SMILES
large_stringlengths
17
56
ID
large_stringlengths
1
7
SELFIES
stringlengths
63
275
SAFE
stringlengths
20
78
CC1(C)C2CCC1(CS(=O)(=O)Nc1ccccc1)C(=O)C2
47859
[C][C][Branch1][C][C][C][C][C][C][Ring1][=Branch1][Branch2][Ring1][C][C][S][=Branch1][C][=O][=Branch1][C][=O][N][C][=C][C][=C][C][=C][Ring1][=Branch1][C][=Branch1][C][=O][C][Ring2][Ring1][C]
CC1(C)C2CCC15C(=O)C2.c14ccccc1.C5S3(=O)=O.N34
Cc1cc(C)c(CNC(=O)NCc2ccco2)c(C)c1
699936
[C][C][=C][C][Branch1][C][C][=C][Branch1][S][C][N][C][=Branch1][C][=O][N][C][C][=C][C][=C][O][Ring1][Branch1][C][Branch1][C][C][=C][Ring2][Ring1][Ring1]
Cc1cc(C)c8c(C)c1.c17ccco1.C34=O.C58.N35.N46.C67
CCOC(=O)C(C#N)C(c1ccco1)c1ccccc1OC
6126
[C][C][O][C][=Branch1][C][=O][C][Branch1][Ring1][C][#N][C][Branch1][Branch2][C][=C][C][=C][O][Ring1][Branch1][C][=C][C][=C][C][=C][Ring1][=Branch1][O][C]
C2(=O)C(C#N)C56.c16ccccc14.c15ccco1.CC3.O23.O4C
O=C(CNC(=O)Cc1ccccc1)NCC(=O)NC1CC1
148066
[O][=C][Branch1][S][C][N][C][=Branch1][C][=O][C][C][=C][C][=C][C][=C][Ring1][=Branch1][N][C][C][=Branch1][C][=O][N][C][C][C][Ring1][Ring1]
c18ccccc1.O=C2C5.C3(=O)C8.C6C4=O.C17CC1.N35.N26.N47
O=C(c1ccccn1)N1CCC(c2nnc(-c3ccccc3)o2)C1
673379
[O][=C][Branch1][=Branch2][C][=C][C][=C][C][=N][Ring1][=Branch1][N][C][C][C][Branch2][Ring1][C][C][=N][N][=C][Branch1][=Branch2][C][=C][C][=C][C][=C][Ring1][=Branch1][O][Ring1][O][C][Ring1][S]
c15ccccn1.N14CCC6C1.c16nnc7o1.c17ccccc1.O=C45
CC(NC1=NS(=O)(=O)c2ccccc21)c1ccc(NC(N)=O)cc1
1229499
[C][C][Branch2][Ring1][Branch1][N][C][=N][S][=Branch1][C][=O][=Branch1][C][=O][C][=C][C][=C][C][=C][Ring1][=Branch1][Ring1][O][C][=C][C][=C][Branch1][#Branch1][N][C][Branch1][C][N][=O][C][=C][Ring1][#Branch2]
N4C1=NS(=O)(=O)c2ccccc21.c16ccc5cc1.CC46.C3(N)=O.N35
O=C(NCc1cccnc1)c1cnc2sc3ncccc3c(=O)n12
1174521
[O][=C][Branch1][O][N][C][C][=C][C][=C][N][=C][Ring1][=Branch1][C][=C][N][=C][S][C][=N][C][=C][C][=C][Ring1][=Branch1][C][=Branch1][C][=O][N][Ring1][=C][Ring1][O]
c16cnc2sc3ncccc3c(=O)n12.c17cccnc1.O=C46.N45.C57
CCC(=O)Nc1cccc(C(=O)OCCN2CCCC2=O)c1
751117
[C][C][C][=Branch1][C][=O][N][C][=C][C][=C][C][Branch1][S][C][=Branch1][C][=O][O][C][C][N][C][C][C][C][Ring1][Branch1][=O][=C][Ring1][P]
c16cccc7c1.N18CCCC1=O.CCC4=O.C37=O.C5C8.N46.O35
NC(=O)C1CCCN(C(=O)c2cc(Cl)ccc2Cl)C1
641612
[N][C][=Branch1][C][=O][C][C][C][C][N][Branch1][P][C][=Branch1][C][=O][C][=C][C][Branch1][C][Cl][=C][C][=C][Ring1][#Branch1][Cl][C][Ring1][S]
c15cc(Cl)ccc1Cl.C14CCCN3C1.NC4=O.C35=O
Cc1csc(NC(=O)c2c[nH]c3c(Cl)cccc3c2=O)n1
1613161
[C][C][=C][S][C][Branch2][Ring1][Branch2][N][C][=Branch1][C][=O][C][=C][NH1][C][=C][Branch1][C][Cl][C][=C][C][=C][Ring1][#Branch1][C][Ring1][O][=O][=N][Ring2][Ring1][Ring2]
c16c[nH]c2c(Cl)cccc2c1=O.Cc1csc5n1.C46=O.N45
CCN1CCOc2ccc(NC(=O)c3ccc(Cl)cc3)cc2C1=O
199864
[C][C][N][C][C][O][C][=C][C][=C][Branch1][P][N][C][=Branch1][C][=O][C][=C][C][=C][Branch1][C][Cl][C][=C][Ring1][#Branch1][C][=C][Ring1][S][C][Ring2][Ring1][Branch1][=O]
N17CCOc2ccc5cc2C1=O.c16ccc(Cl)cc1.C46=O.CC7.N45
Cc1oc(-c2cccs2)nc1C(=O)N1CCOC2CCCC21
738929
[C][C][O][C][Branch1][Branch2][C][=C][C][=C][S][Ring1][Branch1][=N][C][=Ring1][#Branch2][C][=Branch1][C][=O][N][C][C][O][C][C][C][C][C][Ring1][Branch1][Ring1][=Branch2]
N13CCOC2CCCC21.Cc1oc5nc14.c15cccs1.C34=O
CCn1c(SCC(=O)NC2CC2)nnc1-c1cccc(OC)c1
138306
