][N][C][=Branch1][C][=O][C][=C][C][=C][Branch1][O][N][=C][S][C][=C][N][Ring1][Branch1][Ring1][Branch2][S][Ring1][O][=N][Ring2][Ring1][Ring1]
c17cc2c(nc3sccn32)s1.Cn1ccc6n1.C57=O.N56
CN(CCC#N)C(=O)CN1CCn2c(nnc2C2CC2)C1
1900361
[C][N][Branch1][Branch1][C][C][C][#N][C][=Branch1][C][=O][C][N][C][C][N][C][=Branch1][O][=N][N][=C][Ring1][Branch1][C][C][C][Ring1][Ring1][C][Ring1][N]
N15CCn2c6nnc2C1.C4CC#N.C3(=O)C5.CN34.C16CC1
Cn1cc(CCNS(=O)(=O)c2cccc(C(F)(F)F)c2)cn1
575924
[C][N][C][=C][Branch2][Ring1][=N][C][C][N][S][=Branch1][C][=O][=Branch1][C][=O][C][=C][C][=C][C][Branch1][=Branch2][C][Branch1][C][F][Branch1][C][F][F][=C][Ring1][#Branch2][C][=N][Ring2][Ring1][Branch1]
S4(=O)(=O)c1cccc6c1.Cn1cc5cn1.C6(F)(F)F.C5C3.N34
CCOc1ccc(S(=O)(=O)NCCCO)cc1C
458122
[C][C][O][C][=C][C][=C][Branch1][=N][S][=Branch1][C][=O][=Branch1][C][=O][N][C][C][C][O][C][=C][Ring1][=C][C]
c13ccc(S5(=O)=O)cc1C.C4CCO.CC2.O23.N45
Cc1oc2nc(CN3CCc4ccc(Cl)cc4C3)nc(N)c2c1C
1393842
[C][C][O][C][=N][C][Branch2][Ring1][Ring1][C][N][C][C][C][=C][C][=C][Branch1][C][Cl][C][=C][Ring1][#Branch1][C][Ring1][O][=N][C][Branch1][C][N][=C][Ring2][Ring1][Ring1][C][=Ring2][Ring1][=Branch1][C]
Cc1oc2nc6nc(N)c2c1C.N15CCc2ccc(Cl)cc2C1.C56
Cc1ccc(-c2ncco2)cc1NC(=O)NCC(C)Cn1cccn1
1324115
[C][C][=C][C][=C][Branch1][Branch2][C][=N][C][=C][O][Ring1][Branch1][C][=C][Ring1][O][N][C][=Branch1][C][=O][N][C][C][Branch1][C][C][C][N][C][=C][C][=N][Ring1][Branch1]
Cc1ccc8cc16.c18ncco1.C5C(C)C7.n17cccn1.C34=O.N36.N45
NC(=O)Cn1c(Cc2ccc(F)cc2)nc2c(N)cccc21
474045
[N][C][=Branch1][C][=O][C][N][C][Branch1][=N][C][C][=C][C][=C][Branch1][C][F][C][=C][Ring1][#Branch1][=N][C][=C][Branch1][C][N][C][=C][C][=C][Ring1][#Branch1][Ring2][Ring1][C]
n13c4nc2c(N)cccc21.c15ccc(F)cc1.NC(=O)C3.C45
CC(C)(C)NC(=O)C1CCN(S(=O)(=O)Cc2ccccc2)CC1
1798546
[C][C][Branch1][C][C][Branch1][C][C][N][C][=Branch1][C][=O][C][C][C][N][Branch1][P][S][=Branch1][C][=O][=Branch1][C][=O][C][C][=C][C][=C][C][=C][Ring1][=Branch1][C][C][Ring1][S]
C16CCN5CC1.c17ccccc1.S5(=O)(=O)C7.CC4(C)C.C36=O.N34
COc1ccc(-c2noc(CC(=O)N3CCC(C)CC3)n2)cc1
144764
[C][O][C][=C][C][=C][Branch2][Ring1][#Branch2][C][=N][O][C][Branch1][P][C][C][=Branch1][C][=O][N][C][C][C][Branch1][C][C][C][C][Ring1][#Branch1][=N][Ring1][#C][C][=C][Ring2][Ring1][Branch1]
c15ccc7cc1.N14CCC(C)CC1.c17noc6n1.C6C4=O.CO5
CC1CCCC(CNC(=O)NCC(=O)N(C)C)C1
774532
[C][C][C][C][C][C][Branch2][Ring1][C][C][N][C][=Branch1][C][=O][N][C][C][=Branch1][C][=O][N][Branch1][C][C][C][C][Ring1][P]
CC1CCCC7C1.C6C4=O.C23=O.N4(C)C.C57.N25.N36
Cc1[nH]c(C(=O)N(C)C2CC2)c(C)c1C(=O)OC(C)C
619864
[C][C][NH1][C][Branch1][=C][C][=Branch1][C][=O][N][Branch1][C][C][C][C][C][Ring1][Ring1][=C][Branch1][C][C][C][=Ring1][=N][C][=Branch1][C][=O][O][C][Branch1][C][C][C]
Cc1[nH]c7c(C)c18.C47=O.N46C.C16CC1.C38=O.C5(C)C.O35
Cc1cc(C)nc(N2CCCC(C(=O)NC(C)C)C2)n1
103049
[C][C][=C][C][Branch1][C][C][=N][C][Branch2][Ring1][Branch1][N][C][C][C][C][Branch1][O][C][=Branch1][C][=O][N][C][Branch1][C][C][C][C][Ring1][N][=N][Ring2][Ring1][Ring1]
