assay_uid
stringlengths
9
15
positive_smiles
stringlengths
2
615
positive_smiles_hash
stringlengths
64
64
negative_smiles
listlengths
7
7
negative_smiles_hashes
listlengths
7
7
example_weight
float32
1
1.71
chembl:1528623
Cc1ccc(-c2ncccn2)c(C(=O)N2C3CCC2C(COc2ccc(F)cn2)C3)n1
b47932029e434362e66bc6b1a1e4c3339d0c1903959bfdf99bf524f1b57a1fdd
[ "Cc1ccc(C(=O)N2C3CCC2C(Nc2cnc(C(F)(F)F)cn2)C3)c(-n2ccnn2)n1", "O=C(c1cccc(F)c1-c1ccnnc1)N1C2CCC1C(Nc1cnc(C(F)(F)F)cn1)C2", "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1ncc(C(F)(F)F)cn1)C2", "Cc1ccc(C(=O)N2C3CCC2C(COc2ccccn2)C3)c(-n2nccn2)n1", "Cc1ccc(C(=O)N2C3CCC2C(COc2nccc(C(F)(F)F)n2)C3)c(-n2nccn2)n1", "Cc1cc(C)nc(O...
[ "80101f4f7a5fede239dedf39c500921e45c84cb244df3dfb40e7befb00d66ecb", "e921ccd1898af4d7c7829e8120e77c95c1c534456e4d2742ae11c3b3dff3baea", "b97f4a41a5cedfb00c3157f3b9e940376503e4ed11ba86279269eea2696fa398", "8cf62ab90226119046e3cb3a7154a8867bdf1d30da12cf4c73d6c2cf31ce4729", "63e5f5d544ab2dd60cdfe624c583725d7be...
1.644667
chembl:1528623
Cc1ccc(-c2ncccn2)c(C(=O)N2C3CCC2C(COc2ccc(F)cn2)C3)n1
b47932029e434362e66bc6b1a1e4c3339d0c1903959bfdf99bf524f1b57a1fdd
[ "Cc1ccc2nccn2c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "Cc1ccn2ccnc2c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "Cc1ccc(N2CCNCC2)c(C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1ccc(F)cn1)C2", "Cc1nc2sccn2c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1cnc3ccccc3n1)C2", "Cc1ccc(-n2nccn2)...
[ "e958358280dce37a463d061032e29c68a168803e94062a7562d68d020f372796", "515ea2ffa8807a7f0a6787e40ea05eeadb5601cef8c45a785cc877ac4bede677", "0fc0e284b6f14795dd5431215829a32c441f737edc3c5f879773b413a6a92518", "1dc92dac322cafa93f066deaecf37843451f1f38f1f5a093ce6cdff154d24f50", "61611e5a16d66b1b35b9ee02c63c8540270...
1.644667
chembl:1528623
Cc1ccc(-c2ncccn2)c(C(=O)N2C3CCC2C(Nc2cnc4ccccc4n2)C3)n1
aac2072659fb0b7eb5a730cf9ea7e4e307a2efd8c88bdad26ca3640881db297e
[ "Cc1ccc2nccn2c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "Cc1ccn2ccnc2c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "Cc1ccc(N2CCNCC2)c(C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1ccc(F)cn1)C2", "Cc1nc2sccn2c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1cnc3ccccc3n1)C2", "Cc1ccc(-n2nccn2)...
[ "e958358280dce37a463d061032e29c68a168803e94062a7562d68d020f372796", "515ea2ffa8807a7f0a6787e40ea05eeadb5601cef8c45a785cc877ac4bede677", "0fc0e284b6f14795dd5431215829a32c441f737edc3c5f879773b413a6a92518", "1dc92dac322cafa93f066deaecf37843451f1f38f1f5a093ce6cdff154d24f50", "61611e5a16d66b1b35b9ee02c63c8540270...
1.643333
chembl:1528623
Cc1ccc(-c2ncccn2)c(C(=O)N2C3CCC2C(Nc2cnc4ccccc4n2)C3)n1
aac2072659fb0b7eb5a730cf9ea7e4e307a2efd8c88bdad26ca3640881db297e
[ "CCOc1ncc(-c2ccccc2)cc1C(=O)N1C2CCC1C(COc1ccccn1)C2", "COC(=O)c1cnc(NC2CC3CCC2N3C(=O)c2cccc(F)c2-c2ncccn2)cn1", "Cc1ccc(-c2ncccc2C)c(C(=O)N2C3CCC2C(COc2ncc(F)cn2)C3)n1", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(Nc2ccc(F)cn2)C3)n1", "Cc1coc(-c2ccc(C)nc2C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "Cc1ccc2ncc(C)n2c1C(=O)N1C2...
[ "f4fb1ed2df616dcb13ed4bbc598e86e154c2b00f6adece9224846c878b4f2600", "fc30614a06906da50ef26facdc1824dde53eb44f09950784e41ca8bf3375f5cf", "36109ccd9045a0bcccf71ab97db1b74a977cb8ff0ce4e2e3e86e2bc9032ae8c0", "5d4403ad386547bcba1ba024fd2445a3a92b8caff2484185ed0d3b249c84ffc3", "b0b3168b4170993c8431f6ce2280394127f...
1.643333
chembl:1528623
Cc1cc(C)nc(OCC2CC3CCC2N3C(=O)c2c(F)cccc2-c2ncccn2)n1
22137527b5b200e211c08d8cda485777c589940fcc842f20f32d911b249e18fa
[ "CCOc1ncc(-c2ccccc2)cc1C(=O)N1C2CCC1C(COc1ccccn1)C2", "COC(=O)c1cnc(NC2CC3CCC2N3C(=O)c2cccc(F)c2-c2ncccn2)cn1", "Cc1ccc(-c2ncccc2C)c(C(=O)N2C3CCC2C(COc2ncc(F)cn2)C3)n1", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(Nc2ccc(F)cn2)C3)n1", "Cc1coc(-c2ccc(C)nc2C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "Cc1ccc2ncc(C)n2c1C(=O)N1C2...
[ "f4fb1ed2df616dcb13ed4bbc598e86e154c2b00f6adece9224846c878b4f2600", "fc30614a06906da50ef26facdc1824dde53eb44f09950784e41ca8bf3375f5cf", "36109ccd9045a0bcccf71ab97db1b74a977cb8ff0ce4e2e3e86e2bc9032ae8c0", "5d4403ad386547bcba1ba024fd2445a3a92b8caff2484185ed0d3b249c84ffc3", "b0b3168b4170993c8431f6ce2280394127f...
1.643
chembl:1528623
Cc1cc(C)nc(OCC2CC3CCC2N3C(=O)c2c(F)cccc2-c2ncccn2)n1
22137527b5b200e211c08d8cda485777c589940fcc842f20f32d911b249e18fa
[ "COc1cccc(-c2c(C)cnn2C)c1C(=O)N1C2CCC1C(Nc1cnc(C(F)(F)F)cn1)C2", "O=C(c1nc2ccccc2[nH]1)N1C2CCC1C(Nc1cnc(C(F)(F)F)cn1)C2", "Cc1ccc(N2CCN(C)CC2)c(C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "CCOc1ccc(C)nc1C(=O)N1C2CCC1C(Nc1ncc(C(F)(F)F)cn1)C2", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2ccncn2)C3)n1", "Cc1ccc(-n2nccn2)c(C...
[ "6c9cb367b275a634cb4095ebb2ab7f6168d34c9e60f9e5b0ada8b654da7820b6", "ff399b820cb3201b68c2d6b88b386d824aa8686b1bfdffca007e0038fe75d732", "cbb8f3bd86c4cc9f3ebd57d0bdcd6bd5c40685655b02798c55f1bea424dbc256", "40435856f94f24c747098de3efdb17a97a131b832dfc7b041b97990cc471f209", "044d1c0bc4b04fe457f6bf55d8f7cf479e6...
1.643
chembl:1528623
Cc1cccc(-n2nccn2)c1C(=O)N1C2CCC1C(COc1ccc(F)cn1)C2
2b3f831bcb85e7c38d237afc46d78720f543b79b37155bba103c90238932fc3f
[ "COc1cccc(-c2c(C)cnn2C)c1C(=O)N1C2CCC1C(Nc1cnc(C(F)(F)F)cn1)C2", "O=C(c1nc2ccccc2[nH]1)N1C2CCC1C(Nc1cnc(C(F)(F)F)cn1)C2", "Cc1ccc(N2CCN(C)CC2)c(C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "CCOc1ccc(C)nc1C(=O)N1C2CCC1C(Nc1ncc(C(F)(F)F)cn1)C2", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2ccncn2)C3)n1", "Cc1ccc(-n2nccn2)c(C...
[ "6c9cb367b275a634cb4095ebb2ab7f6168d34c9e60f9e5b0ada8b654da7820b6", "ff399b820cb3201b68c2d6b88b386d824aa8686b1bfdffca007e0038fe75d732", "cbb8f3bd86c4cc9f3ebd57d0bdcd6bd5c40685655b02798c55f1bea424dbc256", "40435856f94f24c747098de3efdb17a97a131b832dfc7b041b97990cc471f209", "044d1c0bc4b04fe457f6bf55d8f7cf479e6...
1.642667
chembl:1528623
Cc1cccc(-n2nccn2)c1C(=O)N1C2CCC1C(COc1ccc(F)cn1)C2
2b3f831bcb85e7c38d237afc46d78720f543b79b37155bba103c90238932fc3f
[ "Cc1ccc(-c2ncccc2C)c(C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2ccnn2C)C3)n1", "Cc1ccc(N2CCOCC2)c(C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2cccnn2)C3)n1", "CN(c1cnc(C(F)(F)F)cn1)C1CC2CCC1N2C(=O)c1cccc(F)c1-c1ncccn1", "CCOc1ccnc(Cl)c1C(=O)N1C2CCC1C...
[ "3681e2e80df961ea6c6913cbc4210c3c51d5ed170599dfe37a24d74d93670018", "0d0020e25910a43ee85f87dbcb7222c4e82730d8c8f60343a92a11836ae8069f", "26ed93e3488d6848a5d64cab7d440bd8f08c34ba506e9794bd961ffade785410", "96f2147056fb0dd194524eb0ca901fe41858e297da984fe4b1b75e8bf073d78e", "8e43077cb76b57f77f592c35d9c8814cda8...