[C][C][N][C][Branch1][=N][S][C][C][=Branch1][C][=O][N][C][C][C][Ring1][Ring1][=N][N][=C][Ring1][=N][C][=C][C][=C][C][Branch1][Ring1][O][C][=C][Ring1][Branch2]
n17c8nnc19.c19cccc4c1.C5C3=O.C16CC1.CC7.S58.N36.O4C
CC(=O)NC(C)c1nc2ccccc2n1CCOc1cccc(C)c1
521372
[C][C][=Branch1][C][=O][N][C][Branch1][C][C][C][=N][C][=C][C][=C][C][=C][Ring1][=Branch1][N][Ring1][=Branch2][C][C][O][C][=C][C][=C][C][Branch1][C][C][=C][Ring1][#Branch1]
c18nc2ccccc2n17.c15cccc(C)c1.CC3=O.C68C.C7C4.N36.O45
CN(C(=O)c1nc(-c2cn(C)cn2)n2ccccc12)c1ccccc1
1751131
[C][N][Branch2][Ring1][=C][C][=Branch1][C][=O][C][N][=C][Branch1][O][C][=C][N][Branch1][C][C][C][=N][Ring1][=Branch1][N][C][=C][C][=C][C][=Ring1][#C][Ring1][=Branch1][C][=C][C][=C][C][=C][Ring1][=Branch1]
c15nc6n2ccccc12.c16cn(C)cn1.c14ccccc1.CN34.C35=O
CCCCN(CC)C(=O)Cc1noc2c(C)cc(N)cc12
1138573
[C][C][C][C][N][Branch1][Ring1][C][C][C][=Branch1][C][=O][C][C][=N][O][C][=C][Branch1][C][C][C][=C][Branch1][C][N][C][=C][Ring1][O][Ring1][Branch2]
c16noc2c(C)cc(N)cc12.CCCC4.C3(=O)C6.N345.C5C
COc1ccc2c(C(=O)Nc3nc(C)cs3)cc(=O)oc2c1
559727
[C][O][C][=C][C][=C][C][Branch1][S][C][=Branch1][C][=O][N][C][=N][C][Branch1][C][C][=C][S][Ring1][=Branch1][=C][C][=Branch1][C][=O][O][C][Ring1][S][=C][Ring2][Ring1][Ring2]
c15ccc2c7cc(=O)oc2c1.c16nc(C)cs1.C47=O.CO5.N46
CC(C)NC(=O)NCc1ccc(OCC(N)=O)cc1
699988
[C][C][Branch1][C][C][N][C][=Branch1][C][=O][N][C][C][=C][C][=C][Branch1][Branch2][O][C][C][Branch1][C][N][=O][C][=C][Ring1][O]
c18ccc5cc1.C4C(N)=O.CC6C.C23=O.N26.N37.C78.O45
NC(=O)CCC(=O)N1CCCC(C(=O)c2ccc3ccccc3c2)C1
1610226
[N][C][=Branch1][C][=O][C][C][C][=Branch1][C][=O][N][C][C][C][C][Branch2][Ring1][Ring1][C][=Branch1][C][=O][C][=C][C][=C][C][=C][C][=C][C][Ring1][=Branch1][=C][Ring1][#Branch2][C][Ring2][Ring1][C]
c16ccc2ccccc2c1.NC(=O)CCC4=O.N14CCCC5C1.C56=O
O=C(Cn1cnc2c(oc3ccccc32)c1=O)c1ccc(F)cc1
1690483
[O][=C][Branch2][Ring1][Branch2][C][N][C][=N][C][=C][Branch1][N][O][C][=C][C][=C][C][=C][Ring1][=Branch1][Ring1][=Branch2][C][Ring1][=N][=O][C][=C][C][=C][Branch1][C][F][C][=C][Ring1][#Branch1]
n15cnc2c(oc3ccccc32)c1=O.c14ccc(F)cc1.O=C4C5
Cc1ccc2cnn(CCC(=O)NCc3ccccn3)c2c1
1820850
[C][C][=C][C][=C][C][=N][N][Branch1][P][C][C][C][=Branch1][C][=O][N][C][C][=C][C][=C][C][=N][Ring1][=Branch1][C][Ring1][P][=C][Ring2][Ring1][Branch1]
Cc1ccc2cnn6c2c1.c17ccccn1.C6CC4=O.N45.C57
N#CC1CN(Cc2c[nH]nc2-c2cccnc2)CCO1
1441395
[N][#C][C][C][N][Branch1][P][C][C][=C][NH1][N][=C][Ring1][Branch1][C][=C][C][=C][N][=C][Ring1][=Branch1][C][C][O][Ring2][Ring1][C]
N#CC1CN3CCO1.c14c[nH]nc15.c15cccnc1.C34
O=C(c1ccccc1F)N1CCC(O)(c2cccnc2F)CC1
1025003
[O][=C][Branch1][#Branch2][C][=C][C][=C][C][=C][Ring1][=Branch1][F][N][C][C][C][Branch1][C][O][Branch1][#Branch2][C][=C][C][=C][N][=C][Ring1][=Branch1][F][C][C][Ring1][=C]
N13CCC5(O)CC1.c14ccccc1F.c15cccnc1F.O=C34
N#Cc1ccc(C(=O)Nc2ccn(CCC(N)=O)n2)cc1
1207171
[N][#C][C][=C][C][=C][Branch2][Ring1][=Branch1][C][=Branch1][C][=O][N][C][C][=C][N][Branch1][Branch2][C][C][C][Branch1][C][N][=O][N][=Ring1][#Branch2][C][=C][Ring2][Ring1][Ring1]
N#Cc1ccc5cc1.c14ccn6n1.C6CC(N)=O.C35=O.N34
COc1ccc(N(Cc2ccccc2)C(=O)Cn2cnnn2)cc1
1700404
[C][O][C][=C][C][=C][Branch2][Ring1][=Branch2][N][Branch1][#Branch2][C][C][=C][C][=C][C][=C][Ring1][=Branch1][C][=Branch1][C][=O][C][N][C][=N][N][=N][Ring1][Branch1][C][=C][Ring2][Ring1][=Branch1]
