SMILES
large_stringlengths
17
56
ID
large_stringlengths
1
7
SELFIES
stringlengths
63
275
SAFE
stringlengths
20
78
O=C1CCc2cc(C(=O)Cn3cnc4ccsc4c3=O)ccc2N1
598741
[O][=C][C][C][C][=C][C][Branch2][Ring1][Ring2][C][=Branch1][C][=O][C][N][C][=N][C][C][=C][S][C][=Ring1][Branch1][C][Ring1][=Branch2][=O][=C][C][=C][Ring2][Ring1][Ring1][N][Ring2][Ring1][#Branch1]
O=C1CCc2cc5ccc2N1.n16cnc2ccsc2c1=O.C5(=O)C6
CC1COCCN1C(=O)CN(C)S(C)(=O)=O
600435
[C][C][C][O][C][C][N][Ring1][=Branch1][C][=Branch1][C][=O][C][N][Branch1][C][C][S][Branch1][C][C][=Branch1][C][=O][=O]
CC1COCCN12.C2(=O)C3.S4(C)(=O)=O.N34C
Cc1c(C(=O)Nc2ccc3nn[nH]c3c2)cnn1-c1ccncc1
1396129
[C][C][=C][Branch2][Ring1][Ring1][C][=Branch1][C][=O][N][C][=C][C][=C][N][=N][NH1][C][Ring1][Branch1][=C][Ring1][=Branch2][C][=N][N][Ring1][P][C][=C][C][=N][C][=C][Ring1][=Branch1]
c15ccc2nn[nH]c2c1.Cc1c6cnn17.c17ccncc1.C46=O.N45
CNc1cc(C(=O)N2CCN3CCNC(=O)C3C2)ccn1
879464
[C][N][C][=C][C][Branch2][Ring1][=Branch1][C][=Branch1][C][=O][N][C][C][N][C][C][N][C][=Branch1][C][=O][C][Ring1][#Branch1][C][Ring1][O][=C][C][=N][Ring2][Ring1][Ring1]
N14CCN2CCNC(=O)C2C1.c15cc6ccn1.C46=O.CN5
Cc1cc(NC(=O)c2ccn3cncc3c2)c2ncccc2c1
1411474
[C][C][=C][C][Branch2][Ring1][Ring1][N][C][=Branch1][C][=O][C][C][=C][N][C][=N][C][=C][Ring1][Branch1][C][=Ring1][=Branch2][=C][N][=C][C][=C][C][Ring1][=Branch1][=C][Ring2][Ring1][=Branch1]
Cc1cc5c2ncccc2c1.c16ccn2cncc2c1.C46=O.N45
COc1c(Cl)cccc1NC(=O)c1cnn(C)c1
665540
[C][O][C][=C][Branch1][C][Cl][C][=C][C][=C][Ring1][#Branch1][N][C][=Branch1][C][=O][C][C][=N][N][Branch1][C][C][C][=Ring1][=Branch1]
c13c4cccc1Cl.c15cnn(C)c1.C25=O.CO3.N24
COC(=O)CCc1nc(Cn2cnc(C3CCC3)cc2=O)no1
1344209
[C][O][C][=Branch1][C][=O][C][C][C][=N][C][Branch2][Ring1][Ring1][C][N][C][=N][C][Branch1][#Branch1][C][C][C][C][Ring1][Ring2][=C][C][Ring1][#Branch2][=O][=N][O][Ring1][P]
n15cnc8cc1=O.c16nc7no1.C4(=O)CC6.C18CCC1.CO4.C57
CCN(c1ccccc1)S(=O)(=O)c1ccccc1N
1587346
[C][C][N][Branch1][=Branch2][C][=C][C][=C][C][=C][Ring1][=Branch1][S][=Branch1][C][=O][=Branch1][C][=O][C][=C][C][=C][C][=C][Ring1][=Branch1][N]
S3(=O)(=O)c1ccccc1N.c14ccccc1.N234.CC2
CCN(CC)C(=O)CCC(=O)N(C)c1ccc2nc(C)sc2c1
1300963
[C][C][N][Branch1][Ring1][C][C][C][=Branch1][C][=O][C][C][C][=Branch1][C][=O][N][Branch1][C][C][C][=C][C][=C][N][=C][Branch1][C][C][S][C][Ring1][=Branch1][=C][Ring1][#Branch2]
c17ccc2nc(C)sc2c1.C3(=O)CCC4=O.N356.N47C.CC5.C6C
O=C(NC1CCCC2(C1)OCCO2)c1cc(Cl)ccn1
1926097
[O][=C][Branch2][Ring1][C][N][C][C][C][C][C][Branch1][Ring2][C][Ring1][=Branch1][O][C][C][O][Ring1][=Branch1][C][=C][C][Branch1][C][Cl][=C][C][=N][Ring1][#Branch1]
C14CCCC2(C1)OCCO2.c15cc(Cl)ccn1.O=C35.N34
O=C(Cc1noc2ccccc12)NCc1ccncc1
593088
[O][=C][Branch1][#C][C][C][=N][O][C][=C][C][=C][C][=C][Ring1][=Branch2][Ring1][=Branch1][N][C][C][=C][C][=N][C][=C][Ring1][=Branch1]
c15noc2ccccc12.c16ccncc1.O=C3C5.N34.C46
COCCn1nc(-c2ccc(OC)cc2)cc(C(C)=O)c1=O
1244280
[C][O][C][C][N][N][=C][Branch1][=N][C][=C][C][=C][Branch1][Ring1][O][C][C][=C][Ring1][Branch2][C][=C][Branch1][=Branch1][C][Branch1][C][C][=O][C][Ring1][P][=O]
n16nc7cc5c1=O.c17ccc4cc1.C3C6.C5(C)=O.CO3.O4C
OCc1c(-c2ccncc2)nc2sc(-c3ccccc3)nn12
844583
