SMILES
large_stringlengths
17
56
ID
large_stringlengths
1
7
SELFIES
stringlengths
63
275
SAFE
stringlengths
20
78
O=C(CSc1nnnn1-c1cccc(F)c1)N1CCCCC1
26336
[O][=C][Branch2][Ring1][Branch1][C][S][C][=N][N][=N][N][Ring1][Branch1][C][=C][C][=C][C][Branch1][C][F][=C][Ring1][#Branch1][N][C][C][C][C][C][Ring1][=Branch1]
c14cccc(F)c1.c15nnnn14.N12CCCCC1.O=C2C3.S35
COC(=O)N1CCC(NC(=O)Nc2ccc3ccccc3c2)CC1
1581123
[C][O][C][=Branch1][C][=O][N][C][C][C][Branch2][Ring1][Branch1][N][C][=Branch1][C][=O][N][C][=C][C][=C][C][=C][C][=C][C][Ring1][=Branch1][=C][Ring1][#Branch2][C][C][Ring2][Ring1][Ring2]
c18ccc2ccccc2c1.N15CCC9CC1.C45=O.C67=O.CO4.N69.N78
C=CCOc1cccc(NC(=O)c2ccnc(-n3ccnc3)c2)c1
762623
[C][=C][C][O][C][=C][C][=C][C][Branch2][Ring1][#Branch1][N][C][=Branch1][C][=O][C][=C][C][=N][C][Branch1][Branch2][N][C][=C][N][=C][Ring1][Branch1][=C][Ring1][O][=C][Ring2][Ring1][Ring2]
c16cccc7c1.c18ccnc9c1.n19ccnc1.C=CC5.C48=O.O56.N47
CCC1CN(C(=O)CCC2CC2)CCC(=O)N1Cc1ccccc1
1692646
[C][C][C][C][N][Branch1][N][C][=Branch1][C][=O][C][C][C][C][C][Ring1][Ring1][C][C][C][=Branch1][C][=O][N][Ring1][#C][C][C][=C][C][=C][C][=C][Ring1][=Branch1]
C15CN3CCC(=O)N14.c17ccccc1.C3(=O)CC6.C16CC1.CC5.C47
COc1ccc(C(C)NC(=O)c2cccnc2N)cc1
908974
[C][O][C][=C][C][=C][Branch2][Ring1][Ring1][C][Branch1][C][C][N][C][=Branch1][C][=O][C][=C][C][=C][N][=C][Ring1][=Branch1][N][C][=C][Ring2][Ring1][C]
c14ccc7cc1.c16cccnc1N.C57C.C36=O.CO4.N35
Cn1cc(Br)cc1C(=O)Nc1cc(F)ccc1F
1635623
[C][N][C][=C][Branch1][C][Br][C][=C][Ring1][=Branch1][C][=Branch1][C][=O][N][C][=C][C][Branch1][C][F][=C][C][=C][Ring1][#Branch1][F]
c13cc(F)ccc1F.Cn1cc(Br)cc14.C24=O.N23
O=C(Nc1ccc(Cl)cn1)C1CC1(Cl)Cl
1539374
[O][=C][Branch1][=N][N][C][=C][C][=C][Branch1][C][Cl][C][=N][Ring1][#Branch1][C][C][C][Ring1][Ring1][Branch1][C][Cl][Cl]
c13ccc(Cl)cn1.C14CC1(Cl)Cl.O=C24.N23
COC(=O)c1ccccc1S(=O)(=O)Nc1cc(F)ccc1F
132718
[C][O][C][=Branch1][C][=O][C][=C][C][=C][C][=C][Ring1][=Branch1][S][=Branch1][C][=O][=Branch1][C][=O][N][C][=C][C][Branch1][C][F][=C][C][=C][Ring1][#Branch1][F]
c15ccccc1S3(=O)=O.c14cc(F)ccc1F.C25=O.CO2.N34
CCc1nn(CC(=O)N2CCN(CC)CC2)c(=O)c2cccn12
1797732
[C][C][C][=N][N][Branch2][Ring1][C][C][C][=Branch1][C][=O][N][C][C][N][Branch1][Ring1][C][C][C][C][Ring1][Branch2][C][=Branch1][C][=O][C][=C][C][=C][N][Ring2][Ring1][Branch1][Ring1][Branch1]
c16nn5c(=O)c2cccn12.N13CCN4CC1.C5C3=O.CC6.C4C
CSc1cccc(NCc2c[nH]nc2-c2cccs2)c1
1815362
[C][S][C][=C][C][=C][C][Branch1][P][N][C][C][=C][NH1][N][=C][Ring1][Branch1][C][=C][C][=C][S][Ring1][Branch1][=C][Ring2][Ring1][C]
c16cccc4c1.c15c[nH]nc17.c17cccs1.CS6.N34.C35
CCn1cc(C(=O)N2CCCc3cccc(F)c32)cn1
1068836
[C][C][N][C][=C][Branch2][Ring1][=Branch1][C][=Branch1][C][=O][N][C][C][C][C][=C][C][=C][C][Branch1][C][F][=C][Ring1][#Branch1][Ring1][O][C][=N][Ring2][Ring1][C]
N14CCCc2cccc(F)c21.n16cc5cn1.C45=O.CC6
Cc1csc(C2CN(Cc3ccc(C)s3)CCO2)n1
1436578
[C][C][=C][S][C][Branch2][Ring1][=Branch1][C][C][N][Branch1][N][C][C][=C][C][=C][Branch1][C][C][S][Ring1][=Branch1][C][C][O][Ring1][=N][=N][Ring2][Ring1][C]
C16CN4CCO1.Cc1csc6n1.c15ccc(C)s1.C45
CNS(=O)(=O)Cc1ccccc1CNc1ncnc2ccccc12
422775
[C][N][S][=Branch1][C][=O][=Branch1][C][=O][C][C][=C][C][=C][C][=C][Ring1][=Branch1][C][N][C][=N][C][=N][C][=C][C][=C][C][=C][Ring1][#Branch2][Ring1][=Branch1]
