SMILES
large_stringlengths
17
56
ID
large_stringlengths
1
7
SELFIES
stringlengths
63
275
SAFE
stringlengths
20
78
O=C(Cc1ccon1)Nc1sc2c(c1C(=O)NC1CC1)CCC2
1074642
[O][=C][Branch1][=Branch2][C][C][C][=C][O][N][=Ring1][Branch1][N][C][S][C][=C][Branch1][=C][C][=Ring1][Branch1][C][=Branch1][C][=O][N][C][C][C][Ring1][Ring1][C][C][C][Ring1][N]
c15sc2c(c17)CCC2.c18ccon1.O=C3C8.C47=O.C16CC1.N35.N46
COCCCN1C(=O)CCC1(C)C(=O)NC1CCCC1
348016
[C][O][C][C][C][N][C][=Branch1][C][=O][C][C][C][Ring1][=Branch1][Branch1][C][C][C][=Branch1][C][=O][N][C][C][C][C][C][Ring1][Branch1]
N16C(=O)CCC15C.C14CCCC1.C3CC6.C25=O.CO3.N24
COc1ccc(NC(=O)CCc2ccsc2)cc1S(N)(=O)=O
358652
[C][O][C][=C][C][=C][Branch1][#C][N][C][=Branch1][C][=O][C][C][C][C][=C][S][C][=Ring1][Branch1][C][=C][Ring1][S][S][Branch1][C][N][=Branch1][C][=O][=O]
c14ccc5cc1S(N)(=O)=O.C3(=O)CC6.c16ccsc1.CO4.N35
CN(Cc1ccccn1)C(=O)NCCCn1cccn1
1846301
[C][N][Branch1][#Branch2][C][C][=C][C][=C][C][=N][Ring1][=Branch1][C][=Branch1][C][=O][N][C][C][C][N][C][=C][C][=N][Ring1][Branch1]
c17ccccn1.n16cccn1.C5CC6.CN24.C23=O.C47.N35
NC(=O)NCc1ccc(NC(=O)c2csnn2)cc1
685252
[N][C][=Branch1][C][=O][N][C][C][=C][C][=C][Branch1][=N][N][C][=Branch1][C][=O][C][=C][S][N][=N][Ring1][Branch1][C][=C][Ring1][=C]
c18ccc6cc1.c17csnn1.NC3=O.C47=O.N35.C58.N46
CCC(C)C(=O)NCc1cc(OC)c(OC)c(OC)c1
356396
[C][C][C][Branch1][C][C][C][=Branch1][C][=O][N][C][C][=C][C][Branch1][Ring1][O][C][=C][Branch1][Ring1][O][C][C][Branch1][Ring1][O][C][=C][Ring1][N]
c17cc3c4c5c1.CCC(C)C2=O.N26.C67.O3C.O4C.O5C
CNC(=O)c1cc(N(C)CC(O)COC)ccn1
571678
[C][N][C][=Branch1][C][=O][C][=C][C][Branch1][=N][N][Branch1][C][C][C][C][Branch1][C][O][C][O][C][=C][C][=N][Ring1][=C]
c16cc5ccn1.C4C(O)C3.C26=O.N45C.CN2.O3C
C=CCNC(=O)CCC(O)c1ccc(C(C)C)cc1
1662844
[C][=C][C][N][C][=Branch1][C][=O][C][C][C][Branch1][C][O][C][=C][C][=C][Branch1][=Branch1][C][Branch1][C][C][C][C][=C][Ring1][=Branch2]
C2(=O)CCC4O.c14ccc5cc1.C=CC3.C5(C)C.N23
O=C(NCc1ccccc1Cn1cccn1)C1CCCO1
402501
[O][=C][Branch2][Ring1][Ring1][N][C][C][=C][C][=C][C][=C][Ring1][=Branch1][C][N][C][=C][C][=N][Ring1][Branch1][C][C][C][C][O][Ring1][Branch1]
c16ccccc17.n15cccn1.C14CCCO1.O=C24.N23.C36.C57
COCCN(C)C(=O)Nc1cc(OC)c(OC)cc1Br
676549
[C][O][C][C][N][Branch1][C][C][C][=Branch1][C][=O][N][C][=C][C][Branch1][Ring1][O][C][=C][Branch1][Ring1][O][C][C][=C][Ring1][#Branch2][Br]
c18cc5c6cc1Br.C4C7.N27C.C23=O.CO4.N38.O5C.O6C
Cc1ccc(C)c(NC(=O)c2cncc(Br)c2)c1
1587056
[C][C][=C][C][=C][Branch1][C][C][C][Branch1][P][N][C][=Branch1][C][=O][C][=C][N][=C][C][Branch1][C][Br][=C][Ring1][#Branch1][=C][Ring1][P]
Cc1ccc(C)c4c1.c15cncc(Br)c1.C35=O.N34
COCc1nn(CCNC(=O)C2CCCC2)c(=O)o1
1484314
[C][O][C][C][=N][N][Branch1][#C][C][C][N][C][=Branch1][C][=O][C][C][C][C][C][Ring1][Branch1][C][=Branch1][C][=O][O][Ring1][S]
c18nn7c(=O)o1.C16CCCC1.C7C5.C36=O.CO4.C48.N35
CCOC(=O)C(O)(c1cc(Cl)ccc1O)C(F)(F)F
1100615
[C][C][O][C][=Branch1][C][=O][C][Branch1][C][O][Branch1][=N][C][=C][C][Branch1][C][Cl][=C][C][=C][Ring1][#Branch1][O][C][Branch1][C][F][Branch1][C][F][F]
C2(=O)C4(O)C(F)(F)F.c14cc(Cl)ccc1O.CC3.O23
CCCC1CN(C(=O)CCCOc2cccc(F)c2)CCO1
1908040
