SMILES
large_stringlengths
17
56
ID
large_stringlengths
1
7
SELFIES
stringlengths
63
275
SAFE
stringlengths
20
78
O=C1CN(C(=O)CCS(=O)(=O)c2ccc3c(c2)CCC3)CCN1
603031
[O][=C][C][N][Branch2][Ring1][=N][C][=Branch1][C][=O][C][C][S][=Branch1][C][=O][=Branch1][C][=O][C][=C][C][=C][C][=Branch1][Ring2][=C][Ring1][=Branch1][C][C][C][Ring1][=Branch1][C][C][N][Ring2][Ring1][=Branch1]
C4(=O)CCS(=O)(=O)c1ccc2c(c1)CCC2.O=C1CN4CCN1
CCOc1ccc(NC(=O)NCc2cccnc2OCC)cc1F
1228917
[C][C][O][C][=C][C][=C][Branch2][Ring1][Ring1][N][C][=Branch1][C][=O][N][C][C][=C][C][=C][N][=C][Ring1][=Branch1][O][C][C][C][=C][Ring2][Ring1][Ring2][F]
c18ccc%10cc1F.c1%11cccnc17.C34=O.CC5.O58.N3%10.N49.C9%11.O67.C6C
COCCNC(=O)c1cccc(OCc2ccccc2)c1
135714
[C][O][C][C][N][C][=Branch1][C][=O][C][=C][C][=C][C][Branch1][O][O][C][C][=C][C][=C][C][=C][Ring1][=Branch1][=C][Ring1][=C]
c18cccc6c1.c19ccccc1.C4C7.C38=O.CO4.N37.O56.C59
CCOC(=O)N1CCN(CC(=O)N(c2ccccc2)C(C)C)CC1
1849847
[C][C][O][C][=Branch1][C][=O][N][C][C][N][Branch2][Ring1][=Branch1][C][C][=Branch1][C][=O][N][Branch1][=Branch2][C][=C][C][=C][C][=C][Ring1][=Branch1][C][Branch1][C][C][C][C][C][Ring2][Ring1][Ring1]
N14CCN7CC1.c19ccccc1.C7C5=O.C34=O.N589.C8(C)C.CC6.O36
COCCCCn1nc(-c2ccc(F)cc2)ccc1=O
1346120
[C][O][C][C][C][C][N][N][=C][Branch1][N][C][=C][C][=C][Branch1][C][F][C][=C][Ring1][#Branch1][C][=C][C][Ring1][=N][=O]
n14nc5ccc1=O.c15ccc(F)cc1.C3CCC4.CO3
O=C(CSc1ncc(-c2ccc(F)cc2)o1)NC1CCOCC1
1882390
[O][=C][Branch2][Ring1][#Branch1][C][S][C][=N][C][=C][Branch1][N][C][=C][C][=C][Branch1][C][F][C][=C][Ring1][#Branch1][O][Ring1][N][N][C][C][C][O][C][C][Ring1][=Branch1]
c17ccc(F)cc1.c16ncc7o1.C15CCOCC1.O=C3C4.S46.N35
CCc1nc(C(=O)Nc2ccc3c(ccn3CC(=O)N(C)C)c2)c[nH]1
1216919
[C][C][C][=N][C][Branch2][Ring1][#C][C][=Branch1][C][=O][N][C][=C][C][=C][C][Branch1][S][C][=C][N][Ring1][Branch1][C][C][=Branch1][C][=O][N][Branch1][C][C][C][=C][Ring1][#C][=C][NH1][Ring2][Ring1][#Branch1]
c16ccc2c(ccn28)c1.c19nc7c[nH]1.C8C5=O.C47=O.N5(C)C.CC9.N46
CC(=O)Nc1ccc(C(=O)NCc2noc(C)n2)cc1
1044932
[C][C][=Branch1][C][=O][N][C][=C][C][=C][Branch1][P][C][=Branch1][C][=O][N][C][C][=N][O][C][Branch1][C][C][=N][Ring1][=Branch1][C][=C][Ring1][S]
c16ccc7cc1.c18noc(C)n1.CC3=O.C47=O.N36.N45.C58
CCS(=O)(=O)NCCNc1nc2ccccc2o1
1867102
[C][C][S][=Branch1][C][=O][=Branch1][C][=O][N][C][C][N][C][=N][C][=C][C][=C][C][=C][Ring1][=Branch1][O][Ring1][=Branch2]
c16nc2ccccc2o1.CCS5(=O)=O.C3C4.N35.N46
N#Cc1cccc(NC(=O)c2cnn(-c3cccnc3)c2)c1
1220705
[N][#C][C][=C][C][=C][C][Branch2][Ring1][#Branch1][N][C][=Branch1][C][=O][C][C][=N][N][Branch1][=Branch2][C][=C][C][=C][N][=C][Ring1][=Branch1][C][=Ring1][O][=C][Ring2][Ring1][Ring2]
N#Cc1cccc5c1.c16cnn7c1.c17cccnc1.C46=O.N45
Cc1csc(CCNC(=O)NCc2sccc2C)n1
551958
[C][C][=C][S][C][Branch2][Ring1][C][C][C][N][C][=Branch1][C][=O][N][C][C][S][C][=C][C][=Ring1][Branch1][C][=N][Ring2][Ring1][C]
Cc1csc7n1.c18sccc1C.C7C5.C34=O.N35.N46.C68
O=C(CSc1nc2ccccc2s1)Nc1ccc(O)cc1
68035
[O][=C][Branch1][S][C][S][C][=N][C][=C][C][=C][C][=C][Ring1][=Branch1][S][Ring1][=Branch2][N][C][=C][C][=C][Branch1][C][O][C][=C][Ring1][#Branch1]
c16nc2ccccc2s1.c15ccc(O)cc1.O=C3C4.S46.N35
CCC(C)n1ncc(C(=O)N(C)C2CCCC(C)C2)c1C1CC1
1347515