1.642667
chembl:1528623
O=C(c1cc(F)ccc1-c1cc[nH]n1)N1C2CCC1C(COc1ccc(F)cn1)C2
3f59f60f12e6516ca3bee49cc2c1b0a96108433265bfe78d05b31b700b8772b2
[ "Cc1ccc(-c2ncccc2C)c(C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2ccnn2C)C3)n1", "Cc1ccc(N2CCOCC2)c(C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2cccnn2)C3)n1", "CN(c1cnc(C(F)(F)F)cn1)C1CC2CCC1N2C(=O)c1cccc(F)c1-c1ncccn1", "CCOc1ccnc(Cl)c1C(=O)N1C2CCC1C...
[ "3681e2e80df961ea6c6913cbc4210c3c51d5ed170599dfe37a24d74d93670018", "0d0020e25910a43ee85f87dbcb7222c4e82730d8c8f60343a92a11836ae8069f", "26ed93e3488d6848a5d64cab7d440bd8f08c34ba506e9794bd961ffade785410", "96f2147056fb0dd194524eb0ca901fe41858e297da984fe4b1b75e8bf073d78e", "8e43077cb76b57f77f592c35d9c8814cda8...
1.641667
chembl:1528623
O=C(c1cc(F)ccc1-c1cc[nH]n1)N1C2CCC1C(COc1ccc(F)cn1)C2
3f59f60f12e6516ca3bee49cc2c1b0a96108433265bfe78d05b31b700b8772b2
[ "O=C(c1cccc(F)c1-c1ccnnc1)N1C2CCC1C(Nc1cnc(C(F)(F)F)cn1)C2", "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1ncc(C(F)(F)F)cn1)C2", "Cc1ccc(C(=O)N2C3CCC2C(COc2ccccn2)C3)c(-n2nccn2)n1", "Cc1ccc(C(=O)N2C3CCC2C(COc2nccc(C(F)(F)F)n2)C3)c(-n2nccn2)n1", "Cc1cc(C)nc(OCC2CC3CCC2N3C(=O)c2ccc(C)nc2-n2nccn2)n1", "COc1c(F)cccc1C(=O)N...
[ "e921ccd1898af4d7c7829e8120e77c95c1c534456e4d2742ae11c3b3dff3baea", "b97f4a41a5cedfb00c3157f3b9e940376503e4ed11ba86279269eea2696fa398", "8cf62ab90226119046e3cb3a7154a8867bdf1d30da12cf4c73d6c2cf31ce4729", "63e5f5d544ab2dd60cdfe624c583725d7be7430cefb333c678ec7061b868896b", "2b8c02902d2f3c6a9ccf486c1220ab2b488...
1.641667
chembl:1528623
Cc1cc(C)nc(OCC2CC3CCC2N3C(=O)c2cc(F)ccc2-c2ncccn2)n1
4cf7f1af48589f771dfc5a50d6a49e157f62667b8a184d865ff6663e8cf7fc72
[ "O=C(c1cccc(F)c1-c1ccnnc1)N1C2CCC1C(Nc1cnc(C(F)(F)F)cn1)C2", "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1ncc(C(F)(F)F)cn1)C2", "Cc1ccc(C(=O)N2C3CCC2C(COc2ccccn2)C3)c(-n2nccn2)n1", "Cc1ccc(C(=O)N2C3CCC2C(COc2nccc(C(F)(F)F)n2)C3)c(-n2nccn2)n1", "Cc1cc(C)nc(OCC2CC3CCC2N3C(=O)c2ccc(C)nc2-n2nccn2)n1", "COc1c(F)cccc1C(=O)N...
[ "e921ccd1898af4d7c7829e8120e77c95c1c534456e4d2742ae11c3b3dff3baea", "b97f4a41a5cedfb00c3157f3b9e940376503e4ed11ba86279269eea2696fa398", "8cf62ab90226119046e3cb3a7154a8867bdf1d30da12cf4c73d6c2cf31ce4729", "63e5f5d544ab2dd60cdfe624c583725d7be7430cefb333c678ec7061b868896b", "2b8c02902d2f3c6a9ccf486c1220ab2b488...
1.641
chembl:1528623
Cc1cc(C)nc(OCC2CC3CCC2N3C(=O)c2cc(F)ccc2-c2ncccn2)n1
4cf7f1af48589f771dfc5a50d6a49e157f62667b8a184d865ff6663e8cf7fc72
[ "Cc1ccn2ccnc2c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "Cc1ccc(N2CCNCC2)c(C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1ccc(F)cn1)C2", "Cc1nc2sccn2c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1cnc3ccccc3n1)C2", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2cnccn2)C3)n1", "CCOc1ncc(...
[ "515ea2ffa8807a7f0a6787e40ea05eeadb5601cef8c45a785cc877ac4bede677", "0fc0e284b6f14795dd5431215829a32c441f737edc3c5f879773b413a6a92518", "1dc92dac322cafa93f066deaecf37843451f1f38f1f5a093ce6cdff154d24f50", "61611e5a16d66b1b35b9ee02c63c8540270c28b014f0894789c1a7b8879ceb1c", "09cb13eaf193692e39cc3183c06ceba07a4...
1.641
chembl:1528623
Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2cnc4ccccc4n2)C3)c1
7fbab0ff62f10f6cf06538fac0fafdb304529fb06c4a83d1269241643477bc83
[ "Cc1ccn2ccnc2c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "Cc1ccc(N2CCNCC2)c(C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1ccc(F)cn1)C2", "Cc1nc2sccn2c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1cnc3ccccc3n1)C2", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2cnccn2)C3)n1", "CCOc1ncc(...
[ "515ea2ffa8807a7f0a6787e40ea05eeadb5601cef8c45a785cc877ac4bede677", "0fc0e284b6f14795dd5431215829a32c441f737edc3c5f879773b413a6a92518", "1dc92dac322cafa93f066deaecf37843451f1f38f1f5a093ce6cdff154d24f50", "61611e5a16d66b1b35b9ee02c63c8540270c28b014f0894789c1a7b8879ceb1c", "09cb13eaf193692e39cc3183c06ceba07a4...
1.640667
chembl:1528623
Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2cnc4ccccc4n2)C3)c1
7fbab0ff62f10f6cf06538fac0fafdb304529fb06c4a83d1269241643477bc83
[ "COC(=O)c1cnc(NC2CC3CCC2N3C(=O)c2cccc(F)c2-c2ncccn2)cn1", "Cc1ccc(-c2ncccc2C)c(C(=O)N2C3CCC2C(COc2ncc(F)cn2)C3)n1", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(Nc2ccc(F)cn2)C3)n1", "Cc1coc(-c2ccc(C)nc2C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "Cc1ccc2ncc(C)n2c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "O=C(c1cccc(F)c1-c1ncccn1)N1C2CC...
[ "fc30614a06906da50ef26facdc1824dde53eb44f09950784e41ca8bf3375f5cf", "36109ccd9045a0bcccf71ab97db1b74a977cb8ff0ce4e2e3e86e2bc9032ae8c0", "5d4403ad386547bcba1ba024fd2445a3a92b8caff2484185ed0d3b249c84ffc3", "b0b3168b4170993c8431f6ce2280394127f98fcacb422ca22012ff9ef5c5b861", "6825e7beabb278b00dfc6c7ebdc8c4c9e2f...
1.640667
chembl:1528623
O=C(c1c(F)cccc1-n1nccn1)N1C2CCC1C(COc1ccc(F)cn1)C2
7b3e7c18fe5cbd29bb9b0dd14b18f39929b26f85b922e24757fc15f377cd3ce5
[ "COC(=O)c1cnc(NC2CC3CCC2N3C(=O)c2cccc(F)c2-c2ncccn2)cn1", "Cc1ccc(-c2ncccc2C)c(C(=O)N2C3CCC2C(COc2ncc(F)cn2)C3)n1", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(Nc2ccc(F)cn2)C3)n1", "Cc1coc(-c2ccc(C)nc2C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "Cc1ccc2ncc(C)n2c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "O=C(c1cccc(F)c1-c1ncccn1)N1C2CC...
[ "fc30614a06906da50ef26facdc1824dde53eb44f09950784e41ca8bf3375f5cf", "36109ccd9045a0bcccf71ab97db1b74a977cb8ff0ce4e2e3e86e2bc9032ae8c0", "5d4403ad386547bcba1ba024fd2445a3a92b8caff2484185ed0d3b249c84ffc3", "b0b3168b4170993c8431f6ce2280394127f98fcacb422ca22012ff9ef5c5b861", "6825e7beabb278b00dfc6c7ebdc8c4c9e2f...
1.640667
chembl:1528623
O=C(c1c(F)cccc1-n1nccn1)N1C2CCC1C(COc1ccc(F)cn1)C2
7b3e7c18fe5cbd29bb9b0dd14b18f39929b26f85b922e24757fc15f377cd3ce5
[ "O=C(c1nc2ccccc2[nH]1)N1C2CCC1C(Nc1cnc(C(F)(F)F)cn1)C2", "Cc1ccc(N2CCN(C)CC2)c(C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "CCOc1ccc(C)nc1C(=O)N1C2CCC1C(Nc1ncc(C(F)(F)F)cn1)C2", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2ccncn2)C3)n1", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(Nc2ncc(C(F)(F)F)cn2)C3)n1", "Cc1nc2sccn2c1C(=O)N1C2...
[ "ff399b820cb3201b68c2d6b88b386d824aa8686b1bfdffca007e0038fe75d732", "cbb8f3bd86c4cc9f3ebd57d0bdcd6bd5c40685655b02798c55f1bea424dbc256", "40435856f94f24c747098de3efdb17a97a131b832dfc7b041b97990cc471f209", "044d1c0bc4b04fe457f6bf55d8f7cf479e69aa6c7059d8721b792764429549c6", "89930909d6fa3919baedfc9715ad4ab3890...
1.640667
chembl:1528623
Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2nccc(C(F)(F)F)n2)C3)c1
7efe8d490db333809722397077d169f5d91165f230629cde98c3b5bb76201f37
[ "O=C(c1nc2ccccc2[nH]1)N1C2CCC1C(Nc1cnc(C(F)(F)F)cn1)C2", "Cc1ccc(N2CCN(C)CC2)c(C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "CCOc1ccc(C)nc1C(=O)N1C2CCC1C(Nc1ncc(C(F)(F)F)cn1)C2", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2ccncn2)C3)n1", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(Nc2ncc(C(F)(F)F)cn2)C3)n1", "Cc1nc2sccn2c1C(=O)N1C2...