c14ccc6cc1.c18ccccc1.n17cnnn1.C3(=O)C7.N356.CO4.C58
CCc1nnsc1C(=O)Nc1ccc(N2CCCC2=O)c(OC)c1
356986
[C][C][C][N][=N][S][C][=Ring1][Branch1][C][=Branch1][C][=O][N][C][=C][C][=C][Branch1][=Branch2][N][C][C][C][C][Ring1][Branch1][=O][C][Branch1][Ring1][O][C][=C][Ring1][=C]
c15ccc8c4c1.c17nnsc16.N18CCCC1=O.C36=O.CC7.N35.O4C
CCN(Cc1cccs1)C(=O)NCC1CN2CCCCC2CO1
1396280
[C][C][N][Branch1][=Branch2][C][C][=C][C][=C][S][Ring1][Branch1][C][=Branch1][C][=O][N][C][C][C][N][C][C][C][C][C][Ring1][=Branch1][C][O][Ring1][#Branch2]
C18CN2CCCCC2CO1.c19cccs1.N356.C34=O.CC5.C69.N47.C78
CCCn1cc(NC(=O)Nc2cccc(CN(C)C(C)=O)c2)cn1
1874812
[C][C][C][N][C][=C][Branch2][Ring1][O][N][C][=Branch1][C][=O][N][C][=C][C][=C][C][Branch1][O][C][N][Branch1][C][C][C][Branch1][C][C][=O][=C][Ring1][N][C][=N][Ring2][Ring1][Branch1]
c18cccc%10c1.n19cc7cn1.CCC9.C34=O.N56C.C5(C)=O.N37.N48.C6%10
COc1ccccc1OCC(=O)N(C)c1ccccc1
37088
[C][O][C][=C][C][=C][C][=C][Ring1][=Branch1][O][C][C][=Branch1][C][=O][N][Branch1][C][C][C][=C][C][=C][C][=C][Ring1][=Branch1]
c14ccccc15.c16ccccc1.C3C2=O.N26C.CO4.O35
CSc1ccc(OC(=O)c2cnn(-c3ccncc3)c2C)cc1
1379446
[C][S][C][=C][C][=C][Branch2][Ring1][Branch2][O][C][=Branch1][C][=O][C][C][=N][N][Branch1][=Branch2][C][=C][C][=N][C][=C][Ring1][=Branch1][C][=Ring1][O][C][C][=C][Ring2][Ring1][Branch1]
c18ccc5cc1.c16cnn7c1C.c17ccncc1.C46=O.CS8.O45
CCCCNC(=O)CN1C(=O)C2CCCN2c2ncc(Cl)cc21
1621450
[C][C][C][C][N][C][=Branch1][C][=O][C][N][C][=Branch1][C][=O][C][C][C][C][N][Ring1][Branch1][C][=N][C][=C][Branch1][C][Cl][C][=C][Ring1][#Branch1][Ring1][#C]
C3(=O)CN1C(=O)C2CCCN2c2ncc(Cl)cc21.CCCC4.N34
CN(C)C(=O)N1CCC(C(=O)NCC2(c3ccccc3)CC2)CC1
640495
[C][N][Branch1][C][C][C][=Branch1][C][=O][N][C][C][C][Branch2][Ring1][=Branch1][C][=Branch1][C][=O][N][C][C][Branch1][=Branch2][C][=C][C][=C][C][=C][Ring1][=Branch1][C][C][Ring1][=Branch2][C][C][Ring2][Ring1][Ring1]
N15CCC8CC1.c1%10ccccc1.C19%10CC1.CN4C.C45=O.C68=O.N67.C79
Cc1cc(C)c(NC(=O)C2CCN(C(=O)C3CC3)CC2)c(C)n1
1555703
[C][C][=C][C][Branch1][C][C][=C][Branch2][Ring1][=Branch2][N][C][=Branch1][C][=O][C][C][C][N][Branch1][#Branch2][C][=Branch1][C][=O][C][C][C][Ring1][Ring1][C][C][Ring1][O][C][Branch1][C][C][=N][Ring2][Ring1][=Branch1]
Cc1cc(C)c6c(C)n1.C17CCN5CC1.C47=O.C58=O.C18CC1.N46
N#CCCN(Cc1cccnc1)C(=O)c1ncn(-c2ccccc2)n1
1919497
[N][#C][C][C][N][Branch1][#Branch2][C][C][=C][C][=C][N][=C][Ring1][=Branch1][C][=Branch1][C][=O][C][N][=C][N][Branch1][=Branch2][C][=C][C][=C][C][=C][Ring1][=Branch1][N][=Ring1][O]
c17cccnc1.c16ncn8n1.c18ccccc1.N#CCC4.N345.C36=O.C57
CCCn1cc(-c2nc3cc(C(=O)OC)ccc3[nH]2)c(C)n1
752817
[C][C][C][N][C][=C][Branch2][Ring1][=Branch1][C][=N][C][=C][C][Branch1][#Branch1][C][=Branch1][C][=O][O][C][=C][C][=C][Ring1][#Branch2][NH1][Ring1][=N][C][Branch1][C][C][=N][Ring2][Ring1][Ring1]
c17nc2cc5ccc2[nH]1.n16cc7c(C)n1.CCC6.C45=O.O4C
O=C(CCOCC1CCCO1)Oc1ccc2cn[nH]c2c1
1287402
[O][=C][Branch1][N][C][C][O][C][C][C][C][C][O][Ring1][Branch1][O][C][=C][C][=C][C][=N][NH1][C][Ring1][Branch1][=C][Ring1][=Branch2]
c16ccc2cn[nH]c2c1.O=C3CC4.C17CCCO1.O45.C57.O36
O=C(Cn1nnc(-c2ccc(F)cc2)n1)Nc1cccc(F)c1
26994
[O][=C][Branch2][Ring1][=Branch1][C][N][N][=N][C][Branch1][N][C][=C][C][=C][Branch1][C][F][C][=C][Ring1][#Branch1][=N][Ring1][N][N][C][=C][C][=C][C][Branch1][C][F][=C][Ring1][#Branch1]