[C][C][C][C][C][N][Branch2][Ring1][Ring2][C][=Branch1][C][=O][C][C][C][O][C][=C][C][=C][C][Branch1][C][F][=C][Ring1][#Branch1][C][C][O][Ring2][Ring1][Ring1]
C16CN3CCO1.c15cccc(F)c1.C3(=O)CCC4.CCC6.O45
Cc1ccc(NC(=O)Cn2ccc3c(=O)[nH]ccc32)c(C)c1
449190
[C][C][=C][C][=C][Branch2][Ring1][#Branch1][N][C][=Branch1][C][=O][C][N][C][=C][C][C][=Branch1][C][=O][NH1][C][=C][C][=Ring1][#Branch1][Ring1][#Branch2][C][Branch1][C][C][=C][Ring2][Ring1][Branch1]
n16ccc2c(=O)[nH]ccc21.Cc1ccc5c(C)c1.C4(=O)C6.N45
O=C(NCc1cccc(Cn2cccn2)c1)Nc1ccc2[nH]ccc2c1
941786
[O][=C][Branch2][Ring1][Branch1][N][C][C][=C][C][=C][C][Branch1][=Branch2][C][N][C][=C][C][=N][Ring1][Branch1][=C][Ring1][N][N][C][=C][C][=C][NH1][C][=C][C][Ring1][Branch1][=C][Ring1][=Branch2]
c16ccc2[nH]ccc2c1.c18cccc9c1.n17cccn1.O=C34.N35.C58.C79.N46
CSc1ccc(NC(=O)C2CCCN(S(C)(=O)=O)C2)cc1
259084
[C][S][C][=C][C][=C][Branch2][Ring1][Branch2][N][C][=Branch1][C][=O][C][C][C][C][N][Branch1][=Branch2][S][Branch1][C][C][=Branch1][C][=O][=O][C][Ring1][#Branch2][C][=C][Ring2][Ring1][Ring1]
c17ccc5cc1.C16CCCN4C1.S4(C)(=O)=O.C36=O.CS7.N35
Cc1cc(Nc2cncnc2)n(-c2cccc(Cl)c2)n1
1723529
[C][C][C][=C][Branch1][#Branch2][N][C][=C][N][=C][N][=C][Ring1][=Branch1][N][Branch1][N][C][=C][C][=C][C][Branch1][C][Cl][=C][Ring1][#Branch1][N][=Ring2][Ring1][Ring1]
Cc1cc3n5n1.c15cccc(Cl)c1.c14cncnc1.N34
O=c1c2cc3c(cc2nnn1Cc1ccc(Cl)cc1)OCCO3
433724
[O][=C][C][=C][C][=C][Branch2][Ring1][=Branch1][C][=C][Ring1][=Branch1][N][=N][N][Ring1][#Branch2][C][C][=C][C][=C][Branch1][C][Cl][C][=C][Ring1][#Branch1][O][C][C][O][Ring2][Ring1][Ring1]
O=c1c2cc3c(cc2nnn14)OCCO3.c15ccc(Cl)cc1.C45
Cc1c(C)c(C)c(C(=O)OCc2nnc(C3CC3)o2)c(C)c1C
852992
[C][C][=C][Branch1][C][C][C][Branch1][C][C][=C][Branch2][Ring1][Branch1][C][=Branch1][C][=O][O][C][C][=N][N][=C][Branch1][=Branch1][C][C][C][Ring1][Ring1][O][Ring1][Branch2][C][Branch1][C][C][=C][Ring2][Ring1][Branch1][C]
Cc1c(C)c(C)c6c(C)c1C.c17nnc8o1.C46=O.C18CC1.O45.C57
Cc1ccc(C)c(C(C#N)CCC(=O)N2CCCC2)c1
1124700
[C][C][=C][C][=C][Branch1][C][C][C][Branch2][Ring1][Ring1][C][Branch1][Ring1][C][#N][C][C][C][=Branch1][C][=O][N][C][C][C][C][Ring1][Branch1][=C][Ring2][Ring1][Ring1]
Cc1ccc(C)c4c1.C4(C#N)CCC3=O.N13CCCC1
CCCOC(=O)c1ccc(NCC(=O)NC)cc1
211037
[C][C][C][O][C][=Branch1][C][=O][C][=C][C][=C][Branch1][=Branch2][N][C][C][=Branch1][C][=O][N][C][C][=C][Ring1][N]
c17ccc6cc1.C5C3=O.CCC4.C27=O.O24.N56.N3C
Cc1ccc(-c2noc(-c3cccc(OC(C)C)c3)n2)nn1
1412148
[C][C][=C][C][=C][Branch2][Ring1][#Branch2][C][=N][O][C][Branch1][P][C][=C][C][=C][C][Branch1][#Branch1][O][C][Branch1][C][C][C][=C][Ring1][#Branch2][=N][Ring1][#C][N][=N][Ring2][Ring1][Branch1]
Cc1ccc6nn1.c17cccc5c1.c16noc7n1.C4(C)C.O45
Cn1nc(C(F)(F)F)c(Cl)c1C(=O)NC(C)(C)C
62616
[C][N][N][=C][Branch1][=Branch2][C][Branch1][C][F][Branch1][C][F][F][C][Branch1][C][Cl][=C][Ring1][#Branch2][C][=Branch1][C][=O][N][C][Branch1][C][C][Branch1][C][C][C]
Cn1nc5c(Cl)c14.C5(F)(F)F.C3(C)(C)C.C24=O.N23
CCn1c(=O)[nH]c(=O)c2cc(C(=O)N3CCc4ccccc43)cnc21
1611425
[C][C][N][C][=Branch1][C][=O][NH1][C][=Branch1][C][=O][C][=C][C][Branch2][Ring1][C][C][=Branch1][C][=O][N][C][C][C][=C][C][=C][C][=C][Ring1][=Branch1][Ring1][=Branch2][=C][N][=C][Ring1][P][Ring2][Ring1][#Branch1]
