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1.77M
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240
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stringlengths
44
44
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stringlengths
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stringlengths
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stringlengths
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reactant_001
stringlengths
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reactant_002
stringlengths
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stringlengths
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float64
0
1.49k
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stringlengths
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stringlengths
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float64
-230
30.1k
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float64
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yield_001
float64
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100M
38,952
1,579,049
null
null
null
null
ord_dataset-9741bb5fd93044078df2a45f45733054
2015-01-01T00:04:00
true
The title product (590 mg, yield: 93%) was prepared using a procedure similar to the one described for the synthesis of INTERMEDIATE 24 utilizing (R)-4-(phenylthio)-3-(4-sulfamoyl-2-(trifluoromethylsulfonyl)phenylamino)butanoic acid (INTERMEDIATE 8, 400 mg, 0.8 mmol) and 2-(tert-butyldiphenylsilyloxy)-N-methylethanamin...
CN(CCO[Si](c1ccccc1)(c1ccccc1)C(C)(C)C)C(=O)C[C@H](CSc1ccccc1)Nc1ccc(S(N)(=O)=O)cc1S(=O)(=O)C(F)(F)F
null
CNCCO[Si](c1ccccc1)(c1ccccc1)C(C)(C)C
NS(=O)(=O)c1ccc(N[C@@H](CSc2ccccc2)CC(=O)O)c(S(=O)(=O)C(F)(F)F)c1
null
[C:1]1([S:7][CH2:8][C@H:9]([NH:14][C:15]2[CH:20]=[CH:19][C:18]([S:21](=[O:24])(=[O:23])[NH2:22])=[CH:17][C:16]=2[S:25]([C:28]([F:31])([F:30])[F:29])(=[O:27])=[O:26])[CH2:10][C:11]([OH:13])=O)[CH:6]=[CH:5][CH:4]=[CH:3][CH:2]=1.[Si:32]([O:49][CH2:50][CH2:51][NH:52][CH3:53])([C:45]([CH3:48])([CH3:47])[CH3:46])([C:39]1[CH:...
null
null
null
null
null
null
92.9
650,218
336,298
F[B-](F)(F)F
null
null
null
ord_dataset-65c44df6676d4ce3a1874db5d7958ca9
1996-01-01T00:08:00
true
To a cold (-5° C.) suspension of 4.45 g (16.00 mmol) of compound (19) in 25 ml acetonitrile was added dropwise a suspension of 2.60 g (16.64 mmol) of nitronium tetrafluoroborate in 5 ml of acetonitrile. After ten minutes, the homogenous, light-yellow reaction mixture was poured into water and extracted twice with ethyl...
CC(=O)Nc1ccc([N+](=O)[O-])c2c(Br)ccc(C)c12
null
O=[N+]=O
CC(=O)Nc1cccc2c(Br)ccc(C)c12
null
[Br:1][C:2]1[CH:11]=[CH:10][C:9]([CH3:12])=[C:8]2[C:3]=1[CH:4]=[CH:5][CH:6]=[C:7]2[NH:13][C:14](=[O:16])[CH3:15].F[B-](F)(F)F.[O:22]=[N+:23]=[O:24].O>C(#N)C>[Br:1][C:2]1[CH:11]=[CH:10][C:9]([CH3:12])=[C:8]2[C:3]=1[C:4]([N+:23]([O-:24])=[O:22])=[CH:5][CH:6]=[C:7]2[NH:13][C:14](=[O:16])[CH3:15]
null
CC#N
O
null
null
null
null
270,837
320,044
COc1cccc(C2(O)CCCCC2CN(C)C)c1
Cl
null
null
ord_dataset-0c61835e3a0b4986aabf2b61b708e322
1995-01-01T00:11:00
true
First, tramadol N-oxide was prepared as set forth hereinafter. Tramadol hydrochloride (0.5 mol) was converted its free base in basified water (pH >9) and then extracted with ether. The ether was evaporated to yield the crystalline hydrate of tramadol. The solid was then heated with steam under a high vacuum to remove a...
COc1cccc(C2(O)CCCCC2C[N+](C)(C)[O-])c1
null
O
null
null
[CH3:1][N:2]([CH2:4][CH:5]1[C:10]([OH:19])([C:11]2[CH:16]=[C:15]([O:17][CH3:18])[CH:14]=[CH:13][CH:12]=2)[CH2:9][CH2:8][CH2:7][CH2:6]1)[CH3:3].Cl.[OH2:21]>>[CH3:3][N+:2]([O-:21])([CH2:4][CH:5]1[C:10]([OH:19])([C:11]2[CH:12]=[CH:13][CH:14]=[C:15]([O:17][CH3:18])[CH:16]=2)[CH2:9][CH2:8][CH2:7][CH2:6]1)[CH3:1].[CH3:3][N:2...
null
null
null
null
null
null
null
424,827
56,329
null
null
null
null
ord_dataset-12a0ec4f3cda46e2badc694da2072c39
1979-01-01T00:06:00
true
A solution of dimethyl cyanodithioimidocarbonate (9.0 g, 0.615 mole) and 1,1-dimethylpropargylamine (90% amine, remainder water, 5.68 g, 0.0615 mole) in acetonitrile (125 ml) was stirred at reflux temperature for 13 days. The reaction mixture was evaporated under reduced pressure and the residue chromatographed on sili...
C#CC(C)(C)N=C(NC#N)SC
null
CSC(=NC#N)SC
C#CC(C)(C)N
null
[C:1]([N:3]=[C:4](SC)[S:5][CH3:6])#[N:2].[CH3:9][C:10]([NH2:14])([C:12]#[CH:13])[CH3:11]>C(#N)C>[C:1]([NH:3][C:4](=[N:14][C:10]([CH3:11])([C:12]#[CH:13])[CH3:9])[S:5][CH3:6])#[N:2]
null
CC#N
null
null
null
null
null
723,673
187,577
null
null
null
null
ord_dataset-3ec273742a0345ea916ad5fd071167f2
1989-01-01T00:04:00
true
An amount of 843 g (2.1 mol) of 2-(p-nitrophenoxy]-myristoyl chloride is added dropwise in 60 min to a cooled (0°-5° C.) solution of 525 g (2 mol) of 2-benzamido-4-chloro-5-aminophenol in 6 l of tetrahydrofuran and 220 ml of quninoline. The temperature of the reaction mixture is kept below 10° C. The precipitate of qui...