[ "ff399b820cb3201b68c2d6b88b386d824aa8686b1bfdffca007e0038fe75d732", "cbb8f3bd86c4cc9f3ebd57d0bdcd6bd5c40685655b02798c55f1bea424dbc256", "40435856f94f24c747098de3efdb17a97a131b832dfc7b041b97990cc471f209", "044d1c0bc4b04fe457f6bf55d8f7cf479e69aa6c7059d8721b792764429549c6", "89930909d6fa3919baedfc9715ad4ab3890...
1.640333
chembl:1528623
Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2nccc(C(F)(F)F)n2)C3)c1
7efe8d490db333809722397077d169f5d91165f230629cde98c3b5bb76201f37
[ "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2ccnn2C)C3)n1", "Cc1ccc(N2CCOCC2)c(C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2cccnn2)C3)n1", "CN(c1cnc(C(F)(F)F)cn1)C1CC2CCC1N2C(=O)c1cccc(F)c1-c1ncccn1", "CCOc1ccnc(Cl)c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "Cc1ccc(C(=O)N2C3CCC2C(Nc2cnc(C(F)(F)F...
[ "0d0020e25910a43ee85f87dbcb7222c4e82730d8c8f60343a92a11836ae8069f", "26ed93e3488d6848a5d64cab7d440bd8f08c34ba506e9794bd961ffade785410", "96f2147056fb0dd194524eb0ca901fe41858e297da984fe4b1b75e8bf073d78e", "8e43077cb76b57f77f592c35d9c8814cda81696da4b10d44e2b392e1ca263462", "789d07cde0f56daaa9339ad1aec7b6f6f64...
1.640333
chembl:1528623
Cc1cccc(C(=O)N2C3CCC2C(Nc2ccc(C(F)(F)F)cn2)C3)c1-c1ncco1
d10087a5a654ed14651de327654f5016f9ee727b0ad5f01c4b819eb5f1121a85
[ "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2ccnn2C)C3)n1", "Cc1ccc(N2CCOCC2)c(C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2cccnn2)C3)n1", "CN(c1cnc(C(F)(F)F)cn1)C1CC2CCC1N2C(=O)c1cccc(F)c1-c1ncccn1", "CCOc1ccnc(Cl)c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "Cc1ccc(C(=O)N2C3CCC2C(Nc2cnc(C(F)(F)F...
[ "0d0020e25910a43ee85f87dbcb7222c4e82730d8c8f60343a92a11836ae8069f", "26ed93e3488d6848a5d64cab7d440bd8f08c34ba506e9794bd961ffade785410", "96f2147056fb0dd194524eb0ca901fe41858e297da984fe4b1b75e8bf073d78e", "8e43077cb76b57f77f592c35d9c8814cda81696da4b10d44e2b392e1ca263462", "789d07cde0f56daaa9339ad1aec7b6f6f64...
1.639667
chembl:1528623
Cc1cccc(C(=O)N2C3CCC2C(Nc2ccc(C(F)(F)F)cn2)C3)c1-c1ncco1
d10087a5a654ed14651de327654f5016f9ee727b0ad5f01c4b819eb5f1121a85
[ "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1ncc(C(F)(F)F)cn1)C2", "Cc1ccc(C(=O)N2C3CCC2C(COc2ccccn2)C3)c(-n2nccn2)n1", "Cc1ccc(C(=O)N2C3CCC2C(COc2nccc(C(F)(F)F)n2)C3)c(-n2nccn2)n1", "Cc1cc(C)nc(OCC2CC3CCC2N3C(=O)c2ccc(C)nc2-n2nccn2)n1", "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1ccc(C(F)(F)F)cn1)C2", "Cc1ccc2nccn2c1C(=O)N1C2CCC...
[ "b97f4a41a5cedfb00c3157f3b9e940376503e4ed11ba86279269eea2696fa398", "8cf62ab90226119046e3cb3a7154a8867bdf1d30da12cf4c73d6c2cf31ce4729", "63e5f5d544ab2dd60cdfe624c583725d7be7430cefb333c678ec7061b868896b", "2b8c02902d2f3c6a9ccf486c1220ab2b48822aeafee58748db4e242fef3d04ca", "d94db68cefb332689168cbfd14ab6d50f89...
1.639667
chembl:1528623
Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2ncccc2C(F)(F)F)C3)c1
958b577dc08b0a428da88f902c98f579393a21677c957af8bc1a6972367b18fb
[ "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1ncc(C(F)(F)F)cn1)C2", "Cc1ccc(C(=O)N2C3CCC2C(COc2ccccn2)C3)c(-n2nccn2)n1", "Cc1ccc(C(=O)N2C3CCC2C(COc2nccc(C(F)(F)F)n2)C3)c(-n2nccn2)n1", "Cc1cc(C)nc(OCC2CC3CCC2N3C(=O)c2ccc(C)nc2-n2nccn2)n1", "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1ccc(C(F)(F)F)cn1)C2", "Cc1ccc2nccn2c1C(=O)N1C2CCC...
[ "b97f4a41a5cedfb00c3157f3b9e940376503e4ed11ba86279269eea2696fa398", "8cf62ab90226119046e3cb3a7154a8867bdf1d30da12cf4c73d6c2cf31ce4729", "63e5f5d544ab2dd60cdfe624c583725d7be7430cefb333c678ec7061b868896b", "2b8c02902d2f3c6a9ccf486c1220ab2b48822aeafee58748db4e242fef3d04ca", "d94db68cefb332689168cbfd14ab6d50f89...
1.639
chembl:1528623
Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2ncccc2C(F)(F)F)C3)c1
958b577dc08b0a428da88f902c98f579393a21677c957af8bc1a6972367b18fb
[ "Cc1ccc(N2CCNCC2)c(C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1ccc(F)cn1)C2", "Cc1nc2sccn2c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1cnc3ccccc3n1)C2", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2cnccn2)C3)n1", "CCOc1ncc(-c2ccccc2)cc1C(=O)N1C2CCC1C(COc1ccccn1)C2", "C...
[ "0fc0e284b6f14795dd5431215829a32c441f737edc3c5f879773b413a6a92518", "1dc92dac322cafa93f066deaecf37843451f1f38f1f5a093ce6cdff154d24f50", "61611e5a16d66b1b35b9ee02c63c8540270c28b014f0894789c1a7b8879ceb1c", "09cb13eaf193692e39cc3183c06ceba07a4286fbaeda4627fed41570663984c1", "cd797d064c76d299c8c9b41b2766591a4d5...
1.639
chembl:1528623
Cc1cccc(C(=O)N2C3CCC2C(Nc2cnc(C(F)(F)F)cn2)C3)c1-c1ncco1
060aeb0f7290c4492a0336270168664c8279dc546481d8e1dbe2127211f3c1b7
[ "Cc1ccc(N2CCNCC2)c(C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1ccc(F)cn1)C2", "Cc1nc2sccn2c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1cnc3ccccc3n1)C2", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2cnccn2)C3)n1", "CCOc1ncc(-c2ccccc2)cc1C(=O)N1C2CCC1C(COc1ccccn1)C2", "C...
[ "0fc0e284b6f14795dd5431215829a32c441f737edc3c5f879773b413a6a92518", "1dc92dac322cafa93f066deaecf37843451f1f38f1f5a093ce6cdff154d24f50", "61611e5a16d66b1b35b9ee02c63c8540270c28b014f0894789c1a7b8879ceb1c", "09cb13eaf193692e39cc3183c06ceba07a4286fbaeda4627fed41570663984c1", "cd797d064c76d299c8c9b41b2766591a4d5...
1.639
chembl:1528623
Cc1cccc(C(=O)N2C3CCC2C(Nc2cnc(C(F)(F)F)cn2)C3)c1-c1ncco1
060aeb0f7290c4492a0336270168664c8279dc546481d8e1dbe2127211f3c1b7
[ "Cc1ccc(-c2ncccc2C)c(C(=O)N2C3CCC2C(COc2ncc(F)cn2)C3)n1", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(Nc2ccc(F)cn2)C3)n1", "Cc1coc(-c2ccc(C)nc2C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "Cc1ccc2ncc(C)n2c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "O=C(c1cccc(F)c1-c1ncccn1)N1C2CCC1C(Oc1ncc(C(F)(F)F)cn1)C2", "COc1cccc(-c2c(C)cnn2C)c1C(=O...
[ "36109ccd9045a0bcccf71ab97db1b74a977cb8ff0ce4e2e3e86e2bc9032ae8c0", "5d4403ad386547bcba1ba024fd2445a3a92b8caff2484185ed0d3b249c84ffc3", "b0b3168b4170993c8431f6ce2280394127f98fcacb422ca22012ff9ef5c5b861", "6825e7beabb278b00dfc6c7ebdc8c4c9e2fa78a3f307a24c572c15c2ccfabe79", "98964c15c9acf35c22dc1d014fbffc114c5...
1.639
chembl:1528623
O=C(c1cc(F)ccc1-c1ncccn1)N1C2CCC1C(COc1ccc(F)cn1)C2
d7207e8bed5f155a3340f4f9d54a0d901c8c847e60ed01872e23a3f976426495
[ "Cc1ccc(-c2ncccc2C)c(C(=O)N2C3CCC2C(COc2ncc(F)cn2)C3)n1", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(Nc2ccc(F)cn2)C3)n1", "Cc1coc(-c2ccc(C)nc2C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "Cc1ccc2ncc(C)n2c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "O=C(c1cccc(F)c1-c1ncccn1)N1C2CCC1C(Oc1ncc(C(F)(F)F)cn1)C2", "COc1cccc(-c2c(C)cnn2C)c1C(=O...
[ "36109ccd9045a0bcccf71ab97db1b74a977cb8ff0ce4e2e3e86e2bc9032ae8c0", "5d4403ad386547bcba1ba024fd2445a3a92b8caff2484185ed0d3b249c84ffc3", "b0b3168b4170993c8431f6ce2280394127f98fcacb422ca22012ff9ef5c5b861", "6825e7beabb278b00dfc6c7ebdc8c4c9e2fa78a3f307a24c572c15c2ccfabe79", "98964c15c9acf35c22dc1d014fbffc114c5...