c15ncnc2ccccc12.c16ccccc17.S4(=O)(=O)C6.CN4.C37.N35
Cc1ccc(OCCc2nc(C(C)(C)O)cs2)cc1
1250512
[C][C][=C][C][=C][Branch2][Ring1][Branch1][O][C][C][C][=N][C][Branch1][=Branch2][C][Branch1][C][C][Branch1][C][C][O][=C][S][Ring1][=Branch2][C][=C][Ring2][Ring1][C]
Cc1ccc4cc1.c15nc6cs1.C6(C)(C)O.C3C5.O34
O=C(Nc1c(O)cccc1F)c1csc(-c2ccsc2)n1
1348674
[O][=C][Branch1][=C][N][C][=C][Branch1][C][O][C][=C][C][=C][Ring1][#Branch1][F][C][=C][S][C][Branch1][Branch2][C][C][=C][S][C][=Ring1][Branch1][=N][Ring1][#Branch2]
c14c(O)cccc1F.c15csc6n1.c16ccsc1.O=C35.N34
CN(C(=O)c1ccncc1F)c1ccccc1S(C)(=O)=O
1286234
[C][N][Branch1][=C][C][=Branch1][C][=O][C][=C][C][=N][C][=C][Ring1][=Branch1][F][C][=C][C][=C][C][=C][Ring1][=Branch1][S][Branch1][C][C][=Branch1][C][=O][=O]
c13ccccc1S(C)(=O)=O.c14ccncc1F.CN23.C24=O
CCN(C(=O)Cn1cnc2sc(C)cc2c1=O)c1ccccc1
309636
[C][C][N][Branch2][Ring1][#Branch1][C][=Branch1][C][=O][C][N][C][=N][C][S][C][Branch1][C][C][=C][C][=Ring1][=Branch1][C][Ring1][#Branch2][=O][C][=C][C][=C][C][=C][Ring1][=Branch1]
n16cnc2sc(C)cc2c1=O.c15ccccc1.C3(=O)C6.N345.CC4
CCOc1nnc(CNC2CCc3nc(C)nn3C2)s1
956642
[C][C][O][C][=N][N][=C][Branch2][Ring1][Ring1][C][N][C][C][C][C][=N][C][Branch1][C][C][=N][N][Ring1][=Branch1][C][Ring1][#Branch2][S][Ring1][P]
C17CCc2nc(C)nn2C1.c15nnc8s1.CC4.O45.C68.N67
O=C(Cc1c[nH]c2ccccc12)Nc1cc(-c2ccsc2)no1
1085848
[O][=C][Branch1][#C][C][C][=C][NH1][C][=C][C][=C][C][=C][Ring1][=Branch2][Ring1][=Branch1][N][C][=C][C][Branch1][Branch2][C][C][=C][S][C][=Ring1][Branch1][=N][O][Ring1][#Branch2]
c15c[nH]c2ccccc12.c14cc6no1.c16ccsc1.O=C3C5.N34
CC(Oc1ccccc1)C(=O)N1CCC(c2cc(N)on2)CC1
868452
[C][C][Branch1][#Branch2][O][C][=C][C][=C][C][=C][Ring1][=Branch1][C][=Branch1][C][=O][N][C][C][C][Branch1][O][C][C][=C][Branch1][C][N][O][N][=Ring1][=Branch1][C][C][Ring1][N]
N13CCC6CC1.c15ccccc1.c16cc(N)on1.CC4C3=O.O45
Cn1ccc(S(=O)(=O)N2CCN(c3ncccn3)CC2)c1
802155
[C][N][C][=C][C][Branch2][Ring1][#Branch2][S][=Branch1][C][=O][=Branch1][C][=O][N][C][C][N][Branch1][=Branch2][C][=N][C][=C][C][=N][Ring1][=Branch1][C][C][Ring1][N][=C][Ring2][Ring1][Ring2]
Cn1ccc(S4(=O)=O)c1.N14CCN5CC1.c15ncccn1
COn1ccc2oc(=O)c(NC(=O)c3ccccc3)cc2c1=O
45153
[C][O][N][C][=C][C][O][C][=Branch1][C][=O][C][Branch1][=C][N][C][=Branch1][C][=O][C][=C][C][=C][C][=C][Ring1][=Branch1][=C][C][=Ring1][S][C][Ring2][Ring1][Ring2][=O]
COn1ccc2oc(=O)c5cc2c1=O.c16ccccc1.C46=O.N45
NC(=O)c1cc(NC(=O)c2ccncc2)cc(C(N)=O)c1
132166
[N][C][=Branch1][C][=O][C][=C][C][Branch1][=C][N][C][=Branch1][C][=O][C][=C][C][=N][C][=C][Ring1][=Branch1][=C][C][Branch1][=Branch1][C][Branch1][C][N][=O][=C][Ring2][Ring1][C]
c15cc4cc7c1.c16ccncc1.NC5=O.C36=O.C7(N)=O.N34
CC(C)(CNC(=O)NCc1ccc(F)cc1)N1CCOCC1
440136
[C][C][Branch1][C][C][Branch2][Ring1][Ring2][C][N][C][=Branch1][C][=O][N][C][C][=C][C][=C][Branch1][C][F][C][=C][Ring1][#Branch1][N][C][C][O][C][C][Ring1][=Branch1]
c17ccc(F)cc1.N14CCOCC1.CC4(C)C5.C23=O.N25.N36.C67
O=C(CCSc1nn2cnnc2o1)Nc1ccccc1
821213
[O][=C][Branch1][S][C][C][S][C][=N][N][C][=N][N][=C][Ring1][Branch1][O][Ring1][Branch2][N][C][=C][C][=C][C][=C][Ring1][=Branch1]
c16nn2cnnc2o1.c15ccccc1.O=C3CC4.S46.N35
CC1(CNC(=O)NCC(=O)N2CCCCC2)CCCC1
903650
[C][C][Branch2][Ring1][Branch1][C][N][C][=Branch1][C][=O][N][C][C][=Branch1][C][=O][N][C][C][C][C][C][Ring1][=Branch1][C][C][C][C][Ring2][Ring1][Ring1]
