SMILES
large_stringlengths
17
56
ID
large_stringlengths
1
7
SELFIES
stringlengths
63
275
SAFE
stringlengths
20
78
COc1ccc(S(=O)(=O)NCCCn2ccnc2)c(C)c1C
1793145
[C][O][C][=C][C][=C][Branch2][Ring1][Ring1][S][=Branch1][C][=O][=Branch1][C][=O][N][C][C][C][N][C][=C][N][=C][Ring1][Branch1][C][Branch1][C][C][=C][Ring2][Ring1][Ring1][C]
c13ccc(S5(=O)=O)c(C)c1C.n16ccnc1.C4CC6.CO3.N45
c1ccc(Oc2ccc(CNc3ncn[nH]3)cc2)cc1
1264835
[C][=C][C][=C][Branch2][Ring1][Branch1][O][C][=C][C][=C][Branch1][#Branch2][C][N][C][=N][C][=N][NH1][Ring1][Branch1][C][=C][Ring1][=N][C][=C][Ring2][Ring1][Ring2]
c15ccc8cc1.c1ccc4cc1.c17ncn[nH]1.O45.C68.N67
O=C(CN1CCc2ccccc21)NCC1COCCO1
682540
[O][=C][Branch1][#C][C][N][C][C][C][=C][C][=C][C][=C][Ring1][=Branch1][Ring1][=Branch2][N][C][C][C][O][C][C][O][Ring1][=Branch1]
N14CCc2ccccc21.C16COCCO1.O=C3C4.N35.C56
Cc1cc(C)n(-c2ccc(C(=O)NC(C)CO)cc2)n1
1554915
[C][C][C][=C][Branch1][C][C][N][Branch2][Ring1][=Branch1][C][=C][C][=C][Branch1][N][C][=Branch1][C][=O][N][C][Branch1][C][C][C][O][C][=C][Ring1][=N][N][=Ring2][Ring1][Ring1]
Cc1cc(C)n6n1.c16ccc5cc1.C4(C)CO.C35=O.N34
CN(C)c1ccc(C#CCNC(=O)COc2cccnc2)cc1
1753866
[C][N][Branch1][C][C][C][=C][C][=C][Branch2][Ring1][Ring1][C][#C][C][N][C][=Branch1][C][=O][C][O][C][=C][C][=C][N][=C][Ring1][=Branch1][C][=C][Ring2][Ring1][Ring2]
c17ccc(C#CC6)cc1.c15cccnc1.C3(=O)C4.CN7C.N36.O45
Cc1sc2ncnc(SCCC(=O)Nc3cn[nH]c3)c2c1C
863316
[C][C][S][C][=N][C][=N][C][Branch1][S][S][C][C][C][=Branch1][C][=O][N][C][C][=N][NH1][C][=Ring1][Branch1][=C][Ring1][P][C][=Ring2][Ring1][Ring2][C]
Cc1sc2ncnc7c2c1C.C5CC4=O.c16cn[nH]c1.S57.N46
CCn1ccc(C(=O)Nc2nc3c(Cl)cccc3s2)n1
1613235
[C][C][N][C][=C][C][Branch2][Ring1][=Branch1][C][=Branch1][C][=O][N][C][=N][C][=C][Branch1][C][Cl][C][=C][C][=C][Ring1][#Branch1][S][Ring1][#Branch2][=N][Ring2][Ring1][C]
c15nc2c(Cl)cccc2s1.n17ccc6n1.C46=O.CC7.N45
CCn1c2ccccc2c2cc(CNC(C)C(N)=O)ccc21
740564
[C][C][N][C][=C][C][=C][C][=C][Ring1][=Branch1][C][=C][C][Branch1][N][C][N][C][Branch1][C][C][C][Branch1][C][N][=O][=C][C][=C][Ring1][=N][Ring2][Ring1][Ring2]
n15c2ccccc2c2cc6ccc21.C4(C)C(N)=O.CC5.C36.N34
CCC(C)NC(=O)NC1CC(=O)N(c2ccc(OC)c(OC)c2)C1
90196
[C][C][C][Branch1][C][C][N][C][=Branch1][C][=O][N][C][C][C][=Branch1][C][=O][N][Branch1][P][C][=C][C][=C][Branch1][Ring1][O][C][C][Branch1][Ring1][O][C][=C][Ring1][#Branch2][C][Ring1][S]
c19ccc5c6c1.C18CC(=O)N9C1.CCC7C.C34=O.N37.N48.O5C.O6C
COC(=O)CCN(CC(C)C)C(=O)c1cnc2ccc(C)cn12
1384678
[C][O][C][=Branch1][C][=O][C][C][N][Branch1][#Branch1][C][C][Branch1][C][C][C][C][=Branch1][C][=O][C][=C][N][=C][C][=C][C][Branch1][C][C][=C][N][Ring1][#Branch2][Ring1][#Branch1]
c17cnc2ccc(C)cn12.C3(=O)CC5.C6C(C)C.N456.C47=O.CO3
COc1ccc(NC(=O)Nc2cnn(Cc3ccc(F)cc3)c2)cc1
395672
[C][O][C][=C][C][=C][Branch2][Ring1][N][N][C][=Branch1][C][=O][N][C][C][=N][N][Branch1][=N][C][C][=C][C][=C][Branch1][C][F][C][=C][Ring1][#Branch1][C][=Ring1][=N][C][=C][Ring2][Ring1][#Branch1]
c16ccc7cc1.c1%10ccc(F)cc1.c18cnn9c1.C45=O.CO6.N47.N58.C9%10
CC(C)n1ncc2cc(C(=O)N3CCCC(n4cncn4)C3)cnc21
1880241
[C][C][Branch1][C][C][N][N][=C][C][=C][C][Branch2][Ring1][=Branch1][C][=Branch1][C][=O][N][C][C][C][C][Branch1][Branch2][N][C][=N][C][=N][Ring1][Branch1][C][Ring1][O][=C][N][=C][Ring2][Ring1][Ring1][Ring2][Ring1][=Branch1]