CCCCCCCCCCCCC(Oc1ccc([N+](=O)[O-])cc1)C(=O)Nc1cc(O)c(NC(=O)c2ccccc2)cc1Cl
null
CCCCCCCCCCCCC(Oc1ccc([N+](=O)[O-])cc1)C(=O)Cl
Nc1cc(O)c(NC(=O)c2ccccc2)cc1Cl
null
[N+:1]([C:4]1[CH:26]=[CH:25][C:7]([O:8][CH:9]([CH2:13][CH2:14][CH2:15][CH2:16][CH2:17][CH2:18][CH2:19][CH2:20][CH2:21][CH2:22][CH2:23][CH3:24])[C:10](Cl)=[O:11])=[CH:6][CH:5]=1)([O-:3])=[O:2].[C:27]([NH:35][C:36]1[CH:41]=[C:40]([Cl:42])[C:39]([NH2:43])=[CH:38][C:37]=1[OH:44])(=[O:34])[C:28]1[CH:33]=[CH:32][CH:31]=[CH:3...
null
C1CCOC1
null
null
5
null
null
152,488
194,413
[Na+]
[OH-]
null
null
ord_dataset-b83b16f2fb1a4f8782f3d82c1766cc6b
1989-01-01T00:08:00
true
A mixture of 10.0 g (0.025 mole) of 2-[(7-benzoyl-1H-indol-3-yl)methyl]propanedioic acid diethyl ester in 150 ml of 3N sodium hydroxide was heated at reflux for 18 hr, then treated with charcoal, cooled and filtered. The dark yellow filtrate was acidified by the dropwise addition of 50 ml of concentration hydrochloric ...
O=C(c1ccccc1)c1cccc2c(CC(C(=O)O)C(=O)O)c[nH]c12
null
CCOC(=O)C(Cc1c[nH]c2c(C(=O)c3ccccc3)cccc12)C(=O)OCC
null
null
C([O:3][C:4](=[O:29])[CH:5]([CH2:11][C:12]1[C:20]2[C:15](=[C:16]([C:21](=[O:28])[C:22]3[CH:27]=[CH:26][CH:25]=[CH:24][CH:23]=3)[CH:17]=[CH:18][CH:19]=2)[NH:14][CH:13]=1)[C:6]([O:8]CC)=[O:7])C.C>[OH-].[Na+]>[C:21]([C:16]1[CH:17]=[CH:18][CH:19]=[C:20]2[C:15]=1[NH:14][CH:13]=[C:12]2[CH2:11][CH:5]([C:6]([OH:8])=[O:7])[C:4]...
null
null
null
null
null
null
71.1
227,252
208,521
null
null
null
null
ord_dataset-ac1c7aa04d6c4e588e723e3e05721681
1990-01-01T00:05:00
true
2-ethoxyethyl p-methoxycinnamate or "Cinoxate" according to the common international name, sold under the trade name Giv-Tan F;
COc1ccc(C=CC(=O)OC2CCCCC2)cc1
null
CCOCCOC(=O)C=Cc1ccc(OC)cc1
CCOCCOC(=O)/C=C/c1ccc(OC)cc1
null
[CH3:1][O:2][C:3]1[CH:18]=[CH:17][C:6]([CH:7]=[CH:8][C:9]([O:11][CH2:12][CH2:13]OCC)=[O:10])=[CH:5][CH:4]=1.CCOCCO[C:25](/[CH:27]=[CH:28]/[C:29]1C=CC(OC)=CC=1)=O>>[CH3:1][O:2][C:3]1[CH:4]=[CH:5][C:6]([CH:7]=[CH:8][C:9]([O:11][CH:12]2[CH2:13][CH2:29][CH2:28][CH2:27][CH2:25]2)=[O:10])=[CH:17][CH:18]=1
null
null
null
null
null
null
null
787,400
504,570
O=C([O-])[O-]
[I-]
[K+]
null
ord_dataset-631d58dab387485c8eb0db4c20a232b7
2001-01-01T00:06:00
true
A mixture containing 4-piperazinoindole (0.2 mmole), potassium carbonate (0.5 mmole), potassium iodide (0.08 mmole) and 4-benzyl-5-chloromethyl-2-cyclohexyl oxazole (0.19 mmole) from example 2 was stirred in acetone (2 ml) for 16 hr. The mixture was concentrated in vacuo, water (10 ml) added, and the product extracted ...
c1ccc(Cc2nc(C3CCCCC3)oc2CN2CCN(c3cccc4[nH]ccc34)CC2)cc1
null
c1cc(N2CCNCC2)c2cc[nH]c2c1
ClCc1oc(C2CCCCC2)nc1Cc1ccccc1
null
[N:1]1([C:7]2[CH:15]=[CH:14][CH:13]=[C:12]3[C:8]=2[CH:9]=[CH:10][NH:11]3)[CH2:6][CH2:5][NH:4][CH2:3][CH2:2]1.C(=O)([O-])[O-].[K+].[K+].[I-].[K+].[CH2:24]([C:31]1[N:32]=[C:33]([CH:38]2[CH2:43][CH2:42][CH2:41][CH2:40][CH2:39]2)[O:34][C:35]=1[CH2:36]Cl)[C:25]1[CH:30]=[CH:29][CH:28]=[CH:27][CH:26]=1>CC(C)=O>[CH2:24]([C:31]...
null
CC(C)=O
null
null
null
null
94
568,805
695,760
[H-]
[Na+]
null
null
ord_dataset-a7baa616c65d42559e25ca0ba61e0744
2006-01-01T00:01:00
true
A mixture of 2,4-dichloro-5-methoxyaniline (1.1 g, 5.7 mmol) and 60% sodium hydride (285 mg, 9.9 mmol) in 30 mL of tetrahydrofuran is heated at reflux for 1 hour. The solution is cooled and 4-chloro-2-iodothieno[2,3-b]pyridine-5-carbonitrile (1.0 g, 3.12 mmol) is added. The reaction mixture is heated at reflux for 5 ho...