[O][C][C][=C][Branch1][=Branch2][C][=C][C][=N][C][=C][Ring1][=Branch1][N][=C][S][C][Branch1][=Branch2][C][=C][C][=C][C][=C][Ring1][=Branch1][=N][N][Ring2][Ring1][Ring2][Ring1][O]
c14c5nc2sc6nn12.c15ccncc1.c16ccccc1.OC4
CCC1CN(C(=O)c2c(C)nn(C)c2OC)CCC1c1ccccc1
1065496
[C][C][C][C][N][Branch2][Ring1][Ring2][C][=Branch1][C][=O][C][C][Branch1][C][C][=N][N][Branch1][C][C][C][=Ring1][#Branch1][O][C][C][C][C][Ring1][P][C][=C][C][=C][C][=C][Ring1][=Branch1]
C16CN3CCC17.c15c(C)nn(C)c14.c17ccccc1.C35=O.CC6.O4C
CC(C)(C)OC(=O)NCc1ccc(S(N)(=O)=O)cc1
899873
[C][C][Branch1][C][C][Branch1][C][C][O][C][=Branch1][C][=O][N][C][C][=C][C][=C][Branch1][=Branch2][S][Branch1][C][N][=Branch1][C][=O][=O][C][=C][Ring1][#Branch2]
c16ccc(S(N)(=O)=O)cc1.CC4(C)C.C23=O.O24.N35.C56
CCOc1ccc2nc(C(=O)N(C)Cc3ccccc3)cn2n1
1573661
[C][C][O][C][C][=C][C][=N][C][Branch2][Ring1][C][C][=Branch1][C][=O][N][Branch1][C][C][C][C][=C][C][=C][C][=C][Ring1][=Branch1][=C][N][Ring1][S][N][=Ring2][Ring1][Ring2]
c16ccc2nc8cn2n1.c19ccccc1.C48=O.N47C.CC5.O56.C79
CC(C)COCCC(=O)Nc1ccccc1NC(=O)N1CCCC1
811280
[C][C][Branch1][C][C][C][O][C][C][C][=Branch1][C][=O][N][C][=C][C][=C][C][=C][Ring1][=Branch1][N][C][=Branch1][C][=O][N][C][C][C][C][Ring1][Branch1]
c17ccccc18.C6CC2=O.N14CCCC1.CC(C)C5.C34=O.O56.N27.N38
Cc1cc(CN(C)C(=O)NC(C)c2ccc(C#N)cc2)no1
626181
[C][C][=C][C][Branch2][Ring1][O][C][N][Branch1][C][C][C][=Branch1][C][=O][N][C][Branch1][C][C][C][=C][C][=C][Branch1][Ring1][C][#N][C][=C][Ring1][Branch2][=N][O][Ring2][Ring1][Branch1]
c18ccc(C#N)cc1.Cc1cc7no1.N35C.C34=O.C68C.C57.N46
COC(=O)CN(C(=O)c1ccc(NC(=O)C2CC2C)cc1)C(C)C
1564050
[C][O][C][=Branch1][C][=O][C][N][Branch2][Ring1][#Branch2][C][=Branch1][C][=O][C][=C][C][=C][Branch1][N][N][C][=Branch1][C][=O][C][C][C][Ring1][Ring1][C][C][=C][Ring1][=N][C][Branch1][C][C][C]
c1%10ccc8cc1.C3(=O)C6.C19CC1C.N467.C4%10=O.C59=O.C7(C)C.CO3.N58
O=C1NCC2(CCN(CC(=O)c3ccccc3)CC2)O1
1724679
[O][=C][N][C][C][Branch2][Ring1][#Branch1][C][C][N][Branch1][=C][C][C][=Branch1][C][=O][C][=C][C][=C][C][=C][Ring1][=Branch1][C][C][Ring1][#C][O][Ring2][Ring1][Ring1]
O=C1NCC2(CCN4CC2)O1.c15ccccc1.C4C5=O
Cc1cc(C)c(NC(=O)CN(C)C(=O)c2cnc(C)cn2)c(C)c1
167241
[C][C][=C][C][Branch1][C][C][=C][Branch2][Ring1][#Branch2][N][C][=Branch1][C][=O][C][N][Branch1][C][C][C][=Branch1][C][=O][C][=C][N][=C][Branch1][C][C][C][=N][Ring1][#Branch1][C][Branch1][C][C][=C][Ring2][Ring1][#Branch1]
Cc1cc(C)c6c(C)c1.c17cnc(C)cn1.C3(=O)C5.N45C.C47=O.N36
Cc1ccc(OC2CCN(Cc3cnnn3C)CC2)cc1C
1423893
[C][C][=C][C][=C][Branch2][Ring1][Branch1][O][C][C][C][N][Branch1][#Branch2][C][C][=C][N][=N][N][Ring1][Branch1][C][C][C][Ring1][=N][C][=C][Ring2][Ring1][Ring2][C]
Cc1ccc5cc1C.C14CCN6CC1.c17cnnn1C.O45.C67
CCN(Cc1cccs1)C(=O)Cc1csc(-c2ccccn2)n1
1894781
[C][C][N][Branch1][=Branch2][C][C][=C][C][=C][S][Ring1][Branch1][C][=Branch1][C][=O][C][C][=C][S][C][Branch1][=Branch2][C][=C][C][=C][C][=N][Ring1][=Branch1][=N][Ring1][O]
c17csc8n1.c18ccccn1.c16cccs1.C3(=O)C7.N345.CC4.C56
Cc1cc(C)cc(NC(=O)c2cccc(-n3cccn3)n2)c1
1184261
[C][C][=C][C][Branch1][C][C][=C][C][Branch2][Ring1][#Branch1][N][C][=Branch1][C][=O][C][=C][C][=C][C][Branch1][Branch2][N][C][=C][C][=N][Ring1][Branch1][=N][Ring1][O][=C][Ring2][Ring1][Branch1]
Cc1cc5cc(C)c1.c16cccc7n1.n17cccn1.C46=O.N45
COCC(=O)N(Cc1cccs1)CC1CCCO1
1858703