n17ncc2cc6cnc21.N15CCCC8C1.n18cncn1.CC7C.C56=O
CS(=O)(=O)c1ccc(C(=O)NCCc2cc3ccccc3o2)cc1
1019978
[C][S][=Branch1][C][=O][=Branch1][C][=O][C][=C][C][=C][Branch2][Ring1][Branch1][C][=Branch1][C][=O][N][C][C][C][=C][C][=C][C][=C][C][=C][Ring1][=Branch1][O][Ring1][=Branch2][C][=C][Ring2][Ring1][Ring2]
CS(=O)(=O)c1ccc6cc1.c17cc2ccccc2o1.C46=O.C5C7.N45
Cc1cccc(OCCCNC(=O)Cc2cn3ccsc3n2)c1
371012
[C][C][=C][C][=C][C][Branch2][Ring1][#Branch1][O][C][C][C][N][C][=Branch1][C][=O][C][C][=C][N][C][=C][S][C][Ring1][Branch1][=N][Ring1][Branch2][=C][Ring2][Ring1][=Branch1]
c18cn2ccsc2n1.Cc1cccc6c1.C5CC7.C4(=O)C8.O56.N47
CC(=O)c1ccc(OCCCC(=O)Nc2c(C)cc(C)nc2C)cc1
1539123
[C][C][=Branch1][C][=O][C][=C][C][=C][Branch2][Ring1][=Branch2][O][C][C][C][C][=Branch1][C][=O][N][C][=C][Branch1][C][C][C][=C][Branch1][C][C][N][=C][Ring1][Branch2][C][C][=C][Ring2][Ring1][=Branch1]
c16c(C)cc(C)nc1C.c17ccc5cc1.C4CCC3=O.CC7=O.O45.N36
Cc1cc(NC(=O)NCc2ccccc2OC(F)(F)F)no1
644430
[C][C][=C][C][Branch2][Ring1][=Branch2][N][C][=Branch1][C][=O][N][C][C][=C][C][=C][C][=C][Ring1][=Branch1][O][C][Branch1][C][F][Branch1][C][F][F][=N][O][Ring2][Ring1][Branch1]
c18ccccc15.Cc1cc7no1.O5C(F)(F)F.C34=O.N37.N46.C68
CC1CCCC(C)N1C(=O)C1CN(C(=O)c2ccc(F)c(F)c2)C1
964808
[C][C][C][C][C][C][Branch1][C][C][N][Ring1][#Branch1][C][=Branch1][C][=O][C][C][N][Branch2][Ring1][Ring1][C][=Branch1][C][=O][C][=C][C][=C][Branch1][C][F][C][Branch1][C][F][=C][Ring1][Branch2][C][Ring1][=C]
CC1CCCC(C)N13.c16ccc(F)c(F)c1.C15CN4C1.C35=O.C46=O
COc1ccc(-c2nc3c4ccccc4n(CCC#N)c(=O)n3n2)cc1
403363
[C][O][C][=C][C][=C][Branch2][Ring1][=C][C][N][=C][C][=C][C][=C][C][=C][Ring1][=Branch1][N][Branch1][Branch1][C][C][C][#N][C][=Branch1][C][=O][N][Ring1][#C][N][=Ring2][Ring1][C][C][=C][Ring2][Ring1][Branch2]
c17nc2c3ccccc3n6c(=O)n2n1.c15ccc7cc1.C6CC#N.CO5
CS(=O)(=O)Oc1ccc(C(=O)c2ccc(F)cc2)cc1
513916
[C][S][=Branch1][C][=O][=Branch1][C][=O][O][C][=C][C][=C][Branch1][S][C][=Branch1][C][=O][C][=C][C][=C][Branch1][C][F][C][=C][Ring1][#Branch1][C][=C][Ring1][#C]
c13ccc4cc1.c15ccc(F)cc1.CS(=O)(=O)O3.C45=O
N#CCS(=O)(=O)NCC1(c2cccc(C(F)(F)F)c2)CCC1
1464958
[N][#C][C][S][=Branch1][C][=O][=Branch1][C][=O][N][C][C][Branch2][Ring1][Ring1][C][=C][C][=C][C][Branch1][=Branch2][C][Branch1][C][F][Branch1][C][F][F][=C][Ring1][#Branch2][C][C][C][Ring1][=C]
c17cccc6c1.N#CCS4(=O)=O.C157CCC1.C6(F)(F)F.N34.C35
CC(NC(=O)CCc1ccncc1)c1cccc(N2CCCC2)c1
1309079
[C][C][Branch1][S][N][C][=Branch1][C][=O][C][C][C][=C][C][=N][C][=C][Ring1][=Branch1][C][=C][C][=C][C][Branch1][Branch2][N][C][C][C][C][Ring1][Branch1][=C][Ring1][O]
c16cccc5c1.c17ccncc1.C3(=O)CC7.N15CCCC1.CC46.N34
CCn1nc(C(=O)Nc2ccc(Br)cc2)ccc1=O
217203
[C][C][N][N][=C][Branch1][P][C][=Branch1][C][=O][N][C][=C][C][=C][Branch1][C][Br][C][=C][Ring1][#Branch1][C][=C][C][Ring1][S][=O]
n16nc5ccc1=O.c14ccc(Br)cc1.C35=O.CC6.N34
CCCCCOC(=O)Cn1c(=O)oc2ccccc21
53762
[C][C][C][C][C][O][C][=Branch1][C][=O][C][N][C][=Branch1][C][=O][O][C][=C][C][=C][C][=C][Ring1][=Branch1][Ring1][#Branch2]
n15c(=O)oc2ccccc21.CCCCC4.C3(=O)C5.O34
Cc1cc(C)cc(NC(=O)C(C)N2CCN(C(=O)C(C)(C)C)CC2)c1
1880342
[C][C][=C][C][Branch1][C][C][=C][C][Branch2][Ring1][S][N][C][=Branch1][C][=O][C][Branch1][C][C][N][C][C][N][Branch1][=N][C][=Branch1][C][=O][C][Branch1][C][C][Branch1][C][C][C][C][C][Ring1][N][=C][Ring2][Ring1][Branch2]