n17c(=O)[nH]c(=O)c2cc6cnc21.N15CCc2ccccc21.C56=O.CC7
COc1cccc(C2CCCN2C(=O)COc2ccccc2)c1
751739
[C][O][C][=C][C][=C][C][Branch2][Ring1][=Branch1][C][C][C][C][N][Ring1][Branch1][C][=Branch1][C][=O][C][O][C][=C][C][=C][C][=C][Ring1][=Branch1][=C][Ring2][Ring1][Branch1]
c15cccc7c1.C17CCCN13.c16ccccc1.C3(=O)C4.CO5.O46
COC(=O)C(O)c1c(OC)cc(C)c(Cl)c1C
1114417
[C][O][C][=Branch1][C][=O][C][Branch1][C][O][C][=C][Branch1][Ring1][O][C][C][=C][Branch1][C][C][C][Branch1][C][Cl][=C][Ring1][#Branch2][C]
c14c3cc(C)c(Cl)c1C.C2(=O)C4O.CO2.O3C
CCCCNC(=O)CS(=O)(=O)c1ccc(C(F)(F)F)cn1
635544
[C][C][C][C][N][C][=Branch1][C][=O][C][S][=Branch1][C][=O][=Branch1][C][=O][C][=C][C][=C][Branch1][=Branch2][C][Branch1][C][F][Branch1][C][F][F][C][=N][Ring1][#Branch2]
C2(=O)CS(=O)(=O)c1ccc4cn1.CCCC3.C4(F)(F)F.N23
Cc1n[nH]c(=O)nc1Nc1cccc(C(F)(F)F)c1
1585407
[C][C][=N][NH1][C][=Branch1][C][=O][N][=C][Ring1][#Branch1][N][C][=C][C][=C][C][Branch1][=Branch2][C][Branch1][C][F][Branch1][C][F][F][=C][Ring1][#Branch2]
Cc1n[nH]c(=O)nc12.c13cccc4c1.C4(F)(F)F.N23
Cc1ccc(NCCNC(=O)c2cc3ccccc3oc2=O)nn1
508065
[C][C][=C][C][=C][Branch2][Ring1][Branch2][N][C][C][N][C][=Branch1][C][=O][C][=C][C][=C][C][=C][C][=C][Ring1][=Branch1][O][C][Ring1][#Branch2][=O][N][=N][Ring2][Ring1][#Branch1]
c18cc2ccccc2oc1=O.Cc1ccc7nn1.C5C6.C48=O.N57.N46
O=C(NCc1ccc(-n2cccn2)cc1)NCc1cccs1
444294
[O][=C][Branch2][Ring1][Ring2][N][C][C][=C][C][=C][Branch1][Branch2][N][C][=C][C][=N][Ring1][Branch1][C][=C][Ring1][O][N][C][C][=C][C][=C][S][Ring1][Branch1]
c18ccc9cc1.n19cccn1.c17cccs1.O=C34.N35.C58.N46.C67
O=C(Nc1nc(-c2ccco2)cs1)c1ccc(-n2cccn2)nn1
961272
[O][=C][Branch2][Ring1][C][N][C][=N][C][Branch1][Branch2][C][=C][C][=C][O][Ring1][Branch1][=C][S][Ring1][#Branch2][C][=C][C][=C][Branch1][Branch2][N][C][=C][C][=N][Ring1][Branch1][N][=N][Ring1][O]
c15ccc6nn1.c14nc7cs1.c17ccco1.n16cccn1.O=C35.N34
Cc1cc(=O)[nH]c(SCc2cc(=O)c3ccccc3[nH]2)n1
341595
[C][C][=C][C][=Branch1][C][=O][NH1][C][Branch2][Ring1][Ring2][S][C][C][=C][C][=Branch1][C][=O][C][=C][C][=C][C][=C][Ring1][=Branch1][NH1][Ring1][O][=N][Ring2][Ring1][Ring2]
c15cc(=O)c2ccccc2[nH]1.Cc1cc(=O)[nH]c6n1.S46.C45
CCN(CC(=O)c1ccc(O)cc1)CC(F)(F)F
576456
[C][C][N][Branch1][P][C][C][=Branch1][C][=O][C][=C][C][=C][Branch1][C][O][C][=C][Ring1][#Branch1][C][C][Branch1][C][F][Branch1][C][F][F]
c15ccc(O)cc1.C4C(F)(F)F.C3C5=O.N234.CC2
Cc1c(C(=O)NC2(C)CCOCC2)cnn1-c1ccncc1
1319305
[C][C][=C][Branch1][P][C][=Branch1][C][=O][N][C][Branch1][C][C][C][C][O][C][C][Ring1][#Branch1][C][=N][N][Ring1][#C][C][=C][C][=N][C][=C][Ring1][=Branch1]
Cc1c5cnn16.C14(C)CCOCC1.c16ccncc1.C35=O.N34
Cc1cccc(NC(=O)CCSc2nnc(C(C)(C)C)n2N)c1
1622018
[C][C][=C][C][=C][C][Branch2][Ring1][O][N][C][=Branch1][C][=O][C][C][S][C][=N][N][=C][Branch1][=Branch2][C][Branch1][C][C][Branch1][C][C][C][N][Ring1][=Branch2][N][=C][Ring2][Ring1][=Branch1]
Cc1cccc5c1.c17nnc6n1N.C3(=O)CC4.C6(C)(C)C.N35.S47
Cc1ccccc1-n1nc(C(=O)NCCCN2CCOCC2)nc1C
456077
[C][C][=C][C][=C][C][=C][Ring1][=Branch1][N][N][=C][Branch1][P][C][=Branch1][C][=O][N][C][C][C][N][C][C][O][C][C][Ring1][=Branch1][N][=C][Ring1][P][C]
Cc1ccccc17.n17nc6nc1C.N15CCOCC1.C4CC5.C36=O.N34