1.638667
chembl:1528623
O=C(c1cc(F)ccc1-c1ncccn1)N1C2CCC1C(COc1ccc(F)cn1)C2
d7207e8bed5f155a3340f4f9d54a0d901c8c847e60ed01872e23a3f976426495
[ "Cc1ccc(N2CCN(C)CC2)c(C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "CCOc1ccc(C)nc1C(=O)N1C2CCC1C(Nc1ncc(C(F)(F)F)cn1)C2", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2ccncn2)C3)n1", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(Nc2ncc(C(F)(F)F)cn2)C3)n1", "Cc1nc2sccn2c1C(=O)N1C2CCC1C(Nc1cnc(C(F)(F)F)cn1)C2", "Cc1ccc(-c2ncccc2C)c(C(=O)...
[ "cbb8f3bd86c4cc9f3ebd57d0bdcd6bd5c40685655b02798c55f1bea424dbc256", "40435856f94f24c747098de3efdb17a97a131b832dfc7b041b97990cc471f209", "044d1c0bc4b04fe457f6bf55d8f7cf479e69aa6c7059d8721b792764429549c6", "89930909d6fa3919baedfc9715ad4ab38904f07519acd1e989298aa64d7056e7", "415999c57362169c3175f63f495c5c99c70...
1.638667
chembl:1528623
O=C(c1c(F)cccc1-c1ncccn1)N1C2CCC1C(COc1ccc(F)cn1)C2
44470232a93bf381e4afb0c7d7311d023e5e6c4a9c800426b36f92bb8cbd8ed6
[ "Cc1ccc(N2CCN(C)CC2)c(C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "CCOc1ccc(C)nc1C(=O)N1C2CCC1C(Nc1ncc(C(F)(F)F)cn1)C2", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2ccncn2)C3)n1", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(Nc2ncc(C(F)(F)F)cn2)C3)n1", "Cc1nc2sccn2c1C(=O)N1C2CCC1C(Nc1cnc(C(F)(F)F)cn1)C2", "Cc1ccc(-c2ncccc2C)c(C(=O)...
[ "cbb8f3bd86c4cc9f3ebd57d0bdcd6bd5c40685655b02798c55f1bea424dbc256", "40435856f94f24c747098de3efdb17a97a131b832dfc7b041b97990cc471f209", "044d1c0bc4b04fe457f6bf55d8f7cf479e69aa6c7059d8721b792764429549c6", "89930909d6fa3919baedfc9715ad4ab38904f07519acd1e989298aa64d7056e7", "415999c57362169c3175f63f495c5c99c70...
1.638667
chembl:1528623
O=C(c1c(F)cccc1-c1ncccn1)N1C2CCC1C(COc1ccc(F)cn1)C2
44470232a93bf381e4afb0c7d7311d023e5e6c4a9c800426b36f92bb8cbd8ed6
[ "Cc1ccc(N2CCOCC2)c(C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2cccnn2)C3)n1", "CN(c1cnc(C(F)(F)F)cn1)C1CC2CCC1N2C(=O)c1cccc(F)c1-c1ncccn1", "CCOc1ccnc(Cl)c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "Cc1ccc(C(=O)N2C3CCC2C(Nc2cnc(C(F)(F)F)cn2)C3)c(-n2ccnn2)n1", "O=C(c1cccc(F)c1-c1ccnnc1)N1C...
[ "26ed93e3488d6848a5d64cab7d440bd8f08c34ba506e9794bd961ffade785410", "96f2147056fb0dd194524eb0ca901fe41858e297da984fe4b1b75e8bf073d78e", "8e43077cb76b57f77f592c35d9c8814cda81696da4b10d44e2b392e1ca263462", "789d07cde0f56daaa9339ad1aec7b6f6f6436c22b7d078256809a8484a508068", "80101f4f7a5fede239dedf39c500921e45c...
1.638667
chembl:1528623
O=C(c1cc(Cl)ccc1-n1nccn1)N1C2CCC1C(COc1ccc(F)cn1)C2
2a3fd91d2d1fe6fb6fb92c4b2733b8719c2f7878eea951cd34b4b5eb793bb38c
[ "Cc1ccc(N2CCOCC2)c(C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2cccnn2)C3)n1", "CN(c1cnc(C(F)(F)F)cn1)C1CC2CCC1N2C(=O)c1cccc(F)c1-c1ncccn1", "CCOc1ccnc(Cl)c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "Cc1ccc(C(=O)N2C3CCC2C(Nc2cnc(C(F)(F)F)cn2)C3)c(-n2ccnn2)n1", "O=C(c1cccc(F)c1-c1ccnnc1)N1C...
[ "26ed93e3488d6848a5d64cab7d440bd8f08c34ba506e9794bd961ffade785410", "96f2147056fb0dd194524eb0ca901fe41858e297da984fe4b1b75e8bf073d78e", "8e43077cb76b57f77f592c35d9c8814cda81696da4b10d44e2b392e1ca263462", "789d07cde0f56daaa9339ad1aec7b6f6f6436c22b7d078256809a8484a508068", "80101f4f7a5fede239dedf39c500921e45c...
1.638667
chembl:1528623
O=C(c1cc(Cl)ccc1-n1nccn1)N1C2CCC1C(COc1ccc(F)cn1)C2
2a3fd91d2d1fe6fb6fb92c4b2733b8719c2f7878eea951cd34b4b5eb793bb38c
[ "Cc1ccc(C(=O)N2C3CCC2C(COc2ccccn2)C3)c(-n2nccn2)n1", "Cc1ccc(C(=O)N2C3CCC2C(COc2nccc(C(F)(F)F)n2)C3)c(-n2nccn2)n1", "Cc1cc(C)nc(OCC2CC3CCC2N3C(=O)c2ccc(C)nc2-n2nccn2)n1", "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1ccc(C(F)(F)F)cn1)C2", "Cc1ccc2nccn2c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "Cc1ccn2ccnc2c1C(=O)N1C2CCC1C(COc1c...
[ "8cf62ab90226119046e3cb3a7154a8867bdf1d30da12cf4c73d6c2cf31ce4729", "63e5f5d544ab2dd60cdfe624c583725d7be7430cefb333c678ec7061b868896b", "2b8c02902d2f3c6a9ccf486c1220ab2b48822aeafee58748db4e242fef3d04ca", "d94db68cefb332689168cbfd14ab6d50f89f728034b8e6c8de5187cf86df45d3", "e958358280dce37a463d061032e29c68a16...
1.638667
chembl:1528623
Cc1cccc(C(=O)N2C3CCC2C(COc2ccc(F)cn2)C3)c1-n1nccn1
92ca09d5a5798e61a9b71d64695090c460c54df4fc9072fc8bb2844c65db4f42
[ "Cc1ccc(C(=O)N2C3CCC2C(COc2ccccn2)C3)c(-n2nccn2)n1", "Cc1ccc(C(=O)N2C3CCC2C(COc2nccc(C(F)(F)F)n2)C3)c(-n2nccn2)n1", "Cc1cc(C)nc(OCC2CC3CCC2N3C(=O)c2ccc(C)nc2-n2nccn2)n1", "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1ccc(C(F)(F)F)cn1)C2", "Cc1ccc2nccn2c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "Cc1ccn2ccnc2c1C(=O)N1C2CCC1C(COc1c...
[ "8cf62ab90226119046e3cb3a7154a8867bdf1d30da12cf4c73d6c2cf31ce4729", "63e5f5d544ab2dd60cdfe624c583725d7be7430cefb333c678ec7061b868896b", "2b8c02902d2f3c6a9ccf486c1220ab2b48822aeafee58748db4e242fef3d04ca", "d94db68cefb332689168cbfd14ab6d50f89f728034b8e6c8de5187cf86df45d3", "e958358280dce37a463d061032e29c68a16...
1.637667
chembl:1528623
Cc1cccc(C(=O)N2C3CCC2C(COc2ccc(F)cn2)C3)c1-n1nccn1
92ca09d5a5798e61a9b71d64695090c460c54df4fc9072fc8bb2844c65db4f42
[ "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1ccc(F)cn1)C2", "Cc1nc2sccn2c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1cnc3ccccc3n1)C2", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2cnccn2)C3)n1", "CCOc1ncc(-c2ccccc2)cc1C(=O)N1C2CCC1C(COc1ccccn1)C2", "COC(=O)c1cnc(NC2CC3CCC2N3C(=O)c2cccc(F)c2-c2ncccn2)cn1",...
[ "1dc92dac322cafa93f066deaecf37843451f1f38f1f5a093ce6cdff154d24f50", "61611e5a16d66b1b35b9ee02c63c8540270c28b014f0894789c1a7b8879ceb1c", "09cb13eaf193692e39cc3183c06ceba07a4286fbaeda4627fed41570663984c1", "cd797d064c76d299c8c9b41b2766591a4d5daa2262efeeab5a350f926365283e", "f4fb1ed2df616dcb13ed4bbc598e86e154c...
1.637667
chembl:1528623
O=C(c1cccc(F)c1-c1ncccn1)N1C2CCC1C(Nc1nccn3c(Br)cnc13)C2
9a04f3f2b2dc7056f4848264c3b0f42977dea417c49e03628ec40d46db181a4a
[ "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1ccc(F)cn1)C2", "Cc1nc2sccn2c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1cnc3ccccc3n1)C2", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2cnccn2)C3)n1", "CCOc1ncc(-c2ccccc2)cc1C(=O)N1C2CCC1C(COc1ccccn1)C2", "COC(=O)c1cnc(NC2CC3CCC2N3C(=O)c2cccc(F)c2-c2ncccn2)cn1",...
[ "1dc92dac322cafa93f066deaecf37843451f1f38f1f5a093ce6cdff154d24f50", "61611e5a16d66b1b35b9ee02c63c8540270c28b014f0894789c1a7b8879ceb1c", "09cb13eaf193692e39cc3183c06ceba07a4286fbaeda4627fed41570663984c1", "cd797d064c76d299c8c9b41b2766591a4d5daa2262efeeab5a350f926365283e", "f4fb1ed2df616dcb13ed4bbc598e86e154c...
1.636333
chembl:1528623
O=C(c1cccc(F)c1-c1ncccn1)N1C2CCC1C(Nc1nccn3c(Br)cnc13)C2
9a04f3f2b2dc7056f4848264c3b0f42977dea417c49e03628ec40d46db181a4a
[ "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(Nc2ccc(F)cn2)C3)n1", "Cc1coc(-c2ccc(C)nc2C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "Cc1ccc2ncc(C)n2c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "O=C(c1cccc(F)c1-c1ncccn1)N1C2CCC1C(Oc1ncc(C(F)(F)F)cn1)C2", "COc1cccc(-c2c(C)cnn2C)c1C(=O)N1C2CCC1C(Nc1cnc(C(F)(F)F)cn1)C2", "O=C(c1nc2ccccc2[nH]1)...