[C][O][C][C][=Branch1][C][=O][N][Branch1][=Branch2][C][C][=C][C][=C][S][Ring1][Branch1][C][C][C][C][C][O][Ring1][Branch1]
c17cccs1.C16CCCO1.C3C2=O.N245.CO3.C47.C56
CC(=O)NCc1ccc(C(=O)COc2ccc(C(N)=O)cc2)s1
827777
[C][C][=Branch1][C][=O][N][C][C][=C][C][=C][Branch2][Ring1][=Branch1][C][=Branch1][C][=O][C][O][C][=C][C][=C][Branch1][=Branch1][C][Branch1][C][N][=O][C][=C][Ring1][=Branch2][S][Ring2][Ring1][C]
c15ccc8cc1.c19ccc7s1.C7(=O)C4.CC3=O.C8(N)=O.N36.C69.O45
CC(=O)c1c(C)[nH]c(C(=O)Nc2ccc3[nH]c(=O)[nH]c3c2)c1C
246280
[C][C][=Branch1][C][=O][C][=C][Branch1][C][C][NH1][C][Branch2][Ring1][=Branch1][C][=Branch1][C][=O][N][C][=C][C][=C][NH1][C][=Branch1][C][=O][NH1][C][Ring1][=Branch1][=C][Ring1][#Branch2][=C][Ring2][Ring1][Ring1][C]
c15ccc2[nH]c(=O)[nH]c2c1.c17c(C)[nH]c6c1C.CC7=O.C46=O.N45
C=CCNC(=O)c1cc2c(n(-c3ccccc3)c1=O)CCCC2=O
64206
[C][=C][C][N][C][=Branch1][C][=O][C][=C][C][=C][Branch1][S][N][Branch1][=Branch2][C][=C][C][=C][C][=C][Ring1][=Branch1][C][Ring1][N][=O][C][C][C][C][Ring1][#C][=O]
c16cc2c(n7c1=O)CCCC2=O.c17ccccc1.C=CC5.C46=O.N45
Cc1ccccc1-n1c(N)cc(=O)n(Cc2ccco2)c1=O
11476
[C][C][=C][C][=C][C][=C][Ring1][=Branch1][N][C][Branch1][C][N][=C][C][=Branch1][C][=O][N][Branch1][=Branch2][C][C][=C][C][=C][O][Ring1][Branch1][C][Ring1][=C][=O]
n15c(N)cc(=O)n3c1=O.Cc1ccccc15.c14ccco1.C34
O=S(=O)(CC1CCCCC1)c1nccn1C1CC1
1160010
[O][=S][=Branch1][C][=O][Branch1][#Branch2][C][C][C][C][C][C][C][Ring1][=Branch1][C][=N][C][=C][N][Ring1][Branch1][C][C][C][Ring1][Ring1]
O=S(=O)(C2)c1nccn13.C12CCCCC1.C13CC1
CNC(=O)c1ccc(CN(C(=O)Cc2ccc(C)s2)C2CC2)cc1
780356
[C][N][C][=Branch1][C][=O][C][=C][C][=C][Branch2][Ring1][=Branch2][C][N][Branch1][S][C][=Branch1][C][=O][C][C][=C][C][=C][Branch1][C][C][S][Ring1][=Branch1][C][C][C][Ring1][Ring1][C][=C][Ring2][Ring1][Ring2]
c17ccc9cc1.c18ccc(C)s1.C4(=O)C8.C37=O.N456.C16CC1.CN3.C59
O=C(CNC(=O)c1cccc(F)c1)NCc1cccc2ccccc12
1933283
[O][=C][Branch2][Ring1][C][C][N][C][=Branch1][C][=O][C][=C][C][=C][C][Branch1][C][F][=C][Ring1][#Branch1][N][C][C][=C][C][=C][C][=C][C][=C][C][=C][Ring1][#Branch2][Ring1][=Branch1]
c18cccc2ccccc12.c17cccc(F)c1.O=C3C5.C47=O.N45.N36.C68
COC(=O)c1ccc(C)c(S(=O)(=O)NCCNC(C)=O)c1
436688
[C][O][C][=Branch1][C][=O][C][=C][C][=C][Branch1][C][C][C][Branch1][P][S][=Branch1][C][=O][=Branch1][C][=O][N][C][C][N][C][Branch1][C][C][=O][=C][Ring1][P]
c17ccc(C)c(S6(=O)=O)c1.C27=O.C4C5.C3(C)=O.CO2.N46.N35
CN(Cc1cn[nH]c1)C(=O)c1cc(-c2ccccc2F)on1
954325
[C][N][Branch1][=Branch2][C][C][C][=N][NH1][C][=Ring1][Branch1][C][=Branch1][C][=O][C][C][=C][Branch1][#Branch2][C][=C][C][=C][C][=C][Ring1][=Branch1][F][O][N][=Ring1][N]
c17ccccc1F.c15cc7on1.c16cn[nH]c1.CN34.C35=O.C46
Cc1c(C)c2ccc(NC(=O)c3c(F)cccc3F)cc2[nH]c1=O
1661712
[C][C][=C][Branch1][C][C][C][=C][C][=C][Branch2][Ring1][C][N][C][=Branch1][C][=O][C][=C][Branch1][C][F][C][=C][C][=C][Ring1][#Branch1][F][C][=C][Ring1][P][NH1][C][Ring2][Ring1][=Branch1][=O]
Cc1c(C)c2ccc5cc2[nH]c1=O.c16c(F)cccc1F.C46=O.N45
CC(C)(C)C1CCC(C(=O)N2CCOCC2)CC1
41705
[C][C][Branch1][C][C][Branch1][C][C][C][C][C][C][Branch1][=N][C][=Branch1][C][=O][N][C][C][O][C][C][Ring1][=Branch1][C][C][Ring1][=C]
C15CCC4CC1.N13CCOCC1.CC5(C)C.C34=O
CC(O)CN(C)C(=O)C(C)Oc1cccc(Cl)c1
728605