Cc1cc(C)nc5n1.N15CCCC6C1.C36=O.C4(C)C.N34
Cc1cc(C)cc(N2CCC(C(=O)NCCCOC(C)C)C2=O)c1
736193
[C][C][=C][C][Branch1][C][C][=C][C][Branch2][Ring1][=Branch2][N][C][C][C][Branch1][#C][C][=Branch1][C][=O][N][C][C][C][O][C][Branch1][C][C][C][C][Ring1][#C][=O][=C][Ring2][Ring1][#Branch1]
Cc1cc8cc(C)c1.N18CCC7C1=O.C6CC4.C37=O.C5(C)C.N36.O45
CC(NC(=O)CNc1ccc(C(=O)N(C)C)cc1)c1ccccc1
897782
[C][C][Branch2][Ring1][O][N][C][=Branch1][C][=O][C][N][C][=C][C][=C][Branch1][#Branch2][C][=Branch1][C][=O][N][Branch1][C][C][C][C][=C][Ring1][O][C][=C][C][=C][C][=C][Ring1][=Branch1]
c16ccc7cc1.c18ccccc1.C2(=O)C5.CC48.C37=O.N3(C)C.N24.N56
CC(NC(=O)Nc1ccc(Br)cc1F)c1ccncc1
582323
[C][C][Branch2][Ring1][Ring1][N][C][=Branch1][C][=O][N][C][=C][C][=C][Branch1][C][Br][C][=C][Ring1][#Branch1][F][C][=C][C][=N][C][=C][Ring1][=Branch1]
c15ccc(Br)cc1F.c16ccncc1.CC46.C23=O.N24.N35
COc1cc(OC)cc(C(NC(=O)c2ccc[nH]2)c2nccn2C)c1
1656117
[C][O][C][=C][C][Branch1][Ring1][O][C][=C][C][Branch2][Ring1][Branch2][C][Branch1][=N][N][C][=Branch1][C][=O][C][=C][C][=C][NH1][Ring1][Branch1][C][=N][C][=C][N][Ring1][Branch1][C][=C][Ring2][Ring1][#Branch1]
c14cc5cc9c1.c18nccn1C.c17ccc[nH]1.C689.C37=O.CO4.O5C.N36
CCCn1cc(NC(=O)Nc2ccc(F)c(C(=O)NC)c2)cn1
1875549
[C][C][C][N][C][=C][Branch2][Ring1][#Branch2][N][C][=Branch1][C][=O][N][C][=C][C][=C][Branch1][C][F][C][Branch1][#Branch1][C][=Branch1][C][=O][N][C][=C][Ring1][O][C][=N][Ring2][Ring1][Ring2]
c17ccc(F)c8c1.n19cc6cn1.CCC9.C34=O.C58=O.N36.N47.N5C
CCC(=O)NC(Nc1ccccn1)(C(=O)OC)C(F)(F)F
321941
[C][C][C][=Branch1][C][=O][N][C][Branch1][#Branch2][N][C][=C][C][=C][C][=N][Ring1][=Branch1][Branch1][#Branch1][C][=Branch1][C][=O][O][C][C][Branch1][C][F][Branch1][C][F][F]
C45(C2=O)C(F)(F)F.c16ccccn1.CCC3=O.N34.N56.O2C
CCCn1c(SC(C)C(=O)N(C)C2CCCCC2)n[nH]c1=O
206583
[C][C][C][N][C][Branch2][Ring1][=Branch1][S][C][Branch1][C][C][C][=Branch1][C][=O][N][Branch1][C][C][C][C][C][C][C][C][Ring1][=Branch1][=N][NH1][C][Ring2][Ring1][C][=O]
n16c7n[nH]c1=O.C15CCCCC1.C4(C)C3=O.CCC6.N35C.S47
COc1ccc(N(C)C(=O)c2cccnc2N)cc1
722147
[C][O][C][=C][C][=C][Branch2][Ring1][C][N][Branch1][C][C][C][=Branch1][C][=O][C][=C][C][=C][N][=C][Ring1][=Branch1][N][C][=C][Ring1][P]
c14ccc5cc1.c16cccnc1N.N35C.C36=O.CO4
Cc1nc(CNC(=O)c2ccc3c(c2)OCO3)cs1
565320
[C][C][=N][C][Branch2][Ring1][=Branch1][C][N][C][=Branch1][C][=O][C][=C][C][=C][C][=Branch1][Ring2][=C][Ring1][=Branch1][O][C][O][Ring1][=Branch1][=C][S][Ring2][Ring1][C]
c16ccc2c(c1)OCO2.Cc1nc7cs1.C46=O.C57.N45
O=C(CCCSc1nnc(C2=NC=CC2)o1)c1ccc(F)cc1
1641599
[O][=C][Branch2][Ring1][Branch1][C][C][C][S][C][=N][N][=C][Branch1][Branch2][C][=N][C][=C][C][Ring1][Branch1][O][Ring1][#Branch2][C][=C][C][=C][Branch1][C][F][C][=C][Ring1][#Branch1]
c15nnc(C2=NC=CC2)o1.c14ccc(F)cc1.O=C4CCC3.S35
Cc1cc2ncn(CC(=O)NCCc3ccc(F)cc3)c2cc1C
344656
[C][C][=C][C][N][=C][N][Branch2][Ring1][Ring2][C][C][=Branch1][C][=O][N][C][C][C][=C][C][=C][Branch1][C][F][C][=C][Ring1][#Branch1][C][=Ring2][Ring1][C][C][=C][Ring2][Ring1][=Branch1][C]
Cc1cc2ncn6c2cc1C.c17ccc(F)cc1.C6C4=O.C5C7.N45