Cc1cc6cc(C)c1.N15CCN4CC1.C4(=O)C(C)(C)C.C3(=O)C5C.N36
COC(=O)c1cc(N2CCOCC2)ccc1NC(=O)C1CCC1
1826924
[C][O][C][=Branch1][C][=O][C][=C][C][Branch1][=Branch2][N][C][C][O][C][C][Ring1][=Branch1][=C][C][=C][Ring1][N][N][C][=Branch1][C][=O][C][C][C][C][Ring1][Ring2]
c18cc5ccc16.N15CCOCC1.C17CCC1.C38=O.C47=O.CO3.N46
CCSc1ncc(Cl)c(C(=O)NCCCn2ccnc2)n1
394387
[C][C][S][C][=N][C][=C][Branch1][C][Cl][C][Branch1][S][C][=Branch1][C][=O][N][C][C][C][N][C][=C][N][=C][Ring1][Branch1][=N][Ring2][Ring1][C]
c18ncc(Cl)c6n1.n17ccnc1.C4CC7.C36=O.CC5.S58.N34
Cc1nc(COc2ccc(C(=O)NC(C)C3CCCO3)cc2)no1
530987
[C][C][=N][C][Branch2][Ring1][=N][C][O][C][=C][C][=C][Branch1][P][C][=Branch1][C][=O][N][C][Branch1][C][C][C][C][C][C][O][Ring1][Branch1][C][=C][Ring1][S][=N][O][Ring2][Ring1][#Branch1]
c16ccc8cc1.Cc1nc%10no1.C19CCCO1.C48=O.C79C.C5%10.O56.N47
CCc1nc2n(n1)CCCC2NC1CCCN(c2ccccc2)C1=O
1905586
[C][C][C][N][=C][N][Branch1][Ring2][N][=Ring1][Branch1][C][C][C][C][Ring1][#Branch1][N][C][C][C][C][N][Branch1][=Branch2][C][=C][C][=C][C][=C][Ring1][=Branch1][C][Ring1][N][=O]
c14nc2n(n1)CCCC2N3.C13CCCN5C1=O.c15ccccc1.CC4
O=C(CCc1c(F)cccc1F)N1CCN(C2CCCC2O)CC1
1697368
[O][=C][Branch1][#C][C][C][C][=C][Branch1][C][F][C][=C][C][=C][Ring1][#Branch1][F][N][C][C][N][Branch1][=Branch2][C][C][C][C][C][Ring1][Branch1][O][C][C][Ring1][N]
c15c(F)cccc1F.N13CCN4CC1.C14CCCC1O.O=C3CC5
CCCc1cc(C(=O)N2CCCC2Cn2cc(C)cn2)[nH]n1
990622
[C][C][C][C][C][=C][Branch2][Ring1][#Branch1][C][=Branch1][C][=O][N][C][C][C][C][Ring1][Branch1][C][N][C][=C][Branch1][C][C][C][=N][Ring1][=Branch1][NH1][N][=Ring2][Ring1][Ring1]
c17cc4[nH]n1.N13CCCC16.n15cc(C)cn1.CCC7.C34=O.C56
O=C(Cc1ccsc1)Nc1ccccc1C(=O)NC1CCCC1
367638
[O][=C][Branch1][=Branch2][C][C][C][=C][S][C][=Ring1][Branch1][N][C][=C][C][=C][C][=C][Ring1][=Branch1][C][=Branch1][C][=O][N][C][C][C][C][C][Ring1][Branch1]
c14ccccc16.c17ccsc1.C15CCCC1.O=C2C7.C36=O.N24.N35
CNC(=O)c1ccc(NC(=O)N2CCc3sccc3C2)c(C)c1
1655953
[C][N][C][=Branch1][C][=O][C][=C][C][=C][Branch2][Ring1][Ring1][N][C][=Branch1][C][=O][N][C][C][C][S][C][=C][C][=Ring1][Branch1][C][Ring1][=Branch2][C][Branch1][C][C][=C][Ring2][Ring1][Ring1]
N16CCc2sccc2C1.c18ccc7c(C)c1.C48=O.C56=O.CN4.N57
Cc1cccc(OCCCC(=O)NCc2ccc3c(c2)OCO3)c1
144971
[C][C][=C][C][=C][C][Branch2][Ring1][#Branch2][O][C][C][C][C][=Branch1][C][=O][N][C][C][=C][C][=C][C][=Branch1][Ring2][=C][Ring1][=Branch1][O][C][O][Ring1][=Branch1][=C][Ring2][Ring1][#Branch1]
c18ccc2c(c1)OCO2.Cc1cccc6c1.C5CCC4=O.O56.N47.C78
CC(C)CNC(=O)c1nnc2oc3ccccc3n12
1706655
[C][C][Branch1][C][C][C][N][C][=Branch1][C][=O][C][=N][N][=C][O][C][=C][C][=C][C][=C][Ring1][=Branch1][N][Ring1][N][Ring1][=Branch2]
c16nnc2oc3ccccc3n12.CC(C)C5.C46=O.N45
CNC(=O)c1ccc(C(=O)N(C)C)cc1OC1CC1
1475095
[C][N][C][=Branch1][C][=O][C][=C][C][=C][Branch1][#Branch2][C][=Branch1][C][=O][N][Branch1][C][C][C][C][=C][Ring1][O][O][C][C][C][Ring1][Ring1]
c16ccc7cc15.C26=O.C37=O.N3(C)C.C14CC1.CN2.O45
CC(C)(C)c1ccc(NC(=O)Nc2cc(-n3cncn3)ncn2)cc1
1927543
[C][C][Branch1][C][C][Branch1][C][C][C][=C][C][=C][Branch2][Ring1][Branch2][N][C][=Branch1][C][=O][N][C][=C][C][Branch1][Branch2][N][C][=N][C][=N][Ring1][Branch1][=N][C][=N][Ring1][O][C][=C][Ring2][Ring1][Branch1]
c18ccc7cc1.c16cc9ncn1.n19cncn1.CC8(C)C.C45=O.N47.N56