COc1cc(Nc2c(C#N)cnc3sc(I)cc23)c(Cl)cc1Cl
null
COc1cc(N)c(Cl)cc1Cl
N#Cc1cnc2sc(I)cc2c1Cl
null
[Cl:1][C:2]1[CH:8]=[C:7]([Cl:9])[C:6]([O:10][CH3:11])=[CH:5][C:3]=1[NH2:4].[H-].[Na+].Cl[C:15]1[C:20]([C:21]#[N:22])=[CH:19][N:18]=[C:17]2[S:23][C:24]([I:26])=[CH:25][C:16]=12>O1CCCC1>[Cl:1][C:2]1[CH:8]=[C:7]([Cl:9])[C:6]([O:10][CH3:11])=[CH:5][C:3]=1[NH:4][C:15]1[C:20]([C:21]#[N:22])=[CH:19][N:18]=[C:17]2[S:23][C:24](...
8
C1CCOC1
null
null
25
18.8
null
219,980
1,152,358
[Ni]
null
null
null
ord_dataset-b195433d5c354ddfb6cde0d53c41910f
2012-01-01T00:04:00
true
To a solution of 1-(1,1-dimethylethyl) 2-methyl (2R,5R)-2-(2-cyanoethyl)-5-{4-[(phenylmethyl)oxy]phenyl}-1,2-pyrrolidinedicarboxylate (D49, 215 mg, 0.46 mmol) in methanol (20 mL) was added Raney Nickel (slurry in water, 1 spatula) and the mixture was stirred under a hydrogen atmosphere (6 atm) for 4.5 hours. The cataly...
O=C1NCCC[C@]12CCC(c1ccc(O)cc1)N2
null
COC(=O)[C@]1(CCC#N)CC[C@H](c2ccc(OCc3ccccc3)cc2)N1C(=O)OC(C)(C)C
null
null
[C:1]([CH2:3][CH2:4][C@@:5]1([C:31]([O:33]C)=O)[CH2:9][CH2:8][C@H:7]([C:10]2[CH:15]=[CH:14][C:13]([O:16]CC3C=CC=CC=3)=[CH:12][CH:11]=2)[N:6]1C(OC(C)(C)C)=O)#[N:2].C(O)(C(F)(F)F)=O>CO.[Ni].ClCCl>[OH:16][C:13]1[CH:14]=[CH:15][C:10]([CH:7]2[CH2:8][CH2:9][C@:5]3([CH2:4][CH2:3][CH2:1][NH:2][C:31]3=[O:33])[NH:6]2)=[CH:11][CH...
4.5
ClCCl
CO
O=C(O)C(F)(F)F
0
19.4
null
551,240
1,667,002
CN(C)C(On1nnc2cccnc21)=[N+](C)C
F[P-](F)(F)(F)(F)F
null
null
ord_dataset-9cc455db05a444779921f786a45b21a6
2015-01-01T00:12:00
true
A mixture of 3-amino-4-{(3S)-3-[(tert-butoxycarbonyl)amino]piperidin-1-yl}-6,7-dihydro-5H-cyclopenta[b]pyridin-7-yl acetate (15.0 mg, 0.0384 mmol), 6-[2,6-difluoro-4-(methylsulfonyl)phenyl]-5-fluoropyridine-2-carboxylic acid (15.3 mg, 0.0461 mmol), HATU (36.5 mg, 0.0960 mmol) in DMF (0.09 mL) and DIPEA (14.9 mg, 0.115 ...
CC(=O)OC1CCc2c1ncc(NC(=O)c1ccc(F)c(-c3c(F)cc(S(C)(=O)=O)cc3F)n1)c2N1CCC[C@H](NC(=O)OC(C)(C)C)C1
null
CC(=O)OC1CCc2c1ncc(N)c2N1CCC[C@H](NC(=O)OC(C)(C)C)C1
CS(=O)(=O)c1cc(F)c(-c2nc(C(=O)O)ccc2F)c(F)c1
null
[C:1]([O:4][CH:5]1[C:9]2=[N:10][CH:11]=[C:12]([NH2:28])[C:13]([N:14]3[CH2:19][CH2:18][CH2:17][C@H:16]([NH:20][C:21]([O:23][C:24]([CH3:27])([CH3:26])[CH3:25])=[O:22])[CH2:15]3)=[C:8]2[CH2:7][CH2:6]1)(=[O:3])[CH3:2].[F:29][C:30]1[CH:35]=[C:34]([S:36]([CH3:39])(=[O:38])=[O:37])[CH:33]=[C:32]([F:40])[C:31]=1[C:41]1[N:46]=[...
16
CCN(C(C)C)C(C)C
CN(C)C=O
null
25
null
40.7
185,952
1,355,001
[K+]
[OH-]
null
null
ord_dataset-6034127657614f02860ed057b62b882e
2013-01-01T00:10:00
true
To a stirred suspension of ethyl 1-(2-{[bis(benzyloxy)phosphoryl]oxy}ethyl)-6-{6-[(ethylcarbamoyl)amino]-4-[4-(trifluoromethyl)-1,3-thiazol-2-yl]pyridin-3-yl}-4-oxo-1,4-dihydro-1,8-naphthyridine-3-carboxylate (Example 30, 210 mg, 0.2511 mmol) in ethanol (20 mL), 10% potassium hydroxide (0.2 mL) was added. The reaction ...
