CID
int64
19
167M
SID
int64
842k
144M
IUPAC_Name
stringlengths
6
1.03k
PAIN_flag
stringclasses
2 values
4,116
144,206,179
2,2-dichloro-1,1-difluoro-1-methoxyethane
No
44,820,559
89,449,180
N'-(5-bromo-2-pyridinyl)-N'-[(3,4-dichlorophenyl)methyl]propane-1,3-diamine
No
44,820,549
89,449,181
N'-[(3,4-dichlorophenyl)methyl]-N'-pyridin-2-ylpropane-1,3-diamine
No
44,820,566
89,449,182
N'-(5-bromo-2-pyridinyl)-N'-[(4-chlorophenyl)methyl]propane-1,3-diamine
No
10,785,663
89,449,185
N'-(5-bromo-2-pyridinyl)-N'-[(3,4-dichlorophenyl)methyl]ethane-1,2-diamine
No
44,820,555
89,449,187
N'-(5-bromo-2-pyridinyl)-N'-[(4-methoxyphenyl)methyl]propane-1,3-diamine
No
44,820,570
89,449,200
1-[4-[(5-bromo-2-pyridinyl)-[(4-chlorophenyl)methyl]amino]butyl]-3-[3-(1H-imidazol-5-yl)propyl]thiourea
No
44,820,545
89,449,203
1-[3-[4-bromo-N-[(4-chlorophenyl)methyl]anilino]propyl]-3-[3-(1H-imidazol-5-yl)propyl]thiourea
No
44,820,568
89,449,205
1-[3-[(5-bromo-2-pyridinyl)-[(4-chlorophenyl)methyl]amino]propyl]-3-[3-(1H-imidazol-5-yl)propyl]urea
No
44,820,552
89,449,206
1-[3-[(5-bromopyrimidin-2-yl)-[(4-chlorophenyl)methyl]amino]propyl]-3-[3-(1H-imidazol-5-yl)propyl]thiourea
No
44,820,557
89,449,208
1-[3-[(4-chlorophenyl)methyl-(5-phenyl-2-pyridinyl)amino]propyl]-3-[3-(1H-imidazol-5-yl)propyl]thiourea
No
11,957,540
124,891,649
1-(2,3-dichlorophenyl)ethanamine;hydrochloride
No
24,962,993
81,066,852
methyl (1R,5S)-6-(4-chloro-3-methylphenyl)-8-methyl-4-oxo-3,6,8-triazabicyclo[3.2.1]octane-5-carboxylate
No
810,335
85,146,256
N-(5-amino-1,3-benzothiazol-2-yl)acetamide
No
768,525
85,146,257
1,3-benzothiazole-2,5-diamine
No
815,509
85,146,258
N-(5-nitro-1,3-benzothiazol-2-yl)acetamide
No
25,074,415
85,146,259
2-acetamido-1,3-benzothiazole-5-carboxamide
No
24,962,991
85,146,260
methyl 6-(3-ethoxycarbonylphenyl)-8-methyl-4-oxo-3,6,8-triazabicyclo[3.2.1]octane-5-carboxylate
No
42,609,748
85,147,120
(3R)-3-hydroxy-1-[(2R,10E)-4-oxo-3-oxabicyclo[11.4.0]heptadeca-1(17),10,13,15-tetraen-2-yl]hexane-1,5-dione
No
42,609,752
85,147,123
(3S)-3-hydroxy-1-[(2S,10E)-4-oxo-3-oxabicyclo[11.4.0]heptadeca-1(17),10,13,15-tetraen-2-yl]hexane-1,5-dione
No
42,609,754
85,147,125
(3S)-3-hydroxy-1-[(2R,10E)-4-oxo-3-oxabicyclo[11.4.0]heptadeca-1(17),10,13,15-tetraen-2-yl]hexane-1,5-dione
No
42,609,755
85,147,126
(3S)-3-hydroxy-1-[(2R)-4-oxo-3-oxabicyclo[11.4.0]heptadeca-1(17),13,15-trien-2-yl]hexane-1,5-dione