Cc1ccc(S(=O)(=O)NC2CC3CCC2C3)cc1
1769959
[C][C][=C][C][=C][Branch2][Ring1][Ring2][S][=Branch1][C][=O][=Branch1][C][=O][N][C][C][C][C][C][C][Ring1][=Branch1][C][Ring1][Branch1][C][=C][Ring1][P]
Cc1ccc(S4(=O)=O)cc1.C15CC2CCC1C2.N45
COc1ccc(CNC(=O)C(C)Sc2nc(C)cc(N)n2)cc1
149232
[C][O][C][=C][C][=C][Branch2][Ring1][#Branch2][C][N][C][=Branch1][C][=O][C][Branch1][C][C][S][C][=N][C][Branch1][C][C][=C][C][Branch1][C][N][=N][Ring1][Branch2][C][=C][Ring2][Ring1][Branch1]
c18nc(C)cc(N)n1.c14ccc7cc1.C3(=O)C6C.CO4.C57.N35.S68
COCc1nc(-c2cccc(N3CCCC3=O)c2)cs1
803452
[C][O][C][C][=N][C][Branch2][Ring1][Ring1][C][=C][C][=C][C][Branch1][=Branch2][N][C][C][C][C][Ring1][Branch1][=O][=C][Ring1][N][=C][S][Ring1][P]
c17cccc6c1.c15nc7cs1.N16CCCC1=O.CO4.C45
CN(C(=O)CCc1nc2ccccc2[nH]1)C1CCCCC1
213681
[C][N][Branch2][Ring1][Ring2][C][=Branch1][C][=O][C][C][C][=N][C][=C][C][=C][C][=C][Ring1][=Branch1][NH1][Ring1][=Branch2][C][C][C][C][C][C][Ring1][=Branch1]
c15nc2ccccc2[nH]1.C14CCCCC1.C3(=O)CC5.CN34
CCCCCNC(=O)c1cc2cnn(CC)c2nc1N
1711150
[C][C][C][C][C][N][C][=Branch1][C][=O][C][=C][C][C][=N][N][Branch1][Ring1][C][C][C][=Ring1][#Branch1][N][=C][Ring1][O][N]
c15cc2cnn6c2nc1N.CCCCC4.C35=O.N34.C6C
CCC(NC(=O)c1csc(C)n1)c1cccs1
682565
[C][C][C][Branch1][S][N][C][=Branch1][C][=O][C][=C][S][C][Branch1][C][C][=N][Ring1][=Branch1][C][=C][C][=C][S][Ring1][Branch1]
c14csc(C)n1.c15cccs1.CCC35.C24=O.N23
CCC(CC)N(CCO)C(=O)c1cccc(N)c1
570444
[C][C][C][Branch1][Ring1][C][C][N][Branch1][Ring2][C][C][O][C][=Branch1][C][=O][C][=C][C][=C][C][Branch1][C][N][=C][Ring1][#Branch1]
c15cccc(N)c1.CCC3CC.N234.C4CO.C25=O
Cc1csc(-c2cccc(NC(=O)N(C)Cc3cnn(C)c3)c2)n1
988560
[C][C][=C][S][C][Branch2][Ring1][P][C][=C][C][=C][C][Branch2][Ring1][Branch1][N][C][=Branch1][C][=O][N][Branch1][C][C][C][C][C][=N][N][Branch1][C][C][C][=Ring1][=Branch1][=C][Ring2][Ring1][C][=N][Ring2][Ring1][#Branch1]
c19cccc7c1.Cc1csc9n1.c18cnn(C)c1.C45=O.N56C.N47.C68
CN1C(=O)CCC2(CNS(=O)(=O)c3cccc(F)c3)CCCC12
1574428
[C][N][C][=Branch1][C][=O][C][C][C][Branch2][Ring1][Branch1][C][N][S][=Branch1][C][=O][=Branch1][C][=O][C][=C][C][=C][C][Branch1][C][F][=C][Ring1][#Branch1][C][C][C][C][Ring2][Ring1][=Branch1][Ring1][P]
CN1C(=O)CCC26CCCC12.S5(=O)(=O)c1cccc(F)c1.C46.N45
Cc1ccsc1CN1CCNC(=O)C1C(C)C
1440050
[C][C][C][=C][S][C][=Ring1][Branch1][C][N][C][C][N][C][=Branch1][C][=O][C][Ring1][#Branch1][C][Branch1][C][C][C]
N12CCNC(=O)C13.Cc1ccsc14.C3(C)C.C24
O=C(c1ccsc1)N1CCC2(CC(Nc3cccnc3)CO2)C1
1514227
[O][=C][Branch1][Branch2][C][C][=C][S][C][=Ring1][Branch1][N][C][C][C][Branch2][Ring1][C][C][C][Branch1][#Branch2][N][C][=C][C][=C][N][=C][Ring1][=Branch1][C][O][Ring1][N][C][Ring1][S]
N14CCC2(CC6CO2)C1.c15cccnc1.c17ccsc1.O=C47.N56
O=C(Nc1cc(-c2ccncc2)n[nH]1)c1ccc(Br)cc1
1697246
[O][=C][Branch2][Ring1][Ring1][N][C][=C][C][Branch1][=Branch2][C][=C][C][=N][C][=C][Ring1][=Branch1][=N][NH1][Ring1][O][C][=C][C][=C][Branch1][C][Br][C][=C][Ring1][#Branch1]
c15ccc(Br)cc1.c14cc6n[nH]1.c16ccncc1.O=C35.N34
CC1CCC(NS(=O)(=O)Cc2ccccc2)CC1
183879
[C][C][C][C][C][Branch2][Ring1][C][N][S][=Branch1][C][=O][=Branch1][C][=O][C][C][=C][C][=C][C][=C][Ring1][=Branch1][C][C][Ring1][P]
CC1CCC4CC1.c15ccccc1.S3(=O)(=O)C5.N34
Cc1cc(C)cc(CCC(=O)NCc2nccc(N)n2)c1
1925845