CCNC(=O)Nc1cc(-c2nc(C(F)(F)F)cs2)c(-c2cnc3c(c2)c(=O)c(C(=O)O)cn3CCOP(=O)(OCc2ccccc2)OCc2ccccc2)cn1
null
CCNC(=O)Nc1cc(-c2nc(C(F)(F)F)cs2)c(-c2cnc3c(c2)c(=O)c(C(=O)OCC)cn3CCOP(=O)(OCc2ccccc2)OCc2ccccc2)cn1
null
null
[CH2:1]([O:8][P:9]([O:19][CH2:20][CH2:21][N:22]1[C:31]2[C:26](=[CH:27][C:28]([C:32]3[CH:33]=[N:34][C:35]([NH:47][C:48](=[O:52])[NH:49][CH2:50][CH3:51])=[CH:36][C:37]=3[C:38]3[S:39][CH:40]=[C:41]([C:43]([F:46])([F:45])[F:44])[N:42]=3)=[CH:29][N:30]=2)[C:25](=[O:53])[C:24]([C:54]([O:56]CC)=[O:55])=[CH:23]1)([O:11][CH2:12...
null
CCO
null
null
60
null
73.9
435,543
592,899
null
null
null
null
ord_dataset-278fb6af8a994ac69e4d95e6e6eff756
2003-01-01T00:05:00
true
A solution of 7-methylindoline (10.2 g) in acetic anhydride (25 ml) was refluxed for 30 min. After cooling, the reaction solution was poured into ice water (250 ml) and the resulting crystal was filtered by means of suction, heated and vacuum dried to yield the end product (11.7 g).
CC(=O)N1CCc2cccc(C)c21
null
CC(=O)OC(C)=O
Cc1cccc2c1NCC2
null
[CH3:1][C:2]1[CH:3]=[CH:4][CH:5]=[C:6]2[C:10]=1[NH:9][CH2:8][CH2:7]2.[C:11](OC(=O)C)(=[O:13])[CH3:12]>>[C:11]([N:9]1[C:10]2[C:6](=[CH:5][CH:4]=[CH:3][C:2]=2[CH3:1])[CH2:7][CH2:8]1)(=[O:13])[CH3:12]
null
null
null
null
0
null
null
165,700
621,765
null
null
null
null
ord_dataset-c9f990dde2dc45d0948ecbe037a0d819
2004-01-01T00:01:00
true
(2R,3R,4 R,5R)-4-(acetyloxy)-2-(2,6-dichloro-9H-purin-9-yl)-5-(5-ethylisoxazol-3-yl)tetrahydrofuran-3-yl acetate (125 mg) was dissolved in isopropanol (5 ml) and the solution was treated with diisopropylethylamine (0.06 ml) followed by 1-ethylpropylamine (0.044 ml). The mixture was heated at 50° C. under nitrogen for 1...
CCc1cc([C@H]2O[C@@H](n3cnc4c(NC(CC)CC)nc(Cl)nc43)[C@H](OC(C)=O)[C@@H]2OC(C)=O)no1
null
CCc1cc([C@H]2O[C@@H](n3cnc4c(Cl)nc(Cl)nc43)[C@H](OC(C)=O)[C@@H]2OC(C)=O)no1
CCC(N)CC
null
[C:1]([O:4][C@@H:5]1[C@H:9]([O:10][C:11](=[O:13])[CH3:12])[C@@H:8]([C:14]2[CH:18]=[C:17]([CH2:19][CH3:20])[O:16][N:15]=2)[O:7][C@H:6]1[N:21]1[CH:29]=[N:28][C:27]2[C:22]1=[N:23][C:24]([Cl:31])=[N:25][C:26]=2Cl)(=[O:3])[CH3:2].C(N(C(C)C)CC)(C)C.[CH2:41]([CH:43]([NH2:46])[CH2:44][CH3:45])[CH3:42]>C(O)(C)C>[C:1]([O:4][C@@H...
null
CCN(C(C)C)C(C)C
CC(C)O
null
50
null
null
460,023
1,220,566
CC[SiH](CC)CC
O=C([O-])[O-]
[K+]
null
ord_dataset-dc3bb1b1ac4e4229a3fc28fb559a9777
2012-01-01T00:10:00
true
To a solution of the crude (2R,5R)-2-(tert-butyldiphenylsilanyloxy)-6-oxo-spiro[4.5]de cane-7-carboxylic acid methyl ester (1.65 g) obtained in Step 4 in toluene (1.6 mL) were added trifluoroacetic acid (5 mL) and triethylsilane (0.52 mL) under ice-cooling, followed by stirring the mixture under ice-cooling for 3 hours...
COC(=O)C1CCC[C@]2(CC[C@@H](O[Si](c3ccccc3)(c3ccccc3)C(C)(C)C)C2)C1O
null
COC(=O)C1CCC[C@]2(CC[C@@H](O[Si](c3ccccc3)(c3ccccc3)C(C)(C)C)C2)C1=O
null
null
[CH3:1][O:2][C:3]([CH:5]1[CH2:32][CH2:31][CH2:30][C@@:7]2([CH2:11][C@H:10]([O:12][Si:13]([C:26]([CH3:29])([CH3:28])[CH3:27])([C:20]3[CH:25]=[CH:24][CH:23]=[CH:22][CH:21]=3)[C:14]3[CH:19]=[CH:18][CH:17]=[CH:16][CH:15]=3)[CH2:9][CH2:8]2)[C:6]1=[O:33])=[O:4].FC(F)(F)C(O)=O.C([SiH](CC)CC)C.C(=O)([O-])[O-].[K+].[K+]>C1(C)C=...
null
O=C(O)C(F)(F)F
Cc1ccccc1
O
null
106.2
null
587,458
584,709
null
null
null
null
ord_dataset-cb5dd7a8b94e4f19a9148a1904b0dcb6
2003-01-01T00:03:00
true
Methanesulfonyl chloride (0.94 ml) was added to a solution of ethyl 3-(4-benzyloxyphenyl)lactate (3.32 g), which is the product of Reference example 1(b), in anhydrous dichloromethane (30 ml). To this mixture triethylamine (2.47 ml) was added dropwise in an ice bath. The mixture was stirred at ambient temperature for 3...