[ "5d4403ad386547bcba1ba024fd2445a3a92b8caff2484185ed0d3b249c84ffc3", "b0b3168b4170993c8431f6ce2280394127f98fcacb422ca22012ff9ef5c5b861", "6825e7beabb278b00dfc6c7ebdc8c4c9e2fa78a3f307a24c572c15c2ccfabe79", "98964c15c9acf35c22dc1d014fbffc114c58178b0af6f9a36b9253f576befcda", "6c9cb367b275a634cb4095ebb2ab7f6168d...
1.636333
chembl:1528623
O=C(c1cc(F)ccc1-n1nccn1)N1C2CCC1C(COc1ccc(F)cn1)C2
5e8047b8c2a880ecaf46bf39630a1cededb9d9843be6c8d57a6e561c13065b61
[ "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(Nc2ccc(F)cn2)C3)n1", "Cc1coc(-c2ccc(C)nc2C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "Cc1ccc2ncc(C)n2c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "O=C(c1cccc(F)c1-c1ncccn1)N1C2CCC1C(Oc1ncc(C(F)(F)F)cn1)C2", "COc1cccc(-c2c(C)cnn2C)c1C(=O)N1C2CCC1C(Nc1cnc(C(F)(F)F)cn1)C2", "O=C(c1nc2ccccc2[nH]1)...
[ "5d4403ad386547bcba1ba024fd2445a3a92b8caff2484185ed0d3b249c84ffc3", "b0b3168b4170993c8431f6ce2280394127f98fcacb422ca22012ff9ef5c5b861", "6825e7beabb278b00dfc6c7ebdc8c4c9e2fa78a3f307a24c572c15c2ccfabe79", "98964c15c9acf35c22dc1d014fbffc114c58178b0af6f9a36b9253f576befcda", "6c9cb367b275a634cb4095ebb2ab7f6168d...
1.636
chembl:1528623
O=C(c1cc(F)ccc1-n1nccn1)N1C2CCC1C(COc1ccc(F)cn1)C2
5e8047b8c2a880ecaf46bf39630a1cededb9d9843be6c8d57a6e561c13065b61
[ "CCOc1ccc(C)nc1C(=O)N1C2CCC1C(Nc1ncc(C(F)(F)F)cn1)C2", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2ccncn2)C3)n1", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(Nc2ncc(C(F)(F)F)cn2)C3)n1", "Cc1nc2sccn2c1C(=O)N1C2CCC1C(Nc1cnc(C(F)(F)F)cn1)C2", "Cc1ccc(-c2ncccc2C)c(C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "Cc1ccc(-n2nccn2)c(C(=O)N2C...
[ "40435856f94f24c747098de3efdb17a97a131b832dfc7b041b97990cc471f209", "044d1c0bc4b04fe457f6bf55d8f7cf479e69aa6c7059d8721b792764429549c6", "89930909d6fa3919baedfc9715ad4ab38904f07519acd1e989298aa64d7056e7", "415999c57362169c3175f63f495c5c99c70468338f1f4a4a02d11c65cee361fe", "3681e2e80df961ea6c6913cbc4210c3c51d...
1.636
chembl:1528623
CCOc1ccnc(OCC)c1C(=O)N1C2CCC1C(COc1ccccn1)C2
501b5793db3bbfc5f93ad2661625aa4a88e8267720f5e88ea85cb61b3260b771
[ "CCOc1ccc(C)nc1C(=O)N1C2CCC1C(Nc1ncc(C(F)(F)F)cn1)C2", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2ccncn2)C3)n1", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(Nc2ncc(C(F)(F)F)cn2)C3)n1", "Cc1nc2sccn2c1C(=O)N1C2CCC1C(Nc1cnc(C(F)(F)F)cn1)C2", "Cc1ccc(-c2ncccc2C)c(C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "Cc1ccc(-n2nccn2)c(C(=O)N2C...
[ "40435856f94f24c747098de3efdb17a97a131b832dfc7b041b97990cc471f209", "044d1c0bc4b04fe457f6bf55d8f7cf479e69aa6c7059d8721b792764429549c6", "89930909d6fa3919baedfc9715ad4ab38904f07519acd1e989298aa64d7056e7", "415999c57362169c3175f63f495c5c99c70468338f1f4a4a02d11c65cee361fe", "3681e2e80df961ea6c6913cbc4210c3c51d...
1.635667
chembl:1528623
CCOc1ccnc(OCC)c1C(=O)N1C2CCC1C(COc1ccccn1)C2
501b5793db3bbfc5f93ad2661625aa4a88e8267720f5e88ea85cb61b3260b771
[ "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2cccnn2)C3)n1", "CN(c1cnc(C(F)(F)F)cn1)C1CC2CCC1N2C(=O)c1cccc(F)c1-c1ncccn1", "CCOc1ccnc(Cl)c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "Cc1ccc(C(=O)N2C3CCC2C(Nc2cnc(C(F)(F)F)cn2)C3)c(-n2ccnn2)n1", "O=C(c1cccc(F)c1-c1ccnnc1)N1C2CCC1C(Nc1cnc(C(F)(F)F)cn1)C2", "COc1c(F)cccc1C(=O)N1...
[ "96f2147056fb0dd194524eb0ca901fe41858e297da984fe4b1b75e8bf073d78e", "8e43077cb76b57f77f592c35d9c8814cda81696da4b10d44e2b392e1ca263462", "789d07cde0f56daaa9339ad1aec7b6f6f6436c22b7d078256809a8484a508068", "80101f4f7a5fede239dedf39c500921e45c84cb244df3dfb40e7befb00d66ecb", "e921ccd1898af4d7c7829e8120e77c95c1c...
1.635667
chembl:1528623
COc1cccc(OC)c1C(=O)N1C2CCC1C(COc1ccc(F)cn1)C2
b9a29f95ba5f75064bdfd890b59b66005f010eaac9c6a6d801a5d484f05d2bfb
[ "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2cccnn2)C3)n1", "CN(c1cnc(C(F)(F)F)cn1)C1CC2CCC1N2C(=O)c1cccc(F)c1-c1ncccn1", "CCOc1ccnc(Cl)c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "Cc1ccc(C(=O)N2C3CCC2C(Nc2cnc(C(F)(F)F)cn2)C3)c(-n2ccnn2)n1", "O=C(c1cccc(F)c1-c1ccnnc1)N1C2CCC1C(Nc1cnc(C(F)(F)F)cn1)C2", "COc1c(F)cccc1C(=O)N1...
[ "96f2147056fb0dd194524eb0ca901fe41858e297da984fe4b1b75e8bf073d78e", "8e43077cb76b57f77f592c35d9c8814cda81696da4b10d44e2b392e1ca263462", "789d07cde0f56daaa9339ad1aec7b6f6f6436c22b7d078256809a8484a508068", "80101f4f7a5fede239dedf39c500921e45c84cb244df3dfb40e7befb00d66ecb", "e921ccd1898af4d7c7829e8120e77c95c1c...
1.635333
chembl:1528623
COc1cccc(OC)c1C(=O)N1C2CCC1C(COc1ccc(F)cn1)C2
b9a29f95ba5f75064bdfd890b59b66005f010eaac9c6a6d801a5d484f05d2bfb
[ "Cc1ccc(C(=O)N2C3CCC2C(COc2nccc(C(F)(F)F)n2)C3)c(-n2nccn2)n1", "Cc1cc(C)nc(OCC2CC3CCC2N3C(=O)c2ccc(C)nc2-n2nccn2)n1", "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1ccc(C(F)(F)F)cn1)C2", "Cc1ccc2nccn2c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "Cc1ccn2ccnc2c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "Cc1ccc(N2CCNCC2)c(C(=O)N2C3CCC2C(COc2cccc...
[ "63e5f5d544ab2dd60cdfe624c583725d7be7430cefb333c678ec7061b868896b", "2b8c02902d2f3c6a9ccf486c1220ab2b48822aeafee58748db4e242fef3d04ca", "d94db68cefb332689168cbfd14ab6d50f89f728034b8e6c8de5187cf86df45d3", "e958358280dce37a463d061032e29c68a168803e94062a7562d68d020f372796", "515ea2ffa8807a7f0a6787e40ea05eeadb5...
1.635333
chembl:1528623
Cc1ccc2ccccc2c1C(=O)N1C2CCC1C(COc1ccc(F)cn1)C2
4522a208ceca5cedba7d2b14d1e3efe587fa4c84e02bffa82953009123af48b1
[ "Cc1ccc(C(=O)N2C3CCC2C(COc2nccc(C(F)(F)F)n2)C3)c(-n2nccn2)n1", "Cc1cc(C)nc(OCC2CC3CCC2N3C(=O)c2ccc(C)nc2-n2nccn2)n1", "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1ccc(C(F)(F)F)cn1)C2", "Cc1ccc2nccn2c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "Cc1ccn2ccnc2c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "Cc1ccc(N2CCNCC2)c(C(=O)N2C3CCC2C(COc2cccc...
[ "63e5f5d544ab2dd60cdfe624c583725d7be7430cefb333c678ec7061b868896b", "2b8c02902d2f3c6a9ccf486c1220ab2b48822aeafee58748db4e242fef3d04ca", "d94db68cefb332689168cbfd14ab6d50f89f728034b8e6c8de5187cf86df45d3", "e958358280dce37a463d061032e29c68a168803e94062a7562d68d020f372796", "515ea2ffa8807a7f0a6787e40ea05eeadb5...
1.635
chembl:1528623
Cc1ccc2ccccc2c1C(=O)N1C2CCC1C(COc1ccc(F)cn1)C2
4522a208ceca5cedba7d2b14d1e3efe587fa4c84e02bffa82953009123af48b1
[ "Cc1nc2sccn2c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1cnc3ccccc3n1)C2", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2cnccn2)C3)n1", "CCOc1ncc(-c2ccccc2)cc1C(=O)N1C2CCC1C(COc1ccccn1)C2", "COC(=O)c1cnc(NC2CC3CCC2N3C(=O)c2cccc(F)c2-c2ncccn2)cn1", "Cc1ccc(-c2ncccc2C)c(C(=O)N2C3CCC2C(COc2ncc(F)...