[C][C][Branch1][C][O][C][N][Branch1][C][C][C][=Branch1][C][=O][C][Branch1][C][C][O][C][=C][C][=C][C][Branch1][C][Cl][=C][Ring1][#Branch1]
c14cccc(Cl)c1.C2(=O)C3C.CC(O)C5.N25C.O34
N#Cc1ccc(Cn2nc(-c3ccccc3F)ccc2=O)cc1
599065
[N][#C][C][=C][C][=C][Branch2][Ring1][=Branch1][C][N][N][=C][Branch1][#Branch2][C][=C][C][=C][C][=C][Ring1][=Branch1][F][C][=C][C][Ring1][=N][=O][C][=C][Ring2][Ring1][Branch1]
N#Cc1ccc5cc1.n14nc6ccc1=O.c16ccccc1F.C45
NC(=O)c1cccc(CNC(=O)NCCC2CC3CCC2C3)c1
1225679
[N][C][=Branch1][C][=O][C][=C][C][=C][C][Branch2][Ring1][Branch1][C][N][C][=Branch1][C][=O][N][C][C][C][C][C][C][C][C][Ring1][=Branch1][C][Ring1][Branch1][=C][Ring2][Ring1][Ring2]
c18cccc%10c1.C19CC2CCC1C2.NC8=O.C45=O.C7C9.C6%10.N46.N57
Cc1ncc(C(=O)Nc2ccc(F)c(F)c2)c(N)n1
1885948
[C][C][=N][C][=C][Branch2][Ring1][Ring2][C][=Branch1][C][=O][N][C][=C][C][=C][Branch1][C][F][C][Branch1][C][F][=C][Ring1][Branch2][C][Branch1][C][N][=N][Ring2][Ring1][C]
Cc1ncc5c(N)n1.c14ccc(F)c(F)c1.C35=O.N34
Cc1ccc(C(=O)NCCN2CCCCCC2=O)o1
518744
[C][C][=C][C][=C][Branch2][Ring1][C][C][=Branch1][C][=O][N][C][C][N][C][C][C][C][C][C][Ring1][#Branch1][=O][O][Ring2][Ring1][C]
N16CCCCCC1=O.Cc1ccc5o1.C35=O.C4C6.N34
COCCn1nc(C(=O)Nc2cccc(C)n2)ccc1=O
1828011
[C][O][C][C][N][N][=C][Branch1][P][C][=Branch1][C][=O][N][C][=C][C][=C][C][Branch1][C][C][=N][Ring1][#Branch1][C][=C][C][Ring1][S][=O]
n17nc6ccc1=O.c15cccc(C)n1.C4C7.C36=O.CO4.N35
CC(Sc1nnnn1C1CC1)C(=O)N(C)c1ccc(F)c(F)c1
769131
[C][C][Branch1][=C][S][C][=N][N][=N][N][Ring1][Branch1][C][C][C][Ring1][Ring1][C][=Branch1][C][=O][N][Branch1][C][C][C][=C][C][=C][Branch1][C][F][C][Branch1][C][F][=C][Ring1][Branch2]
c14ccc(F)c(F)c1.c16nnnn15.CC3C2=O.C15CC1.N24C.S36
Cc1ccc(CCC(=O)NCCC(=O)Nc2cccc(C)n2)cc1
807994
[C][C][=C][C][=C][Branch2][Ring1][#Branch2][C][C][C][=Branch1][C][=O][N][C][C][C][=Branch1][C][=O][N][C][=C][C][=C][C][Branch1][C][C][=N][Ring1][#Branch1][C][=C][Ring2][Ring1][#Branch1]
Cc1ccc7cc1.c16cccc(C)n1.C7CC3=O.C5CC4=O.N35.N46
COc1ccc(OC)c(C(C)NC(=O)c2c(F)cccc2F)c1
388103
[C][O][C][=C][C][=C][Branch1][Ring1][O][C][C][Branch2][Ring1][=Branch1][C][Branch1][C][C][N][C][=Branch1][C][=O][C][=C][Branch1][C][F][C][=C][C][=C][Ring1][#Branch1][F][=C][Ring2][Ring1][Branch1]
c14ccc5c8c1.c17c(F)cccc1F.C68C.C37=O.CO4.O5C.N36
CC1CN(C(=O)C2CC(=O)N(CCc3ccccc3)C2)CC(C)O1
717370
[C][C][C][N][Branch2][Ring1][O][C][=Branch1][C][=O][C][C][C][=Branch1][C][=O][N][Branch1][O][C][C][C][=C][C][=C][C][=C][Ring1][=Branch1][C][Ring1][=C][C][C][Branch1][C][C][O][Ring2][Ring1][#Branch1]
CC1CN4CC(C)O1.C15CC(=O)N6C1.c17ccccc1.C45=O.C6C7
C=CCCCN(C)C(=O)C1CCN(c2ccc3nncn3n2)CC1
1119603
[C][=C][C][C][C][N][Branch1][C][C][C][=Branch1][C][=O][C][C][C][N][Branch1][=C][C][C][=C][C][=N][N][=C][N][Ring1][Branch1][N][=Ring1][=Branch2][C][C][Ring1][#C]
c16ccc2nncn2n1.C17CCN6CC1.C=CCCC5.N45C.C47=O
Cc1ccc2c(c1)NC(=O)C(C)(C(=O)Nc1ccccc1)O2
1821128
[C][C][=C][C][=C][C][=Branch1][Ring2][=C][Ring1][=Branch1][N][C][=Branch1][C][=O][C][Branch1][C][C][Branch1][=C][C][=Branch1][C][=O][N][C][=C][C][=C][C][=C][Ring1][=Branch1][O][Ring2][Ring1][C]
Cc1ccc2c(c1)NC(=O)C5(C)O2.c14ccccc1.C35=O.N34
COc1cc(CO)ccc1OCCc1cccc(C)c1
554771
[C][O][C][=C][C][Branch1][Ring1][C][O][=C][C][=C][Ring1][Branch2][O][C][C][C][=C][C][=C][C][Branch1][C][C][=C][Ring1][#Branch1]
c13cc5ccc14.c16cccc(C)c1.C2C6.CO3.C5O.O24