c16ccc(F)cc1.c14cccc(F)c1.n15nnc6n1.O=C3C5.N34
COCC(C)NC(=O)C1(c2cccc(Cl)c2)CC1
400133
[C][O][C][C][Branch1][C][C][N][C][=Branch1][C][=O][C][Branch1][N][C][=C][C][=C][C][Branch1][C][Cl][=C][Ring1][#Branch1][C][C][Ring1][#Branch2]
c17cccc(Cl)c1.C4C5C.C167CC1.C36=O.CO4.N35
O=C1CCCc2[nH]c(=O)c(C(=O)N3CCCCC3)cc21
255312
[O][=C][C][C][C][C][NH1][C][=Branch1][C][=O][C][Branch1][=N][C][=Branch1][C][=O][N][C][C][C][C][C][Ring1][=Branch1][=C][C][=Ring1][#C][Ring2][Ring1][Ring1]
O=C1CCCc2[nH]c(=O)c5cc21.N14CCCCC1.C45=O
COCCc1nc(N)cc(Nc2ccccc2F)n1
694028
[C][O][C][C][C][=N][C][Branch1][C][N][=C][C][Branch1][O][N][C][=C][C][=C][C][=C][Ring1][=Branch1][F][=N][Ring1][#C]
c16nc4cc(N)n1.c15ccccc1F.C3C6.CO3.N45
CCCn1ccc(C(=O)N2CCN(c3ccc(F)cc3)CC2)n1
396544
[C][C][C][N][C][=C][C][Branch2][Ring1][#Branch2][C][=Branch1][C][=O][N][C][C][N][Branch1][N][C][=C][C][=C][Branch1][C][F][C][=C][Ring1][#Branch1][C][C][Ring1][=N][=N][Ring2][Ring1][Ring2]
N14CCN5CC1.c15ccc(F)cc1.n17ccc6n1.CCC7.C46=O
O=C(CNCC(F)(F)F)NC1CCN(c2cccc(Cl)c2)C1
1217563
[O][=C][Branch1][N][C][N][C][C][Branch1][C][F][Branch1][C][F][F][N][C][C][C][N][Branch1][N][C][=C][C][=C][C][Branch1][C][Cl][=C][Ring1][#Branch1][C][Ring1][N]
c16cccc(Cl)c1.C17CCN6C1.C5C(F)(F)F.O=C3C4.N45.N37
CC(=O)N(CCc1ccccc1)CC(=O)NC(C)C
1377909
[C][C][=Branch1][C][=O][N][Branch1][O][C][C][C][=C][C][=C][C][=C][Ring1][=Branch1][C][C][=Branch1][C][=O][N][C][Branch1][C][C][C]
c17ccccc1.C5C3=O.CC2=O.N245.C4C7.C6(C)C.N36
CN(Cc1ccccc1)C(=O)CNC(=O)c1ccc2cc[nH]c2n1
1168237
[C][N][Branch1][#Branch2][C][C][=C][C][=C][C][=C][Ring1][=Branch1][C][=Branch1][C][=O][C][N][C][=Branch1][C][=O][C][=C][C][=C][C][=C][NH1][C][Ring1][Branch1][=N][Ring1][=Branch2]
c17ccc2cc[nH]c2n1.c18ccccc1.C3(=O)C6.CN35.C47=O.C58.N46
COc1ccc(C)cc1NC(=O)c1nc(-c2ccncc2)no1
144303
[C][O][C][=C][C][=C][Branch1][C][C][C][=C][Ring1][#Branch1][N][C][=Branch1][C][=O][C][=N][C][Branch1][=Branch2][C][=C][C][=N][C][=C][Ring1][=Branch1][=N][O][Ring1][O]
c14ccc(C)cc15.c16nc7no1.c17ccncc1.C36=O.CO4.N35
CN(C)c1ccc(NC(=O)CCc2ccc(F)c(F)c2)cn1
438315
[C][N][Branch1][C][C][C][=C][C][=C][Branch2][Ring1][=Branch1][N][C][=Branch1][C][=O][C][C][C][=C][C][=C][Branch1][C][F][C][Branch1][C][F][=C][Ring1][Branch2][C][=N][Ring2][Ring1][Ring1]
c16ccc(F)c(F)c1.c14ccc5cn1.C3(=O)CC6.CN4C.N35
CN(C(=O)c1[nH]c2ccc(Cl)cc2c1Cl)C1CC1
674035
[C][N][Branch2][Ring1][=Branch1][C][=Branch1][C][=O][C][NH1][C][=C][C][=C][Branch1][C][Cl][C][=C][Ring1][#Branch1][C][=Ring1][#Branch2][Cl][C][C][C][Ring1][Ring1]
c15[nH]c2ccc(Cl)cc2c1Cl.CN34.C35=O.C14CC1
O=C(Cc1ccc(F)c(F)c1)Nc1nnc(C(F)F)s1
1297084
[O][=C][Branch1][S][C][C][=C][C][=C][Branch1][C][F][C][Branch1][C][F][=C][Ring1][Branch2][N][C][=N][N][=C][Branch1][=Branch1][C][Branch1][C][F][F][S][Ring1][Branch2]
c15ccc(F)c(F)c1.c13nnc4s1.O=C2C5.C4(F)F.N23
O=C(C1CC1)N(CCn1cccn1)c1nc2c(Cl)cccc2s1
363333
[O][=C][Branch1][=Branch1][C][C][C][Ring1][Ring1][N][Branch1][#Branch2][C][C][N][C][=C][C][=N][Ring1][Branch1][C][=N][C][=C][Branch1][C][Cl][C][=C][C][=C][Ring1][#Branch1][S][Ring1][#Branch2]
c15nc2c(Cl)cccc2s1.n17cccn1.O=C36.C16CC1.N345.C4C7
Cc1cc(C)n2nc(C)c(C(=O)N(C)CCOCC3CC3)c2n1
1305804
[C][C][C][=C][Branch1][C][C][N][N][=C][Branch1][C][C][C][Branch2][Ring1][C][C][=Branch1][C][=O][N][Branch1][C][C][C][C][O][C][C][C][C][Ring1][Ring1][=C][Ring1][P][N][=Ring2][Ring1][=Branch1]