[ "61611e5a16d66b1b35b9ee02c63c8540270c28b014f0894789c1a7b8879ceb1c", "09cb13eaf193692e39cc3183c06ceba07a4286fbaeda4627fed41570663984c1", "cd797d064c76d299c8c9b41b2766591a4d5daa2262efeeab5a350f926365283e", "f4fb1ed2df616dcb13ed4bbc598e86e154c2b00f6adece9224846c878b4f2600", "fc30614a06906da50ef26facdc1824dde53...
1.635
chembl:1528623
O=C(c1cccc2ccccc12)N1C2CCC1C(COc1ccc(F)cn1)C2
3267e2f8b2b05998130564f308471c49e7d3074c4494919df05d4fd7124bfe6e
[ "Cc1nc2sccn2c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1cnc3ccccc3n1)C2", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2cnccn2)C3)n1", "CCOc1ncc(-c2ccccc2)cc1C(=O)N1C2CCC1C(COc1ccccn1)C2", "COC(=O)c1cnc(NC2CC3CCC2N3C(=O)c2cccc(F)c2-c2ncccn2)cn1", "Cc1ccc(-c2ncccc2C)c(C(=O)N2C3CCC2C(COc2ncc(F)...
[ "61611e5a16d66b1b35b9ee02c63c8540270c28b014f0894789c1a7b8879ceb1c", "09cb13eaf193692e39cc3183c06ceba07a4286fbaeda4627fed41570663984c1", "cd797d064c76d299c8c9b41b2766591a4d5daa2262efeeab5a350f926365283e", "f4fb1ed2df616dcb13ed4bbc598e86e154c2b00f6adece9224846c878b4f2600", "fc30614a06906da50ef26facdc1824dde53...
1.634667
chembl:1528623
O=C(c1cccc2ccccc12)N1C2CCC1C(COc1ccc(F)cn1)C2
3267e2f8b2b05998130564f308471c49e7d3074c4494919df05d4fd7124bfe6e
[ "Cc1coc(-c2ccc(C)nc2C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "Cc1ccc2ncc(C)n2c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "O=C(c1cccc(F)c1-c1ncccn1)N1C2CCC1C(Oc1ncc(C(F)(F)F)cn1)C2", "COc1cccc(-c2c(C)cnn2C)c1C(=O)N1C2CCC1C(Nc1cnc(C(F)(F)F)cn1)C2", "O=C(c1nc2ccccc2[nH]1)N1C2CCC1C(Nc1cnc(C(F)(F)F)cn1)C2", "Cc1ccc(N2CCN(C)CC2)...
[ "b0b3168b4170993c8431f6ce2280394127f98fcacb422ca22012ff9ef5c5b861", "6825e7beabb278b00dfc6c7ebdc8c4c9e2fa78a3f307a24c572c15c2ccfabe79", "98964c15c9acf35c22dc1d014fbffc114c58178b0af6f9a36b9253f576befcda", "6c9cb367b275a634cb4095ebb2ab7f6168d34c9e60f9e5b0ada8b654da7820b6", "ff399b820cb3201b68c2d6b88b386d824aa...
1.634667
chembl:1528623
COc1cccc(-c2ncccn2)c1C(=O)N1C2CCC1C(Nc1cnc(C(F)(F)F)cn1)C2
07af980624881ef3a23caa6afecc8b2c5c7a87694698f1c627892cbbc5330bd5
[ "Cc1coc(-c2ccc(C)nc2C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "Cc1ccc2ncc(C)n2c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "O=C(c1cccc(F)c1-c1ncccn1)N1C2CCC1C(Oc1ncc(C(F)(F)F)cn1)C2", "COc1cccc(-c2c(C)cnn2C)c1C(=O)N1C2CCC1C(Nc1cnc(C(F)(F)F)cn1)C2", "O=C(c1nc2ccccc2[nH]1)N1C2CCC1C(Nc1cnc(C(F)(F)F)cn1)C2", "Cc1ccc(N2CCN(C)CC2)...
[ "b0b3168b4170993c8431f6ce2280394127f98fcacb422ca22012ff9ef5c5b861", "6825e7beabb278b00dfc6c7ebdc8c4c9e2fa78a3f307a24c572c15c2ccfabe79", "98964c15c9acf35c22dc1d014fbffc114c58178b0af6f9a36b9253f576befcda", "6c9cb367b275a634cb4095ebb2ab7f6168d34c9e60f9e5b0ada8b654da7820b6", "ff399b820cb3201b68c2d6b88b386d824aa...
1.633667
chembl:1528623
COc1cccc(-c2ncccn2)c1C(=O)N1C2CCC1C(Nc1cnc(C(F)(F)F)cn1)C2
07af980624881ef3a23caa6afecc8b2c5c7a87694698f1c627892cbbc5330bd5
[ "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2ccncn2)C3)n1", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(Nc2ncc(C(F)(F)F)cn2)C3)n1", "Cc1nc2sccn2c1C(=O)N1C2CCC1C(Nc1cnc(C(F)(F)F)cn1)C2", "Cc1ccc(-c2ncccc2C)c(C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2ccnn2C)C3)n1", "Cc1ccc(N2CCOCC2)c(C(=O)N2C3C...
[ "044d1c0bc4b04fe457f6bf55d8f7cf479e69aa6c7059d8721b792764429549c6", "89930909d6fa3919baedfc9715ad4ab38904f07519acd1e989298aa64d7056e7", "415999c57362169c3175f63f495c5c99c70468338f1f4a4a02d11c65cee361fe", "3681e2e80df961ea6c6913cbc4210c3c51d5ed170599dfe37a24d74d93670018", "0d0020e25910a43ee85f87dbcb7222c4e82...
1.633667
chembl:1528623
Cc1cc(-c2ccc(C)nc2C(=O)N2C3CCC2C(COc2ccc(F)cn2)C3)on1
cfb03841b690d9f56783c69bf943ed48e9e8633182e4229579409cb111f84c54
[ "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2ccncn2)C3)n1", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(Nc2ncc(C(F)(F)F)cn2)C3)n1", "Cc1nc2sccn2c1C(=O)N1C2CCC1C(Nc1cnc(C(F)(F)F)cn1)C2", "Cc1ccc(-c2ncccc2C)c(C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2ccnn2C)C3)n1", "Cc1ccc(N2CCOCC2)c(C(=O)N2C3C...
[ "044d1c0bc4b04fe457f6bf55d8f7cf479e69aa6c7059d8721b792764429549c6", "89930909d6fa3919baedfc9715ad4ab38904f07519acd1e989298aa64d7056e7", "415999c57362169c3175f63f495c5c99c70468338f1f4a4a02d11c65cee361fe", "3681e2e80df961ea6c6913cbc4210c3c51d5ed170599dfe37a24d74d93670018", "0d0020e25910a43ee85f87dbcb7222c4e82...
1.633667
chembl:1528623
Cc1cc(-c2ccc(C)nc2C(=O)N2C3CCC2C(COc2ccc(F)cn2)C3)on1
cfb03841b690d9f56783c69bf943ed48e9e8633182e4229579409cb111f84c54
[ "CN(c1cnc(C(F)(F)F)cn1)C1CC2CCC1N2C(=O)c1cccc(F)c1-c1ncccn1", "CCOc1ccnc(Cl)c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "Cc1ccc(C(=O)N2C3CCC2C(Nc2cnc(C(F)(F)F)cn2)C3)c(-n2ccnn2)n1", "O=C(c1cccc(F)c1-c1ccnnc1)N1C2CCC1C(Nc1cnc(C(F)(F)F)cn1)C2", "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1ncc(C(F)(F)F)cn1)C2", "Cc1ccc(C(=O)N2C3CCC...
[ "8e43077cb76b57f77f592c35d9c8814cda81696da4b10d44e2b392e1ca263462", "789d07cde0f56daaa9339ad1aec7b6f6f6436c22b7d078256809a8484a508068", "80101f4f7a5fede239dedf39c500921e45c84cb244df3dfb40e7befb00d66ecb", "e921ccd1898af4d7c7829e8120e77c95c1c534456e4d2742ae11c3b3dff3baea", "b97f4a41a5cedfb00c3157f3b9e94037650...
1.633667
chembl:1528623
O=C(c1cccc(F)c1-c1cnccn1)N1C2CCC1C(Nc1cnc(C(F)(F)F)cn1)C2
bb6f4ed77d45228b53aaafae868309e2c82040ecc8b050b91b40cc45f43e0cd4
[ "CN(c1cnc(C(F)(F)F)cn1)C1CC2CCC1N2C(=O)c1cccc(F)c1-c1ncccn1", "CCOc1ccnc(Cl)c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "Cc1ccc(C(=O)N2C3CCC2C(Nc2cnc(C(F)(F)F)cn2)C3)c(-n2ccnn2)n1", "O=C(c1cccc(F)c1-c1ccnnc1)N1C2CCC1C(Nc1cnc(C(F)(F)F)cn1)C2", "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1ncc(C(F)(F)F)cn1)C2", "Cc1ccc(C(=O)N2C3CCC...
[ "8e43077cb76b57f77f592c35d9c8814cda81696da4b10d44e2b392e1ca263462", "789d07cde0f56daaa9339ad1aec7b6f6f6436c22b7d078256809a8484a508068", "80101f4f7a5fede239dedf39c500921e45c84cb244df3dfb40e7befb00d66ecb", "e921ccd1898af4d7c7829e8120e77c95c1c534456e4d2742ae11c3b3dff3baea", "b97f4a41a5cedfb00c3157f3b9e94037650...
1.632667
chembl:1528623
O=C(c1cccc(F)c1-c1cnccn1)N1C2CCC1C(Nc1cnc(C(F)(F)F)cn1)C2
bb6f4ed77d45228b53aaafae868309e2c82040ecc8b050b91b40cc45f43e0cd4
[ "Cc1cc(C)nc(OCC2CC3CCC2N3C(=O)c2ccc(C)nc2-n2nccn2)n1", "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1ccc(C(F)(F)F)cn1)C2", "Cc1ccc2nccn2c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "Cc1ccn2ccnc2c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "Cc1ccc(N2CCNCC2)c(C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1ccc(F)cn1)C2", "Cc...
[ "2b8c02902d2f3c6a9ccf486c1220ab2b48822aeafee58748db4e242fef3d04ca", "d94db68cefb332689168cbfd14ab6d50f89f728034b8e6c8de5187cf86df45d3", "e958358280dce37a463d061032e29c68a168803e94062a7562d68d020f372796", "515ea2ffa8807a7f0a6787e40ea05eeadb5601cef8c45a785cc877ac4bede677", "0fc0e284b6f14795dd5431215829a32c441...