CC18CCCC1.N15CCCCC1.C7C5=O.C34=O.C68.N36.N47
CN(Cc1ccc(C2CC(=O)Nc3n[nH]cc32)o1)S(C)(=O)=O
1856450
[C][N][Branch2][Ring1][O][C][C][=C][C][=C][Branch1][P][C][C][C][=Branch1][C][=O][N][C][=N][NH1][C][=C][Ring1][Branch1][Ring1][#Branch2][O][Ring1][#C][S][Branch1][C][C][=Branch1][C][=O][=O]
c16ccc(C2CC(=O)Nc3n[nH]cc32)o1.S5(C)(=O)=O.CN45.C46
O=C(NCc1ccncc1)Nc1cccc(OCC(F)F)n1
1550702
[O][=C][Branch1][O][N][C][C][=C][C][=N][C][=C][Ring1][=Branch1][N][C][=C][C][=C][C][Branch1][Branch2][O][C][C][Branch1][C][F][F][=N][Ring1][O]
c17cccc5n1.c18ccncc1.C4C(F)F.O=C23.N26.C68.N37.O45
CCCC(=O)NCc1cccc(CN2CCCC2=O)c1
1702366
[C][C][C][C][=Branch1][C][=O][N][C][C][=C][C][=C][C][Branch1][#Branch2][C][N][C][C][C][C][Ring1][Branch1][=O][=C][Ring1][=N]
c16cccc7c1.N15CCCC1=O.CCCC3=O.N34.C46.C57
CCS(=O)(=O)N1CCOC2C(Oc3ccccn3)CCC21
1489945
[C][C][S][=Branch1][C][=O][=Branch1][C][=O][N][C][C][O][C][C][Branch1][#Branch2][O][C][=C][C][=C][C][=N][Ring1][=Branch1][C][C][C][Ring1][N][Ring1][S]
N16CCOC2C5CCC21.c14ccccn1.CCS6(=O)=O.O45
CCc1ccsc1C(=O)N1CCCC(CNC(N)=O)C1
664244
[C][C][C][C][=C][S][C][=Ring1][Branch1][C][=Branch1][C][=O][N][C][C][C][C][Branch1][Branch2][C][N][C][Branch1][C][N][=O][C][Ring1][O]
N12CCCC6C1.c17ccsc15.C25=O.C3(N)=O.CC7.C46.N34
CN(CC(=O)NCC(=O)N1CCCC1)c1ccc2ccccc2c1
1717901
[C][N][Branch2][Ring1][Ring1][C][C][=Branch1][C][=O][N][C][C][=Branch1][C][=O][N][C][C][C][C][Ring1][Branch1][C][=C][C][=C][C][=C][C][=C][C][Ring1][=Branch1][=C][Ring1][#Branch2]
c17ccc2ccccc2c1.N14CCCC1.C5C3=O.C6C4=O.CN57.N36
CCOC(=O)CN(C(=O)Nc1ccc(F)cc1)C(C)C
1640032
[C][C][O][C][=Branch1][C][=O][C][N][Branch1][P][C][=Branch1][C][=O][N][C][=C][C][=C][Branch1][C][F][C][=C][Ring1][#Branch1][C][Branch1][C][C][C]
c18ccc(F)cc1.C2(=O)C6.N367.C34=O.C7(C)C.CC5.O25.N48
CCOC(=O)c1sc(NC(=O)c2ccccc2O)nc1C
123494
[C][C][O][C][=Branch1][C][=O][C][S][C][Branch1][#C][N][C][=Branch1][C][=O][C][=C][C][=C][C][=C][Ring1][=Branch1][O][=N][C][=Ring1][#C][C]
c17sc6nc1C.c18ccccc1O.C37=O.C48=O.CC5.O35.N46
CN(Cc1cc(-c2ccncc2)no1)c1nnc(C2CCC2)o1
1453825
[C][N][Branch2][Ring1][Ring1][C][C][=C][C][Branch1][=Branch2][C][=C][C][=N][C][=C][Ring1][=Branch1][=N][O][Ring1][O][C][=N][N][=C][Branch1][#Branch1][C][C][C][C][Ring1][Ring2][O][Ring1][=Branch2]
c15cc7no1.c17ccncc1.c14nnc6o1.C16CCC1.CN34.C35
O=C(Nc1cccc2c1OCCO2)C1CCCN1C(=O)c1ccco1
1235392
[O][=C][Branch1][S][N][C][=C][C][=C][C][=C][Ring1][=Branch1][O][C][C][O][Ring1][=Branch1][C][C][C][C][N][Ring1][Branch1][C][=Branch1][C][=O][C][=C][C][=C][O][Ring1][Branch1]
c15cccc2c1OCCO2.C16CCCN14.c17ccco1.O=C36.C47=O.N35
CCc1cccc(CC)c1NC(=O)C1CC(=O)N(C2CCCC2)C1
1620843
[C][C][C][=C][C][=C][C][Branch1][Ring1][C][C][=C][Ring1][Branch2][N][C][=Branch1][C][=O][C][C][C][=Branch1][C][=O][N][Branch1][Branch2][C][C][C][C][C][Ring1][Branch1][C][Ring1][O]
c16cccc7c14.C15CC(=O)N8C1.C18CCCC1.C35=O.CC6.C7C.N34
CC(C)CN1CC(C(=O)N2Cc3cnn(CCO)c3C2)CC1=O
910892
[C][C][Branch1][C][C][C][N][C][C][Branch2][Ring1][=Branch1][C][=Branch1][C][=O][N][C][C][C][=N][N][Branch1][Ring2][C][C][O][C][=Ring1][Branch2][C][Ring1][O][C][C][Ring2][Ring1][C][=O]
N14Cc2cnn6c2C1.N17CC5CC1=O.CC(C)C7.C45=O.C6CO
CNC(=O)C1CCCN1S(=O)(=O)c1ccc2ccccc2c1
159384
[C][N][C][=Branch1][C][=O][C][C][C][C][N][Ring1][Branch1][S][=Branch1][C][=O][=Branch1][C][=O][C][=C][C][=C][C][=C][C][=C][C][Ring1][=Branch1][=C][Ring1][#Branch2]