[C][C][C][Branch1][C][C][N][N][=C][C][Branch2][Ring1][Ring2][C][=Branch1][C][=O][N][Branch1][C][C][C][C][C][C][C][Branch1][C][C][C][Ring1][#Branch1][=C][Ring1][S][C][C][C][Ring1][Ring1]
n16ncc5c17.C14CCCC(C)C1.CCC6C.C35=O.N34C.C17CC1
N#CCCNS(=O)(=O)c1ccc2c(c1)CC(=O)N2
787269
[N][#C][C][C][N][S][=Branch1][C][=O][=Branch1][C][=O][C][=C][C][=C][C][=Branch1][Ring2][=C][Ring1][=Branch1][C][C][=Branch1][C][=O][N][Ring1][#Branch1]
S4(=O)(=O)c1ccc2c(c1)CC(=O)N2.N#CCC3.N34
CC(=O)Nc1ccc(C(=O)c2cc3cc4c(cc3o2)OCO4)cc1
816349
[C][C][=Branch1][C][=O][N][C][=C][C][=C][Branch2][Ring1][=Branch2][C][=Branch1][C][=O][C][=C][C][=C][C][=C][Branch1][Branch2][C][=C][Ring1][=Branch1][O][Ring1][=Branch2][O][C][O][Ring1][Branch2][C][=C][Ring2][Ring1][Ring2]
c17cc2cc3c(cc2o1)OCO3.c16ccc8cc1.CC5=O.C78=O.N56
CCNC(=O)C(C)NC(=O)CN(C)C(=O)c1cccs1
617972
[C][C][N][C][=Branch1][C][=O][C][Branch1][C][C][N][C][=Branch1][C][=O][C][N][Branch1][C][C][C][=Branch1][C][=O][C][=C][C][=C][S][Ring1][Branch1]
C2(=O)C6C.c18cccs1.C3(=O)C7.N47C.C48=O.CC5.N25.N36
Cc1cc2cc(NC(=O)N3CCCCC3c3cccnc3)ccc2o1
1924454
[C][C][=C][C][=C][C][Branch2][Ring1][=Branch1][N][C][=Branch1][C][=O][N][C][C][C][C][C][Ring1][=Branch1][C][=C][C][=C][N][=C][Ring1][=Branch1][=C][C][=C][Ring2][Ring1][Branch1][O][Ring2][Ring1][Branch2]
Cc1cc2cc6ccc2o1.N15CCCCC17.c17cccnc1.C45=O.N46
CCN(CC)C(=O)N1CCN(CC(=O)NC2CCCC(C)C2)CC1
1092445
[C][C][N][Branch1][Ring1][C][C][C][=Branch1][C][=O][N][C][C][N][Branch2][Ring1][C][C][C][=Branch1][C][=O][N][C][C][C][C][C][Branch1][C][C][C][Ring1][#Branch1][C][C][Ring1][P]
N14CCN8CC1.C19CCCC(C)C1.C8C5=O.N367.C34=O.CC6.C7C.N59
CCOc1cc(C#N)c(Br)cc1OCC(=O)OC
62197
[C][C][O][C][=C][C][Branch1][Ring1][C][#N][=C][Branch1][C][Br][C][=C][Ring1][=Branch2][O][C][C][=Branch1][C][=O][O][C]
c15cc(C#N)c(Br)cc16.C4C2=O.CC3.O35.O46.O2C
COc1ccc(NC(=O)C(C)Oc2cccc(C)c2)cc1OC
79159
[C][O][C][=C][C][=C][Branch2][Ring1][=Branch1][N][C][=Branch1][C][=O][C][Branch1][C][C][O][C][=C][C][=C][C][Branch1][C][C][=C][Ring1][#Branch1][C][=C][Ring2][Ring1][Ring1][O][C]
c15ccc8cc17.c16cccc(C)c1.C3(=O)C4C.CO5.N38.O46.O7C
C=CCCNc1ccc(C(=O)N2CCCC(C)C2)cc1C
1150154
[C][=C][C][C][N][C][=C][C][=C][Branch1][S][C][=Branch1][C][=O][N][C][C][C][C][Branch1][C][C][C][Ring1][#Branch1][C][=C][Ring1][#C][C]
c15ccc6cc1C.N13CCCC(C)C1.C=CCC4.C36=O.N45
N#Cc1cccc(COC(=O)c2cccc(C#N)c2)c1
1601816
[N][#C][C][=C][C][=C][C][Branch2][Ring1][Ring1][C][O][C][=Branch1][C][=O][C][=C][C][=C][C][Branch1][Ring1][C][#N][=C][Ring1][Branch2][=C][Ring2][Ring1][C]
N#Cc1cccc6c1.c15cccc(C#N)c1.C35=O.C46.O34
Cc1sc(CNC(=O)c2cnccn2)nc1-c1ccccc1
810259
[C][C][S][C][Branch1][#C][C][N][C][=Branch1][C][=O][C][=C][N][=C][C][=N][Ring1][=Branch1][=N][C][=Ring1][#C][C][=C][C][=C][C][=C][Ring1][=Branch1]
Cc1sc6nc17.c15cnccn1.c17ccccc1.C35=O.C46.N34
CN(Cc1cc(Br)cs1)CC(O)c1ccccc1F
830129
[C][N][Branch1][N][C][C][=C][C][Branch1][C][Br][=C][S][Ring1][=Branch1][C][C][Branch1][C][O][C][=C][C][=C][C][=C][Ring1][=Branch1][F]
c15ccccc1F.c14cc(Br)cs1.C3C5O.CN23.C24
O=C(Nc1ccc2[nH]ncc2c1)c1cnn2ncccc12
1714634
[O][=C][Branch1][#C][N][C][=C][C][=C][NH1][N][=C][C][Ring1][Branch1][=C][Ring1][=Branch2][C][C][=N][N][N][=C][C][=C][C][=Ring1][=Branch2][Ring1][=Branch1]
c14ccc2[nH]ncc2c1.c15cnn2ncccc12.O=C35.N34
O=C(Nc1cc(C(F)(F)F)c[nH]c1=O)N(CCCCO)C1CC1
1310212