1.632667
chembl:1528623
Cc1cccc(OCC2CC3CCC2N3C(=O)c2nc(C)ccc2-n2nccn2)n1
319f4c904d6fef08a20419b951c801f896f91dc6dd68da12af328f681fd574d9
[ "Cc1cc(C)nc(OCC2CC3CCC2N3C(=O)c2ccc(C)nc2-n2nccn2)n1", "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1ccc(C(F)(F)F)cn1)C2", "Cc1ccc2nccn2c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "Cc1ccn2ccnc2c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "Cc1ccc(N2CCNCC2)c(C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1ccc(F)cn1)C2", "Cc...
[ "2b8c02902d2f3c6a9ccf486c1220ab2b48822aeafee58748db4e242fef3d04ca", "d94db68cefb332689168cbfd14ab6d50f89f728034b8e6c8de5187cf86df45d3", "e958358280dce37a463d061032e29c68a168803e94062a7562d68d020f372796", "515ea2ffa8807a7f0a6787e40ea05eeadb5601cef8c45a785cc877ac4bede677", "0fc0e284b6f14795dd5431215829a32c441...
1.632667
chembl:1528623
Cc1cccc(OCC2CC3CCC2N3C(=O)c2nc(C)ccc2-n2nccn2)n1
319f4c904d6fef08a20419b951c801f896f91dc6dd68da12af328f681fd574d9
[ "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1cnc3ccccc3n1)C2", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2cnccn2)C3)n1", "CCOc1ncc(-c2ccccc2)cc1C(=O)N1C2CCC1C(COc1ccccn1)C2", "COC(=O)c1cnc(NC2CC3CCC2N3C(=O)c2cccc(F)c2-c2ncccn2)cn1", "Cc1ccc(-c2ncccc2C)c(C(=O)N2C3CCC2C(COc2ncc(F)cn2)C3)n1", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C...
[ "09cb13eaf193692e39cc3183c06ceba07a4286fbaeda4627fed41570663984c1", "cd797d064c76d299c8c9b41b2766591a4d5daa2262efeeab5a350f926365283e", "f4fb1ed2df616dcb13ed4bbc598e86e154c2b00f6adece9224846c878b4f2600", "fc30614a06906da50ef26facdc1824dde53eb44f09950784e41ca8bf3375f5cf", "36109ccd9045a0bcccf71ab97db1b74a977...
1.632667
chembl:1528623
Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2ccc(Br)cn2)C3)n1
1bad046e47e176692296cba4356b332561b5f35dceaf7afc311f7e0319a2891c
[ "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1cnc3ccccc3n1)C2", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2cnccn2)C3)n1", "CCOc1ncc(-c2ccccc2)cc1C(=O)N1C2CCC1C(COc1ccccn1)C2", "COC(=O)c1cnc(NC2CC3CCC2N3C(=O)c2cccc(F)c2-c2ncccn2)cn1", "Cc1ccc(-c2ncccc2C)c(C(=O)N2C3CCC2C(COc2ncc(F)cn2)C3)n1", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C...
[ "09cb13eaf193692e39cc3183c06ceba07a4286fbaeda4627fed41570663984c1", "cd797d064c76d299c8c9b41b2766591a4d5daa2262efeeab5a350f926365283e", "f4fb1ed2df616dcb13ed4bbc598e86e154c2b00f6adece9224846c878b4f2600", "fc30614a06906da50ef26facdc1824dde53eb44f09950784e41ca8bf3375f5cf", "36109ccd9045a0bcccf71ab97db1b74a977...
1.632333
chembl:1528623
Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2ccc(Br)cn2)C3)n1
1bad046e47e176692296cba4356b332561b5f35dceaf7afc311f7e0319a2891c
[ "Cc1ccc2ncc(C)n2c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "O=C(c1cccc(F)c1-c1ncccn1)N1C2CCC1C(Oc1ncc(C(F)(F)F)cn1)C2", "COc1cccc(-c2c(C)cnn2C)c1C(=O)N1C2CCC1C(Nc1cnc(C(F)(F)F)cn1)C2", "O=C(c1nc2ccccc2[nH]1)N1C2CCC1C(Nc1cnc(C(F)(F)F)cn1)C2", "Cc1ccc(N2CCN(C)CC2)c(C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "CCOc1ccc(C)nc1C(=...
[ "6825e7beabb278b00dfc6c7ebdc8c4c9e2fa78a3f307a24c572c15c2ccfabe79", "98964c15c9acf35c22dc1d014fbffc114c58178b0af6f9a36b9253f576befcda", "6c9cb367b275a634cb4095ebb2ab7f6168d34c9e60f9e5b0ada8b654da7820b6", "ff399b820cb3201b68c2d6b88b386d824aa8686b1bfdffca007e0038fe75d732", "cbb8f3bd86c4cc9f3ebd57d0bdcd6bd5c40...
1.632333
chembl:1528623
O=C(c1cccc(F)c1-n1nccn1)N1C2CCC1C(COc1cccc(C(F)(F)F)n1)C2
cea19ee59ae858ab274580636cf38760e9e604e20faa5ef224be6dd78eb57dd3
[ "Cc1ccc2ncc(C)n2c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "O=C(c1cccc(F)c1-c1ncccn1)N1C2CCC1C(Oc1ncc(C(F)(F)F)cn1)C2", "COc1cccc(-c2c(C)cnn2C)c1C(=O)N1C2CCC1C(Nc1cnc(C(F)(F)F)cn1)C2", "O=C(c1nc2ccccc2[nH]1)N1C2CCC1C(Nc1cnc(C(F)(F)F)cn1)C2", "Cc1ccc(N2CCN(C)CC2)c(C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "CCOc1ccc(C)nc1C(=...
[ "6825e7beabb278b00dfc6c7ebdc8c4c9e2fa78a3f307a24c572c15c2ccfabe79", "98964c15c9acf35c22dc1d014fbffc114c58178b0af6f9a36b9253f576befcda", "6c9cb367b275a634cb4095ebb2ab7f6168d34c9e60f9e5b0ada8b654da7820b6", "ff399b820cb3201b68c2d6b88b386d824aa8686b1bfdffca007e0038fe75d732", "cbb8f3bd86c4cc9f3ebd57d0bdcd6bd5c40...
1.632
chembl:1528623
O=C(c1cccc(F)c1-n1nccn1)N1C2CCC1C(COc1cccc(C(F)(F)F)n1)C2
cea19ee59ae858ab274580636cf38760e9e604e20faa5ef224be6dd78eb57dd3
[ "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(Nc2ncc(C(F)(F)F)cn2)C3)n1", "Cc1nc2sccn2c1C(=O)N1C2CCC1C(Nc1cnc(C(F)(F)F)cn1)C2", "Cc1ccc(-c2ncccc2C)c(C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2ccnn2C)C3)n1", "Cc1ccc(N2CCOCC2)c(C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "Cc1ccc(-n2nccn2)c(C(=O)N2C3C...
[ "89930909d6fa3919baedfc9715ad4ab38904f07519acd1e989298aa64d7056e7", "415999c57362169c3175f63f495c5c99c70468338f1f4a4a02d11c65cee361fe", "3681e2e80df961ea6c6913cbc4210c3c51d5ed170599dfe37a24d74d93670018", "0d0020e25910a43ee85f87dbcb7222c4e82730d8c8f60343a92a11836ae8069f", "26ed93e3488d6848a5d64cab7d440bd8f08...
1.632
chembl:1528623
CCOc1ncc2ccccc2c1C(=O)N1C2CCC1C(COc1ccccn1)C2
6c4d09b14d5163f2b06856fe2614c5b25437b930ec0e7fe8ba2911a7a7ce988f
[ "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(Nc2ncc(C(F)(F)F)cn2)C3)n1", "Cc1nc2sccn2c1C(=O)N1C2CCC1C(Nc1cnc(C(F)(F)F)cn1)C2", "Cc1ccc(-c2ncccc2C)c(C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "Cc1ccc(-n2nccn2)c(C(=O)N2C3CCC2C(COc2ccnn2C)C3)n1", "Cc1ccc(N2CCOCC2)c(C(=O)N2C3CCC2C(COc2ccccn2)C3)n1", "Cc1ccc(-n2nccn2)c(C(=O)N2C3C...
[ "89930909d6fa3919baedfc9715ad4ab38904f07519acd1e989298aa64d7056e7", "415999c57362169c3175f63f495c5c99c70468338f1f4a4a02d11c65cee361fe", "3681e2e80df961ea6c6913cbc4210c3c51d5ed170599dfe37a24d74d93670018", "0d0020e25910a43ee85f87dbcb7222c4e82730d8c8f60343a92a11836ae8069f", "26ed93e3488d6848a5d64cab7d440bd8f08...
1.632
chembl:1528623
CCOc1ncc2ccccc2c1C(=O)N1C2CCC1C(COc1ccccn1)C2
6c4d09b14d5163f2b06856fe2614c5b25437b930ec0e7fe8ba2911a7a7ce988f
[ "CCOc1ccnc(Cl)c1C(=O)N1C2CCC1C(COc1ccccn1)C2", "Cc1ccc(C(=O)N2C3CCC2C(Nc2cnc(C(F)(F)F)cn2)C3)c(-n2ccnn2)n1", "O=C(c1cccc(F)c1-c1ccnnc1)N1C2CCC1C(Nc1cnc(C(F)(F)F)cn1)C2", "COc1c(F)cccc1C(=O)N1C2CCC1C(Nc1ncc(C(F)(F)F)cn1)C2", "Cc1ccc(C(=O)N2C3CCC2C(COc2ccccn2)C3)c(-n2nccn2)n1", "Cc1ccc(C(=O)N2C3CCC2C(COc2nc...
[ "789d07cde0f56daaa9339ad1aec7b6f6f6436c22b7d078256809a8484a508068", "80101f4f7a5fede239dedf39c500921e45c84cb244df3dfb40e7befb00d66ecb", "e921ccd1898af4d7c7829e8120e77c95c1c534456e4d2742ae11c3b3dff3baea", "b97f4a41a5cedfb00c3157f3b9e940376503e4ed11ba86279269eea2696fa398", "8cf62ab90226119046e3cb3a7154a8867bd...