S4(=O)(=O)c1ccc2ccccc2c1.C15CCCN14.C35=O.CN3
Cc1nn(C)c(C)c1C(=O)NC(C)c1cccc2ccccc12
247688
[C][C][=N][N][Branch1][C][C][C][Branch1][C][C][=C][Ring1][#Branch1][C][=Branch1][C][=O][N][C][Branch1][C][C][C][=C][C][=C][C][=C][C][=C][C][=C][Ring1][#Branch2][Ring1][=Branch1]
c16cccc2ccccc12.Cc1nn(C)c(C)c15.C35=O.C46C.N34
CCCCCN(Cc1ccc(F)cc1)C(=O)c1ccc(=O)n(C)n1
825591
[C][C][C][C][C][N][Branch1][=N][C][C][=C][C][=C][Branch1][C][F][C][=C][Ring1][#Branch1][C][=Branch1][C][=O][C][C][=C][C][=Branch1][C][=O][N][Branch1][C][C][N][=Ring1][Branch2]
c15ccc(=O)n(C)n1.c16ccc(F)cc1.CCCCC3.N234.C25=O.C46
Cc1nc(CCNC(=O)c2c[nH]nc2-c2ccccc2Cl)cs1
1903227
[C][C][=N][C][Branch2][Ring1][Branch2][C][C][N][C][=Branch1][C][=O][C][=C][NH1][N][=C][Ring1][Branch1][C][=C][C][=C][C][=C][Ring1][=Branch1][Cl][=C][S][Ring2][Ring1][=Branch1]
c17ccccc1Cl.Cc1nc6cs1.c15c[nH]nc17.C6C4.C35=O.N34
Cc1cccc(CNC(=O)c2cccc(N)c2)c1C
1262113
[C][C][=C][C][=C][C][Branch2][Ring1][C][C][N][C][=Branch1][C][=O][C][=C][C][=C][C][Branch1][C][N][=C][Ring1][#Branch1][=C][Ring1][P][C]
Cc1cccc6c1C.c15cccc(N)c1.C35=O.C46.N34
CCCc1cc(NCC2CCc3nnc(CC)n3C2)n2ncnc2n1
941772
[C][C][C][C][C][=C][Branch2][Ring1][Ring2][N][C][C][C][C][C][=N][N][=C][Branch1][Ring1][C][C][N][Ring1][#Branch1][C][Ring1][O][N][N][=C][N][=C][Ring1][Branch1][N][=Ring2][Ring1][=Branch1]
c16cc5n2ncnc2n1.C18CCc2nnc7n2C1.CCC6.N45.C48.C7C
Cc1ccc(C)c(NC(=O)C(C)n2nnc(C(N)=O)c2C)c1
840304
[C][C][=C][C][=C][Branch1][C][C][C][Branch2][Ring1][=Branch2][N][C][=Branch1][C][=O][C][Branch1][C][C][N][N][=N][C][Branch1][=Branch1][C][Branch1][C][N][=O][=C][Ring1][Branch2][C][=C][Ring2][Ring1][Branch1]
Cc1ccc(C)c4c1.n16nnc5c1C.C3(=O)C6C.C5(N)=O.N34
Cc1cccc(OC(=O)c2sccc2-n2cnnn2)c1
576788
[C][C][=C][C][=C][C][Branch2][Ring1][Ring2][O][C][=Branch1][C][=O][C][S][C][=C][C][=Ring1][Branch1][N][C][=N][N][=N][Ring1][Branch1][=C][Ring2][Ring1][Ring1]
Cc1cccc4c1.c15sccc16.n16cnnn1.C35=O.O34
COCCn1cc(CCC(=O)Nc2ccn(C)n2)c2ccccc21
1896138
[C][O][C][C][N][C][=C][Branch2][Ring1][C][C][C][C][=Branch1][C][=O][N][C][C][=C][N][Branch1][C][C][N][=Ring1][=Branch1][C][=C][C][=C][C][=C][Ring1][=Branch1][Ring2][Ring1][Ring2]
n16cc7c2ccccc21.c15ccn(C)n1.C7CC3=O.C4C6.CO4.N35
O=C(Nc1ccc(OCC2CCOC2)cc1)c1ccc2nccn2c1
1079699
[O][=C][Branch2][Ring1][Branch1][N][C][=C][C][=C][Branch1][#Branch2][O][C][C][C][C][O][C][Ring1][Branch1][C][=C][Ring1][=N][C][C][=C][C][=N][C][=C][N][Ring1][Branch1][C][=Ring1][=Branch2]
c17ccc2nccn2c1.c16ccc5cc1.C18CCOC1.O=C37.N36.O45.C48
CN(Cc1ccc2c(c1)OCCO2)C(=O)c1ccc(Cl)cc1
361921
[C][N][Branch2][Ring1][C][C][C][=C][C][=C][C][=Branch1][Ring2][=C][Ring1][=Branch1][O][C][C][O][Ring1][#Branch1][C][=Branch1][C][=O][C][=C][C][=C][Branch1][C][Cl][C][=C][Ring1][#Branch1]
c16ccc2c(c1)OCCO2.c15ccc(Cl)cc1.CN34.C35=O.C46
CC(NC(=O)c1ccc(S(C)(=O)=O)cc1)c1nnc2ccccn12
733071
[C][C][Branch2][Ring1][Branch2][N][C][=Branch1][C][=O][C][=C][C][=C][Branch1][=Branch2][S][Branch1][C][C][=Branch1][C][=O][=O][C][=C][Ring1][#Branch2][C][=N][N][=C][C][=C][C][=C][N][Ring1][=Branch2][Ring1][=Branch1]
c15ccc(S(C)(=O)=O)cc1.c16nnc2ccccn12.CC46.C35=O.N34
CC(NC(=O)c1ccco1)C(=O)NC(C)c1ccc2c(c1)OCO2
264260
[C][C][Branch1][=N][N][C][=Branch1][C][=O][C][=C][C][=C][O][Ring1][Branch1][C][=Branch1][C][=O][N][C][Branch1][C][C][C][=C][C][=C][C][=Branch1][Ring2][=C][Ring1][=Branch1][O][C][O][Ring1][=Branch1]