[O][=C][Branch2][Ring1][Branch1][N][C][=C][C][Branch1][=Branch2][C][Branch1][C][F][Branch1][C][F][F][=C][NH1][C][Ring1][#Branch2][=O][N][Branch1][=Branch1][C][C][C][C][O][C][C][C][Ring1][Ring1]
c15cc7c[nH]c1=O.C4CCCO.C7(F)(F)F.O=C23.N346.C16CC1.N25
Cc1ncc(NS(=O)(=O)Cc2ccccc2)c(C)c1Cl
1509319
[C][C][=N][C][=C][Branch2][Ring1][C][N][S][=Branch1][C][=O][=Branch1][C][=O][C][C][=C][C][=C][C][=C][Ring1][=Branch1][C][Branch1][C][C][=C][Ring2][Ring1][C][Cl]
Cc1ncc4c(C)c1Cl.c15ccccc1.S3(=O)(=O)C5.N34
CCCc1nnc(NC(=O)c2ccc3nc(C)c(C)nc3c2)s1
1629155
[C][C][C][C][=N][N][=C][Branch2][Ring1][#Branch2][N][C][=Branch1][C][=O][C][=C][C][=C][N][=C][Branch1][C][C][C][Branch1][C][C][=N][C][Ring1][Branch2][=C][Ring1][N][S][Ring2][Ring1][Ring2]
c16ccc2nc(C)c(C)nc2c1.c17nnc5s1.CCC7.C46=O.N45
COc1ccc(Br)cc1CN1CCN(C(C)=O)CC1
1801635
[C][O][C][=C][C][=C][Branch1][C][Br][C][=C][Ring1][#Branch1][C][N][C][C][N][Branch1][=Branch1][C][Branch1][C][C][=O][C][C][Ring1][=Branch2]
c13ccc(Br)cc15.N14CCN2CC1.C2(C)=O.CO3.C45
NS(=O)(=O)CCNC(=O)c1ccc(-n2cccc2)cc1
774963
[N][S][=Branch1][C][=O][=Branch1][C][=O][C][C][N][C][=Branch1][C][=O][C][=C][C][=C][Branch1][Branch2][N][C][=C][C][=C][Ring1][Branch1][C][=C][Ring1][O]
c15ccc6cc1.NS(=O)(=O)CC4.n16cccc1.C35=O.N34
CCC(CO)NS(=O)(=O)c1ccc(C(C)(C)C)cc1
213765
[C][C][C][Branch1][Ring1][C][O][N][S][=Branch1][C][=O][=Branch1][C][=O][C][=C][C][=C][Branch1][=Branch2][C][Branch1][C][C][Branch1][C][C][C][C][=C][Ring1][#Branch2]
S3(=O)(=O)c1ccc4cc1.CCC2CO.C4(C)(C)C.N23
CCC(NC(=O)c1cc(S(N)(=O)=O)c(C)o1)c1nccs1
1308710
[C][C][C][Branch2][Ring1][#Branch2][N][C][=Branch1][C][=O][C][=C][C][Branch1][=Branch2][S][Branch1][C][N][=Branch1][C][=O][=O][=C][Branch1][C][C][O][Ring1][#Branch2][C][=N][C][=C][S][Ring1][Branch1]
c14cc(S(N)(=O)=O)c(C)o1.c15nccs1.CCC35.C24=O.N23
CCC1c2ccsc2CCN1C(=O)c1cncnc1
1873275
[C][C][C][C][C][=C][S][C][=Ring1][Branch1][C][C][N][Ring1][=Branch2][C][=Branch1][C][=O][C][=C][N][=C][N][=C][Ring1][=Branch1]
CCC1c2ccsc2CCN13.c14cncnc1.C34=O
O=C(COC(=O)CC1CC2CCC1C2)NCc1ccc2c(c1)OCO2
115685
[O][=C][Branch2][Ring1][Ring1][C][O][C][=Branch1][C][=O][C][C][C][C][C][C][C][Ring1][=Branch1][C][Ring1][Branch1][N][C][C][=C][C][=C][C][=Branch1][Ring2][=C][Ring1][=Branch1][O][C][O][Ring1][=Branch1]
c18ccc2c(c1)OCO2.C17CC2CCC1C2.O=C4C5.C3(=O)C7.O35.N46.C68
COC(=O)NCC(=O)NCC(C)c1ccccc1
660102
[C][O][C][=Branch1][C][=O][N][C][C][=Branch1][C][=O][N][C][C][Branch1][C][C][C][=C][C][=C][C][=C][Ring1][=Branch1]
c17ccccc1.C5C4=O.C6C7C.C23=O.CO2.N35.N46
Cc1ccc(C)c(Cn2ccnc2CN(C(=O)C2CCC2)C(C)C)c1
135545
[C][C][=C][C][=C][Branch1][C][C][C][Branch2][Ring1][N][C][N][C][=C][N][=C][Ring1][Branch1][C][N][Branch1][O][C][=Branch1][C][=O][C][C][C][C][Ring1][Ring2][C][Branch1][C][C][C][=C][Ring2][Ring1][Branch2]
Cc1ccc(C)c9c1.n17ccnc18.C16CCC1.N345.C36=O.C5(C)C.C79.C48
CC(C)[S+]([O-])c1ccc(C(=O)Nc2ccccn2)cc1
1176989
[C][C][Branch1][C][C][S+1][Branch1][C][O-1][C][=C][C][=C][Branch1][=C][C][=Branch1][C][=O][N][C][=C][C][=C][C][=N][Ring1][=Branch1][C][=C][Ring1][#C]
CC(C)[S+]([O-])c1ccc5cc1.c14ccccn1.C35=O.N34
Cc1ccc(C(=O)N(C)Cc2ccc(O)cc2)cc1S(C)(=O)=O
734930
[C][C][=C][C][=C][Branch2][Ring1][Branch1][C][=Branch1][C][=O][N][Branch1][C][C][C][C][=C][C][=C][Branch1][C][O][C][=C][Ring1][#Branch1][C][=C][Ring2][Ring1][C][S][Branch1][C][C][=Branch1][C][=O][=O]
Cc1ccc5cc1S(C)(=O)=O.c16ccc(O)cc1.C35=O.N34C.C46