CCOC(=O)C(Cc1ccc(OCc2ccccc2)cc1)OS(C)(=O)=O
null
CCOC(=O)C(O)Cc1ccc(OCc2ccccc2)cc1
CS(=O)(=O)Cl
null
[CH3:1][S:2](Cl)(=[O:4])=[O:3].[CH2:6]([O:13][C:14]1[CH:19]=[CH:18][C:17]([CH2:20][CH:21]([OH:27])[C:22]([O:24][CH2:25][CH3:26])=[O:23])=[CH:16][CH:15]=1)[C:7]1[CH:12]=[CH:11][CH:10]=[CH:9][CH:8]=1.C(N(CC)CC)C>ClCCl>[CH2:6]([O:13][C:14]1[CH:19]=[CH:18][C:17]([CH2:20][CH:21]([O:27][S:2]([CH3:1])(=[O:4])=[O:3])[C:22]([O:...
3
CCN(CC)CC
ClCCl
null
25
null
null
257,838
870,677
[I-]
null
null
null
ord_dataset-c31cb9b44c404c10ba3aa533aa079e2b
2009-01-01T00:03:00
true
As described for example 84b, 2-(4-methyl-imidazol-1-yl)-5-trifluoromethoxy benzonitrile (+regioisomer) was reacted with Eschenmoser's salt in DMF for 24 h at 90° C. Evaporation of the solvent, aqueous workup and chromatography afforded the title compound as a colorless oil that was sufficiently pure to be used in the ...
Cc1ncn(-c2ccc(OC(F)(F)F)cc2C#N)c1CN(C)C
null
Cc1cn(-c2ccc(OC(F)(F)F)cc2C#N)cn1
C=[N+](C)C
null
[CH3:1][C:2]1[N:3]=[CH:4][N:5]([C:7]2[CH:14]=[CH:13][C:12]([O:15][C:16]([F:19])([F:18])[F:17])=[CH:11][C:8]=2[C:9]#[N:10])[CH:6]=1.[CH3:20][N+:21]([CH3:23])=[CH2:22].[I-]>CN(C=O)C>[CH3:20][N:21]([CH2:23][C:6]1[N:5]([C:7]2[CH:14]=[CH:13][C:12]([O:15][C:16]([F:19])([F:17])[F:18])=[CH:11][C:8]=2[C:9]#[N:10])[CH:4]=[N:3][C...
null
CN(C)C=O
null
null
null
null
38
33,451
910,370
null
null
null
null
ord_dataset-46d216f2c4374ef5b9df90427e2a4cd4
2009-01-01T00:09:00
true
This compound was made in the following manner: 50 mg of 3-(S)-benzyl-1-(2′-chloro-5′-methyl-biphenyl-4-ylmethyl)-piperazine was dissolved in THF, 2 equiv. of acetylchloride and 2 equiv. of N,N-diisopropylethylamine were added. The reaction was stirred at room temperature overnight. The reaction was diluted with DCM, w...
CC(=O)N1CCN(Cc2ccc(-c3cc(C)ccc3Cl)cc2)C[C@@H]1Cc1ccccc1
null
CC(=O)Cl
Cc1ccc(Cl)c(-c2ccc(CN3CCN[C@@H](Cc4ccccc4)C3)cc2)c1
null
[CH2:1]([C@@H:8]1[NH:13][CH2:12][CH2:11][N:10]([CH2:14][C:15]2[CH:20]=[CH:19][C:18]([C:21]3[CH:26]=[C:25]([CH3:27])[CH:24]=[CH:23][C:22]=3[Cl:28])=[CH:17][CH:16]=2)[CH2:9]1)[C:2]1[CH:7]=[CH:6][CH:5]=[CH:4][CH:3]=1.[C:29](Cl)(=[O:31])[CH3:30].C(N(CC)C(C)C)(C)C>C1COCC1.C(Cl)Cl>[CH2:1]([C@H:8]1[CH2:9][N:10]([CH2:14][C:15]...
8
CCN(C(C)C)C(C)C
ClCCl
C1CCOC1
25
null
null
885,386
1,755,849
[O-][Cl+3]([O-])([O-])O
null
null
null
ord_dataset-97eb2ab57fec4160922caae33b54d956
2016-01-01T00:08:00
true
To a solution of 2,6-dichloro-4-methylnicotinic acid (1.00 g, 4.85 mmol, 1 equiv) in tert-butyl acetate (24 mL) was added 70% perchloric acid (0.88 mL, 14.56 mmol, 3 equiv). After 1 h, reaction was diluted with DCM, washed cautiously with saturated aqueous sodium bicarbonate solution, dried (Na2SO4), and concentrated i...
Cc1cc(Cl)nc(Cl)c1C(=O)OC(C)(C)C
null
Cc1cc(Cl)nc(Cl)c1C(=O)O
null
null
[Cl:1][C:2]1[N:10]=[C:9]([Cl:11])[CH:8]=[C:7]([CH3:12])[C:3]=1[C:4]([OH:6])=[O:5].Cl(O)(=O)(=O)=O>C(OC(C)(C)C)(=O)C.C(Cl)Cl>[Cl:1][C:2]1[N:10]=[C:9]([Cl:11])[CH:8]=[C:7]([CH3:12])[C:3]=1[C:4]([O:6][C:3]([CH3:7])([CH3:4])[CH3:2])=[O:5]
1
CC(=O)OC(C)(C)C
ClCCl
null
null
190.4
null
701,363
1,118,058
null
null
null
null
ord_dataset-4226e9b4f9f845db967ed997270dcafc
2011-01-01T00:12:00
true
3-{1-[5-chloro-2-(trifluoromethyl)benzyl]-1,2,3,4-tetrahydropyrido[2,3-b]pyrazin-7-yl}benzoic acid was reacted with 4-phenylpiperidine as in General Procedure 10 to give the title compound. LCMS: m/z=590.98 (M+H+); retention time=1.03 minutes.