1.632
chembl:1535880
NC(=O)C(CCC(=O)O)NC(=O)C(CC(=O)O)NC(=O)CCc1ccc(-c2ccc(-c3ccccc3)cc2)cc1
8e89d3c265ac11fb2de4e7400fbbc7c470e852764262213c47f23d464430fdb0
[ "O=C(O)CCC(NC(=O)CCc1ccc(-c2ccccc2)cc1)C(=O)N1CCCC(CC(=O)O)C1", "NC(=O)C(CCC(=O)O)NC(=O)C(CCC(=O)O)NC(=O)CCc1ccc(-c2cccc(Cl)c2)cc1", "NC(=O)C(CCC(=O)O)NC(=O)C(CCC(=O)O)NC(=O)CCc1ccc(-c2cccc(C(=O)O)c2)cc1", "NC(=O)C(CCC(=O)O)NC(=O)C(CCC(=O)O)NC(=O)CCc1cc(-c2ccccc2)no1", "NC(=O)CCC(NC(=O)C(CCC(N)=O)NC(=O)CCc1...
[ "bcc49f01ba08faab2ed28c520f94a41a1b30a3f973aea75a81453ed26ae2358f", "b29e8c6b12595ffefe492ce920c37a2b0711309bdd6702a2c9497c1586883541", "4b35f85afc8249fd1c52ab99e610ff54ceafb313f14241a5c18f0bc46a160670", "2044dfc27bb11124e3d7f521b4af09125ad8a7c33a2d5f17cfb10a5f8e7e0a66", "52bd50101096ced90daf88027ed8b3bd6e9...
1.66
chembl:1535880
NC(=O)C(CCC(=O)O)NC(=O)C(CC(=O)O)NC(=O)CCc1ccc(-c2ccc(-c3ccccc3)cc2)cc1
8e89d3c265ac11fb2de4e7400fbbc7c470e852764262213c47f23d464430fdb0
[ "CC(NC(=O)C(CCC(=O)O)NC(=O)CCc1ccc(-c2ccccc2)cc1)C(N)=O", "NC(=O)CCC(NC(=O)C(CCC(=O)O)NC(=O)CCc1ccc(-c2cc(-c3ccccc3)cs2)cc1)C(N)=O", "NC(=O)C(CCC(=O)O)NC(=O)C(CCC(=O)O)NC(=O)CCc1ccc(COc2ccccc2)cc1", "NC(=O)CCC(NC(=O)CCc1ccc(-c2cc(-c3ccccc3)cs2)cc1)C(=O)NC(CCC(=O)O)C(N)=O", "NCCCCC(NC(=O)C(CCC(=O)O)NC(=O)CCc...
[ "5e05d238936509355581f4555e224f4f75ae7d6e59a647a72a0094413bd95b3a", "08b95b5a66463ca766c57a11a7b58ddafb26c1f00bdd17d76af89fc318a593a4", "87ed094d488a20f2383776ebd5d37e91c56a15e82eb4049b3624aa7781387058", "b6818b4a2358ee61cf3a991e8ab23af1e1f48ee6df127290f22c25e43b753edb", "a87dfb15727b454f62f7ddae4e0b72aaed6...
1.66
chembl:1535880
O=C(O)CCC(NC(=O)CCc1ccc(-c2ccc(-c3ccccc3)cc2)cc1)C(=O)Nc1cccc(CC(=O)O)c1
2f4067f36f417b3671802836134418834e192f8e67db7a457e8edb72e3279ba2
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chembl:1535880
O=C(O)CCC(NC(=O)CCc1ccc(-c2ccc(-c3ccccc3)cc2)cc1)C(=O)Nc1cccc(CC(=O)O)c1
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chembl:1535880
NC(=O)C(CCC(=O)O)NC(=O)C(CCC(=O)O)NC(=O)CCc1cc(-c2ccc(-c3cccc(Cl)c3)cc2)no1
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1.640333
chembl:1535880
NC(=O)C(CCC(=O)O)NC(=O)C(CCC(=O)O)NC(=O)CCc1cc(-c2ccc(-c3cccc(Cl)c3)cc2)no1
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1.640333
chembl:1535880
NC(=O)C(CCC(=O)O)NC(=O)C(CCC(=O)O)NC(=O)CCc1ccc(-c2ccc(-c3ccccc3)cc2)cc1
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1.639667
chembl:1535880
NC(=O)C(CCC(=O)O)NC(=O)C(CCC(=O)O)NC(=O)CCc1ccc(-c2ccc(-c3ccccc3)cc2)cc1
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chembl:1535880
CCC(NC(=O)CCc1cc(-c2ccc(-c3ccccc3)cc2)no1)C(=O)NC(CCC(=O)O)C(N)=O
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chembl:1535880
CCC(NC(=O)CCc1cc(-c2ccc(-c3ccccc3)cc2)no1)C(=O)NC(CCC(=O)O)C(N)=O
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1.637
chembl:1535880
NC(=O)C(CC(=O)O)NC(=O)C(CC(=O)O)NC(=O)CCc1cc(-c2ccc(-c3cccc(Cl)c3)cc2)no1
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1.635667
chembl:1535880
NC(=O)C(CC(=O)O)NC(=O)C(CC(=O)O)NC(=O)CCc1cc(-c2ccc(-c3cccc(Cl)c3)cc2)no1
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1.635667
chembl:1535880
CCC(NC(=O)CCc1ccc(-c2nc3ccccc3s2)cc1)C(=O)NC(CCC(=O)O)C(N)=O
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1.635333
chembl:1535880
CCC(NC(=O)CCc1ccc(-c2nc3ccccc3s2)cc1)C(=O)NC(CCC(=O)O)C(N)=O
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1.635333
chembl:1535880
NC(=O)CCC(NC(=O)C(CCC(=O)O)NC(=O)CCc1cc(-c2ccc(-c3ccccc3)cc2)no1)C(N)=O
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1.632667
chembl:1535880
NC(=O)CCC(NC(=O)C(CCC(=O)O)NC(=O)CCc1cc(-c2ccc(-c3ccccc3)cc2)no1)C(N)=O
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1.632667
chembl:1535880
NC(=O)C(CCC(=O)O)NC(=O)C(CCC(=O)O)NC(=O)CCc1ccc(-c2ccc(-c3ccccc3)s2)cc1
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1.632333
chembl:1535880
NC(=O)C(CCC(=O)O)NC(=O)C(CCC(=O)O)NC(=O)CCc1ccc(-c2ccc(-c3ccccc3)s2)cc1
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chembl:1535880
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chembl:1535880
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chembl:1535880
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chembl:1535880
NC(=O)C(CCC(=O)O)NC(=O)C(CO)NC(=O)CCc1ccc(-c2ccc(-c3ccccc3)cc2)cc1
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1.631333
chembl:1535880
NC(=O)C(CCC(=O)O)NC(=O)CCc1cc(-c2ccc(-c3cccc(Cl)c3)cc2)no1
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chembl:1535880
NC(=O)C(CCC(=O)O)NC(=O)CCc1cc(-c2ccc(-c3cccc(Cl)c3)cc2)no1
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chembl:1535880
NC(=O)C(CCCC(=O)O)NC(=O)C(CCC(=O)O)NC(=O)CCc1cc(-c2ccc(-c3cccc(Cl)c3)cc2)no1
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1.629667
chembl:1535880
NC(=O)C(CCCC(=O)O)NC(=O)C(CCC(=O)O)NC(=O)CCc1cc(-c2ccc(-c3cccc(Cl)c3)cc2)no1
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chembl:1535880
CC(NC(=O)CCc1ccc(-c2ccc(-c3ccccc3)cc2)cc1)C(=O)NC(CCC(=O)O)C(N)=O
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1.628333
chembl:1535880
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1.628333
chembl:1535880
NC(=O)C(CC(=O)O)NC(=O)C(CCC(=O)O)NC(=O)CCc1ccc(-c2ccc(-c3ccccc3)cc2)cc1
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1.626
chembl:1535880
NC(=O)C(CC(=O)O)NC(=O)C(CCC(=O)O)NC(=O)CCc1ccc(-c2ccc(-c3ccccc3)cc2)cc1
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1.626
chembl:1535880
CC(C)CC(NC(=O)CCc1ccc(-c2ccc(-c3ccccc3)cc2)cc1)C(=O)NC(CCC(=O)O)C(N)=O
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1.623
chembl:1535880
CC(C)CC(NC(=O)CCc1ccc(-c2ccc(-c3ccccc3)cc2)cc1)C(=O)NC(CCC(=O)O)C(N)=O
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chembl:1535880
O=C(O)CCC(NC(=O)CCc1ccc(-c2ccc(-c3ccccc3)cc2)cc1)C(=O)N1CCCC(CC(=O)O)C1
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1.621333
chembl:1535880
O=C(O)CCC(NC(=O)CCc1ccc(-c2ccc(-c3ccccc3)cc2)cc1)C(=O)N1CCCC(CC(=O)O)C1
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1.621333
chembl:1535880
CC(NC(=O)C(CCC(=O)O)NC(=O)CCc1ccc(-c2ccc(-c3ccccc3)cc2)cc1)C(N)=O
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1.620667
chembl:1535880
CC(NC(=O)C(CCC(=O)O)NC(=O)CCc1ccc(-c2ccc(-c3ccccc3)cc2)cc1)C(N)=O
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1.620667
chembl:1535880
NC(=O)C(CC(=O)O)NC(=O)C(CCC(=O)O)NC(=O)CCc1cc(-c2ccc(-c3cccc(Cl)c3)cc2)no1
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1.620333
chembl:1535880
NC(=O)C(CC(=O)O)NC(=O)C(CCC(=O)O)NC(=O)CCc1cc(-c2ccc(-c3cccc(Cl)c3)cc2)no1
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1.620333
chembl:1535880
NC(=O)CCC(NC(=O)C(CCC(=O)O)NC(=O)CCc1ccc(-c2ccc(-c3ccccc3)cc2)cc1)C(N)=O
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1.620333
chembl:1535880
NC(=O)CCC(NC(=O)C(CCC(=O)O)NC(=O)CCc1ccc(-c2ccc(-c3ccccc3)cc2)cc1)C(N)=O
748339e6b6b30751e4a444f1209e4ec92ffc68a0db4a9ef948c1190545d9c68f
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1.620333
chembl:1535880
NC(=O)C(CCC(=O)O)NC(=O)C(Cc1ccc(O)cc1)NC(=O)CCc1ccc(-c2ccc(-c3ccccc3)cc2)cc1
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1.62
chembl:1535880
NC(=O)C(CCC(=O)O)NC(=O)C(Cc1ccc(O)cc1)NC(=O)CCc1ccc(-c2ccc(-c3ccccc3)cc2)cc1
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1.62