Cc1nc(C)c(CC(=O)NCCCN(C)c2ccccc2)c(=O)[nH]1
415573
[C][C][=N][C][Branch1][C][C][=C][Branch2][Ring1][=Branch1][C][C][=Branch1][C][=O][N][C][C][C][N][Branch1][C][C][C][=C][C][=C][C][=C][Ring1][=Branch1][C][=Branch1][C][=O][NH1][Ring2][Ring1][#Branch1]
Cc1nc(C)c7c(=O)[nH]1.c16ccccc1.C7C3=O.C4CC5.N56C.N34
Cc1n[nH]c(C)c1N1CCN(Cc2cc(F)ccc2F)CC1
777204
[C][C][=N][NH1][C][Branch1][C][C][=C][Ring1][=Branch1][N][C][C][N][Branch1][=C][C][C][=C][C][Branch1][C][F][=C][C][=C][Ring1][#Branch1][F][C][C][Ring1][#C]
c15cc(F)ccc1F.Cc1n[nH]c(C)c14.N14CCN3CC1.C35
Cc1noc(C)c1CNc1cccc(S(=O)(=O)C2CCCC2)c1
385194
[C][C][=N][O][C][Branch1][C][C][=C][Ring1][=Branch1][C][N][C][=C][C][=C][C][Branch1][#C][S][=Branch1][C][=O][=Branch1][C][=O][C][C][C][C][C][Ring1][Branch1][=C][Ring1][=C]
c14cccc(S(=O)(=O)C2CCCC2)c1.Cc1noc(C)c15.C35.N34
CCCNC(=O)c1ccc(F)c(S(=O)(=O)NC(C)(C)C)c1
407787
[C][C][C][N][C][=Branch1][C][=O][C][=C][C][=C][Branch1][C][F][C][Branch1][P][S][=Branch1][C][=O][=Branch1][C][=O][N][C][Branch1][C][C][Branch1][C][C][C][=C][Ring1][#C]
c16ccc(F)c(S5(=O)=O)c1.C4(C)(C)C.CCC3.C26=O.N23.N45
CC(NC(=O)c1cc(C2CC2)[nH]n1)c1ccc2c(c1)NC(=O)CO2
448322
[C][C][Branch2][Ring1][Ring2][N][C][=Branch1][C][=O][C][C][=C][Branch1][=Branch1][C][C][C][Ring1][Ring1][NH1][N][=Ring1][Branch2][C][=C][C][=C][C][=Branch1][Ring2][=C][Ring1][=Branch1][N][C][=Branch1][C][=O][C][O][Ring1][Branch2]
c16ccc2c(c1)NC(=O)CO2.c15cc7[nH]n1.CC46.C35=O.C17CC1.N34
CC(=O)Nc1ccc(CC(=O)OCC(=O)NC(C)C)cc1
157151
[C][C][=Branch1][C][=O][N][C][=C][C][=C][Branch2][Ring1][C][C][C][=Branch1][C][=O][O][C][C][=Branch1][C][=O][N][C][Branch1][C][C][C][C][=C][Ring1][P]
c17ccc8cc1.C8C2=O.C5C4=O.CC3=O.C6(C)C.N37.O25.N46
Cc1noc(-c2cccc(=O)n2CC(=O)Nc2ccccc2F)n1
1855148
[C][C][=N][O][C][Branch2][Ring1][O][C][=C][C][=C][C][=Branch1][C][=O][N][Ring1][#Branch1][C][C][=Branch1][C][=O][N][C][=C][C][=C][C][=C][Ring1][=Branch1][F][=N][Ring2][Ring1][#Branch1]
c16cccc(=O)n15.c14ccccc1F.Cc1noc6n1.C5C3=O.N34
Cc1nc2ccccn2c(=O)c1NC(=O)CCCc1ccccc1
90268
[C][C][N][=C][C][=C][C][=C][N][Ring1][=Branch1][C][=Branch1][C][=O][C][=Ring1][O][N][C][=Branch1][C][=O][C][C][C][C][=C][C][=C][C][=C][Ring1][=Branch1]
Cc1nc2ccccn2c(=O)c14.C3(=O)CCC5.c15ccccc1.N34
O=c1ccc(CNc2cccc(OC(F)F)c2)c[nH]1
1264749
[O][=C][C][=C][C][Branch2][Ring1][Ring1][C][N][C][=C][C][=C][C][Branch1][#Branch1][O][C][Branch1][C][F][F][=C][Ring1][#Branch2][=C][NH1][Ring2][Ring1][C]
O=c1ccc6c[nH]1.c15cccc3c1.O3C(F)F.C46.N45
CCCCN(C)C(=O)c1cnc(-c2ccccc2)nc1N
1138145
[C][C][C][C][N][Branch1][C][C][C][=Branch1][C][=O][C][=C][N][=C][Branch1][=Branch2][C][=C][C][=C][C][=C][Ring1][=Branch1][N][=C][Ring1][N][N]
c15cnc6nc1N.c16ccccc1.CCCC4.N34C.C35=O
CCCOCC(=O)N1CCN(Cc2nc(N)c3ccccc3n2)CC1
891353
[C][C][C][O][C][C][=Branch1][C][=O][N][C][C][N][Branch2][Ring1][Ring1][C][C][=N][C][Branch1][C][N][=C][C][=C][C][=C][C][Ring1][=Branch1][=N][Ring1][O][C][C][Ring2][Ring1][C]
c18nc(N)c2ccccc2n1.N14CCN7CC1.C6C4=O.CCC5.O56.C78
Cc1ccc(OC(C)C(=O)Nc2cccnc2N(C)C)cc1
442820
[C][C][=C][C][=C][Branch2][Ring1][Branch2][O][C][Branch1][C][C][C][=Branch1][C][=O][N][C][=C][C][=C][N][=C][Ring1][=Branch1][N][Branch1][C][C][C][C][=C][Ring2][Ring1][Branch1]
Cc1ccc5cc1.c17cccnc16.C4(C)C3=O.N6(C)C.O45.N37
Brc1cccc(OCCCN2CCOCC2)c1
1796917