O=C(c1cccc(-c2cnc3c(c2)N(Cc2cc(Cl)ccc2C(F)(F)F)CCN3)c1)N1CCC(c2ccccc2)CC1
null
c1ccc(C2CCNCC2)cc1
O=C(O)c1cccc(-c2cnc3c(c2)N(Cc2cc(Cl)ccc2C(F)(F)F)CCN3)c1
null
[Cl:1][C:2]1[CH:3]=[CH:4][C:5]([C:28]([F:31])([F:30])[F:29])=[C:6]([CH:27]=1)[CH2:7][N:8]1[CH2:13][CH2:12][NH:11][C:10]2[N:14]=[CH:15][C:16]([C:18]3[CH:19]=[C:20]([CH:24]=[CH:25][CH:26]=3)[C:21](O)=[O:22])=[CH:17][C:9]1=2.[C:32]1([CH:38]2[CH2:43][CH2:42][NH:41][CH2:40][CH2:39]2)[CH:37]=[CH:36][CH:35]=[CH:34][CH:33]=1>>...
null
null
null
null
null
null
null
396,337
276,504
O=S(=O)(OS(=O)(=O)C(F)(F)F)C(F)(F)F
null
null
null
ord_dataset-02ee2261663048188cf6d85d2cc96e3f
1993-01-01T00:09:00
true
A solution of trifluoromethanesulfonic anhydride (0.954 g, 3.38 mmol) in methylene chloride (5 ml) was cooled to -78° C. under nitrogen, and a solution of 2-n-butyl-1-(2-chlorophenyl)methyl-5-(2-hydroxyethyl)-1H-imidazole (0.9 g, 3.07 mmol), diisopropylethylamine (0.44 g. 3.38 mmol) and methylene chloride (10 ml) was a...
CCCCc1ncc(CCN[C@@H](Cc2ccccc2)C(=O)OC)n1Cc1ccccc1Cl
null
COC(=O)[C@@H](N)Cc1ccccc1
CCCCc1ncc(CCO)n1Cc1ccccc1Cl
null
FC(F)(F)S(OS(C(F)(F)F)(=O)=O)(=O)=O.[CH2:16]([C:20]1[N:21]([CH2:28][C:29]2[CH:34]=[CH:33][CH:32]=[CH:31][C:30]=2[Cl:35])[C:22]([CH2:25][CH2:26]O)=[CH:23][N:24]=1)[CH2:17][CH2:18][CH3:19].C(N(C(C)C)CC)(C)C.[CH3:45][O:46][C:47](=[O:57])[C@H:48]([CH2:50][C:51]1[CH:56]=[CH:55][CH:54]=[CH:53][CH:52]=1)[NH2:49]>C(Cl)Cl>[CH3:...
0.25
CCN(C(C)C)C(C)C
ClCCl
null
-78
null
64.6
383,228
1,709,383
null
null
null
null
ord_dataset-3f2a531ffbae4b9eb1048afcd7953beb
2016-01-01T00:04:00
true
The title compound was prepared using 6-bromo-3-phenoxy-4-(trifluoromethyl)quinolin-2(1H)-one (Intermediate 8, step a) in place of 6-bromo-3-(4-chlorophenoxy)-4-(trifluoromethyl)quinolin-2(1H)-one (Intermediate 7, step c) according to the procedure described in Intermediate 7, step d.
FC(F)(F)c1c(Oc2ccccc2)c(Cl)nc2ccc(Br)cc12
null
O=c1[nH]c2ccc(Br)cc2c(C(F)(F)F)c1Oc1ccc(Cl)cc1
O=c1[nH]c2ccc(Br)cc2c(C(F)(F)F)c1Oc1ccccc1
null
[Br:1][C:2]1[CH:3]=[C:4]2[C:9](=[CH:10][CH:11]=1)[NH:8][C:7](=O)[C:6]([O:13][C:14]1[CH:19]=[CH:18][CH:17]=[CH:16][CH:15]=1)=[C:5]2[C:20]([F:23])([F:22])[F:21].BrC1C=C2C(=CC=1)NC(=O)C(OC1C=CC([Cl:43])=CC=1)=C2C(F)(F)F>>[Br:1][C:2]1[CH:3]=[C:4]2[C:9](=[CH:10][CH:11]=1)[N:8]=[C:7]([Cl:43])[C:6]([O:13][C:14]1[CH:19]=[CH:18...
null
null
null
null
null
null
null
352,605
188,369
null
null
null
null
ord_dataset-3ec273742a0345ea916ad5fd071167f2
1989-01-01T00:04:00
true
A solution of 3-butyl-6-hydrazino-1-(4-methoxybenzyl)uracil 0.64 g, 2 mM) and ethyl isothiocyanate (0.53 ml, 6 mM) in DMF (6 ml) was stirred at 90° C. for 14 hours and then at 110° C. for 14 hours. To the solution was added water (2 ml) and the mixture was cooled to give crystals. Recrystallization from DMF/ethanol/wat...
CCCCn1c(=O)c2c(NCC)n[nH]c2n(Cc2ccc(OC)cc2)c1=O
null
CCN=C=S
CCCCn1c(=O)cc(NN)n(Cc2ccc(OC)cc2)c1=O
null
[CH2:1]([N:5]1[C:10](=[O:11])[CH:9]=[C:8]([NH:12][NH2:13])[N:7]([CH2:14][C:15]2[CH:20]=[CH:19][C:18]([O:21][CH3:22])=[CH:17][CH:16]=2)[C:6]1=[O:23])[CH2:2][CH2:3][CH3:4].[CH2:24]([N:26]=[C:27]=S)[CH3:25].O>CN(C=O)C>[CH2:1]([N:5]1[C:10](=[O:11])[C:9]2[C:27]([NH:26][CH2:24][CH3:25])=[N:13][NH:12][C:8]=2[N:7]([CH2:14][C:1...