[C][C][=C][C][Branch1][C][C][=C][C][Branch2][Ring1][Ring2][C][C][C][=Branch1][C][=O][N][C][C][=N][C][=C][C][Branch1][C][N][=N][Ring1][#Branch1][=C][Ring2][Ring1][Ring2]
Cc1cc6cc(C)c1.c15nccc(N)n1.C6CC3=O.N34.C45
Cc1ccc(C(=O)NC(C)(C)c2nc(C)c(C)s2)cc1C
1119139
[C][C][=C][C][=C][Branch2][Ring1][#Branch2][C][=Branch1][C][=O][N][C][Branch1][C][C][Branch1][C][C][C][=N][C][Branch1][C][C][=C][Branch1][C][C][S][Ring1][#Branch1][C][=C][Ring2][Ring1][Ring1][C]
Cc1ccc5cc1C.c16nc(C)c(C)s1.C46(C)C.C35=O.N34
Cc1noc(C)c1CNc1ccc(C(=O)Nc2ccccc2)nn1
1019697
[C][C][=N][O][C][Branch1][C][C][=C][Ring1][=Branch1][C][N][C][=C][C][=C][Branch1][=C][C][=Branch1][C][=O][N][C][=C][C][=C][C][=C][Ring1][=Branch1][N][=N][Ring1][#C]
Cc1noc(C)c18.c15ccc7nn1.c16ccccc1.C37=O.C48.N45.N36
COc1ccc(CN2CC(C)OCC2C)cc1OCCCC#N
1420093
[C][O][C][=C][C][=C][Branch1][=C][C][N][C][C][Branch1][C][C][O][C][C][Ring1][#Branch1][C][C][=C][Ring1][#C][O][C][C][C][C][#N]
c14ccc7cc15.N16CC(C)OCC1C.C3CCC#N.CO4.C67.O35
Cc1ccccc1NC(=O)C(C)Sc1nnnn1-c1ccccc1
78358
[C][C][=C][C][=C][C][=C][Ring1][=Branch1][N][C][=Branch1][C][=O][C][Branch1][C][C][S][C][=N][N][=N][N][Ring1][Branch1][C][=C][C][=C][C][=C][Ring1][=Branch1]
Cc1ccccc14.c16nnnn15.c15ccccc1.C2(=O)C3C.N24.S36
COCC(NC(=O)c1cc(Br)ccc1F)C(N)=O
1325156
[C][O][C][C][Branch2][Ring1][C][N][C][=Branch1][C][=O][C][=C][C][Branch1][C][Br][=C][C][=C][Ring1][#Branch1][F][C][Branch1][C][N][=O]
c15cc(Br)ccc1F.C3C4C(N)=O.C25=O.CO3.N24
CC(C)(C)C(=O)N1CCCC(c2nc3ccccc3[nH]2)C1
442099
[C][C][Branch1][C][C][Branch1][C][C][C][=Branch1][C][=O][N][C][C][C][C][Branch1][=C][C][=N][C][=C][C][=C][C][=C][Ring1][=Branch1][NH1][Ring1][=Branch2][C][Ring1][#C]
c15nc2ccccc2[nH]1.N14CCCC5C1.CC(C)(C)C4=O
Cc1cc2ccccc2n2c(=O)n(CC(=O)N(C(C)C)C(C)C)nc12
223784
[C][C][=C][C][=C][C][=C][C][=C][Ring1][=Branch1][N][C][=Branch1][C][=O][N][Branch2][Ring1][Ring1][C][C][=Branch1][C][=O][N][Branch1][=Branch1][C][Branch1][C][C][C][C][Branch1][C][C][C][N][=C][Ring2][Ring1][Branch2][Ring1][S]
Cc1cc2ccccc2n2c(=O)n6nc12.C6C3=O.N345.C4(C)C.C5(C)C
O=C(NCCn1nnn(-c2ccccc2)c1=O)C1CCC1
1699087
[O][=C][Branch2][Ring1][=Branch1][N][C][C][N][N][=N][N][Branch1][=Branch2][C][=C][C][=C][C][=C][Ring1][=Branch1][C][Ring1][O][=O][C][C][C][C][Ring1][Ring2]
n16nnn7c1=O.c17ccccc1.C15CCC1.O=C35.C4C6.N34
O=S(=O)(NCc1ccoc1)c1ccc(F)cc1
612203
[O][=S][=Branch1][C][=O][Branch1][#Branch2][N][C][C][C][=C][O][C][=Ring1][Branch1][C][=C][C][=C][Branch1][C][F][C][=C][Ring1][#Branch1]
O=S3(=O)c1ccc(F)cc1.c14ccoc1.N23.C24
CNC(=O)c1cc(Cl)ccc1NC(=O)c1cc(C(N)=O)cs1
739962
[C][N][C][=Branch1][C][=O][C][=C][C][Branch1][C][Cl][=C][C][=C][Ring1][#Branch1][N][C][=Branch1][C][=O][C][=C][C][Branch1][=Branch1][C][Branch1][C][N][=O][=C][S][Ring1][Branch2]
c16cc(Cl)ccc14.c15cc7cs1.C26=O.C35=O.C7(N)=O.CN2.N34
Cc1ncc(C(=O)NCCNC(=O)c2ccoc2)s1
881375
[C][C][=N][C][=C][Branch2][Ring1][Ring2][C][=Branch1][C][=O][N][C][C][N][C][=Branch1][C][=O][C][C][=C][O][C][=Ring1][Branch1][S][Ring2][Ring1][C]
Cc1ncc7s1.c18ccoc1.C37=O.C5C6.C48=O.N35.N46
O=C(COc1ccc(F)cc1)Nc1noc(-c2cccs2)n1
282631
[O][=C][Branch1][=C][C][O][C][=C][C][=C][Branch1][C][F][C][=C][Ring1][#Branch1][N][C][=N][O][C][Branch1][Branch2][C][=C][C][=C][S][Ring1][Branch1][=N][Ring1][#Branch2]
c15ccc(F)cc1.c16noc7n1.c17cccs1.O=C3C4.O45.N36
COCCNC(=O)NC(C)c1ccc(-n2ccnc2C)cc1
1727468