[Br][C][=C][C][=C][C][Branch1][=N][O][C][C][C][N][C][C][O][C][C][Ring1][=Branch1][=C][Ring1][S]
Brc1cccc4c1.N15CCOCC1.C3CC5.O34
COc1cc(CN(Cc2cc(F)ccc2C#N)C2CC2)ccc1O
1369753
[C][O][C][=C][C][Branch2][Ring1][Branch2][C][N][Branch1][#C][C][C][=C][C][Branch1][C][F][=C][C][=C][Ring1][#Branch1][C][#N][C][C][C][Ring1][Ring1][=C][C][=C][Ring2][Ring1][Branch1][O]
c18cc(F)ccc1C#N.c13cc7ccc1O.N456.C16CC1.CO3.C47.C58
Cc1cnc(C(=O)NCCOc2ccc(C(C)(C)C)cc2)cn1
349866
[C][C][=C][N][=C][Branch2][Ring1][O][C][=Branch1][C][=O][N][C][C][O][C][=C][C][=C][Branch1][=Branch2][C][Branch1][C][C][Branch1][C][C][C][C][=C][Ring1][#Branch2][C][=N][Ring2][Ring1][=Branch1]
Cc1cnc7cn1.c15ccc8cc1.C8(C)(C)C.C37=O.C6C4.N36.O45
CCOC(=O)C1CCCN(C(=O)c2nccc3cccc(N)c23)C1
1530493
[C][C][O][C][=Branch1][C][=O][C][C][C][C][N][Branch2][Ring1][=Branch1][C][=Branch1][C][=O][C][=N][C][=C][C][=C][C][=C][C][Branch1][C][N][=C][Ring1][O][Ring1][#Branch1][C][Ring2][Ring1][Ring1]
c17nccc2cccc(N)c12.C18CCCN5C1.C48=O.C57=O.CC6.O46
Cc1ccc(-c2ncco2)cc1NC(=O)CCc1cccnc1
1339492
[C][C][=C][C][=C][Branch1][Branch2][C][=N][C][=C][O][Ring1][Branch1][C][=C][Ring1][O][N][C][=Branch1][C][=O][C][C][C][=C][C][=C][N][=C][Ring1][=Branch1]
Cc1ccc6cc14.c15cccnc1.c16ncco1.C3(=O)CC5.N34
CCN(C(=O)CCNC(=O)OC(C)(C)C)c1ccc(C)cc1C
1187977
[C][C][N][Branch2][Ring1][Branch1][C][=Branch1][C][=O][C][C][N][C][=Branch1][C][=O][O][C][Branch1][C][C][Branch1][C][C][C][C][=C][C][=C][Branch1][C][C][C][=C][Ring1][#Branch1][C]
c18ccc(C)cc1C.C3(=O)CC7.C5(C)(C)C.N368.C24=O.CC6.N47.O25
Cc1nc2cc(C(=O)N3CCc4sccc4C3)ccc2s1
339297
[C][C][=N][C][=C][C][Branch2][Ring1][C][C][=Branch1][C][=O][N][C][C][C][S][C][=C][C][=Ring1][Branch1][C][Ring1][=Branch2][=C][C][=C][Ring1][P][S][Ring2][Ring1][Ring2]
Cc1nc2cc6ccc2s1.N15CCc2sccc2C1.C56=O
CCn1ncnc1CN1CC(NS(=O)(=O)N(C)C)C(C2CC2)C1
1416040
[C][C][N][N][=C][N][=C][Ring1][Branch1][C][N][C][C][Branch1][=C][N][S][=Branch1][C][=O][=Branch1][C][=O][N][Branch1][C][C][C][C][Branch1][=Branch1][C][C][C][Ring1][Ring1][C][Ring1][#C]
N13CC4C(C2CC2)C1.N4S(=O)(=O)N(C)C.n15ncnc16.CC5.C36
CC(Cc1ccsc1)n1c(=O)[nH]c2ccccc2c1=O
659237
[C][C][Branch1][=Branch2][C][C][C][=C][S][C][=Ring1][Branch1][N][C][=Branch1][C][=O][NH1][C][=C][C][=C][C][=C][Ring1][=Branch1][C][Ring1][O][=O]
n13c(=O)[nH]c2ccccc2c1=O.c14ccsc1.CC3C4
Cc1cc(C)n2nc(SCc3nc(N)c4ccccc4n3)nc2n1
1780809
[C][C][C][=C][Branch1][C][C][N][N][=C][Branch2][Ring1][Ring2][S][C][C][=N][C][Branch1][C][N][=C][C][=C][C][=C][C][Ring1][=Branch1][=N][Ring1][O][N][=C][Ring2][Ring1][C][N][=Ring2][Ring1][#Branch1]
Cc1cc(C)n2nc7nc2n1.c16nc(N)c2ccccc2n1.S57.C56
CCC(C)C(C)NC(=O)Nc1ccc(C(=O)NC)c(Cl)c1
1581098
[C][C][C][Branch1][C][C][C][Branch1][C][C][N][C][=Branch1][C][=O][N][C][=C][C][=C][Branch1][#Branch1][C][=Branch1][C][=O][N][C][C][Branch1][C][Cl][=C][Ring1][O]
c16ccc7c(Cl)c1.CCC(C)C5C.C23=O.C47=O.N25.N36.N4C
Cc1ccc(Cl)c(OC(=O)Cn2c(=O)[nH]c3ccccc3c2=O)c1
1085854
[C][C][=C][C][=C][Branch1][C][Cl][C][Branch2][Ring1][=Branch2][O][C][=Branch1][C][=O][C][N][C][=Branch1][C][=O][NH1][C][=C][C][=C][C][=C][Ring1][=Branch1][C][Ring1][O][=O][=C][Ring2][Ring1][#Branch1]
n16c(=O)[nH]c2ccccc2c1=O.Cc1ccc(Cl)c5c1.C4(=O)C6.O45
Cn1nc2n(c1=O)CCN(CCn1nc3ccccn3c1=O)C2
1396318
[C][N][N][=C][N][Branch1][Branch1][C][Ring1][Branch1][=O][C][C][N][Branch1][P][C][C][N][N][=C][C][=C][C][=C][N][Ring1][=Branch1][C][Ring1][=Branch2][=O][C][Ring2][Ring1][Ring2]