14
O
CN(C)C=O
null
null
null
70
912,230
965,217
CC(=O)O[BH-](OC(C)=O)OC(C)=O
[Na+]
[OH-]
null
ord_dataset-03ba810b7f464a06b5d8787af2e8b64e
2010-01-01T00:06:00
true
To a solution of 3-[5-(6-Methyl-pyridin-3-yl)-2,4-dioxo-3,4-dihydro-2H-pyrimidin-1-yl]-propionaldehyde (Prep59, 90 mg, 0.35 mmol), (1S,5R)-1-(4-trifluoromethyl-phenyl)-3-aza-bicyclo[3.1.0]hexane (Prep4, 71 mg, 0.31 mmol) and AcOH (21 mg, 0.35 mmol) in dichloroethane (2 mL), NaBH(AcO)3 (77 mg, 0.36 mmol) was added porti...
Cc1ccc(-c2cn(CCCN3C[C@@H]4C[C@]4(c4ccc(C(F)(F)F)cc4)C3)c(=O)[nH]c2=O)cn1
Cl
Cc1ccc(-c2cn(CCC=O)c(=O)[nH]c2=O)cn1
CC(Cl)Cl
FC(F)(F)c1ccc([C@@]23CNC[C@@H]2C3)cc1
[CH3:1][C:2]1[N:7]=[CH:6][C:5]([C:8]2[C:9](=[O:19])[NH:10][C:11](=[O:18])[N:12]([CH2:14][CH2:15][CH:16]=O)[CH:13]=2)=[CH:4][CH:3]=1.[F:20][C:21]([F:35])([F:34])[C:22]1[CH:27]=[CH:26][C:25]([C@:28]23[CH2:33][C@H:32]2[CH2:31][NH:30][CH2:29]3)=[CH:24][CH:23]=1.CC(O)=O.[BH-](OC(C)=O)(OC(C)=O)OC(C)=O.[Na+].[OH-].[Na+].[Cl:5...
0.75
CC(=O)O
null
null
0
40
null
508,022
22,450
N#CCCl
null
null
null
ord_dataset-19b9e29d593f4660ab77c07b459da9bb
1977-01-01T00:04:00
true
A mixture of 7-methoxy-2-tetralone (472 g., 2.68 mole), pyrrolidine (241 g., 3.40 mole) and benzene (2.5l) was refluxed under nitrogen with water separation (Dean-Stark trap) for 2 hrs. and then distilled for a further 1 hr. (1.2l) of distillate). Chloroacetonitrile (324 g., 4.30 mole) was added during 15 mins. and the...
COc1ccc2c(c1)C(CC#N)C(=O)CC2
null
C1CCNC1
COc1ccc2c(c1)CC(=O)CC2
null
[CH3:1][O:2][C:3]1[CH:12]=[C:11]2[C:6]([CH2:7][CH2:8][C:9](=[O:13])[CH2:10]2)=[CH:5][CH:4]=1.[NH:14]1CC[CH2:16][CH2:15]1.C1C=CC=CC=1.ClCC#N>O>[CH3:1][O:2][C:3]1[CH:12]=[C:11]2[C:6]([CH2:7][CH2:8][C:9](=[O:13])[CH:10]2[CH2:16][C:15]#[N:14])=[CH:5][CH:4]=1
8
O
c1ccccc1
null
null
null
null
737,433
1,025,907
null
null
null
null
ord_dataset-136cfada6ce247b4919085a57363459e
2011-01-01T00:01:00
true
4,5-Dimethyl-thiazol-2-ylamine and 2-(2-bromo-ethoxy)-1,1,1,-trifluoro-ethane were mixed and heated at 65° C. for 4 hours. The residue was triturated with hexane to afford the title compound. MS (ESI+) m/z 255 (M+H)+.
Br
Cc1sc(=N)n(CCOCC(F)(F)F)c1C
FC(F)(F)COCCBr
Cc1nc(N)sc1C
null
[CH3:1][C:2]1[N:3]=[C:4]([NH2:8])[S:5][C:6]=1[CH3:7].[Br:9][CH2:10][CH2:11][O:12][CH2:13][C:14]([F:17])([F:16])[F:15]>>[BrH:9].[CH3:1][C:2]1[N:3]([CH2:10][CH2:11][O:12][CH2:13][C:14]([F:17])([F:16])[F:15])[C:4](=[NH:8])[S:5][C:6]=1[CH3:7]
null
null
null
null
65
null
null
840,860
1,320,599
null
null
null
null
ord_dataset-2d6edb8ffd434003bb508360153bd9bb
2013-01-01T00:07:00
true
To a solution of methyl 2-amino-6-[4-fluoro-3-({[3-(trifluoromethyl)phenyl]acetyl}amino)phenoxy]-1,3-benzothiazole-7-carboxylate (2.50 mg, 4.81 mmol) in tetrahydrofuran (20 mL) were added pyridine (770 μL, 9.62 mmol) and cyclopropanecarbonyl chloride (790 μL, 8.66 mmol), and the mixture was stirred at room temperature ...
COC(=O)c1c(Oc2ccc(F)c(NC(=O)Cc3cccc(C(F)(F)F)c3)c2)ccc2nc(NC(=O)C3CC3)sc12
null
COC(=O)c1c(Oc2ccc(F)c(NC(=O)Cc3cccc(C(F)(F)F)c3)c2)ccc2nc(N)sc12
O=C(Cl)C1CC1
null
[NH2:1][C:2]1[S:3][C:4]2[C:10]([C:11]([O:13][CH3:14])=[O:12])=[C:9]([O:15][C:16]3[CH:21]=[CH:20][C:19]([F:22])=[C:18]([NH:23][C:24](=[O:36])[CH2:25][C:26]4[CH:31]=[CH:30][CH:29]=[C:28]([C:32]([F:35])([F:34])[F:33])[CH:27]=4)[CH:17]=3)[CH:8]=[CH:7][C:5]=2[N:6]=1.N1C=CC=CC=1.[CH:43]1([C:46](Cl)=[O:47])[CH2:45][CH2:44]1>O...