c18ccc2c(c1)OCO2.CC5C4=O.c17ccco1.C37=O.C68C.N35.N46
CC(C)(C)C(=O)N1CCC(C(=O)OCc2ccccc2C#N)CC1
150280
[C][C][Branch1][C][C][Branch1][C][C][C][=Branch1][C][=O][N][C][C][C][Branch1][P][C][=Branch1][C][=O][O][C][C][=C][C][=C][C][=C][Ring1][=Branch1][C][#N][C][C][Ring2][Ring1][C]
c17ccccc1C#N.N14CCC6CC1.CC(C)(C)C4=O.C36=O.O35.C57
Cc1ccn(CC(=O)c2cc(C)n(CCC(C)C)c2C)c(=O)c1
1195977
[C][C][C][=C][N][Branch2][Ring1][#Branch2][C][C][=Branch1][C][=O][C][C][=C][Branch1][C][C][N][Branch1][Branch2][C][C][C][Branch1][C][C][C][C][=Ring1][O][C][C][=Branch1][C][=O][C][=Ring2][Ring1][=Branch1]
Cc1ccn4c(=O)c1.c13cc(C)n5c1C.C5CC(C)C.C4C3=O
Cc1ccn2cc(C(=O)Nc3ccc(NS(C)(=O)=O)cc3)nc2c1
211450
[C][C][C][=C][N][C][=C][Branch2][Ring1][=Branch2][C][=Branch1][C][=O][N][C][=C][C][=C][Branch1][#Branch2][N][S][Branch1][C][C][=Branch1][C][=O][=O][C][=C][Ring1][O][N][=C][Ring2][Ring1][Ring1][C][=Ring2][Ring1][#Branch1]
Cc1ccn2cc8nc2c1.c16ccc7cc1.S5(C)(=O)=O.C48=O.N46.N57
CCCN1C(=O)CCc2cc(NC(=O)c3ccsc3)ccc21
1088319
[C][C][C][N][C][=Branch1][C][=O][C][C][C][=C][C][Branch1][=N][N][C][=Branch1][C][=O][C][C][=C][S][C][=Ring1][Branch1][=C][C][=C][Ring1][=C][Ring2][Ring1][Ring1]
CCCN1C(=O)CCc2cc5ccc21.c16ccsc1.C46=O.N45
CC(C(=O)Nc1cc(S(=O)(=O)N(C)C)ccc1F)n1cccn1
1079893
[C][C][Branch2][Ring1][=N][C][=Branch1][C][=O][N][C][=C][C][Branch1][=N][S][=Branch1][C][=O][=Branch1][C][=O][N][Branch1][C][C][C][=C][C][=C][Ring1][N][F][N][C][=C][C][=N][Ring1][Branch1]
c14cc(S3(=O)=O)ccc1F.CC5C2=O.n15cccn1.N3(C)C.N24
Cc1ccc(CC(=O)NCC(O)c2ccc(Cl)cc2Cl)cn1
995016
[C][C][=C][C][=C][Branch2][Ring1][Branch2][C][C][=Branch1][C][=O][N][C][C][Branch1][C][O][C][=C][C][=C][Branch1][C][Cl][C][=C][Ring1][#Branch1][Cl][C][=N][Ring2][Ring1][Branch1]
c16ccc(Cl)cc1Cl.Cc1ccc5cn1.C5C3=O.C4C6O.N34
CC(C)Oc1ccc(CCNC(=O)Nc2ccnn2C(C)C)cc1
584423
[C][C][Branch1][C][C][O][C][=C][C][=C][Branch2][Ring1][Branch1][C][C][N][C][=Branch1][C][=O][N][C][=C][C][=N][N][Ring1][Branch1][C][Branch1][C][C][C][C][=C][Ring2][Ring1][Ring2]
c16ccc%10cc1.c18ccnn19.CC5C.C%10C7.C34=O.C9(C)C.O56.N37.N48
CCOCC(=O)Nc1nc(-c2c[nH]c(C(=O)OC)c2)cs1
1059172
[C][C][O][C][C][=Branch1][C][=O][N][C][=N][C][Branch1][S][C][=C][NH1][C][Branch1][#Branch1][C][=Branch1][C][=O][O][C][=C][Ring1][=Branch2][=C][S][Ring1][=C]
c17nc9cs1.c19c[nH]c8c1.C6C4=O.C38=O.CC5.O56.N47.O3C
CCC(C)(C)NS(=O)(=O)c1ccc(S(=O)(=O)NC)cc1
591540
[C][C][C][Branch1][C][C][Branch1][C][C][N][S][=Branch1][C][=O][=Branch1][C][=O][C][=C][C][=C][Branch1][#Branch2][S][=Branch1][C][=O][=Branch1][C][=O][N][C][C][=C][Ring1][O]
S3(=O)(=O)c1ccc(S4(=O)=O)cc1.CCC2(C)C.N23.N4C
CNc1snc(C)c1C(=O)Nc1ccc2nc(C)oc2c1
1218396
[C][N][C][S][N][=C][Branch1][C][C][C][=Ring1][=Branch1][C][=Branch1][C][=O][N][C][=C][C][=C][N][=C][Branch1][C][C][O][C][Ring1][=Branch1][=C][Ring1][#Branch2]
c15ccc2nc(C)oc2c1.c14snc(C)c16.C36=O.CN4.N35
COc1ccc(OC)c(-n2cnnc2CN2CCOCC2)c1
918008
[C][O][C][=C][C][=C][Branch1][Ring1][O][C][C][Branch1][P][N][C][=N][N][=C][Ring1][Branch1][C][N][C][C][O][C][C][Ring1][=Branch1][=C][Ring2][Ring1][Ring2]
c13ccc4c7c1.n17cnnc16.N15CCOCC1.CO3.O4C.C56
CCN(CCO)S(=O)(=O)c1ccc(C(F)(F)F)cc1
496536
[C][C][N][Branch1][Ring2][C][C][O][S][=Branch1][C][=O][=Branch1][C][=O][C][=C][C][=C][Branch1][=Branch2][C][Branch1][C][F][Branch1][C][F][F][C][=C][Ring1][#Branch2]