Cn1nc2n(c1=O)CCN4C2.n15nc2ccccn2c1=O.C4C5
O=C(CCCNC(=O)c1cc2sccc2[nH]1)Nc1ccccc1
1167952
[O][=C][Branch2][Ring1][Branch1][C][C][C][N][C][=Branch1][C][=O][C][=C][C][S][C][=C][C][=Ring1][Branch1][NH1][Ring1][Branch2][N][C][=C][C][=C][C][=C][Ring1][=Branch1]
c17cc2sccc2[nH]1.O=C3CCC5.c16ccccc1.C47=O.N45.N36
Cc1ccc(-c2nc(CC(=O)NC(C3CC3)C3CC3)cs2)o1
1880881
[C][C][=C][C][=C][Branch2][Ring1][=C][C][=N][C][Branch2][Ring1][Ring2][C][C][=Branch1][C][=O][N][C][Branch1][=Branch1][C][C][C][Ring1][Ring1][C][C][C][Ring1][Ring1][=C][S][Ring1][S][O][Ring2][Ring1][Branch1]
Cc1ccc9o1.c19nc6cs1.C6C4=O.C578.C17CC1.C18CC1.N45
COCc1nc(C)cc(N(C)C2CCN(CC(F)(F)F)C2=O)n1
1075645
[C][O][C][C][=N][C][Branch1][C][C][=C][C][Branch2][Ring1][Branch2][N][Branch1][C][C][C][C][C][N][Branch1][#Branch2][C][C][Branch1][C][F][Branch1][C][F][F][C][Ring1][#Branch2][=O][=N][Ring2][Ring1][Ring2]
c17nc4cc(C)n1.C15CCN6C1=O.C6C(F)(F)F.N45C.CO3.C37
COc1ccc(OCCNC(=O)c2ccc(-n3cncn3)nc2)cc1
1203305
[C][O][C][=C][C][=C][Branch2][Ring1][#Branch2][O][C][C][N][C][=Branch1][C][=O][C][=C][C][=C][Branch1][Branch2][N][C][=N][C][=N][Ring1][Branch1][N][=C][Ring1][O][C][=C][Ring2][Ring1][#Branch1]
c16ccc7cc1.c19ccc%10nc1.n1%10cncn1.C5C8.C49=O.CO6.O57.N48
CCC(C)C(NC(=O)c1sc(C)nc1C)C(N)=O
939946
[C][C][C][Branch1][C][C][C][Branch1][P][N][C][=Branch1][C][=O][C][S][C][Branch1][C][C][=N][C][=Ring1][=Branch1][C][C][Branch1][C][N][=O]
CCC(C)C3C(N)=O.c14sc(C)nc1C.C24=O.N23
CC1CCN(C(=O)c2ccc3ncnc(N4CCCCC4)c3c2)CC1
1088382
[C][C][C][C][N][Branch2][Ring1][=N][C][=Branch1][C][=O][C][=C][C][=C][N][=C][N][=C][Branch1][=Branch2][N][C][C][C][C][C][Ring1][=Branch1][C][Ring1][N][=C][Ring1][S][C][C][Ring2][Ring1][Branch2]
c17ccc2ncnc6c2c1.CC1CCN5CC1.N16CCCCC1.C57=O
CCn1c(=O)c2c(nc3n(-c4ccc(C)cc4)c(C)cn23)n(C)c1=O
87085
[C][C][N][C][=Branch1][C][=O][C][=C][Branch2][Ring1][O][N][=C][N][Branch1][N][C][=C][C][=C][Branch1][C][C][C][=C][Ring1][#Branch1][C][Branch1][C][C][=C][N][Ring1][S][Ring1][=N][N][Branch1][C][C][C][Ring2][Ring1][=Branch1][=O]
n15c(=O)c2c(nc3n6c(C)cn23)n(C)c1=O.c16ccc(C)cc1.CC5
CC(C(=O)NCc1cccc(OCC#N)c1)c1ccsc1
1182735
[C][C][Branch2][Ring1][Branch1][C][=Branch1][C][=O][N][C][C][=C][C][=C][C][Branch1][Branch1][O][C][C][#N][=C][Ring1][#Branch2][C][C][=C][S][C][=Ring1][Branch1]
c17cccc4c1.CC6C2=O.c16ccsc1.C3C#N.N25.C57.O34
CCC(NC(=O)c1cnc(C)cn1)c1ccc(Cl)cc1
358312
[C][C][C][Branch1][P][N][C][=Branch1][C][=O][C][=C][N][=C][Branch1][C][C][C][=N][Ring1][#Branch1][C][=C][C][=C][Branch1][C][Cl][C][=C][Ring1][#Branch1]
c14cnc(C)cn1.c15ccc(Cl)cc1.CCC35.C24=O.N23
CCc1nn(-c2ccccc2)c(NC(=O)c2ccc(C)[nH]c2=O)c1C
754666
[C][C][C][=N][N][Branch1][=Branch2][C][=C][C][=C][C][=C][Ring1][=Branch1][C][Branch2][Ring1][C][N][C][=Branch1][C][=O][C][=C][C][=C][Branch1][C][C][NH1][C][Ring1][#Branch1][=O][=C][Ring2][Ring1][=Branch1][C]
c16nn7c4c1C.c15ccc(C)[nH]c1=O.c17ccccc1.C35=O.CC6.N34
Cc1[nH]ncc1CCCNC(=O)N1CCN(S(C)(=O)=O)CC1
1221346
[C][C][NH1][N][=C][C][=Ring1][Branch1][C][C][C][N][C][=Branch1][C][=O][N][C][C][N][Branch1][=Branch2][S][Branch1][C][C][=Branch1][C][=O][=O][C][C][Ring1][#Branch2]
N13CCN5CC1.Cc1[nH]ncc16.C6CC4.S5(C)(=O)=O.C23=O.N24
Cc1nc2nc(N)nn2c(C)c1CCC(=O)N1CCCC1
295466