COCCNc1c(-c2ccc(O)cc2)nc2cccc(C)n12
99436
[C][O][C][C][N][C][=C][Branch1][N][C][=C][C][=C][Branch1][C][O][C][=C][Ring1][#Branch1][N][=C][C][=C][C][=C][Branch1][C][C][N][Ring1][P][Ring1][#Branch1]
c15c6nc2cccc(C)n12.c16ccc(O)cc1.C3C4.CO3.N45
CC(C)OCCC(=O)Nc1cc(Cl)ccc1O
1685333
[C][C][Branch1][C][C][O][C][C][C][=Branch1][C][=O][N][C][=C][C][Branch1][C][Cl][=C][C][=C][Ring1][#Branch1][O]
c15cc(Cl)ccc1O.C4CC2=O.CC3C.O34.N25
O=C(NC1CCN(c2ccc(C(F)(F)F)cn2)CC1)c1ccoc1
533911
[O][=C][Branch2][Ring1][#C][N][C][C][C][N][Branch2][Ring1][Ring1][C][=C][C][=C][Branch1][=Branch2][C][Branch1][C][F][Branch1][C][F][F][C][=N][Ring1][#Branch2][C][C][Ring1][S][C][C][=C][O][C][=Ring1][Branch1]
C15CCN4CC1.c14ccc7cn1.c16ccoc1.C7(F)(F)F.O=C36.N35
O=C(CSc1nc2ncccc2[nH]1)Nc1ccccc1F
1772119
[O][=C][Branch1][S][C][S][C][=N][C][=N][C][=C][C][=C][Ring1][=Branch1][NH1][Ring1][=Branch2][N][C][=C][C][=C][C][=C][Ring1][=Branch1][F]
c16nc2ncccc2[nH]1.c15ccccc1F.O=C3C4.S46.N35
CCCOc1ccccc1Cn1c(=O)oc(=O)c2ccccc21
125735
[C][C][C][O][C][=C][C][=C][C][=C][Ring1][=Branch1][C][N][C][=Branch1][C][=O][O][C][=Branch1][C][=O][C][=C][C][=C][C][=C][Ring1][=Branch1][Ring1][N]
n15c(=O)oc(=O)c2ccccc21.c14ccccc16.CCC3.O34.C56
NC(=O)C1CCN(S(=O)(=O)c2cncc(Cl)c2)CC1
1464255
[N][C][=Branch1][C][=O][C][C][C][N][Branch2][Ring1][Ring1][S][=Branch1][C][=O][=Branch1][C][=O][C][=C][N][=C][C][Branch1][C][Cl][=C][Ring1][#Branch1][C][C][Ring1][S]
S3(=O)(=O)c1cncc(Cl)c1.C14CCN3CC1.NC4=O
Cc1nc(NCc2ccco2)sc1C(=O)NCc1ccncc1
598746
[C][C][N][=C][Branch1][#Branch2][N][C][C][=C][C][=C][O][Ring1][Branch1][S][C][=Ring1][N][C][=Branch1][C][=O][N][C][C][=C][C][=N][C][=C][Ring1][=Branch1]
Cc1nc6sc17.c19ccncc1.c18ccco1.C37=O.N46.C48.N35.C59
Cc1nc(C(C)(C)NCc2cccc(F)c2F)sc1C
1133006
[C][C][N][=C][Branch2][Ring1][=Branch1][C][Branch1][C][C][Branch1][C][C][N][C][C][=C][C][=C][C][Branch1][C][F][=C][Ring1][#Branch1][F][S][C][=Ring2][Ring1][C][C]
c16cccc(F)c1F.Cc1nc5sc1C.C35(C)C.N34.C46
O=C1OCCN1CCSc1nc2ccccc2[nH]1
405082
[O][=C][O][C][C][N][Ring1][Branch1][C][C][S][C][=N][C][=C][C][=C][C][=C][Ring1][=Branch1][NH1][Ring1][=Branch2]
c15nc2ccccc2[nH]1.O=C1OCCN14.C4C3.S35
Cc1ccsc1CNC(=O)Cn1c(=O)sc2ccccc21
1214301
[C][C][C][=C][S][C][=Ring1][Branch1][C][N][C][=Branch1][C][=O][C][N][C][=Branch1][C][=O][S][C][=C][C][=C][C][=C][Ring1][=Branch1][Ring1][#Branch2]
n15c(=O)sc2ccccc21.Cc1ccsc16.C3(=O)C5.C46.N34
C=CCn1c(C)cc(C(=O)CSc2nnc(-c3ccco3)o2)c1C
57958
[C][=C][C][N][C][Branch1][C][C][=C][C][Branch2][Ring1][#Branch1][C][=Branch1][C][=O][C][S][C][=N][N][=C][Branch1][Branch2][C][=C][C][=C][O][Ring1][Branch1][O][Ring1][#Branch2][=C][Ring2][Ring1][Ring2][C]
n16c(C)cc5c1C.c17nnc8o1.c18ccco1.C5(=O)C4.C=CC6.S47
Cc1nn(C)c(C)c1Cc1ccc(NC(=O)C(C)C)cc1
36679
[C][C][=N][N][Branch1][C][C][C][Branch1][C][C][=C][Ring1][#Branch1][C][C][=C][C][=C][Branch1][O][N][C][=Branch1][C][=O][C][Branch1][C][C][C][C][=C][Ring1][N]
Cc1nn(C)c(C)c14.c15ccc3cc1.C2(=O)C(C)C.C45.N23
Cc1ncc(CNC(=O)Cn2nc(C)c3ccccc3c2=O)s1
1571669
[C][C][=N][C][=C][Branch2][Ring1][#Branch2][C][N][C][=Branch1][C][=O][C][N][N][=C][Branch1][C][C][C][=C][C][=C][C][=C][Ring1][=Branch1][C][Ring1][O][=O][S][Ring2][Ring1][=Branch1]