O=C(C1CCCN(c2ncnc3c2CCC3)C1)N1CCOCC1
806866
[O][=C][Branch2][Ring1][Branch2][C][C][C][C][N][Branch1][=C][C][=N][C][=N][C][=C][Ring1][=Branch1][C][C][C][Ring1][Branch1][C][Ring1][#C][N][C][C][O][C][C][Ring1][=Branch1]
c15ncnc2c1CCC2.C16CCCN5C1.N14CCOCC1.O=C46
Cc1cnn(CCC(=O)NC(C)c2cccc(C(F)(F)F)c2)c1
1234684
[C][C][C][=N][N][Branch2][Ring1][=C][C][C][C][=Branch1][C][=O][N][C][Branch1][C][C][C][=C][C][=C][C][Branch1][=Branch2][C][Branch1][C][F][Branch1][C][F][F][=C][Ring1][#Branch2][C][=Ring2][Ring1][=Branch1]
c16cccc7c1.Cc1cnn5c1.C5CC3=O.C7(F)(F)F.C46C.N34
CCN(CC)c1nc2sc(C(=O)N(C)C)cc2s1
660430
[C][C][N][Branch1][Ring1][C][C][C][=N][C][S][C][Branch1][#Branch2][C][=Branch1][C][=O][N][Branch1][C][C][C][=C][C][=Ring1][#Branch2][S][Ring1][=N]
c16nc2sc7cc2s1.N456.C37=O.N3(C)C.CC4.C5C
CCC(C)NC(=O)C(NC(=O)Nc1ccccc1)C(C)C
1687772
[C][C][C][Branch1][C][C][N][C][=Branch1][C][=O][C][Branch1][#C][N][C][=Branch1][C][=O][N][C][=C][C][=C][C][=C][Ring1][=Branch1][C][Branch1][C][C][C]
C2(=O)C6C(C)C.c17ccccc1.CCC5C.C34=O.N25.N36.N47
COC(CNC(=O)c1cnc2ccc(C)cn12)C(C)(C)C
1394776
[C][O][C][Branch2][Ring1][#Branch1][C][N][C][=Branch1][C][=O][C][=C][N][=C][C][=C][C][Branch1][C][C][=C][N][Ring1][#Branch2][Ring1][#Branch1][C][Branch1][C][C][Branch1][C][C][C]
c16cnc2ccc(C)cn12.C4(C5)C(C)(C)C.C36=O.CO4.N35
Cc1nn(C)c(C)c1C1CCCN1Cc1nc(-c2cccs2)no1
1078839
[C][C][=N][N][Branch1][C][C][C][Branch1][C][C][=C][Ring1][#Branch1][C][C][C][C][N][Ring1][Branch1][C][C][=N][C][Branch1][Branch2][C][=C][C][=C][S][Ring1][Branch1][=N][O][Ring1][#Branch2]
Cc1nn(C)c(C)c15.C15CCCN13.c14nc6no1.c16cccs1.C34
Cc1nn(-c2ccc(F)cc2)cc1CNC(=O)N1CCNC(=O)C1C
1208023
[C][C][=N][N][Branch1][N][C][=C][C][=C][Branch1][C][F][C][=C][Ring1][#Branch1][C][=C][Ring1][N][C][N][C][=Branch1][C][=O][N][C][C][N][C][=Branch1][C][=O][C][Ring1][#Branch1][C]
N14CCNC(=O)C1C.Cc1nn7cc16.c17ccc(F)cc1.C34=O.C56.N35
Cc1ncn(CC(=O)Nc2cccc(Cl)c2)c(=O)c1C
858485
[C][C][N][=C][N][Branch2][Ring1][C][C][C][=Branch1][C][=O][N][C][=C][C][=C][C][Branch1][C][Cl][=C][Ring1][#Branch1][C][=Branch1][C][=O][C][=Ring2][Ring1][C][C]
Cc1ncn5c(=O)c1C.c14cccc(Cl)c1.C5C3=O.N34
C=CCNC(=O)Nc1ccc(C)cc1OCC(=O)N(C)C
772406
[C][=C][C][N][C][=Branch1][C][=O][N][C][=C][C][=C][Branch1][C][C][C][=C][Ring1][#Branch1][O][C][C][=Branch1][C][=O][N][Branch1][C][C][C]
c18ccc(C)cc16.C5C4=O.C=CC7.C23=O.N4(C)C.N27.N38.O56
Cc1cccc(C(=O)NCC(=O)NCC2CCCO2)c1
1811429
[C][C][=C][C][=C][C][Branch2][Ring1][Ring2][C][=Branch1][C][=O][N][C][C][=Branch1][C][=O][N][C][C][C][C][C][O][Ring1][Branch1][=C][Ring2][Ring1][Ring1]
Cc1cccc7c1.C18CCCO1.C5C4=O.C37=O.N35.N46.C68
O=C(NC1CCN(C(=O)C2CC2(Cl)Cl)CC1)c1ccsc1
1574767
[O][=C][Branch2][Ring1][=Branch2][N][C][C][C][N][Branch1][=C][C][=Branch1][C][=O][C][C][C][Ring1][Ring1][Branch1][C][Cl][Cl][C][C][Ring1][=N][C][C][=C][S][C][=Ring1][Branch1]
C15CCN4CC1.C16CC1(Cl)Cl.c17ccsc1.O=C37.C46=O.N35
O=C(OCc1cccc(F)c1)c1ccc(-n2ccnn2)cc1
1359928
[O][=C][Branch1][=C][O][C][C][=C][C][=C][C][Branch1][C][F][=C][Ring1][#Branch1][C][=C][C][=C][Branch1][Branch2][N][C][=C][N][=N][Ring1][Branch1][C][=C][Ring1][O]
c16cccc(F)c1.c15ccc7cc1.n17ccnn1.O=C35.O34.C46
COCC(C)Nc1ncnc(Nc2cc(Cl)ccc2C)c1N
537799