No
42,609,756
85,147,127
(3S)-3-hydroxy-1-[(1S,6Z)-3-oxo-1,4,5,8-tetrahydro-2-benzoxecin-1-yl]hexane-1,5-dione
No
42,609,771
85,147,128
(3R)-3-hydroxy-1-[(1R,4R,6Z)-4-methyl-3-oxo-1,4,5,8-tetrahydro-2-benzoxecin-1-yl]hexane-1,5-dione
No
24,963,006
85,147,129
(3R)-3-hydroxy-1-[(1S,6Z)-3-oxo-1,4,5,8-tetrahydro-2-benzoxecin-1-yl]hexane-1,5-dione
No
24,963,007
85,147,130
(3R)-3-hydroxy-1-[(1R,6Z)-3-oxo-1,4,5,8-tetrahydro-2-benzoxecin-1-yl]hexane-1,5-dione
No
42,609,741
85,147,131
(3R)-3-hydroxy-1-[(2S)-4-oxo-3-oxabicyclo[9.4.0]pentadeca-1(15),11,13-trien-2-yl]hexane-1,5-dione
No
42,609,747
85,147,133
(3S)-1-[(1R,4R)-4-ethyl-3-oxo-1,4,5,6,7,8-hexahydro-2-benzoxecin-1-yl]-3-hydroxyhexane-1,5-dione
No
42,609,743
85,147,135
(3S)-3-hydroxy-1-[(2R)-4-oxo-3-oxabicyclo[9.4.0]pentadeca-1(15),11,13-trien-2-yl]hexane-1,5-dione
No
42,609,772
85,147,136
(3S)-3-hydroxy-1-[(1S,4R,6Z)-4-methyl-3-oxo-1,4,5,8-tetrahydro-2-benzoxecin-1-yl]hexane-1,5-dione
No
42,609,781
85,147,137
(3R)-3-hydroxy-1-[(2R)-4-oxo-3-oxabicyclo[10.4.0]hexadeca-1(16),12,14-trien-2-yl]hexane-1,5-dione
No
42,609,782
85,147,138
(3S)-3-hydroxy-1-[(2S)-4-oxo-3-oxabicyclo[10.4.0]hexadeca-1(16),12,14-trien-2-yl]hexane-1,5-dione
No
42,621,523
85,272,373
(3S)-1-[(1S,4S,6Z)-4-ethyl-3-oxo-1,4,5,8-tetrahydro-2-benzoxecin-1-yl]-3-hydroxyhexane-1,5-dione
No
42,621,525
85,272,399
(3R)-1-[(1S,4R,6Z)-4-ethyl-3-oxo-1,4,5,8-tetrahydro-2-benzoxecin-1-yl]-3-hydroxyhexane-1,5-dione
No
42,621,526
85,272,400
(3R)-1-[(1S,4R)-4-ethyl-3-oxo-1,4,5,6,7,8-hexahydro-2-benzoxecin-1-yl]-3-hydroxyhexane-1,5-dione
No
42,621,527
85,272,401
(3S)-1-[(1R,4S,6Z)-4-ethyl-3-oxo-1,4,5,8-tetrahydro-2-benzoxecin-1-yl]-3-hydroxyhexane-1,5-dione
No
42,609,742
85,272,525
(3S)-3-hydroxy-1-[(2S)-4-oxo-3-oxabicyclo[9.4.0]pentadeca-1(15),11,13-trien-2-yl]hexane-1,5-dione
No
42,609,744
85,272,526
(3S)-1-[(1S,4R,6Z)-4-ethyl-3-oxo-1,4,5,8-tetrahydro-2-benzoxecin-1-yl]-3-hydroxyhexane-1,5-dione
No
42,609,746
85,272,527
(3S)-1-[(1S,4R)-4-ethyl-3-oxo-1,4,5,6,7,8-hexahydro-2-benzoxecin-1-yl]-3-hydroxyhexane-1,5-dione
No
42,609,758
85,272,528
(3R)-3-hydroxy-1-[(1S)-3-oxo-1,4,5,6,7,8-hexahydro-2-benzoxecin-1-yl]hexane-1,5-dione
No
42,609,759
85,272,529
(3R)-3-hydroxy-1-[(1R)-3-oxo-1,4,5,6,7,8-hexahydro-2-benzoxecin-1-yl]hexane-1,5-dione
No
42,609,760
85,272,530