S4(=O)(=O)c1ccc5cc1.C5(F)(F)F.N234.C3CO.CC2
COCCCCNS(=O)(=O)c1ccnc(N)c1
721400
[C][O][C][C][C][C][N][S][=Branch1][C][=O][=Branch1][C][=O][C][=C][C][=N][C][Branch1][C][N][=C][Ring1][#Branch1]
S4(=O)(=O)c1ccnc(N)c1.C2CCC3.CO2.N34
COc1cc(-c2cc(OC)c3c(C)oc(C)c3c(=O)c2)ccc1O
6747
[C][O][C][=C][C][Branch2][Ring1][N][C][C][=C][Branch1][Ring1][O][C][C][=C][Branch1][C][C][O][C][Branch1][C][C][=C][Ring1][#Branch1][C][=Branch1][C][=O][C][=Ring1][#C][=C][C][=C][Ring2][Ring1][Branch1][O]
c16cc5c2c(C)oc(C)c2c(=O)c1.c14cc6ccc1O.CO4.O5C
CC1(NS(=O)(=O)c2ccc(F)cc2)Cc2ccccc2C1
1743472
[C][C][Branch2][Ring1][Ring2][N][S][=Branch1][C][=O][=Branch1][C][=O][C][=C][C][=C][Branch1][C][F][C][=C][Ring1][#Branch1][C][C][=C][C][=C][C][=C][Ring1][=Branch1][C][Ring2][Ring1][Ring2]
CC13Cc2ccccc2C1.S4(=O)(=O)c1ccc(F)cc1.N34
CC(=O)NCCNC(=O)Cc1cccc(OCC#N)c1
1338560
[C][C][=Branch1][C][=O][N][C][C][N][C][=Branch1][C][=O][C][C][=C][C][=C][C][Branch1][Branch1][O][C][C][#N][=C][Ring1][#Branch2]
c18cccc5c1.C3(=O)C8.CC2=O.C6C7.C4C#N.N26.N37.O45
CC(=O)c1c(C)[nH]c(C(=O)Nc2ccc(C(F)(F)F)cc2)c1C
250676
[C][C][=Branch1][C][=O][C][=C][Branch1][C][C][NH1][C][Branch2][Ring1][Branch2][C][=Branch1][C][=O][N][C][=C][C][=C][Branch1][=Branch2][C][Branch1][C][F][Branch1][C][F][F][C][=C][Ring1][#Branch2][=C][Ring2][Ring1][Ring1][C]
c16c(C)[nH]c5c1C.c14ccc7cc1.C7(F)(F)F.CC6=O.C35=O.N34
COc1cccc(CC(=O)NCCc2n[nH]c(-c3ccccc3)n2)c1
1636116
[C][O][C][=C][C][=C][C][Branch2][Ring1][#Branch2][C][C][=Branch1][C][=O][N][C][C][C][=N][NH1][C][Branch1][=Branch2][C][=C][C][=C][C][=C][Ring1][=Branch1][=N][Ring1][O][=C][Ring2][Ring1][#Branch1]
c15cccc8c1.c17n[nH]c9n1.c19ccccc1.C8C4=O.C6C7.CO5.N46
O=C(CCc1ccccc1O)N1CCN(C(=O)N2CCCCC2)CC1
1802589
[O][=C][Branch1][N][C][C][C][=C][C][=C][C][=C][Ring1][=Branch1][O][N][C][C][N][Branch1][=N][C][=Branch1][C][=O][N][C][C][C][C][C][Ring1][=Branch1][C][C][Ring1][=C]
c16ccccc1O.N13CCN4CC1.N15CCCCC1.O=C3CC6.C45=O
Cc1ccc(NC(=O)COC(=O)CC2C=CCC2)cc1C
148326
[C][C][=C][C][=C][Branch2][Ring1][Ring2][N][C][=Branch1][C][=O][C][O][C][=Branch1][C][=O][C][C][C][=C][C][C][Ring1][Branch1][C][=C][Ring2][Ring1][Ring1][C]
Cc1ccc6cc1C.C17C=CCC1.C4(=O)C5.C3(=O)C7.N46.O35
CC(=O)N1CCc2cc(CNC(=O)Nc3cc(F)ccc3F)ccc21
864700
[C][C][=Branch1][C][=O][N][C][C][C][=C][C][Branch2][Ring1][Ring2][C][N][C][=Branch1][C][=O][N][C][=C][C][Branch1][C][F][=C][C][=C][Ring1][#Branch1][F][=C][C][=C][Ring2][Ring1][Ring1][Ring2][Ring1][=Branch1]
N14CCc2cc9ccc21.c18cc(F)ccc1F.CC4=O.C56=O.C79.N57.N68
COc1ccc(CC(=O)N(C)Cc2nc3ccccc3s2)cc1
114552
[C][O][C][=C][C][=C][Branch2][Ring1][Branch2][C][C][=Branch1][C][=O][N][Branch1][C][C][C][C][=N][C][=C][C][=C][C][=C][Ring1][=Branch1][S][Ring1][=Branch2][C][=C][Ring2][Ring1][Branch1]
c17nc2ccccc2s1.c15ccc8cc1.C8C4=O.N46C.CO5.C67
CC(C)(C)c1cnc(Cn2c(S(C)(=O)=O)nc3ccccc32)o1
943749
[C][C][Branch1][C][C][Branch1][C][C][C][=C][N][=C][Branch2][Ring1][=Branch2][C][N][C][Branch1][=Branch2][S][Branch1][C][C][=Branch1][C][=O][=O][=N][C][=C][C][=C][C][=C][Ring1][=Branch1][Ring1][=N][O][Ring2][Ring1][Ring1]
n14c(S(C)(=O)=O)nc2ccccc21.c15cnc6o1.CC5(C)C.C46
COc1ccc(C2CC(=O)NC3=C2C(=O)OC3(C)C)cc1OC(C)C
1023928