[C][C][=N][C][=N][C][Branch1][C][N][=N][N][Ring1][=Branch1][C][Branch1][C][C][=C][Ring1][O][C][C][C][=Branch1][C][=O][N][C][C][C][C][Ring1][Branch1]
Cc1nc2nc(N)nn2c(C)c14.C4CC3=O.N13CCCC1
COC(=O)C1CN(S(C)(=O)=O)CCN1C(=O)C1CCCCC1
87479
[C][O][C][=Branch1][C][=O][C][C][N][Branch1][=Branch2][S][Branch1][C][C][=Branch1][C][=O][=O][C][C][N][Ring1][#Branch2][C][=Branch1][C][=O][C][C][C][C][C][C][Ring1][=Branch1]
C15CN4CCN13.C16CCCCC1.S4(C)(=O)=O.C25=O.C36=O.CO2
CCOc1ccccc1-n1nnc(CO)c1-c1ccncc1
839172
[C][C][O][C][=C][C][=C][C][=C][Ring1][=Branch1][N][N][=N][C][Branch1][Ring1][C][O][=C][Ring1][#Branch1][C][=C][C][=N][C][=C][Ring1][=Branch1]
c13ccccc15.n15nnc4c16.c16ccncc1.CC2.O23.C4O
CCCc1noc(C2CCN(C(=O)CCOC)CC2)n1
538422
[C][C][C][C][=N][O][C][Branch2][Ring1][Ring1][C][C][C][N][Branch1][=Branch2][C][=Branch1][C][=O][C][C][O][C][C][C][Ring1][N][=N][Ring1][P]
C16CCN3CC1.c15noc6n1.C3(=O)CC4.CCC5.O4C
Cc1ccc(CN2CCN(C(=O)CC(C)C)CC2)cc1
1795844
[C][C][=C][C][=C][Branch2][Ring1][=Branch1][C][N][C][C][N][Branch1][O][C][=Branch1][C][=O][C][C][Branch1][C][C][C][C][C][Ring1][N][C][=C][Ring2][Ring1][Ring1]
Cc1ccc5cc1.N14CCN3CC1.C3(=O)CC(C)C.C45
COc1cccc(C(=O)NC(C)C(=O)OC2CCCC2)c1F
1394910
[C][O][C][=C][C][=C][C][Branch2][Ring1][=Branch1][C][=Branch1][C][=O][N][C][Branch1][C][C][C][=Branch1][C][=O][O][C][C][C][C][C][Ring1][Branch1][=C][Ring2][Ring1][Ring1][F]
c16cccc8c1F.C7(C)C3=O.C15CCCC1.C48=O.CO6.N47.O35
COc1cc(C(=O)NCC(C)C)cc(OC)c1OC
22206
[C][O][C][=C][C][Branch1][N][C][=Branch1][C][=O][N][C][C][Branch1][C][C][C][=C][C][Branch1][Ring1][O][C][=C][Ring1][#C][O][C]
c13cc7cc4c15.C6C(C)C.C27=O.CO3.N26.O4C.O5C
Cc1ccnc(N2CCc3[nH]nc(-c4cccc(F)c4)c3C2)n1
1686974
[C][C][=C][C][=N][C][Branch2][Ring1][O][N][C][C][C][NH1][N][=C][Branch1][N][C][=C][C][=C][C][Branch1][C][F][=C][Ring1][#Branch1][C][=Ring1][N][C][Ring1][S][=N][Ring2][Ring1][=Branch1]
N15CCc2[nH]nc6c2C1.Cc1ccnc5n1.c16cccc(F)c1
CCc1cc(C(=O)N2CCCC(CCO)C2)sc1C
729079
[C][C][C][C][=C][Branch2][Ring1][C][C][=Branch1][C][=O][N][C][C][C][C][Branch1][Ring2][C][C][O][C][Ring1][=Branch2][S][C][=Ring1][S][C]
c16cc4sc1C.N13CCCC5C1.C34=O.C5CO.CC6
CC1CCN(C(=O)CN(C)C(=O)c2cccs2)C(C)C1
1715196
[C][C][C][C][N][Branch2][Ring1][Branch1][C][=Branch1][C][=O][C][N][Branch1][C][C][C][=Branch1][C][=O][C][=C][C][=C][S][Ring1][Branch1][C][Branch1][C][C][C][Ring2][Ring1][Ring1]
CC1CCN3C(C)C1.c16cccs1.C3(=O)C5.N45C.C46=O
COc1ccc(CN(C)C(=O)c2ccc(C(F)(F)F)nc2)cc1
1052556
[C][O][C][=C][C][=C][Branch2][Ring1][N][C][N][Branch1][C][C][C][=Branch1][C][=O][C][=C][C][=C][Branch1][=Branch2][C][Branch1][C][F][Branch1][C][F][F][N][=C][Ring1][#Branch2][C][=C][Ring2][Ring1][Branch1]
c14ccc8cc1.c16ccc7nc1.C7(F)(F)F.N35C.C36=O.CO4.C58
CCc1nc2cc3c(cc2n1CC(=O)Nc1ccccc1)OCCO3
1680209
[C][C][C][=N][C][=C][C][=C][Branch2][Ring1][=Branch1][C][=C][Ring1][=Branch1][N][Ring1][=Branch2][C][C][=Branch1][C][=O][N][C][=C][C][=C][C][=C][Ring1][=Branch1][O][C][C][O][Ring2][Ring1][Ring1]
c17nc2cc3c(cc2n16)OCCO3.c15ccccc1.C6C4=O.CC7.N45
CC1OCCN(Cc2ccc(C(=O)N(C)C)[nH]2)C1C
1443332
[C][C][O][C][C][N][Branch2][Ring1][Ring2][C][C][=C][C][=C][Branch1][#Branch2][C][=Branch1][C][=O][N][Branch1][C][C][C][NH1][Ring1][#Branch2][C][Ring1][P][C]
CC1OCCN4C1C.c16ccc5[nH]1.C35=O.N3(C)C.C46
CCCc1cc(C(=O)N2CCN(Cc3cc(C)no3)CC2)[nH]n1
1654912