[C][O][C][C][Branch1][C][C][N][C][=N][C][=N][C][Branch1][=C][N][C][=C][C][Branch1][C][Cl][=C][C][=C][Ring1][#Branch1][C][=C][Ring1][#C][N]
c15ncnc6c1N.c17cc(Cl)ccc1C.C3C4C.CO3.N45.N67
COc1cccc(C(=O)CSc2nnc(C)o2)c1
651609
[C][O][C][=C][C][=C][C][Branch1][P][C][=Branch1][C][=O][C][S][C][=N][N][=C][Branch1][C][C][O][Ring1][=Branch1][=C][Ring1][S]
c13cccc5c1.c16nnc(C)o1.C5(=O)C4.CO3.S46
Cc1ccc2nc(C)c(C)c(C(=O)N(C)Cc3cnc(N)nc3)c2c1
1471762
[C][C][=C][C][=C][N][=C][Branch1][C][C][C][Branch1][C][C][=C][Branch2][Ring1][Branch1][C][=Branch1][C][=O][N][Branch1][C][C][C][C][=C][N][=C][Branch1][C][N][N][=C][Ring1][#Branch1][C][Ring2][Ring1][Ring2][=C][Ring2][Ring1][Branch2]
Cc1ccc2nc(C)c(C)c6c2c1.c17cnc(N)nc1.C46=O.N45C.C57
O=C(c1cc(-n2cnnn2)ccc1O)N1CCOC2CCCCC21
1686057
[O][=C][Branch2][Ring1][Ring1][C][=C][C][Branch1][Branch2][N][C][=N][N][=N][Ring1][Branch1][=C][C][=C][Ring1][O][O][N][C][C][O][C][C][C][C][C][C][Ring1][=Branch1][Ring1][#Branch2]
N13CCOC2CCCCC21.c14cc5ccc1O.n15cnnn1.O=C34
O=C(NCCCN1CCc2ccccc21)N1CCOCC1
1628155
[O][=C][Branch2][Ring1][C][N][C][C][C][N][C][C][C][=C][C][=C][C][=C][Ring1][=Branch1][Ring1][=Branch2][N][C][C][O][C][C][Ring1][=Branch1]
N16CCc2ccccc21.N14CCOCC1.C5CC6.O=C34.N35
Cc1cnc(C(=O)Nc2cccc(C#Cc3cccs3)c2)cn1
245438
[C][C][=C][N][=C][Branch2][Ring1][=Branch2][C][=Branch1][C][=O][N][C][=C][C][=C][C][Branch1][#Branch2][C][#C][C][=C][C][=C][S][Ring1][Branch1][=C][Ring1][=N][C][=N][Ring2][Ring1][=Branch1]
c15cccc(C#Cc2cccs2)c1.Cc1cnc6cn1.C46=O.N45
COc1ccc2c(c1)OCC1=C2CCC2(C)C(=O)CCC=C12
288959
[C][O][C][=C][C][=C][C][=Branch1][Ring2][=C][Ring1][=Branch1][O][C][C][=C][Ring1][#Branch1][C][C][C][Branch1][C][C][C][=Branch1][C][=O][C][C][C][=C][Ring1][N][Ring1][Branch2]
c13ccc2c(c1)OCC1=C2CCC2(C)C(=O)CCC=C12.CO3
CC(Oc1ccccc1Cl)C(=O)Nc1ccn(CC(N)=O)n1
1673853
[C][C][Branch1][O][O][C][=C][C][=C][C][=C][Ring1][=Branch1][Cl][C][=Branch1][C][=O][N][C][C][=C][N][Branch1][#Branch1][C][C][Branch1][C][N][=O][N][=Ring1][=Branch2]
c14ccccc1Cl.c15ccn6n1.CC3C2=O.C6C(N)=O.O34.N25
CC(C)CNC(=O)NCc1cccc(C(=O)NCC2CCCO2)c1
851955
[C][C][Branch1][C][C][C][N][C][=Branch1][C][=O][N][C][C][=C][C][=C][C][Branch1][=C][C][=Branch1][C][=O][N][C][C][C][C][C][O][Ring1][Branch1][=C][Ring1][#C]
c1%11cccc9c1.C1%10CCCO1.CC(C)C6.C34=O.C59=O.N36.N47.C7%11.N58.C8%10
COC(=O)NC1=Nc2ccc(Cl)cc2NS1
49406
[C][O][C][=Branch1][C][=O][N][C][=N][C][=C][C][=C][Branch1][C][Cl][C][=C][Ring1][#Branch1][N][S][Ring1][O]
N4C1=Nc2ccc(Cl)cc2NS1.C34=O.CO3
CNc1ncc(S(=O)(=O)NC2CCCCC2)cc1C
1582424
[C][N][C][=N][C][=C][Branch1][P][S][=Branch1][C][=O][=Branch1][C][=O][N][C][C][C][C][C][C][Ring1][=Branch1][C][=C][Ring1][S][C]
c14ncc(S3(=O)=O)cc1C.C15CCCCC1.CN4.N35
O=C(NCC(=O)N1CCCC1)Nc1cc(Cl)ccc1F
1825213
[O][=C][Branch1][=C][N][C][C][=Branch1][C][=O][N][C][C][C][C][Ring1][Branch1][N][C][=C][C][Branch1][C][Cl][=C][C][=C][Ring1][#Branch1][F]
c16cc(Cl)ccc1F.N14CCCC1.C5C4=O.O=C23.N25.N36
O=C(Nc1cccc(OC(=O)C2CC=CCC2)c1)C1CC1
617587
[O][=C][Branch2][Ring1][=Branch2][N][C][=C][C][=C][C][Branch1][=C][O][C][=Branch1][C][=O][C][C][C][=C][C][C][Ring1][=Branch1][=C][Ring1][#C][C][C][C][Ring1][Ring1]
c16cccc5c1.C18CC=CCC1.O=C47.C38=O.C17CC1.N46.O35
Cc1cccc(NC(=O)Oc2cccc3cccnc23)c1
24980
[C][C][=C][C][=C][C][Branch2][Ring1][Branch1][N][C][=Branch1][C][=O][O][C][=C][C][=C][C][=C][C][=C][N][=C][Ring1][#Branch2][Ring1][=Branch1][=C][Ring2][Ring1][Ring2]