n16nc(C)c2ccccc2c1=O.Cc1ncc7s1.C4(=O)C6.C57.N45
CC(NC(=O)Cc1ccc2c(c1)CCO2)c1nc2c(s1)CCCC2
1690262
[C][C][Branch2][Ring1][=Branch1][N][C][=Branch1][C][=O][C][C][=C][C][=C][C][=Branch1][Ring2][=C][Ring1][=Branch1][C][C][O][Ring1][=Branch1][C][=N][C][=C][Branch1][Ring2][S][Ring1][Branch1][C][C][C][C][Ring1][#Branch1]
c16ccc2c(c1)CCO2.c15nc2c(s1)CCCC2.C3(=O)C6.CC45.N34
CC(=O)Oc1ccc(C(=O)Nc2nc(C)cc(C)n2)cc1
60508
[C][C][=Branch1][C][=O][O][C][=C][C][=C][Branch2][Ring1][Ring2][C][=Branch1][C][=O][N][C][=N][C][Branch1][C][C][=C][C][Branch1][C][C][=N][Ring1][Branch2][C][=C][Ring1][P]
c16nc(C)cc(C)n1.c15ccc7cc1.CC3=O.C47=O.O35.N46
CCC(=O)Nc1ccc(SCc2cccnc2)cc1
1801511
[C][C][C][=Branch1][C][=O][N][C][=C][C][=C][Branch1][O][S][C][C][=C][C][=C][N][=C][Ring1][=Branch1][C][=C][Ring1][=C]
c15ccc7cc1.c16cccnc1.CCC3=O.N35.S47.C46
CC(C)Cn1ccc2cc(NC(=O)NC(C)(CO)CO)ccc21
1482057
[C][C][Branch1][C][C][C][N][C][=C][C][=C][C][Branch1][P][N][C][=Branch1][C][=O][N][C][Branch1][C][C][Branch1][Ring1][C][O][C][O][=C][C][=C][Ring1][S][Ring2][Ring1][Ring1]
n17ccc2cc6ccc21.C5(C)(CO)CO.CC(C)C7.C34=O.N36.N45
CCOc1cc(-c2ncc(CO)s2)ccc1OC
838105
[C][C][O][C][=C][C][Branch1][N][C][=N][C][=C][Branch1][Ring1][C][O][S][Ring1][#Branch1][=C][C][=C][Ring1][=N][O][C]
c14cc7ccc15.c17ncc6s1.CC3.O34.C6O.O5C
Cc1nn(C)c(C)c1CC(=O)Nc1ccc[nH]c1=O
1697581
[C][C][=N][N][Branch1][C][C][C][Branch1][C][C][=C][Ring1][#Branch1][C][C][=Branch1][C][=O][N][C][=C][C][=C][NH1][C][Ring1][=Branch1][=O]
Cc1nn(C)c(C)c14.c13ccc[nH]c1=O.C4C2=O.N23
Cc1cccc(N(CCC(N)=O)CC(=O)N(C)c2ccccc2)c1
1125790
[C][C][=C][C][=C][C][Branch2][Ring1][N][N][Branch1][Branch2][C][C][C][Branch1][C][N][=O][C][C][=Branch1][C][=O][N][Branch1][C][C][C][=C][C][=C][C][=C][Ring1][=Branch1][=C][Ring2][Ring1][#Branch1]
Cc1cccc6c1.c17ccccc1.C4CC(N)=O.C5C3=O.N456.N37C
C=C(C)CN(CC)C(=O)c1cccnc1OCC(F)F
1347081
[C][=C][Branch1][C][C][C][N][Branch1][Ring1][C][C][C][=Branch1][C][=O][C][=C][C][=C][N][=C][Ring1][=Branch1][O][C][C][Branch1][C][F][F]
c17cccnc14.C=C(C)C5.C3C(F)F.N256.C27=O.C6C.O34
CCNC(=O)c1ccc(CNC(=O)NC2CCCCCC2)cc1
634910
[C][C][N][C][=Branch1][C][=O][C][=C][C][=C][Branch1][P][C][N][C][=Branch1][C][=O][N][C][C][C][C][C][C][C][Ring1][#Branch1][C][=C][Ring2][Ring1][C]
c19ccc%10cc1.C18CCCCCC1.C39=O.C45=O.CC6.N36.C7%10.N47.N58
Cc1cccc(C(O)c2cc(F)c3c(c2)CCC(=O)N3)c1
799997
[C][C][=C][C][=C][C][Branch2][Ring1][O][C][Branch1][C][O][C][=C][C][Branch1][C][F][=C][C][=Branch1][Ring2][=C][Ring1][#Branch1][C][C][C][=Branch1][C][=O][N][Ring1][Branch2][=C][Ring2][Ring1][Ring2]
c15cc(F)c2c(c1)CCC(=O)N2.Cc1cccc4c1.C45O
CCC(CC)NC(=O)NCc1ccc(OC)c(O)c1
1648772
[C][C][C][Branch1][Ring1][C][C][N][C][=Branch1][C][=O][N][C][C][=C][C][=C][Branch1][Ring1][O][C][C][Branch1][C][O][=C][Ring1][=Branch2]
c17ccc4c(O)c1.CCC5CC.C23=O.N25.N36.C67.O4C
CCc1ocnc1C(=O)Nc1nc(-c2ccc3c(c2)COC3)cs1
1900303
[C][C][C][O][C][=N][C][=Ring1][Branch1][C][=Branch1][C][=O][N][C][=N][C][Branch1][S][C][=C][C][=C][C][=Branch1][Ring2][=C][Ring1][=Branch1][C][O][C][Ring1][=Branch1][=C][S][Ring1][=C]
c18ccc2c(c1)COC2.c17ocnc16.c15nc8cs1.C46=O.CC7.N45
CCOC(=O)C(N)Cc1cc(C)c(Cl)cc1O
1110226