[C][O][C][C][N][C][=Branch1][C][=O][N][C][Branch1][C][C][C][=C][C][=C][Branch1][=Branch2][N][C][=C][N][=C][Ring1][Branch1][C][C][=C][Ring1][N]
c18ccc9cc1.n19ccnc1C.C5C6.C34=O.C78C.CO5.N36.N47
Cc1[nH]c(=O)[nH]c(=O)c1CCC(=O)Nc1cccc(Cl)c1Cl
1790686
[C][C][NH1][C][=Branch1][C][=O][NH1][C][=Branch1][C][=O][C][=Ring1][Branch2][C][C][C][=Branch1][C][=O][N][C][=C][C][=C][C][Branch1][C][Cl][=C][Ring1][#Branch1][Cl]
Cc1[nH]c(=O)[nH]c(=O)c14.c13cccc(Cl)c1Cl.C4CC2=O.N23
CCc1cc2c(C)cc(=O)oc2cc1OC(=O)Cc1c(C)noc1C
608325
[C][C][C][=C][C][C][Branch1][C][C][=C][C][=Branch1][C][=O][O][C][=Ring1][Branch2][C][=C][Ring1][N][O][C][=Branch1][C][=O][C][C][C][Branch1][C][C][=N][O][C][=Ring1][=Branch1][C]
c15cc2c(C)cc(=O)oc2cc14.c16c(C)noc1C.C3(=O)C6.CC5.O34
O=C(Nc1nnc(C2CC2)s1)c1cccnc1N1CCCCC1
519758
[O][=C][Branch1][S][N][C][=N][N][=C][Branch1][=Branch1][C][C][C][Ring1][Ring1][S][Ring1][Branch2][C][=C][C][=C][N][=C][Ring1][=Branch1][N][C][C][C][C][C][Ring1][=Branch1]
c16cccnc15.c14nnc7s1.N15CCCCC1.O=C36.C17CC1.N34
COC(=O)CCn1c(=O)c2cccn2c2ccc(F)cc21
331362
[C][O][C][=Branch1][C][=O][C][C][N][C][=Branch1][C][=O][C][=C][C][=C][N][Ring1][Branch1][C][=C][C][=C][Branch1][C][F][C][=C][Ring1][#Branch1][Ring1][#C]
n14c(=O)c2cccn2c2ccc(F)cc21.C3(=O)CC4.CO3
CCN(C(=O)CCCS(=O)(=O)N1CCCC1)c1cccc(F)c1
1755319
[C][C][N][Branch2][Ring1][=Branch1][C][=Branch1][C][=O][C][C][C][S][=Branch1][C][=O][=Branch1][C][=O][N][C][C][C][C][Ring1][Branch1][C][=C][C][=C][C][Branch1][C][F][=C][Ring1][#Branch1]
C2(=O)CCCS4(=O)=O.c15cccc(F)c1.N14CCCC1.N235.CC3
COCCCNC(=O)CN(C)C(=O)c1cc2c(F)cccc2s1
808808
[C][O][C][C][C][N][C][=Branch1][C][=O][C][N][Branch1][C][C][C][=Branch1][C][=O][C][=C][C][=C][Branch1][C][F][C][=C][C][=C][Ring1][#Branch1][S][Ring1][#Branch2]
c18cc2c(F)cccc2s1.C5CC6.C3(=O)C7.N47C.C48=O.CO5.N36
Cc1cc2c(cc1Br)N(Cc1n[nH]c(=O)[nH]1)CCC2
1320730
[C][C][=C][C][=C][Branch1][=Branch1][C][=C][Ring1][=Branch1][Br][N][Branch1][N][C][C][=N][NH1][C][=Branch1][C][=O][NH1][Ring1][=Branch1][C][C][C][Ring1][S]
Cc1cc2c(cc1Br)N3CCC2.c14n[nH]c(=O)[nH]1.C34
CC(=O)N1CCc2cc(C(=O)OCc3ccc(C#N)cc3)ccc21
410743
[C][C][=Branch1][C][=O][N][C][C][C][=C][C][Branch2][Ring1][Ring1][C][=Branch1][C][=O][O][C][C][=C][C][=C][Branch1][Ring1][C][#N][C][=C][Ring1][Branch2][=C][C][=C][Ring2][Ring1][C][Ring2][Ring1][Branch1]
N15CCc2cc7ccc21.c18ccc(C#N)cc1.CC5=O.C47=O.O46.C68
COC1CCCN(C(=O)c2cc3ccccc3n2C)C1
1113035
[C][O][C][C][C][C][N][Branch2][Ring1][Ring1][C][=Branch1][C][=O][C][=C][C][=C][C][=C][C][=C][Ring1][=Branch1][N][Ring1][=Branch2][C][C][Ring2][Ring1][C]
c16cc2ccccc2n1C.C15CCCN4C1.C46=O.CO5
CC(OC(=O)c1ccc(O)cc1)C(=O)c1ccccc1
73187
[C][C][Branch1][P][O][C][=Branch1][C][=O][C][=C][C][=C][Branch1][C][O][C][=C][Ring1][#Branch1][C][=Branch1][C][=O][C][=C][C][=C][C][=C][Ring1][=Branch1]
c14ccc(O)cc1.c15ccccc1.CC3C5=O.C24=O.O23
COC(=O)N1CCCC(C(=O)N2C(C)CCCC2c2ccccc2)C1
1219071
[C][O][C][=Branch1][C][=O][N][C][C][C][C][Branch2][Ring1][Branch2][C][=Branch1][C][=O][N][C][Branch1][C][C][C][C][C][C][Ring1][#Branch1][C][=C][C][=C][C][=C][Ring1][=Branch1][C][Ring2][Ring1][Branch1]
N15C7CCCC1C.N14CCCC6C1.c17ccccc1.C34=O.C56=O.CO3
Cc1noc(C)c1CCC(=O)N1CCN(Cc2cccc(F)c2)CC1
1697001
[C][C][=N][O][C][Branch1][C][C][=C][Ring1][=Branch1][C][C][C][=Branch1][C][=O][N][C][C][N][Branch1][=N][C][C][=C][C][=C][C][Branch1][C][F][=C][Ring1][#Branch1][C][C][Ring1][=C]