[C][C][C][C][C][=C][Branch2][Ring1][#Branch2][C][=Branch1][C][=O][N][C][C][N][Branch1][N][C][C][=C][C][Branch1][C][C][=N][O][Ring1][=Branch1][C][C][Ring1][=N][NH1][N][=Ring2][Ring1][Ring2]
N14CCN5CC1.c17cc6[nH]n1.c18cc(C)no1.CCC7.C46=O.C58
O=C(Cn1ccc2ccccc21)NCC1CC2C=CC1C2
424303
[O][=C][Branch1][#C][C][N][C][=C][C][=C][C][=C][C][=C][Ring1][=Branch1][Ring1][=Branch2][N][C][C][C][C][C][=C][C][Ring1][=Branch1][C][Ring1][Branch1]
n15ccc2ccccc21.C16CC2C=CC1C2.O=C3C5.N34.C46
Cc1nc(NC(=O)c2csnn2)sc1Cc1ccccc1F
817266
[C][C][N][=C][Branch1][=N][N][C][=Branch1][C][=O][C][=C][S][N][=N][Ring1][Branch1][S][C][=Ring1][=N][C][C][=C][C][=C][C][=C][Ring1][=Branch1][F]
Cc1nc4sc16.c17ccccc1F.c15csnn1.C35=O.N34.C67
COc1ccc(Nc2ncnc3sccc23)cc1OC
74155
[C][O][C][=C][C][=C][Branch1][#C][N][C][=N][C][=N][C][S][C][=C][C][Ring1][=Branch2][=Ring1][Branch1][C][=C][Ring1][S][O][C]
c16ncnc2sccc12.c14ccc7cc15.CO4.N67.O5C
CCn1c(C)nnc1SCCNC(=O)c1cncnc1C
1565539
[C][C][N][C][Branch1][C][C][=N][N][=C][Ring1][=Branch1][S][C][C][N][C][=Branch1][C][=O][C][=C][N][=C][N][=C][Ring1][=Branch1][C]
n16c7nnc1C.c15cncnc1C.C4C3.C25=O.CC6.S47.N23
O=C(Nc1cccc(-c2cn[nH]c2)c1)c1cnc2sccn2c1=O
1914700
[O][=C][Branch2][Ring1][Ring1][N][C][=C][C][=C][C][Branch1][Branch2][C][C][=N][NH1][C][=Ring1][Branch1][=C][Ring1][O][C][=C][N][=C][S][C][=C][N][Ring1][Branch1][C][Ring1][=Branch2][=O]
c15cnc2sccn2c1=O.c14cccc6c1.c16cn[nH]c1.O=C35.N34
CCCNS(=O)(=O)c1ccc(CC(C)C)cc1
259762
[C][C][C][N][S][=Branch1][C][=O][=Branch1][C][=O][C][=C][C][=C][Branch1][#Branch1][C][C][Branch1][C][C][C][C][=C][Ring1][#Branch2]
S3(=O)(=O)c1ccc4cc1.C4C(C)C.CCC2.N23
NS(=O)(=O)N1CCN(Cc2ccc(Cl)cc2Cl)CC1
1834331
[N][S][=Branch1][C][=O][=Branch1][C][=O][N][C][C][N][Branch1][=C][C][C][=C][C][=C][Branch1][C][Cl][C][=C][Ring1][#Branch1][Cl][C][C][Ring1][#C]
NS(=O)(=O)N1CCN3CC1.c14ccc(Cl)cc1Cl.C34
Cc1ccc(C(=O)N2CCC(c3ccccc3)CC2)c(=O)[nH]1
1077402
[C][C][=C][C][=C][Branch2][Ring1][#Branch1][C][=Branch1][C][=O][N][C][C][C][Branch1][=Branch2][C][=C][C][=C][C][=C][Ring1][=Branch1][C][C][Ring1][N][C][=Branch1][C][=O][NH1][Ring2][Ring1][Branch1]
Cc1ccc5c(=O)[nH]1.N14CCC6CC1.c16ccccc1.C45=O
Nc1cccc(C(O)CCC(=O)N2CCCc3ccccc32)c1
714543
[N][C][=C][C][=C][C][Branch2][Ring1][=Branch2][C][Branch1][C][O][C][C][C][=Branch1][C][=O][N][C][C][C][C][=C][C][=C][C][=C][Ring1][=Branch1][Ring1][#Branch2][=C][Ring2][Ring1][=Branch1]
N14CCCc2ccccc21.Nc1cccc5c1.C5(O)CCC4=O
Cc1cc(C)n(CCCNC(=O)c2cc3ccc(F)cc3n2C)n1
544397
[C][C][C][=C][Branch1][C][C][N][Branch2][Ring1][#Branch2][C][C][C][N][C][=Branch1][C][=O][C][=C][C][=C][C][=C][Branch1][C][F][C][=C][Ring1][#Branch1][N][Ring1][#Branch2][C][N][=Ring2][Ring1][#Branch1]
c16cc2ccc(F)cc2n1C.Cc1cc(C)n7n1.C7CC5.C46=O.N45
O=C(c1cc(-c2ccncc2)on1)N1CCC(=Cc2ccccc2)CC1
1910912
[O][=C][Branch2][Ring1][C][C][C][=C][Branch1][=Branch2][C][=C][C][=N][C][=C][Ring1][=Branch1][O][N][=Ring1][O][N][C][C][C][=Branch1][#Branch2][=C][C][=C][C][=C][C][=C][Ring1][=Branch1][C][C][Ring1][=N]
N13CCC=5CC1.C=5c1ccccc1.c14cc6on1.c16ccncc1.O=C34
CCn1c(C2CC(=O)N(C3CCCC3)C2)nc2ccccc21
521219
[C][C][N][C][Branch2][Ring1][Ring2][C][C][C][=Branch1][C][=O][N][Branch1][Branch2][C][C][C][C][C][Ring1][Branch1][C][Ring1][O][=N][C][=C][C][=C][C][=C][Ring1][=Branch1][Ring2][Ring1][Ring2]
n14c6nc2ccccc21.C16CC(=O)N5C1.C15CCCC1.CC4