[C][C][O][C][=Branch1][C][=O][C][Branch1][C][N][C][C][=C][C][Branch1][C][C][=C][Branch1][C][Cl][C][=C][Ring1][Branch2][O]
c14cc(C)c(Cl)cc1O.C2(=O)C(N)C4.CC3.O23
CC(=O)Nc1ccc(S(=O)(=O)N(C)Cc2ccc(C)o2)cc1
76596
[C][C][=Branch1][C][=O][N][C][=C][C][=C][Branch2][Ring1][#Branch1][S][=Branch1][C][=O][=Branch1][C][=O][N][Branch1][C][C][C][C][=C][C][=C][Branch1][C][C][O][Ring1][=Branch1][C][=C][Ring2][Ring1][C]
c16ccc(S5(=O)=O)cc1.c17ccc(C)o1.CC3=O.N45C.N36.C47
FC(F)(F)c1cccc(-n2nc(C3CC3)nc2CC2CCOC2)c1
1506248
[F][C][Branch1][C][F][Branch1][C][F][C][=C][C][=C][C][Branch2][Ring1][#Branch1][N][N][=C][Branch1][=Branch1][C][C][C][Ring1][Ring1][N][=C][Ring1][Branch2][C][C][C][C][O][C][Ring1][Branch1][=C][Ring2][Ring1][Ring2]
c16cccc7c1.n17nc8nc14.C15CCOC1.FC6(F)F.C18CC1.C45
Cc1noc(-c2ccc(C(=O)Nc3ncc(C(N)=O)s3)cc2)n1
1544356
[C][C][=N][O][C][Branch2][Ring1][#C][C][=C][C][=C][Branch2][Ring1][Ring2][C][=Branch1][C][=O][N][C][=N][C][=C][Branch1][=Branch1][C][Branch1][C][N][=O][S][Ring1][Branch2][C][=C][Ring1][P][=N][Ring2][Ring1][=Branch1]
c18ccc7cc1.Cc1noc8n1.c15ncc6s1.C47=O.C6(N)=O.N45
Cc1cccc(-c2noc(C(=O)NCc3ccco3)c2N)c1
1133631
[C][C][=C][C][=C][C][Branch2][Ring1][Branch2][C][=N][O][C][Branch1][=C][C][=Branch1][C][=O][N][C][C][=C][C][=C][O][Ring1][Branch1][=C][Ring1][=C][N][=C][Ring2][Ring1][Branch1]
Cc1cccc8c1.c18noc6c1N.c17ccco1.C46=O.N45.C57
CCCOc1c(C(=O)OC)sc2ccc(NC(=O)NC)cc12
865717
[C][C][C][O][C][=C][Branch1][#Branch1][C][=Branch1][C][=O][O][C][S][C][=C][C][=C][Branch1][Branch2][N][C][=Branch1][C][=O][N][C][C][=C][Ring2][Ring1][C][Ring1][O]
c17c9sc2ccc8cc12.CCC6.C39=O.C45=O.O67.O3C.N48.N5C
NC(=O)c1cccc(OC(=O)C2CC2c2ccccc2Cl)c1
1709382
[N][C][=Branch1][C][=O][C][=C][C][=C][C][Branch2][Ring1][Ring2][O][C][=Branch1][C][=O][C][C][C][Ring1][Ring1][C][=C][C][=C][C][=C][Ring1][=Branch1][Cl][=C][Ring2][Ring1][Ring1]
c16cccc4c1.c17ccccc1Cl.C15CC17.NC6=O.C35=O.O34
CNc1ccc(N(C)S(=O)(=O)N(C)C)cc1Cl
1118364
[C][N][C][=C][C][=C][Branch1][P][N][Branch1][C][C][S][=Branch1][C][=O][=Branch1][C][=O][N][Branch1][C][C][C][C][=C][Ring1][=C][Cl]
c12ccc3cc1Cl.N3(C)S(=O)(=O)N(C)C.CN2
CCCCN(C)C(=O)Nc1cccc(OCC(=O)N(C)C)c1
1706191
[C][C][C][C][N][Branch1][C][C][C][=Branch1][C][=O][N][C][=C][C][=C][C][Branch1][N][O][C][C][=Branch1][C][=O][N][Branch1][C][C][C][=C][Ring1][=N]
c18cccc6c1.CCCC7.C5C4=O.N27C.C23=O.N4(C)C.N38.O56
N#Cc1ccc(COC(=O)Cc2ccc(F)cc2)cc1
119395
[N][#C][C][=C][C][=C][Branch2][Ring1][Ring1][C][O][C][=Branch1][C][=O][C][C][=C][C][=C][Branch1][C][F][C][=C][Ring1][#Branch1][C][=C][Ring2][Ring1][C]
N#Cc1ccc5cc1.c16ccc(F)cc1.C3(=O)C6.C45.O34
CCOC(C)C(=O)N(C)CC(=O)Nc1cccc(Cl)c1
1001494
[C][C][O][C][Branch1][C][C][C][=Branch1][C][=O][N][Branch1][C][C][C][C][=Branch1][C][=O][N][C][=C][C][=C][C][Branch1][C][Cl][=C][Ring1][#Branch1]
c17cccc(Cl)c1.C5(C)C2=O.C6C3=O.N26C.CC4.O45.N37
COC(=O)C=C(C)c1cncc(-c2ccccc2OC)c1
1252042
[C][O][C][=Branch1][C][=O][C][=C][Branch1][C][C][C][=C][N][=C][C][Branch1][O][C][=C][C][=C][C][=C][Ring1][=Branch1][O][C][=C][Ring1][=C]
C=5(C)c1cncc6c1.c16ccccc14.C3(=O)C=5.CO3.O4C
CC(C)(NC(=O)c1ccc(-n2ccnn2)cc1)c1nccs1
1354433