[C][O][C][=C][C][=C][Branch2][Ring1][Branch2][C][C][C][=Branch1][C][=O][N][C][=C][Ring1][#Branch1][C][=Branch1][C][=O][O][C][Ring1][=Branch1][Branch1][C][C][C][C][=C][Ring2][Ring1][Ring1][O][C][Branch1][C][C][C]
C17CC(=O)NC2=C1C(=O)OC2(C)C.c15ccc7cc16.C4(C)C.CO5.O46
CCc1nnc(NC(=O)CCn2c(=O)n(CC)c3ccccc32)s1
206360
[C][C][C][=N][N][=C][Branch2][Ring1][N][N][C][=Branch1][C][=O][C][C][N][C][=Branch1][C][=O][N][Branch1][Ring1][C][C][C][=C][C][=C][C][=C][Ring1][=Branch1][Ring1][N][S][Ring2][Ring1][=Branch1]
n16c(=O)n7c2ccccc21.c18nnc5s1.C4(=O)CC6.CC8.N45.C7C
C=CCOC(=O)c1nnc2c(-c3ccc(F)cc3)c(C)nn2c1C
335434
[C][=C][C][O][C][=Branch1][C][=O][C][N][=N][C][=C][Branch1][N][C][=C][C][=C][Branch1][C][F][C][=C][Ring1][#Branch1][C][Branch1][C][C][=N][N][Ring1][=N][C][=Ring1][P][C]
c16nnc2c7c(C)nn2c1C.c17ccc(F)cc1.C=CC5.C46=O.O45
CCOC(=O)C1CCCN(C(=O)c2cccc(F)c2N)C1
1251903
[C][C][O][C][=Branch1][C][=O][C][C][C][C][N][Branch1][P][C][=Branch1][C][=O][C][=C][C][=C][C][Branch1][C][F][=C][Ring1][#Branch1][N][C][Ring1][S]
c17cccc(F)c1N.C16CCCN4C1.C36=O.C47=O.CC5.O35
Cc1cccc(C2(C(=O)Nc3cnn(CC(N)=O)c3)CCCC2)c1
931297
[C][C][=C][C][=C][C][Branch2][Ring1][#C][C][Branch2][Ring1][Branch1][C][=Branch1][C][=O][N][C][C][=N][N][Branch1][#Branch1][C][C][Branch1][C][N][=O][C][=Ring1][=Branch2][C][C][C][C][Ring1][P][=C][Ring2][Ring1][#Branch1]
Cc1cccc8c1.C168CCCC1.c15cnn7c1.C7C(N)=O.C46=O.N45
Cc1noc(C)c1CC(=O)N1CCCc2c(F)cc(F)cc21
563562
[C][C][=N][O][C][Branch1][C][C][=C][Ring1][=Branch1][C][C][=Branch1][C][=O][N][C][C][C][C][=C][Branch1][C][F][C][=C][Branch1][C][F][C][=C][Ring1][Branch2][Ring1][N]
N13CCCc2c(F)cc(F)cc21.Cc1noc(C)c14.C4C3=O
CCN1C(=O)CCc2cc(NC(=O)c3cccc(C)c3)ccc21
294571
[C][C][N][C][=Branch1][C][=O][C][C][C][=C][C][Branch1][P][N][C][=Branch1][C][=O][C][=C][C][=C][C][Branch1][C][C][=C][Ring1][#Branch1][=C][C][=C][Ring1][S][Ring2][Ring1][Branch1]
CCN1C(=O)CCc2cc5ccc21.c16cccc(C)c1.C46=O.N45
N#Cc1ccccc1NC(=O)Cn1nc2ccccn2c1=O
327563
[N][#C][C][=C][C][=C][C][=C][Ring1][=Branch1][N][C][=Branch1][C][=O][C][N][N][=C][C][=C][C][=C][N][Ring1][=Branch1][C][Ring1][=Branch2][=O]
n15nc2ccccn2c1=O.N#Cc1ccccc14.C3(=O)C5.N34
CCS(=O)(=O)N1CCc2c(nnn2CC2CC2)C1COC
1493069
[C][C][S][=Branch1][C][=O][=Branch1][C][=O][N][C][C][C][=C][Branch1][N][N][=N][N][Ring1][Branch1][C][C][C][C][Ring1][Ring1][C][Ring1][=N][C][O][C]
N14CCc2c(nnn25)C1C3.CCS4(=O)=O.C16CC1.C56.O3C
NS(=O)(=O)C1CCN(C(=O)NCc2ccc3c(c2)OCO3)C1
1922560
[N][S][=Branch1][C][=O][=Branch1][C][=O][C][C][C][N][Branch2][Ring1][=Branch1][C][=Branch1][C][=O][N][C][C][=C][C][=C][C][=Branch1][Ring2][=C][Ring1][=Branch1][O][C][O][Ring1][=Branch1][C][Ring2][Ring1][C]
NS(=O)(=O)C1CCN4C1.c17ccc2c(c1)OCO2.C45=O.N56.C67
CS(=O)(=O)N1CCCC1C(=O)NCC(F)(F)F
564121
[C][S][=Branch1][C][=O][=Branch1][C][=O][N][C][C][C][C][Ring1][Branch1][C][=Branch1][C][=O][N][C][C][Branch1][C][F][Branch1][C][F][F]
N14CCCC15.C3C(F)(F)F.CS4(=O)=O.C25=O.N23
Cc1cc(Oc2ccccc2)nc(C2CCCN(C(=O)C3CC3)C2)n1
1873371
[C][C][=C][C][Branch1][#Branch2][O][C][=C][C][=C][C][=C][Ring1][=Branch1][=N][C][Branch2][Ring1][Ring2][C][C][C][C][N][Branch1][#Branch2][C][=Branch1][C][=O][C][C][C][Ring1][Ring1][C][Ring1][O][=N][Ring2][Ring1][Branch2]
Cc1cc5nc8n1.C18CCCN4C1.c16ccccc1.C47=O.C17CC1.O56
CNC(=O)CCCC(O)c1ccc2c(c1)OCCO2
705801
[C][N][C][=Branch1][C][=O][C][C][C][C][Branch1][C][O][C][=C][C][=C][C][=Branch1][Ring2][=C][Ring1][=Branch1][O][C][C][O][Ring1][#Branch1]