(3S)-3-hydroxy-1-[(1S)-3-oxo-1,4,5,6,7,8-hexahydro-2-benzoxecin-1-yl]hexane-1,5-dione
No
42,609,761
85,272,531
(3S)-3-hydroxy-1-[(1R)-3-oxo-1,4,5,6,7,8-hexahydro-2-benzoxecin-1-yl]hexane-1,5-dione
No
42,609,762
85,272,532
(3R)-3-hydroxy-1-[(1S,4S,6Z)-4-methyl-3-oxo-1,4,5,8-tetrahydro-2-benzoxecin-1-yl]hexane-1,5-dione
No
42,609,763
85,272,533
(3R)-3-hydroxy-1-[(1R,4S,6Z)-4-methyl-3-oxo-1,4,5,8-tetrahydro-2-benzoxecin-1-yl]hexane-1,5-dione
No
42,609,764
85,272,534
(3S)-3-hydroxy-1-[(1S,4S,6Z)-4-methyl-3-oxo-1,4,5,8-tetrahydro-2-benzoxecin-1-yl]hexane-1,5-dione
No
42,609,765
85,272,535
(3S)-3-hydroxy-1-[(1R,4S,6Z)-4-methyl-3-oxo-1,4,5,8-tetrahydro-2-benzoxecin-1-yl]hexane-1,5-dione
No
42,609,767
85,272,536
(3R)-3-hydroxy-1-[(1R,4S)-4-methyl-3-oxo-1,4,5,6,7,8-hexahydro-2-benzoxecin-1-yl]hexane-1,5-dione
No
42,609,768
85,272,537
(3S)-3-hydroxy-1-[(1S,4S)-4-methyl-3-oxo-1,4,5,6,7,8-hexahydro-2-benzoxecin-1-yl]hexane-1,5-dione
No
42,609,770
85,272,538
(3R)-3-hydroxy-1-[(1S,4R,6Z)-4-methyl-3-oxo-1,4,5,8-tetrahydro-2-benzoxecin-1-yl]hexane-1,5-dione
No
42,609,773
85,272,539
(3S)-3-hydroxy-1-[(1R,4R,6Z)-4-methyl-3-oxo-1,4,5,8-tetrahydro-2-benzoxecin-1-yl]hexane-1,5-dione
No
42,609,774
85,272,540
(3R)-3-hydroxy-1-[(1S,4R)-4-methyl-3-oxo-1,4,5,6,7,8-hexahydro-2-benzoxecin-1-yl]hexane-1,5-dione
No
42,609,775
85,272,541
(3R)-3-hydroxy-1-[(1R,4R)-4-methyl-3-oxo-1,4,5,6,7,8-hexahydro-2-benzoxecin-1-yl]hexane-1,5-dione
No
42,609,776
85,272,542
(3S)-3-hydroxy-1-[(1S,4R)-4-methyl-3-oxo-1,4,5,6,7,8-hexahydro-2-benzoxecin-1-yl]hexane-1,5-dione
No
42,609,778
85,272,543
(3R)-1-[(1R,4R,6Z)-4-ethyl-3-oxo-1,4,5,8-tetrahydro-2-benzoxecin-1-yl]-3-hydroxyhexane-1,5-dione
No
42,609,779
85,272,544
(3R)-1-[(1R,4R)-4-ethyl-3-oxo-1,4,5,6,7,8-hexahydro-2-benzoxecin-1-yl]-3-hydroxyhexane-1,5-dione
No
16,196,965
24,841,411
methyl (5Z)-4-[2-[[5-(1,3-dihydroxypropan-2-yl)-3-[2-[(3Z)-3-ethylidene-5-methoxycarbonyl-2-[3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-4H-pyran-4-yl]acetyl]oxy-2-methylcyclopentyl]methoxy]-2-oxoethyl]-5-ethylidene-6-[3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-4H-pyran-3-carboxylate
No
23,843,932
24,841,412
N-[(9E,21E,33E)-15,27-diacetamido-7,19,31-trihydroxy-10,22,34-trimethyl-2,8,14,20,26,32-hexaoxo-1,13,25-trioxa-7,19,31-triazacyclohexatriaconta-9,21,33-trien-3-yl]acetamide
No
6,451,074
24,841,413