[C][C][Branch1][C][C][Branch2][Ring1][#Branch1][N][C][=Branch1][C][=O][C][=C][C][=C][Branch1][Branch2][N][C][=C][N][=N][Ring1][Branch1][C][=C][Ring1][O][C][=N][C][=C][S][Ring1][Branch1]
c15ccc7cc1.n17ccnn1.c16nccs1.CC46C.C35=O.N34
COCCN(CC(C)C)c1ccc(F)cc1C(C)O
568716
[C][O][C][C][N][Branch1][#Branch1][C][C][Branch1][C][C][C][C][=C][C][=C][Branch1][C][F][C][=C][Ring1][#Branch1][C][Branch1][C][C][O]
c15ccc(F)cc16.C4C(C)C.C2C3.N345.C6(C)O.CO2
C=CCNC(=O)CSc1ncc(-c2ccccc2)o1
803489
[C][=C][C][N][C][=Branch1][C][=O][C][S][C][=N][C][=C][Branch1][=Branch2][C][=C][C][=C][C][=C][Ring1][=Branch1][O][Ring1][O]
c16ncc7o1.c17ccccc1.C3(=O)C5.C=CC4.N34.S56
CCC(C)Sc1ccc(NCc2nnc(C3CCC3)o2)c(C)c1
1902596
[C][C][C][Branch1][C][C][S][C][=C][C][=C][Branch2][Ring1][C][N][C][C][=N][N][=C][Branch1][#Branch1][C][C][C][C][Ring1][Ring2][O][Ring1][=Branch2][C][Branch1][C][C][=C][Ring2][Ring1][C]
c18ccc6c(C)c1.c17nnc9o1.CCC5C.C19CCC1.S58.N46.C47
CCn1nnnc1SCC(=O)Nc1cccc(Cl)c1
27606
[C][C][N][N][=N][N][=C][Ring1][Branch1][S][C][C][=Branch1][C][=O][N][C][=C][C][=C][C][Branch1][C][Cl][=C][Ring1][#Branch1]
c14cccc(Cl)c1.n15nnnc16.C3C2=O.CC5.S36.N24
CCC(C)NC(=O)CCC(O)c1cc(F)ccc1OC
709018
[C][C][C][Branch1][C][C][N][C][=Branch1][C][=O][C][C][C][Branch1][C][O][C][=C][C][Branch1][C][F][=C][C][=C][Ring1][#Branch1][O][C]
c15cc(F)ccc13.C2(=O)CCC5O.CCC4C.N24.O3C
CS(=O)(=O)N1CC(C(=O)Nc2ccc(Cl)cc2)C1
1866338
[C][S][=Branch1][C][=O][=Branch1][C][=O][N][C][C][Branch1][P][C][=Branch1][C][=O][N][C][=C][C][=C][Branch1][C][Cl][C][=C][Ring1][#Branch1][C][Ring1][=C]
c15ccc(Cl)cc1.N14CC6C1.CS4(=O)=O.C36=O.N35
Cc1cnc2n(c1=O)CC(C(=O)NCc1ccco1)CS2
1398762
[C][C][=C][N][=C][N][Branch1][Branch1][C][Ring1][=Branch1][=O][C][C][Branch1][=C][C][=Branch1][C][=O][N][C][C][=C][C][=C][O][Ring1][Branch1][C][S][Ring1][P]
Cc1cnc2n(c1=O)CC5CS2.c16ccco1.C35=O.N34.C46
CS(=O)(=O)Nc1cccc(Br)c1
19363
[C][S][=Branch1][C][=O][=Branch1][C][=O][N][C][=C][C][=C][C][Branch1][C][Br][=C][Ring1][#Branch1]
c13cccc(Br)c1.CS2(=O)=O.N23
NC(=O)c1c(NC(=O)COC(=O)c2ccco2)sc2c1CCC2
122251
[N][C][=Branch1][C][=O][C][=C][Branch2][Ring1][Ring1][N][C][=Branch1][C][=O][C][O][C][=Branch1][C][=O][C][=C][C][=C][O][Ring1][Branch1][S][C][=C][Ring1][P][C][C][C][Ring1][Branch1]
c18c6sc2c1CCC2.c17ccco1.C4(=O)C5.NC8=O.C37=O.N46.O35
CCC(C)C(=O)N1CCCC(C(=O)N2CCCC2(C)C)C1
1152836
[C][C][C][Branch1][C][C][C][=Branch1][C][=O][N][C][C][C][C][Branch1][S][C][=Branch1][C][=O][N][C][C][C][C][Ring1][Branch1][Branch1][C][C][C][C][Ring1][#C]
N13CCCC5C1.N14CCCC1(C)C.CCC(C)C3=O.C45=O
CS(=O)(=O)NC1CCN(C(=O)c2cccc3cn[nH]c23)CC1
1825813
[C][S][=Branch1][C][=O][=Branch1][C][=O][N][C][C][C][N][Branch2][Ring1][C][C][=Branch1][C][=O][C][=C][C][=C][C][C][=N][NH1][C][Ring1][=Branch2][=Ring1][Branch1][C][C][Ring1][P]
c17cccc2cn[nH]c12.C16CCN4CC1.CS5(=O)=O.C47=O.N56
CC(C)C(CC#N)OC(=O)C1CC(=O)N(c2ccc3c(c2)OCO3)C1
1022827
[C][C][Branch1][C][C][C][Branch1][Ring2][C][C][#N][O][C][=Branch1][C][=O][C][C][C][=Branch1][C][=O][N][Branch1][S][C][=C][C][=C][C][=Branch1][Ring2][=C][Ring1][=Branch1][O][C][O][Ring1][=Branch1][C][Ring1][#C]
c17ccc2c(c1)OCO2.CC(C)C5CC#N.C16CC(=O)N7C1.C46=O.O45
Cc1noc(C)c1CCC(=O)N1CCCCCC1c1cccn1C
1826931