Cc1cc(C)n2nc(C)c8c2n1.C48=O.N47C.C7C5.C19CC1.O56.C69
CCS(=O)(=O)N1CCC(c2nc3c4ccccc4ncn3n2)CC1
64071
[C][C][S][=Branch1][C][=O][=Branch1][C][=O][N][C][C][C][Branch2][Ring1][Ring2][C][N][=C][C][=C][C][=C][C][=C][Ring1][=Branch1][N][=C][N][Ring1][#Branch2][N][=Ring1][=N][C][C][Ring2][Ring1][Ring1]
c16nc2c3ccccc3ncn2n1.N15CCC6CC1.CCS5(=O)=O
CCCC(C)(C)NC(=O)CNC(=O)NCc1ccco1
723206
[C][C][C][C][Branch1][C][C][Branch1][C][C][N][C][=Branch1][C][=O][C][N][C][=Branch1][C][=O][N][C][C][=C][C][=C][O][Ring1][Branch1]
CCCC5(C)C.c18ccco1.C2(=O)C6.C34=O.N25.N36.N47.C78
COc1ccc(OCc2nc(C#N)c(NCc3ccco3)o2)cc1
13365
[C][O][C][=C][C][=C][Branch2][Ring1][=Branch2][O][C][C][=N][C][Branch1][Ring1][C][#N][=C][Branch1][#Branch2][N][C][C][=C][C][=C][O][Ring1][Branch1][O][Ring1][=C][C][=C][Ring2][Ring1][=Branch1]
c19nc(C#N)c8o1.c15ccc6cc1.c1%10ccco1.CO5.O46.C49.N78.C7%10
COc1ccc(NC(=O)CC(C)C)cc1-n1cccc1
833855
[C][O][C][=C][C][=C][Branch1][N][N][C][=Branch1][C][=O][C][C][Branch1][C][C][C][C][=C][Ring1][=N][N][C][=C][C][=C][Ring1][Branch1]
c13ccc4cc15.C2(=O)CC(C)C.n15cccc1.CO3.N24
Cc1cc(C)cc(NC(=O)c2ccc3oc(=O)n(C)c3c2)c1
863509
[C][C][=C][C][Branch1][C][C][=C][C][Branch2][Ring1][=Branch2][N][C][=Branch1][C][=O][C][=C][C][=C][O][C][=Branch1][C][=O][N][Branch1][C][C][C][Ring1][#Branch1][=C][Ring1][O][=C][Ring2][Ring1][Branch1]
c16ccc2oc(=O)n(C)c2c1.Cc1cc5cc(C)c1.C46=O.N45
COc1ncccc1N(C)C(=O)c1ccc([S+]([O-])C(C)C)cc1
1214268
[C][O][C][=N][C][=C][C][=C][Ring1][=Branch1][N][Branch1][C][C][C][=Branch1][C][=O][C][=C][C][=C][Branch1][#Branch2][S+1][Branch1][C][O-1][C][Branch1][C][C][C][C][=C][Ring1][O]
c15ccc([S+]([O-])C(C)C)cc1.c13ncccc14.N24C.C25=O.CO3
CCc1noc(-c2ccc(SCC(=O)NC(C)C)nc2)n1
869662
[C][C][C][=N][O][C][Branch2][Ring1][#Branch1][C][=C][C][=C][Branch1][=N][S][C][C][=Branch1][C][=O][N][C][Branch1][C][C][C][N][=C][Ring1][=C][=N][Ring2][Ring1][Ring1]
c18ccc7nc1.c16noc8n1.C5C3=O.C4(C)C.CC6.S57.N34
COc1ccc(OC(=O)CNC(=O)C(C)(C)C)cc1
1047805
[C][O][C][=C][C][=C][Branch2][Ring1][Ring2][O][C][=Branch1][C][=O][C][N][C][=Branch1][C][=O][C][Branch1][C][C][Branch1][C][C][C][C][=C][Ring1][P]
c14ccc5cc1.C3(=O)C(C)(C)C.C2(=O)C6.CO4.O25.N36
CC1(C)CCC(CNC(=O)C2CCCN2C(=O)c2ccccn2)CC1
1323596
[C][C][Branch1][C][C][C][C][C][Branch2][Ring1][#Branch2][C][N][C][=Branch1][C][=O][C][C][C][C][N][Ring1][Branch1][C][=Branch1][C][=O][C][=C][C][=C][C][=N][Ring1][=Branch1][C][C][Ring2][Ring1][Branch2]
CC1(C)CCC8CC1.C16CCCN14.c17ccccn1.C36=O.C47=O.C58.N35
Cc1oncc1C(=O)N1CCCc2cccc(O)c21
850398
[C][C][O][N][=C][C][=Ring1][Branch1][C][=Branch1][C][=O][N][C][C][C][C][=C][C][=C][C][Branch1][C][O][=C][Ring1][#Branch1][Ring1][O]
N13CCCc2cccc(O)c21.Cc1oncc14.C34=O
Cc1cc(CN(C)Cc2coc(C(C)C)n2)ccn1
1569330
[C][C][=C][C][Branch2][Ring1][Branch1][C][N][Branch1][C][C][C][C][=C][O][C][Branch1][=Branch1][C][Branch1][C][C][C][=N][Ring1][Branch2][=C][C][=N][Ring2][Ring1][C]
Cc1cc7ccn1.c15coc6n1.N34C.C6(C)C.C37.C45
N#CCn1c(-c2ccccc2)nc2cc3c(cc21)OCO3
422436
[N][#C][C][N][C][Branch1][=Branch2][C][=C][C][=C][C][=C][Ring1][=Branch1][=N][C][=C][C][=C][Branch1][#Branch1][C][=C][Ring1][=Branch1][Ring1][#C][O][C][O][Ring1][#Branch1]
n14c5nc2cc3c(cc21)OCO3.c15ccccc1.N#CC4
COc1cc(OC)cc(C(=O)NCC(=O)N(C)CC(F)(F)F)c1