c16cccc2cccnc12.Cc1cccc7c1.C45=O.N57.O46
O=C(CN1CCOCC1)Nc1ccccc1Br
1799781
[O][=C][Branch1][#Branch2][C][N][C][C][O][C][C][Ring1][=Branch1][N][C][=C][C][=C][C][=C][Ring1][=Branch1][Br]
c14ccccc1Br.N13CCOCC1.O=C2C3.N24
CCn1cnnc1CNC(=O)COc1ccc(C(C)(C)C)cc1
625563
[C][C][N][C][=N][N][=C][Ring1][Branch1][C][N][C][=Branch1][C][=O][C][O][C][=C][C][=C][Branch1][=Branch2][C][Branch1][C][C][Branch1][C][C][C][C][=C][Ring1][#Branch2]
c14ccc8cc1.n16cnnc17.C2(=O)C3.C8(C)(C)C.CC6.C57.N25.O34
Cc1cnc(C(=O)Nc2cc(C(C)(C)C)no2)cn1
1640595
[C][C][=C][N][=C][Branch2][Ring1][#Branch1][C][=Branch1][C][=O][N][C][=C][C][Branch1][=Branch2][C][Branch1][C][C][Branch1][C][C][C][=N][O][Ring1][=Branch2][C][=N][Ring2][Ring1][C]
Cc1cnc5cn1.c14cc6no1.C6(C)(C)C.C35=O.N34
CCCC1CN(C(=O)c2cc(C3CC3)nc3c2c(=O)[nH]n3C)CCO1
1732391
[C][C][C][C][C][N][Branch2][Ring1][=N][C][=Branch1][C][=O][C][=C][C][Branch1][=Branch1][C][C][C][Ring1][Ring1][=N][C][=C][Ring1][=Branch2][C][=Branch1][C][=O][NH1][N][Ring1][=Branch1][C][C][C][O][Ring2][Ring1][=Branch1]
c15cc7nc2c1c(=O)[nH]n2C.C16CN4CCO1.CCC6.C45=O.C17CC1
CCC(C)(C)NC(=O)C(C)N1CCN(C(=O)c2ccc(C)cc2)CC1
732943
[C][C][C][Branch1][C][C][Branch1][C][C][N][C][=Branch1][C][=O][C][Branch1][C][C][N][C][C][N][Branch1][S][C][=Branch1][C][=O][C][=C][C][=C][Branch1][C][C][C][=C][Ring1][#Branch1][C][C][Ring1][#C]
N16CCN4CC1.c17ccc(C)cc1.CCC5(C)C.C3(=O)C6C.C47=O.N35
O=C(Nc1ccccc1C(=O)OCC1CCCO1)c1ccco1
374494
[O][=C][Branch2][Ring1][#Branch1][N][C][=C][C][=C][C][=C][Ring1][=Branch1][C][=Branch1][C][=O][O][C][C][C][C][C][O][Ring1][Branch1][C][=C][C][=C][O][Ring1][Branch1]
c15ccccc17.C18CCCO1.c16ccco1.O=C36.C27=O.N35.O24.C48
CCNC(=O)C(C)NC(=O)c1cc(N)ccc1F
483165
[C][C][N][C][=Branch1][C][=O][C][Branch1][C][C][N][C][=Branch1][C][=O][C][=C][C][Branch1][C][N][=C][C][=C][Ring1][#Branch1][F]
c16cc(N)ccc1F.C2(=O)C5C.C36=O.CC4.N24.N35
Cc1ccc(OCC(=O)Nc2cccc(Oc3cnccn3)c2)cc1
423409
[C][C][=C][C][=C][Branch2][Ring1][O][O][C][C][=Branch1][C][=O][N][C][=C][C][=C][C][Branch1][#Branch2][O][C][=C][N][=C][C][=N][Ring1][=Branch1][=C][Ring1][=N][C][=C][Ring2][Ring1][Branch2]
Cc1ccc7cc1.c19cccc8c1.c16cnccn1.C5C4=O.O57.N49.O68
CCCn1c(C)cc(-c2csc(NC(=O)C3CCCO3)n2)c1C
1687158
[C][C][C][N][C][Branch1][C][C][=C][C][Branch2][Ring1][=Branch1][C][=C][S][C][Branch1][=N][N][C][=Branch1][C][=O][C][C][C][C][O][Ring1][Branch1][=N][Ring1][=N][=C][Ring2][Ring1][Ring1][C]
n17c(C)cc8c1C.c18csc5n1.C16CCCO1.CCC7.C46=O.N45
COC(=O)C(c1ccc(F)cc1)N1CCN(Cc2ccncc2)CC1
1481574
[C][O][C][=Branch1][C][=O][C][Branch1][N][C][=C][C][=C][Branch1][C][F][C][=C][Ring1][#Branch1][N][C][C][N][Branch1][#Branch2][C][C][=C][C][=N][C][=C][Ring1][=Branch1][C][C][Ring1][=N]
c16ccc(F)cc1.N14CCN5CC1.c17ccncc1.C3(=O)C46.CO3.C57
CC(O)c1nc2ccccc2n1CC(O)COc1ccccc1
102305
[C][C][Branch1][C][O][C][=N][C][=C][C][=C][C][=C][Ring1][=Branch1][N][Ring1][=Branch2][C][C][Branch1][C][O][C][O][C][=C][C][=C][C][=C][Ring1][=Branch1]
c16nc2ccccc2n15.c14ccccc1.C5C(O)C3.CC6O.O34
CC(C)n1ccnc1-c1cc(NCc2ccccn2)nc2[nH]ccc12
1696610
[C][C][Branch1][C][C][N][C][=C][N][=C][Ring1][Branch1][C][=C][C][Branch1][O][N][C][C][=C][C][=C][C][=N][Ring1][=Branch1][=N][C][NH1][C][=C][C][Ring1][P][=Ring1][Branch1]