Cc1noc(C)c15.N13CCN4CC1.c16cccc(F)c1.C5CC3=O.C46
CN(C)C(=O)C1CCCN1c1cc(F)ccc1N
729996
[C][N][Branch1][C][C][C][=Branch1][C][=O][C][C][C][C][N][Ring1][Branch1][C][=C][C][Branch1][C][F][=C][C][=C][Ring1][#Branch1][N]
c13cc(F)ccc1N.C14CCCN13.CN2C.C24=O
Cc1nc(N2CCC(C(=O)NCCCOC(C)C)CC2)sc1C
1459234
[C][C][N][=C][Branch2][Ring1][=Branch2][N][C][C][C][Branch1][#C][C][=Branch1][C][=O][N][C][C][C][O][C][Branch1][C][C][C][C][C][Ring1][S][S][C][=Ring2][Ring1][Branch1][C]
Cc1nc7sc1C.N17CCC8CC1.C6CC4.C38=O.C5(C)C.N36.O45
CC(=O)c1ccc(NC(=O)c2cc(-c3ccc(C)cc3)[nH]n2)cc1
241932
[C][C][=Branch1][C][=O][C][=C][C][=C][Branch2][Ring1][#Branch2][N][C][=Branch1][C][=O][C][C][=C][Branch1][N][C][=C][C][=C][Branch1][C][C][C][=C][Ring1][#Branch1][NH1][N][=Ring1][N][C][=C][Ring2][Ring1][Branch1]
c17ccc5cc1.c18ccc(C)cc1.c16cc8[nH]n1.CC7=O.C46=O.N45
O=C(c1ccc(F)cc1F)N1CC(c2nc(-c3ccco3)no2)C1
1520670
[O][=C][Branch1][=N][C][=C][C][=C][Branch1][C][F][C][=C][Ring1][#Branch1][F][N][C][C][Branch1][P][C][=N][C][Branch1][Branch2][C][=C][C][=C][O][Ring1][Branch1][=N][O][Ring1][#Branch2][C][Ring1][=C]
c15ccc(F)cc1F.c17nc6no1.N14CC7C1.c16ccco1.O=C45
Nc1cc(-c2ccco2)nn(CC(=O)Nc2ccccc2Cl)c1=O
303867
[N][C][=C][C][Branch1][Branch2][C][=C][C][=C][O][Ring1][Branch1][=N][N][Branch1][S][C][C][=Branch1][C][=O][N][C][=C][C][=C][C][=C][Ring1][=Branch1][Cl][C][Ring2][Ring1][=Branch1][=O]
Nc1cc6nn5c1=O.c14ccccc1Cl.c16ccco1.C5C3=O.N34
O=C(Cc1nnc(-c2cnccn2)o1)Nc1cc(Cl)ccc1F
870834
[O][=C][Branch2][Ring1][Ring1][C][C][=N][N][=C][Branch1][=Branch2][C][=C][N][=C][C][=N][Ring1][=Branch1][O][Ring1][O][N][C][=C][C][Branch1][C][Cl][=C][C][=C][Ring1][#Branch1][F]
c14cc(Cl)ccc1F.c15nnc6o1.c16cnccn1.O=C3C5.N34
Cc1ccccc1CN(C)C(=O)NCc1cc(=O)[nH]c2ccccc12
1282226
[C][C][=C][C][=C][C][=C][Ring1][=Branch1][C][N][Branch1][C][C][C][=Branch1][C][=O][N][C][C][=C][C][=Branch1][C][=O][NH1][C][=C][C][=C][C][=C][Ring1][O][Ring1][=Branch1]
c18cc(=O)[nH]c2ccccc12.Cc1ccccc17.N35C.C34=O.C57.N46.C68
CCCn1nnnc1Cn1c(=O)c(C(F)(F)F)nc2ccccc21
437802
[C][C][C][N][N][=N][N][=C][Ring1][Branch1][C][N][C][=Branch1][C][=O][C][Branch1][=Branch2][C][Branch1][C][F][Branch1][C][F][F][=N][C][=C][C][=C][C][=C][Ring1][=Branch1][Ring1][#C]
n14c(=O)c6nc2ccccc21.n13nnnc15.C6(F)(F)F.CCC3.C45
CCOC(=O)CCC(=O)N1CCC(Oc2ccc(C)nn2)CC1
1502114
[C][C][O][C][=Branch1][C][=O][C][C][C][=Branch1][C][=O][N][C][C][C][Branch1][=N][O][C][=C][C][=C][Branch1][C][C][N][=N][Ring1][#Branch1][C][C][Ring1][=C]
C3(=O)CCC4=O.N14CCC7CC1.c16ccc(C)nn1.CC5.O35.O67
CC(CNC(=O)CCC(=O)c1ccc(Cl)cc1)N1CCOCC1
634913
[C][C][Branch2][Ring1][Branch2][C][N][C][=Branch1][C][=O][C][C][C][=Branch1][C][=O][C][=C][C][=C][Branch1][C][Cl][C][=C][Ring1][#Branch1][N][C][C][O][C][C][Ring1][=Branch1]
C2(=O)CCC5=O.c15ccc(Cl)cc1.N13CCOCC1.CC3C4.N24
O=C1OCCN1Cc1sccc1Br
586224
[O][=C][O][C][C][N][Ring1][Branch1][C][C][S][C][=C][C][=Ring1][Branch1][Br]
O=C1OCCN12.c13sccc1Br.C23
CC(=O)N(C)Cc1cccc(NC(=O)CCn2cncn2)c1
1807834
[C][C][=Branch1][C][=O][N][Branch1][C][C][C][C][=C][C][=C][C][Branch1][#C][N][C][=Branch1][C][=O][C][C][N][C][=N][C][=N][Ring1][Branch1][=C][Ring1][S]
c18cccc6c1.C4(=O)CC7.n17cncn1.CC3=O.N35C.C58.N46
CC(O)CN1CCN(CC(=O)NCCc2ccc(Cl)cc2)CC1
952969