[C][C][=N][O][C][Branch1][C][C][=C][Ring1][=Branch1][C][C][C][=Branch1][C][=O][N][C][C][C][C][C][C][Ring1][#Branch1][C][=C][C][=C][N][Ring1][Branch1][C]
N12CCCCCC14.Cc1noc(C)c13.c14cccn1C.C3CC2=O
CCNC(=O)c1cc(=O)c2cc(CC)cc(N)c2o1
1132591
[C][C][N][C][=Branch1][C][=O][C][=C][C][=Branch1][C][=O][C][=C][C][Branch1][Ring1][C][C][=C][C][Branch1][C][N][=C][Ring1][=Branch2][O][Ring1][=C]
c15cc(=O)c2cc6cc(N)c2o1.C35=O.CC4.N34.C6C
Cn1cc(-c2ccnc(NCc3ccc4c(c3)OCCCO4)n2)cn1
365876
[C][N][C][=C][Branch2][Ring1][S][C][=C][C][=N][C][Branch2][Ring1][Ring2][N][C][C][=C][C][=C][C][=Branch1][Ring2][=C][Ring1][=Branch1][O][C][C][C][O][Ring1][Branch2][=N][Ring2][Ring1][Ring1][C][=N][Ring2][Ring1][Branch2]
c17ccc2c(c1)OCCCO2.c18ccnc6n1.Cn1cc8cn1.N56.C57
CCOC(=O)Cc1ccc(-c2nn3cnnc3s2)cc1Cl
1645513
[C][C][O][C][=Branch1][C][=O][C][C][=C][C][=C][Branch1][=N][C][=N][N][C][=N][N][=C][Ring1][Branch1][S][Ring1][Branch2][C][=C][Ring1][=C][Cl]
c16ccc7cc1Cl.c17nn2cnnc2s1.C4(=O)C6.CC5.O45
O=C(CCC1CCOCC1)N1CCc2ccc(Cl)cc2C1
1387376
[O][=C][Branch1][O][C][C][C][C][C][O][C][C][Ring1][=Branch1][N][C][C][C][=C][C][=C][Branch1][C][Cl][C][=C][Ring1][#Branch1][C][Ring1][O]
N13CCc2ccc(Cl)cc2C1.C14CCOCC1.O=C3CC4
COc1ccc(-c2nc(C)sc2Cc2nnc(N)o2)cc1OC
388685
[C][O][C][=C][C][=C][Branch2][Ring1][=Branch1][C][N][=C][Branch1][C][C][S][C][=Ring1][=Branch1][C][C][=N][N][=C][Branch1][C][N][O][Ring1][=Branch1][C][=C][Ring2][Ring1][Ring1][O][C]
c13ccc7cc14.c17nc(C)sc15.c16nnc(N)o1.CO3.C56.O4C
CCCCC(NC(=O)c1ccncc1F)c1ccc(OC)cc1
1182075
[C][C][C][C][C][Branch1][#C][N][C][=Branch1][C][=O][C][=C][C][=N][C][=C][Ring1][=Branch1][F][C][=C][C][=C][Branch1][Ring1][O][C][C][=C][Ring1][Branch2]
c15ccncc1F.c16ccc3cc1.CCCCC46.C25=O.N24.O3C
CCCn1c(SC(C)C(=O)c2ccc(CC)cc2)n[nH]c1=O
157278
[C][C][C][N][C][Branch2][Ring1][=Branch1][S][C][Branch1][C][C][C][=Branch1][C][=O][C][=C][C][=C][Branch1][Ring1][C][C][C][=C][Ring1][Branch2][=N][NH1][C][Ring2][Ring1][C][=O]
n15c7n[nH]c1=O.c14ccc6cc1.C3(C)C4=O.CCC5.S37.C6C
CN(CCC(F)(F)F)C(=O)CSc1ccc(C(F)(F)F)cn1
1571357
[C][N][Branch1][O][C][C][C][Branch1][C][F][Branch1][C][F][F][C][=Branch1][C][=O][C][S][C][=C][C][=C][Branch1][=Branch2][C][Branch1][C][F][Branch1][C][F][F][C][=N][Ring1][#Branch2]
c16ccc5cn1.C3CC(F)(F)F.C2(=O)C4.C5(F)(F)F.CN23.S46
CCCCn1ncc(NC(=O)Nc2cc(F)ccc2OC)c1C
1918999
[C][C][C][C][N][N][=C][C][Branch2][Ring1][Ring2][N][C][=Branch1][C][=O][N][C][=C][C][Branch1][C][F][=C][C][=C][Ring1][#Branch1][O][C][=C][Ring2][Ring1][C][C]
c17cc(F)ccc15.n18ncc6c1C.CCCC8.C34=O.N36.N47.O5C
Cn1nc(-c2ccc(Cl)cc2Cl)cc(CO)c1=O
1243774
[C][N][N][=C][Branch1][=N][C][=C][C][=C][Branch1][C][Cl][C][=C][Ring1][#Branch1][Cl][C][=C][Branch1][Ring1][C][O][C][Ring1][S][=O]
Cn1nc4cc3c1=O.c14ccc(Cl)cc1Cl.C3O
CCc1nnc2n1CCN(C(=O)c1cc(Cl)c[nH]1)C2
936079
[C][C][C][=N][N][=C][N][Ring1][Branch1][C][C][N][Branch1][#C][C][=Branch1][C][=O][C][=C][C][Branch1][C][Cl][=C][NH1][Ring1][=Branch1][C][Ring1][=C]
c15nnc2n1CCN3C2.c14cc(Cl)c[nH]1.C34=O.CC5
COc1ccc(NC(=O)CCc2ccccc2F)cc1OC
1617944
[C][O][C][=C][C][=C][Branch1][P][N][C][=Branch1][C][=O][C][C][C][=C][C][=C][C][=C][Ring1][=Branch1][F][C][=C][Ring2][Ring1][C][O][C]
c14ccc6cc15.c17ccccc1F.C3(=O)CC7.CO4.N36.O5C