1683853
[C][O][C][=C][C][Branch1][Ring1][O][C][=C][C][Branch2][Ring1][Branch2][C][=Branch1][C][=O][N][C][C][=Branch1][C][=O][N][Branch1][C][C][C][C][Branch1][C][F][Branch1][C][F][F][=C][Ring2][Ring1][Branch1]
c14cc5cc8c1.C7C(F)(F)F.C6C3=O.C28=O.N37C.CO4.O5C.N26
COCC(C)NC(=O)CSc1nnc(-c2cccc(C)c2)n1C
204191
[C][O][C][C][Branch1][C][C][N][C][=Branch1][C][=O][C][S][C][=N][N][=C][Branch1][N][C][=C][C][=C][C][Branch1][C][C][=C][Ring1][#Branch1][N][Ring1][N][C]
c17nnc8n1C.c18cccc(C)c1.C4C5C.C3(=O)C6.CO4.N35.S67
Cc1c(C(=O)NC(C)CCN2CCOCC2)cnn1-c1ccncc1
1393690
[C][C][=C][Branch2][Ring1][Ring2][C][=Branch1][C][=O][N][C][Branch1][C][C][C][C][N][C][C][O][C][C][Ring1][=Branch1][C][=N][N][Ring2][Ring1][C][C][=C][C][=N][C][=C][Ring1][=Branch1]
Cc1c6cnn17.N15CCOCC1.c17ccncc1.C4(C)CC5.C36=O.N34
Cc1ccc2[nH]cc(NC(=O)NCc3ccco3)c(=O)c2c1
184988
[C][C][=C][C][=C][NH1][C][=C][Branch1][#C][N][C][=Branch1][C][=O][N][C][C][=C][C][=C][O][Ring1][Branch1][C][=Branch1][C][=O][C][Ring1][P][=C][Ring2][Ring1][Branch1]
Cc1ccc2[nH]cc7c(=O)c2c1.c18ccco1.C45=O.N47.N56.C68
CCC(C(=O)N1CCN(c2ccccc2OC)C(=O)C1)n1cccc1
1722128
[C][C][C][Branch2][Ring1][N][C][=Branch1][C][=O][N][C][C][N][Branch1][O][C][=C][C][=C][C][=C][Ring1][=Branch1][O][C][C][=Branch1][C][=O][C][Ring1][#C][N][C][=C][C][=C][Ring1][Branch1]
N13CCN6C(=O)C1.c16ccccc14.CCC5C3=O.n15cccc1.O4C
COc1ccc(-c2nc(C(=O)N(C)Cc3ccc(C)o3)cs2)cc1
479125
[C][O][C][=C][C][=C][Branch2][Ring1][=C][C][=N][C][Branch2][Ring1][Ring2][C][=Branch1][C][=O][N][Branch1][C][C][C][C][=C][C][=C][Branch1][C][C][O][Ring1][=Branch1][=C][S][Ring1][S][C][=C][Ring2][Ring1][=Branch1]
c15ccc9cc1.c19nc7cs1.c18ccc(C)o1.C47=O.N46C.CO5.C68
COCc1nc2nccc(-c3cccc4ccccc34)n2n1
786131
[C][O][C][C][N][=C][N][=C][C][=C][Branch1][#C][C][=C][C][=C][C][=C][C][=C][C][=C][Ring1][#Branch2][Ring1][=Branch1][N][Ring1][S][N][=Ring2][Ring1][Ring1]
c16nc2nccc7n2n1.c17cccc2ccccc12.CO5.C56
CSc1cc(C(=O)Nc2ccc(F)cc2Cl)ccn1
1537575
[C][S][C][=C][C][Branch2][Ring1][C][C][=Branch1][C][=O][N][C][=C][C][=C][Branch1][C][F][C][=C][Ring1][#Branch1][Cl][=C][C][=N][Ring1][P]
c14ccc(F)cc1Cl.c16cc5ccn1.C35=O.CS6.N34
CC1=C(C(=O)N2CCCC(CCC(=O)NC3CC3)C2)OCCO1
228538
[C][C][=C][Branch2][Ring1][O][C][=Branch1][C][=O][N][C][C][C][C][Branch1][=N][C][C][C][=Branch1][C][=O][N][C][C][C][Ring1][Ring1][C][Ring1][=C][O][C][C][O][Ring2][Ring1][=Branch1]
CC1=C(C4=O)OCCO1.N14CCCC7C1.C7CC5=O.C16CC1.N56
CCCS(=O)(=O)c1ccc2[nH]c(=O)cc(C)c2c1
1682059
[C][C][C][S][=Branch1][C][=O][=Branch1][C][=O][C][=C][C][=C][NH1][C][=Branch1][C][=O][C][=C][Branch1][C][C][C][Ring1][Branch2][=C][Ring1][N]
CCCS(=O)(=O)c1ccc2[nH]c(=O)cc(C)c2c1
CC(=O)Nc1ccc(C(=O)NC2CCCc3ccccc32)cc1
115643
[C][C][=Branch1][C][=O][N][C][=C][C][=C][Branch2][Ring1][Ring2][C][=Branch1][C][=O][N][C][C][C][C][C][=C][C][=C][C][=C][Ring1][=Branch1][Ring1][#Branch2][C][=C][Ring2][Ring1][Ring1]
N5C1CCCc2ccccc21.c16ccc7cc1.CC4=O.C57=O.N46
Cn1cnc(CNC(=O)NCCOc2ccc(Cl)cn2)n1
1409285
[C][N][C][=N][C][Branch2][Ring1][=Branch1][C][N][C][=Branch1][C][=O][N][C][C][O][C][=C][C][=C][Branch1][C][Cl][C][=N][Ring1][#Branch1][=N][Ring2][Ring1][Ring2]
c16ccc(Cl)cn1.Cn1cnc9n1.C34=O.C8C5.C79.N37.N48.O56
CCc1onc(C)c1NC(=O)C(NC(=O)OC)C(C)C
1326523
[C][C][C][O][N][=C][Branch1][C][C][C][=Ring1][=Branch1][N][C][=Branch1][C][=O][C][Branch1][Branch2][N][C][=Branch1][C][=O][O][C][C][Branch1][C][C][C]