[C][C][Branch1][C][O][C][N][C][C][N][Branch2][Ring1][Ring2][C][C][=Branch1][C][=O][N][C][C][C][=C][C][=C][Branch1][C][Cl][C][=C][Ring1][#Branch1][C][C][Ring2][Ring1][Ring1]
N14CCN5CC1.c17ccc(Cl)cc1.CC(O)C4.C5C3=O.C6C7.N36
CC(C(=O)N1CCn2cnnc2C1)n1nnc2ccccc21
1794301
[C][C][Branch2][Ring1][C][C][=Branch1][C][=O][N][C][C][N][C][=N][N][=C][Ring1][Branch1][C][Ring1][=Branch2][N][N][=N][C][=C][C][=C][C][=C][Ring1][=Branch1][Ring1][=Branch2]
N13CCn2cnnc2C1.n14nnc2ccccc21.CC4C3=O
O=C(Cc1ccccn1)N1Cc2ccnn2CC(COCC2CC2)C1
1510878
[O][=C][Branch1][#Branch2][C][C][=C][C][=C][C][=N][Ring1][=Branch1][N][C][C][=C][C][=N][N][Ring1][Branch1][C][C][Branch1][=Branch2][C][O][C][C][C][C][Ring1][Ring1][C][Ring1][S]
N13Cc2ccnn2CC7C1.c16ccccn1.O=C3C6.C18CC1.C47.O45.C58
CC(C)CN(CC#Cc1ccccc1)C(=O)CCNS(C)(=O)=O
752214
[C][C][Branch1][C][C][C][N][Branch1][N][C][C][#C][C][=C][C][=C][C][=C][Ring1][=Branch1][C][=Branch1][C][=O][C][C][N][S][Branch1][C][C][=Branch1][C][=O][=O]
C4C#Cc1ccccc1.C2(=O)CC5.CC(C)C3.S6(C)(=O)=O.N234.N56
Cc1noc(C)c1CN(C)C(=O)C1(c2cccc(Cl)c2)CCC1
635140
[C][C][=N][O][C][Branch1][C][C][=C][Ring1][=Branch1][C][N][Branch1][C][C][C][=Branch1][C][=O][C][Branch1][N][C][=C][C][=C][C][Branch1][C][Cl][=C][Ring1][#Branch1][C][C][C][Ring1][O]
Cc1noc(C)c16.c17cccc(Cl)c1.C157CCC1.N34C.C35=O.C46
CC(=O)N(CCc1ccccc1)CC(=O)NC(C)c1c(C)noc1C
1386033
[C][C][=Branch1][C][=O][N][Branch1][O][C][C][C][=C][C][=C][C][=C][Ring1][=Branch1][C][C][=Branch1][C][=O][N][C][Branch1][C][C][C][C][Branch1][C][C][=N][O][C][=Ring1][=Branch1][C]
c18c(C)noc1C.c17ccccc1.C5C3=O.CC2=O.N245.C4C7.C68C.N36
Cc1ccccc1CNC(=O)CNc1cccc(C(N)=O)c1C
764432
[C][C][=C][C][=C][C][=C][Ring1][=Branch1][C][N][C][=Branch1][C][=O][C][N][C][=C][C][=C][C][Branch1][=Branch1][C][Branch1][C][N][=O][=C][Ring1][=Branch2][C]
c15cccc6c1C.Cc1ccccc17.C2(=O)C4.C6(N)=O.C37.N23.N45
CN(CCC#N)C(=O)CSc1nnnn1C1CC1
240759
[C][N][Branch1][Branch1][C][C][C][#N][C][=Branch1][C][=O][C][S][C][=N][N][=N][N][Ring1][Branch1][C][C][C][Ring1][Ring1]
c16nnnn15.C3CC#N.C2(=O)C4.CN23.C15CC1.S46
CC(O)CNC(=O)C(C)Oc1ccc(F)cc1Br
1758022
[C][C][Branch1][C][O][C][N][C][=Branch1][C][=O][C][Branch1][C][C][O][C][=C][C][=C][Branch1][C][F][C][=C][Ring1][#Branch1][Br]
c14ccc(F)cc1Br.C2(=O)C3C.CC(O)C5.N25.O34
O=C(Cc1ccc(O)cc1)N1CCN(CCO)CC1
458491
[O][=C][Branch1][=N][C][C][=C][C][=C][Branch1][C][O][C][=C][Ring1][#Branch1][N][C][C][N][Branch1][Ring2][C][C][O][C][C][Ring1][=Branch2]
c14ccc(O)cc1.N12CCN3CC1.O=C2C4.C3CO
Nc1nccc(C2CCCN(c3ncccn3)C2)n1
1698573
[N][C][=N][C][=C][C][Branch2][Ring1][Ring1][C][C][C][C][N][Branch1][=Branch2][C][=N][C][=C][C][=N][Ring1][=Branch1][C][Ring1][N][=N][Ring2][Ring1][C]
Nc1nccc5n1.C15CCCN4C1.c14ncccn1
CC(CNC(=O)Cn1cnc2ccccc2c1=O)c1ccccc1
153176
[C][C][Branch2][Ring1][#Branch1][C][N][C][=Branch1][C][=O][C][N][C][=N][C][=C][C][=C][C][=C][Ring1][=Branch1][C][Ring1][#Branch2][=O][C][=C][C][=C][C][=C][Ring1][=Branch1]
n15cnc2ccccc2c1=O.c16ccccc1.CC6C4.C3(=O)C5.N34
COc1ccc(C2C3=C(COC3=O)Nc3[nH]nc(C)c32)c(OC)c1
1620485
[C][O][C][=C][C][=C][Branch2][Ring1][=Branch2][C][C][=C][Branch1][#Branch1][C][O][C][Ring1][Branch1][=O][N][C][NH1][N][=C][Branch1][C][C][C][=Ring1][=Branch1][Ring1][=C][C][Branch1][Ring1][O][C][=C][Ring2][Ring1][=Branch1]
c14ccc(C2C3=C(COC3=O)Nc3[nH]nc(C)c32)c5c1.CO4.O5C