c14ccc2c(c1)OCCO2.C3(=O)CCCC4O.CN3
CC12CN(C(=O)c3ccc(F)cc3)C3(C#N)CC1CCC23C
35390
[C][C][C][N][Branch1][S][C][=Branch1][C][=O][C][=C][C][=C][Branch1][C][F][C][=C][Ring1][#Branch1][C][Branch1][Ring1][C][#N][C][C][Ring1][P][C][C][C][Ring2][Ring1][Ring2][Ring1][Branch2][C]
CC12CN4C3(C#N)CC1CCC23C.c15ccc(F)cc1.C45=O
Cc1noc(C)c1CC(C)C(=O)NC1CC1c1cccc(Cl)c1
1708622
[C][C][=N][O][C][Branch1][C][C][=C][Ring1][=Branch1][C][C][Branch1][C][C][C][=Branch1][C][=O][N][C][C][C][Ring1][Ring1][C][=C][C][=C][C][Branch1][C][Cl][=C][Ring1][#Branch1]
Cc1noc(C)c14.c15cccc(Cl)c1.C4C(C)C2=O.C13CC15.N23
O=C(NCCc1ccccc1)C1CCCN(C(=O)N2CCCC2)C1
810637
[O][=C][Branch1][N][N][C][C][C][=C][C][=C][C][=C][Ring1][=Branch1][C][C][C][C][N][Branch1][N][C][=Branch1][C][=O][N][C][C][C][C][Ring1][Branch1][C][Ring1][=N]
C17CCCN4C1.c18ccccc1.N15CCCC1.O=C37.C6C8.C45=O.N36
COC(=O)N1CCC(NC(=O)C(C)Sc2ccccc2)CC1
784457
[C][O][C][=Branch1][C][=O][N][C][C][C][Branch2][Ring1][Ring1][N][C][=Branch1][C][=O][C][Branch1][C][C][S][C][=C][C][=C][C][=C][Ring1][=Branch1][C][C][Ring2][Ring1][C]
N14CCC7CC1.c18ccccc1.C5(=O)C6C.C34=O.CO3.N57.S68
COc1cccc2[nH]c3c(N4CCCC(C)C4)ncnc3c12
35016
[C][O][C][=C][C][=C][C][NH1][C][=C][Branch1][N][N][C][C][C][C][Branch1][C][C][C][Ring1][#Branch1][N][=C][N][=C][Ring1][=N][C][Ring2][Ring1][Ring2][=Ring1][S]
c15cccc2[nH]c3c6ncnc3c12.N16CCCC(C)C1.CO5
Cc1nnnn1-c1cccc(NC(=O)NCc2ccccn2)c1
610945
[C][C][=N][N][=N][N][Ring1][Branch1][C][=C][C][=C][C][Branch1][S][N][C][=Branch1][C][=O][N][C][C][=C][C][=C][C][=N][Ring1][=Branch1][=C][Ring1][P]
c18cccc6c1.Cc1nnnn18.c17ccccn1.C34=O.N36.N45.C57
Cc1ccc2nc(C)cc(C(=O)N3CCOCC3)c2c1
445405
[C][C][=C][C][=C][N][=C][Branch1][C][C][C][=C][Branch1][=N][C][=Branch1][C][=O][N][C][C][O][C][C][Ring1][=Branch1][C][Ring1][#C][=C][Ring2][Ring1][Ring1]
Cc1ccc2nc(C)cc5c2c1.N14CCOCC1.C45=O
C#CCCNC(=O)c1ccc(Oc2ccccc2)cc1
968023
[C][#C][C][C][N][C][=Branch1][C][=O][C][=C][C][=C][Branch1][#Branch2][O][C][=C][C][=C][C][=C][Ring1][=Branch1][C][=C][Ring1][=N]
c17ccc4cc1.c15ccccc1.C#CCC6.C37=O.N36.O45
CC(C)N=c1ccccn1C(=O)CN1C(=O)COc2ccccc21
212585
[C][C][Branch1][C][C][N][=C][C][=C][C][=C][N][Ring1][=Branch1][C][=Branch1][C][=O][C][N][C][=Branch1][C][=O][C][O][C][=C][C][=C][C][=C][Ring1][=Branch1][Ring1][O]
CC(C)N=c1ccccn1C(=O)CN1C(=O)COc2ccccc21
O=C1CN(C(=O)CS(=O)(=O)c2ccc(Cl)cc2)CCN1
790577
[O][=C][C][N][Branch2][Ring1][Branch2][C][=Branch1][C][=O][C][S][=Branch1][C][=O][=Branch1][C][=O][C][=C][C][=C][Branch1][C][Cl][C][=C][Ring1][#Branch1][C][C][N][Ring2][Ring1][Ring1]
C3(=O)CS(=O)(=O)c1ccc(Cl)cc1.O=C1CN3CCN1
COCCOc1ccc(NC(=O)NCC(F)(F)F)cc1
624234
[C][O][C][C][O][C][=C][C][=C][Branch1][S][N][C][=Branch1][C][=O][N][C][C][Branch1][C][F][Branch1][C][F][F][C][=C][Ring1][#C]
c16ccc8cc1.C7C(F)(F)F.C4C5.C23=O.CO4.O56.N28.N37
O=C(c1cc2ccccc2[nH]1)N(CCO)Cc1ccccc1
1553274
[O][=C][Branch1][=C][C][=C][C][=C][C][=C][C][=C][Ring1][=Branch1][NH1][Ring1][=Branch2][N][Branch1][Ring2][C][C][O][C][C][=C][C][=C][C][=C][Ring1][=Branch1]
c16cc2ccccc2[nH]1.c17ccccc1.O=C36.N345.C4CO.C57
NC(=O)C1CCN(C(=O)c2ccc3sccc3c2)CC1
1460139
[N][C][=Branch1][C][=O][C][C][C][N][Branch2][Ring1][C][C][=Branch1][C][=O][C][=C][C][=C][S][C][=C][C][Ring1][Branch1][=C][Ring1][=Branch2][C][C][Ring1][P]
c16ccc2sccc2c1.C15CCN4CC1.NC5=O.C46=O