c17onc(C)c16.C3(=O)C5C(C)C.C24=O.CC7.N36.N45.O2C
COc1cccc(CNc2ncc(C(N)=O)cc2Cl)c1
654725
[C][O][C][=C][C][=C][C][Branch2][Ring1][Ring1][C][N][C][=N][C][=C][Branch1][=Branch1][C][Branch1][C][N][=O][C][=C][Ring1][=Branch2][Cl][=C][Ring2][Ring1][C]
c15ncc6cc1Cl.c13cccc7c1.C6(N)=O.CO3.C47.N45
Cc1ccc(S(=O)(=O)N(C)C(C)(C)C#N)cc1C
787366
[C][C][=C][C][=C][Branch2][Ring1][Branch1][S][=Branch1][C][=O][=Branch1][C][=O][N][Branch1][C][C][C][Branch1][C][C][Branch1][C][C][C][#N][C][=C][Ring1][S][C]
Cc1ccc(S3(=O)=O)cc1C.C2(C)(C)C#N.N23C
C=CCNC(=O)CCc1ccc(S(=O)(=O)N2CCCC2)cc1
1785662
[C][=C][C][N][C][=Branch1][C][=O][C][C][C][=C][C][=C][Branch1][#C][S][=Branch1][C][=O][=Branch1][C][=O][N][C][C][C][C][Ring1][Branch1][C][=C][Ring1][=C]
c16ccc(S5(=O)=O)cc1.C3(=O)CC6.N15CCCC1.C=CC4.N34
Cc1occc1C(=O)Nc1cccc(N2CCNC2=O)c1
519222
[C][C][O][C][=C][C][=Ring1][Branch1][C][=Branch1][C][=O][N][C][=C][C][=C][C][Branch1][=Branch2][N][C][C][N][C][Ring1][Branch1][=O][=C][Ring1][N]
c14cccc6c1.Cc1occc15.N16CCNC1=O.C35=O.N34
C#CCN1CCN(C(=O)NCCc2c[nH]c3ccc(F)cc23)CC1
1736209
[C][#C][C][N][C][C][N][Branch2][Ring1][Branch2][C][=Branch1][C][=O][N][C][C][C][=C][NH1][C][=C][C][=C][Branch1][C][F][C][=C][Ring1][#Branch2][Ring1][#Branch1][C][C][Ring2][Ring1][Branch1]
c18c[nH]c2ccc(F)cc12.N16CCN4CC1.C#CC6.C45=O.C7C8.N57
CCNC(=O)c1cccc(CNS(=O)(=O)N2CCCCC2)c1
767338
[C][C][N][C][=Branch1][C][=O][C][=C][C][=C][C][Branch2][Ring1][C][C][N][S][=Branch1][C][=O][=Branch1][C][=O][N][C][C][C][C][C][Ring1][=Branch1][=C][Ring1][P]
N5S(=O)(=O)N1CCCCC1.c16cccc7c1.C36=O.CC4.N34.C57
Cc1n[nH]c(C)c1S(=O)(=O)Nc1cccc2cccnc12
299742
[C][C][=N][NH1][C][Branch1][C][C][=C][Ring1][=Branch1][S][=Branch1][C][=O][=Branch1][C][=O][N][C][=C][C][=C][C][=C][C][=C][N][=C][Ring1][#Branch2][Ring1][=Branch1]
Cc1n[nH]c(C)c1S3(=O)=O.c14cccc2cccnc12.N34
CC(C)CC(=O)N1CCN(C(=O)c2cc(Cl)ccn2)CC1
498106
[C][C][Branch1][C][C][C][C][=Branch1][C][=O][N][C][C][N][Branch1][S][C][=Branch1][C][=O][C][=C][C][Branch1][C][Cl][=C][C][=N][Ring1][#Branch1][C][C][Ring1][#C]
N13CCN4CC1.c15cc(Cl)ccn1.CC(C)CC3=O.C45=O
Cn1cc(CC(=O)Nc2ccc(Oc3ccc(Cl)cn3)cc2)cn1
1237250
[C][N][C][=C][Branch2][Ring1][=N][C][C][=Branch1][C][=O][N][C][=C][C][=C][Branch1][=N][O][C][=C][C][=C][Branch1][C][Cl][C][=N][Ring1][#Branch1][C][=C][Ring1][=C][C][=N][Ring2][Ring1][#Branch1]
c17ccc6cc1.c15ccc(Cl)cn1.Cn1cc8cn1.C8C4=O.N47.O56
CCC(C)C(=O)NC1CCN(C(=O)Cc2cccc(OC)c2)CC1
1683441
[C][C][C][Branch1][C][C][C][=Branch1][C][=O][N][C][C][C][N][Branch2][Ring1][C][C][=Branch1][C][=O][C][C][=C][C][=C][C][Branch1][Ring1][O][C][=C][Ring1][Branch2][C][C][Ring1][P]
C16CCN4CC1.c17cccc5c1.CCC(C)C3=O.C4(=O)C7.N36.O5C
COCCN1CCN(Cc2nc(C)no2)CC1=O
1412661
[C][O][C][C][N][C][C][N][Branch1][N][C][C][=N][C][Branch1][C][C][=N][O][Ring1][=Branch1][C][C][Ring1][=N][=O]
N15CCN4CC1=O.c16nc(C)no1.C3C5.CO3.C46
Cn1ccc(NC(=O)NCC2(c3ccccc3)CCCC2)n1
1050938
[C][N][C][=C][C][Branch2][Ring1][=Branch2][N][C][=Branch1][C][=O][N][C][C][Branch1][=Branch2][C][=C][C][=C][C][=C][Ring1][=Branch1][C][C][C][C][Ring1][O][=N][Ring2][Ring1][Branch1]
Cn1ccc7n1.C189CCCC1.c19ccccc1.C45=O.N47.N56.C68
O=C(Nc1ccccc1)C(C(F)(F)F)C(F)(F)F
54904
[O][=C][Branch1][#Branch2][N][C][=C][C][=C][C][=C][Ring1][=Branch1][C][Branch1][=Branch2][C][Branch1][C][F][Branch1][C][F][F][C][Branch1][C][F][Branch1][C][F][F]