c17cc4nc2[nH]ccc12.n15ccnc17.c16ccccn1.CC5C.N34.C36
CCn1cc2c(n1)C(COC)CN(C(=O)c1cc(C)nn1CC)C2
1929137
[C][C][N][C][=C][C][=Branch1][Ring2][=N][Ring1][Branch1][C][Branch1][Ring2][C][O][C][C][N][Branch1][P][C][=Branch1][C][=O][C][=C][C][Branch1][C][C][=N][N][Ring1][=Branch1][C][C][C][Ring2][Ring1][Ring2]
n16cc2c(n1)C(C4)CN3C2.c15cc(C)nn17.C35=O.CC6.O4C.C7C
Cc1nn(-c2ccccc2)c(C)c1CN(C)C(=O)c1cccs1
1632855
[C][C][=N][N][Branch1][=Branch2][C][=C][C][=C][C][=C][Ring1][=Branch1][C][Branch1][C][C][=C][Ring1][N][C][N][Branch1][C][C][C][=Branch1][C][=O][C][=C][C][=C][S][Ring1][Branch1]
Cc1nn7c(C)c16.c17ccccc1.c15cccs1.N34C.C35=O.C46
CN(C)c1ccc(NC(=O)c2ccc(Cl)cc2F)nc1
693954
[C][N][Branch1][C][C][C][=C][C][=C][Branch2][Ring1][C][N][C][=Branch1][C][=O][C][=C][C][=C][Branch1][C][Cl][C][=C][Ring1][#Branch1][F][N][=C][Ring1][P]
c16ccc(Cl)cc1F.c15ccc4nc1.CN5C.C36=O.N34
CCCn1c(=O)n(Cc2ccco2)c(=O)c2sccc21
1599508
[C][C][C][N][C][=Branch1][C][=O][N][Branch1][=Branch2][C][C][=C][C][=C][O][Ring1][Branch1][C][=Branch1][C][=O][C][S][C][=C][C][=Ring1][Branch1][Ring1][P]
n13c(=O)n4c(=O)c2sccc21.c15ccco1.CCC3.C45
O=C(c1c[nH]c(=O)cn1)N1CCCCC1CCO
496206
[O][=C][Branch1][N][C][=C][NH1][C][=Branch1][C][=O][C][=N][Ring1][#Branch1][N][C][C][C][C][C][Ring1][=Branch1][C][C][O]
c13c[nH]c(=O)cn1.N12CCCCC14.O=C23.C4CO
Cc1cc(C2CCCN(C(=O)Cc3ccc4c(c3)CCO4)C2)n[nH]1
1725680
[C][C][=C][C][Branch2][Ring1][P][C][C][C][C][N][Branch2][Ring1][Branch1][C][=Branch1][C][=O][C][C][=C][C][=C][C][=Branch1][Ring2][=C][Ring1][=Branch1][C][C][O][Ring1][=Branch1][C][Ring2][Ring1][C][=N][NH1][Ring2][Ring1][#Branch1]
c16ccc2c(c1)CCO2.C17CCCN5C1.Cc1cc7n[nH]1.C5(=O)C6
CC(C)C(=O)N1CCCc2cc(C(=O)CN)ccc21
1067007
[C][C][Branch1][C][C][C][=Branch1][C][=O][N][C][C][C][C][=C][C][Branch1][#Branch1][C][=Branch1][C][=O][C][N][=C][C][=C][Ring1][#Branch2][Ring1][=C]
N13CCCc2cc4ccc21.CC(C)C3=O.C4(=O)CN
CC=CCOC(=O)c1cc(S(=O)(=O)NCC)ccc1C
1641896
[C][C][=C][C][O][C][=Branch1][C][=O][C][=C][C][Branch1][O][S][=Branch1][C][=O][=Branch1][C][=O][N][C][C][=C][C][=C][Ring1][N][C]
c16cc(S5(=O)=O)ccc1C.C=7C3.C26=O.CC=7.O23.N45.C4C
Cc1ccccc1OCc1nc(CCCO)cs1
553314
[C][C][=C][C][=C][C][=C][Ring1][=Branch1][O][C][C][=N][C][Branch1][Branch1][C][C][C][O][=C][S][Ring1][=Branch2]
Cc1ccccc13.c14nc5cs1.C5CCO.O23.C24
CCCc1nnc(NC(=O)c2sc(C)cc2OC)s1
1875101
[C][C][C][C][=N][N][=C][Branch2][Ring1][C][N][C][=Branch1][C][=O][C][S][C][Branch1][C][C][=C][C][=Ring1][=Branch1][O][C][S][Ring1][S]
c16sc(C)cc14.c17nnc5s1.CCC7.C36=O.N35.O4C
CCN1CCN(C(=O)Cc2ccc(OC)cc2)CC1
320085
[C][C][N][C][C][N][Branch2][Ring1][C][C][=Branch1][C][=O][C][C][=C][C][=C][Branch1][Ring1][O][C][C][=C][Ring1][Branch2][C][C][Ring1][P]
N15CCN3CC1.c16ccc4cc1.C3(=O)C6.CC5.O4C
Cc1ccccc1C(CC(=O)NCCC(C)C)NC(N)=O
1066780
[C][C][=C][C][=C][C][=C][Ring1][=Branch1][C][Branch1][=C][C][C][=Branch1][C][=O][N][C][C][C][Branch1][C][C][C][N][C][Branch1][C][N][=O]
Cc1ccccc16.C46CC2=O.C5CC(C)C.C3(N)=O.N25.N34
CCOc1ccc(C(=O)Nc2cnc3c(cnn3C(C)C)c2)cc1
240241
[C][C][O][C][=C][C][=C][Branch2][Ring1][#Branch2][C][=Branch1][C][=O][N][C][=C][N][=C][C][Branch1][O][C][=N][N][Ring1][Branch1][C][Branch1][C][C][C][=C][Ring1][N][C][=C][Ring2][Ring1][Branch1]
c17cnc2c(cnn29)c1.c16ccc8cc1.C48=O.C9(C)C.CC5.O56.N47