(6aR,9R,9aR)-9-acetyl-3-[(1E,3E,5S)-3,5-dimethylhepta-1,3-dienyl]-6a-methyl-9,9a-dihydrofuro[2,3-h]isochromene-6,8-dione
No
15,674,942
24,841,416
(2R)-7-hydroxy-8-(2-hydroxyethyl)-5-methoxy-2-methyl-2,3-dihydrochromen-4-one
No
15,649,435
24,841,417
3-benzyl-4-methyl-1,3-dihydro-1,4-benzodiazepine-2,5-dione
No
11,958,880
24,841,418
3-hydroxy-3-methyl-5-oxo-5-[[3,4,5-trihydroxy-6-[6-methoxy-2-oxo-3-(2-oxochromen-7-yl)oxychromen-7-yl]oxyoxan-2-yl]methoxy]pentanoic acid
No
16,196,967
24,841,419
(2R,3S)-3-hydroxy-5-[(2S)-2-hydroxypropyl]-2-methyl-2,3-dihydropyran-6-one
No
348,130
24,841,421
5-hydroxy-2-(4-hydroxyphenyl)-7-methoxy-2,3-dihydrochromen-4-one
No
16,196,968
24,841,422
2-(2,3-dihydroxy-5-methylphenoxy)-5-methylbenzene-1,3-diol
PAIN
4,485,701
24,841,424
3,4-dimethyl-2,5-bis(3,4,5-trimethoxyphenyl)oxolane
No
160,115
24,841,426
5,6,8-trihydroxy-2-methyl-9-(5,6,8-trihydroxy-2-methyl-4-oxo-2,3-dihydrobenzo[g]chromen-9-yl)-2,3-dihydrobenzo[g]chromen-4-one
No
5,379,262
24,841,427
3,5-dihydroxy-6,7,8-trimethoxy-2-phenylchromen-4-one
No
638,759
24,841,429
3-hydroxy-1-(4-hydroxyphenyl)propan-1-one
No
16,196,969
24,841,430
4-hydroxy-3,3,5-trimethyl-4-[(E)-3-[3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxybut-1-enyl]cyclohexan-1-one
No
301,798
24,841,431
5,7-dihydroxy-2-(4-hydroxyphenyl)-6-methyl-2,3-dihydrochromen-4-one
No
16,196,970
24,841,432
methyl (2R,4aR,4bS,10aS,10bS,12aR)-6,10b-dihydroxy-2,4b,7,7,10a,12a-hexamethyl-12-methylidene-1,4,5,8-tetraoxo-4a,9,10,11-tetrahydronaphtho[1,2-h]isochromene-2-carboxylate
No
5,351,523
24,841,433
2-[4-[3-(4-hydroxy-3-methoxyphenyl)-1,3,3a,4,6,6a-hexahydrofuro[3,4-c]furan-6-yl]-2-methoxyphenoxy]-6-(hydroxymethyl)oxane-3,4,5-triol
No
5,748,551
24,841,434
7-hydroxy-3-(4-hydroxyphenyl)-5-methoxychromen-4-one
No
16,196,971
24,841,435
[2-hydroxy-2-(2-hydroxy-4-methylphenyl)-3-(2-methylpropanoyloxy)propyl] 2-methylpropanoate
No
16,196,972
24,841,436
(5S,8S)-8-benzoyl-2-[(Z,1S,2S)-1,2-dihydroxyhex-3-enyl]-9-hydroxy-8-methoxy-3-methyl-1-oxa-7-azaspiro[4.4]non-2-ene-4,6-dione
No
641,785
24,841,437
(E)-1-(2,4-dihydroxy-6-methoxyphenyl)-3-phenylprop-2-en-1-one
No
5,280,448
24,841,438
7-hydroxy-3-(3-hydroxy-4-methoxyphenyl)chromen-4-one
No
73,525
24,841,439
(3S,3'R)-4-methyl-3'-phenylspiro[1H-1,4-benzodiazepine-3,2'-oxirane]-2,5-dione
No
16,196,973
24,841,440
2-(2-acetyl-3,5-dihydroxyphenyl)acetic acid
No
16,196,974