O=C2C(C(F)(F)F)C(F)(F)F.c13ccccc1.N23
CC(C)Oc1ccc(C(=O)NC2(C#N)CCC3(CC2)OCCO3)cn1
1195483
[C][C][Branch1][C][C][O][C][=C][C][=C][Branch2][Ring1][#Branch2][C][=Branch1][C][=O][N][C][Branch1][Ring1][C][#N][C][C][C][Branch1][Branch1][C][C][Ring1][Branch2][O][C][C][O][Ring1][#Branch1][C][=N][Ring2][Ring1][Branch1]
C17(C#N)CCC2(CC1)OCCO2.c16ccc8cn1.CC5C.C48=O.O56.N47
COCCOc1ccccc1NC(=O)c1cc(C)sc1C
779128
[C][O][C][C][O][C][=C][C][=C][C][=C][Ring1][=Branch1][N][C][=Branch1][C][=O][C][C][=C][Branch1][C][C][S][C][=Ring1][=Branch1][C]
c15ccccc16.c17cc(C)sc1C.C3C4.C27=O.CO3.O45.N26
CCN(CCc1nc2ccc(F)cc2[nH]1)C(=O)Cc1cccnc1
912072
[C][C][N][Branch2][Ring1][Ring1][C][C][C][=N][C][=C][C][=C][Branch1][C][F][C][=C][Ring1][#Branch1][NH1][Ring1][#Branch2][C][=Branch1][C][=O][C][C][=C][C][=C][N][=C][Ring1][=Branch1]
c16nc2ccc(F)cc2[nH]1.c17cccnc1.C3(=O)C7.N345.C5C6.CC4
CC(C)c1ccccc1OCC(=O)NCc1ccccc1
33754
[C][C][Branch1][C][C][C][=C][C][=C][C][=C][Ring1][=Branch1][O][C][C][=Branch1][C][=O][N][C][C][=C][C][=C][C][=C][Ring1][=Branch1]
c16ccccc14.c17ccccc1.C3C2=O.CC6C.O34.N25.C57
CCC(C(=O)NCc1ccc(S(N)(=O)=O)cc1)c1ccccc1
1773887
[C][C][C][Branch2][Ring1][=Branch2][C][=Branch1][C][=O][N][C][C][=C][C][=C][Branch1][=Branch2][S][Branch1][C][N][=Branch1][C][=O][=O][C][=C][Ring1][#Branch2][C][=C][C][=C][C][=C][Ring1][=Branch1]
c15ccc(S(N)(=O)=O)cc1.CCC4C2=O.c14ccccc1.N23.C35
COCCN1CCN(C(=O)NCC(C)Cn2cccn2)CC1=O
1444917
[C][O][C][C][N][C][C][N][Branch2][Ring1][Ring1][C][=Branch1][C][=O][N][C][C][Branch1][C][C][C][N][C][=C][C][=N][Ring1][Branch1][C][C][Ring2][Ring1][C][=O]
N18CCN3CC1=O.C6C(C)C7.n17cccn1.C5C8.C34=O.CO5.N46
N#Cc1ccc(NC(=O)COC(=O)CCC2CCCCC2)cc1
71895
[N][#C][C][=C][C][=C][Branch2][Ring1][=Branch1][N][C][=Branch1][C][=O][C][O][C][=Branch1][C][=O][C][C][C][C][C][C][C][C][Ring1][=Branch1][C][=C][Ring2][Ring1][Branch1]
N#Cc1ccc6cc1.C17CCCCC1.C3(=O)CC7.C4(=O)C5.N46.O35
CC(C)CC(NC(=O)c1cc(C(N)=O)cs1)c1ccccc1
737427
[C][C][Branch1][C][C][C][C][Branch2][Ring1][Ring2][N][C][=Branch1][C][=O][C][=C][C][Branch1][=Branch1][C][Branch1][C][N][=O][=C][S][Ring1][Branch2][C][=C][C][=C][C][=C][Ring1][=Branch1]
CC(C)CC36.c14cc5cs1.c16ccccc1.C24=O.C5(N)=O.N23
C#CCN(Cc1cccc(C)n1)C(=O)c1cn(-c2ccccc2)nn1
1022160
[C][#C][C][N][Branch1][=N][C][C][=C][C][=C][C][Branch1][C][C][=N][Ring1][#Branch1][C][=Branch1][C][=O][C][=C][N][Branch1][=Branch2][C][=C][C][=C][C][=C][Ring1][=Branch1][N][=N][Ring1][O]
c17cccc(C)n1.c16cn8nn1.c18ccccc1.C#CC4.N345.C36=O.C57
CC(C)(C)CC(=O)NCc1csc(C2CC2)n1
950229
[C][C][Branch1][C][C][Branch1][C][C][C][C][=Branch1][C][=O][N][C][C][=C][S][C][Branch1][=Branch1][C][C][C][Ring1][Ring1][=N][Ring1][Branch2]
CC(C)(C)CC3=O.c15csc6n1.C16CC1.N34.C45
O=C(NCCNC(=O)c1ccc2c(c1)COCO2)c1ccccc1
1051268
[O][=C][Branch2][Ring1][=Branch2][N][C][C][N][C][=Branch1][C][=O][C][=C][C][=C][C][=Branch1][Ring2][=C][Ring1][=Branch1][C][O][C][O][Ring1][#Branch1][C][=C][C][=C][C][=C][Ring1][=Branch1]
c18ccc2c(c1)COCO2.c17ccccc1.O=C37.C5C6.C48=O.N35.N46
CCNC(=O)NC1CCC(OC(=O)c2cccn2C)CC1
1859013
[C][C][N][C][=Branch1][C][=O][N][C][C][C][C][Branch1][=C][O][C][=Branch1][C][=O][C][=C][C][=C][N][Ring1][Branch1][C][C][C][Ring1][#C]
C18CCC6CC1.c19cccn1C.C45=O.C39=O.CC7.N47.N58.O36