24,841,441
2-(3,4-dihydroxyphenyl)-7-hydroxy-8-(3-methylbut-2-enyl)-2,3-dihydrochromen-4-one
PAIN
14,583,237
24,841,443
5-chloro-9-(3-hydroxy-2-methylbutanoyl)-6a-methyl-3-[(E)-3-methylpent-1-enyl]-9,9a-dihydrofuro[2,3-h]isochromene-6,8-dione
PAIN
10,958,572
24,841,444
5-methoxy-8,8-dimethyl-2-phenylpyrano[2,3-h]chromen-4-one
No
5,282,074
24,841,445
3-(2,4-dihydroxyphenyl)-5,7-dihydroxychromen-4-one
No
11,217,464
24,841,446
4-(3-hydroxypropyl)benzene-1,2-diol
PAIN
6,438,437
24,841,448
(1R,3E,6R,7E,9S,11E,13R,14S,16R,17S,18R,19S)-6-hydroxy-19-(1H-indol-3-ylmethyl)-7,9,16,17-tetramethyl-15-oxa-20-azatetracyclo[11.8.0.01,18.014,16]henicosa-3,7,11-triene-2,5,21-trione
No
14,286,542
24,841,449
(3E,9E)-5,6-dihydroxy-9,13,14-trimethyl-16-(2-methylpropyl)-17-azatricyclo[9.7.0.01,15]octadeca-3,9,12-triene-2,18-dione
No
136,417
24,841,450
2-(3,4-dimethoxyphenyl)-5-hydroxy-3,6,7,8-tetramethoxychromen-4-one
No
6,426,860
24,841,451
2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-6-[3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]chromen-4-one
PAIN
3,951
24,841,453
5,7-dihydroxy-2-(4-hydroxyphenyl)-6,8-bis(3-methylbut-2-enyl)-2,3-dihydrochromen-4-one
No
5,467,708
24,841,456
4-[[2-[(E)-3-hydroxybut-1-enyl]-5-oxooxolan-3-yl]amino]benzaldehyde
No
14,730,864
24,841,457
2-phenylmethoxy-6-[(3,4,5-trihydroxyoxan-2-yl)oxymethyl]oxane-3,4,5-triol
No
375,148
24,841,459
3,8-dimethyl-3-(4-methylpent-3-enyl)-11H-pyrano[3,2-a]carbazol-9-ol
No
11,081,347
24,841,460
(2S,3R,5R,10R,13R,14S,17S)-2,3,14-trihydroxy-10,13-dimethyl-17-[(2R,3R)-2,3,6-trihydroxy-6-methylheptan-2-yl]-2,3,4,5,9,11,12,15,16,17-decahydro-1H-cyclopenta[a]phenanthren-6-one
No
11,447,214
24,841,462
2-hexyl-3-methylidenebutanedioic acid
No
9,842,429
24,841,463
6-hydroxy-2-(1-hydroxy-3-methylbutyl)-1-methoxy-8-methyl-10H-benzo[b][1,5]benzodioxocin-12-one
No
9,799,192
24,841,464
(4R,6S,8S,9Z,11E)-16-chloro-17,19-dihydroxy-4-methyl-3,7-dioxatricyclo[13.4.0.06,8]nonadeca-1(15),9,11,16,18-pentaene-2,13-dione
No
130,919
24,841,465
2,10,15,23-tetrazapentacyclo[12.9.0.02,11.04,9.017,22]tricosa-1(23),4,6,8,10,17,19,21-octaene-3,16-dione
No
483,513
24,841,467
4-(2,3-dihydroxy-3-methylbutoxy)furo[3,2-g]chromen-7-one
No
12,313,332
24,841,470
5,7-dihydroxy-2-(4-hydroxyphenyl)-3-[3,4,5-trihydroxy-6-[(3,4,5-trihydroxy-6-methyloxan-2-yl)oxymethyl]oxan-2-yl]oxychromen-4-one
No