12
c1ccncc1
CCOC(C)=O
C1CCOC1
25
null
79.6
481,568
970,863
null
null
null
null
ord_dataset-03ba810b7f464a06b5d8787af2e8b64e
2010-01-01T00:06:00
true
The title compound was prepared from N-(5-iodo-2,3-dihydro-1H-inden-2-yl)-2-propanesulfonamide and [3-(aminosulfonyl)phenyl]boronic acid (WO2003004472) in a similar manner to Example 1.
CC(C)S(O)(O)NC1Cc2ccc(-c3cccc(S(N)(=O)=O)c3)cc2C1
null
CC(C)S(=O)(=O)NC1Cc2ccc(I)cc2C1
NS(=O)(=O)c1cccc(B(O)O)c1
null
I[C:2]1[CH:3]=[C:4]2[C:8](=[CH:9][CH:10]=1)[CH2:7][CH:6]([NH:11][S:12]([CH:15]([CH3:17])[CH3:16])(=[O:14])=[O:13])[CH2:5]2.[NH2:18][S:19]([C:22]1[CH:23]=[C:24](B(O)O)[CH:25]=[CH:26][CH:27]=1)(=[O:21])=[O:20]>>[OH:13][S:12]([NH:11][CH:6]1[CH2:5][C:4]2[C:8](=[CH:9][CH:10]=[C:2]([C:26]3[CH:27]=[C:22]([S:19]([NH2:18])(=[O:...
null
null
null
null
null
null
null
7,417
64,192
Cl
[Al+3]
[Cl-]
null
ord_dataset-b1bf0950b5cb430abbb1d80744f5df84
1980-01-01T00:03:00
true
To a solution maintained at 0° C. of 12.5 g of the ester obtained according to (a) and 8.79 g thiophene-2-carboxylic acid chloride in 130 ml methylene chloride, there are added little by little 7.9 g aluminium chloride. The mixture is then maintained at reflux temperature for 6 hours and then poured into a mixture of i...
COC(=O)COc1ccc(C(=O)c2cccs2)c2c1CCCC2
null
O=C(Cl)c1cccs1
COC(=O)COc1cccc2c1CCCC2
null
[C:1]1([O:11][CH2:12][C:13]([O:15][CH3:16])=[O:14])[C:10]2[CH2:9][CH2:8][CH2:7][CH2:6][C:5]=2[CH:4]=[CH:3][CH:2]=1.[S:17]1[CH:21]=[CH:20][CH:19]=[C:18]1[C:22](Cl)=[O:23].[Cl-].[Al+3].[Cl-].[Cl-].Cl>C(Cl)Cl>[C:18]1([C:22]([C:4]2[C:5]3[CH2:6][CH2:7][CH2:8][CH2:9][C:10]=3[C:1]([O:11][CH2:12][C:13]([O:15][CH3:16])=[O:14])=...
null
ClCCl
null
null
null
85
null
371,507
66,295
null
null
null
null
ord_dataset-8af141577c90485cb9c91079a5ef96b3
1980-01-01T00:05:00
true
A mixture of ethyl N-(6-amino-5-chloro-2-pyridyl)carbamate (64.7 g., 0.3 mole), dimethylamine (45 g., 1.0 mole) and 300 ml. of ethanol is heated at 120° C. for 24 hours in a pressure vessel. The reaction mixture is then concentrated in vacuo and 68 g. of brown solid is obtained. Recrystallization from n-butyl chloride ...
CN(C)C(=O)Nc1ccc(Cl)c(N)n1
null
CNC
CCOC(=O)Nc1ccc(Cl)c(N)n1
null
[NH2:1][C:2]1[N:7]=[C:6]([NH:8][C:9](=[O:13])OCC)[CH:5]=[CH:4][C:3]=1[Cl:14].[CH3:15][NH:16][CH3:17]>C(O)C>[CH3:15][N:16]([CH3:17])[C:9]([NH:8][C:6]1[CH:5]=[CH:4][C:3]([Cl:14])=[C:2]([NH2:1])[N:7]=1)=[O:13]
null
CCO
null
null
null
null
null
391,247
406,435
null
null
null
null
ord_dataset-d5bb2294ac964841b8ffc9e0a34e93af
1998-01-01T00:07:00
true
Compound 14g is prepared in a manner similar to that used for preparation of Compound 14 h using previously prepared Compound 13 and 2-thienylcarbonylmethyl chloride.
CC(C)(C)OC(=O)NC1C(=O)N(CC(=O)c2cccs2)c2ccccc2N(CC(=O)c2cccs2)C1=O
null
CC(C)(C)OC(=O)NC1C(=O)Nc2ccccc2NC1=O
O=C(CCl)c1cccs1
null
[C:1]([O:5][C:6]([NH:8][CH:9]1[C:15](=[O:16])[NH:14][C:13]2[CH:17]=[CH:18][CH:19]=[CH:20][C:12]=2[NH:11][C:10]1=[O:21])=[O:7])([CH3:4])([CH3:3])[CH3:2].[S:22]1[CH:26]=[CH:25][CH:24]=[C:23]1[C:27]([CH2:29]Cl)=[O:28]>>[S:22]1[CH:26]=[CH:25][CH:24]=[C:23]1[C:27]([CH2:29][N:14]1[C:13]2[CH:17]=[CH:18][CH:19]=[CH:20][C:12]=2...
null
null
null
null
null
null
null
835,433
752,824
CCN=C=NCCCN(C)C
Cl
On1nnc2ccccc21
null
ord_dataset-844a22e1fcab44a5b59c5e2922b2855a
2007-01-01T00:01:00
true
2′-Methyl-5′-(5-methyl-1,3,4-oxadiazol-2-yl)-1,1′-biphenyl-4-carboxylic acid (11.3 mg, 0.034 mmol), HOBT (6.0 mg, 0.044 mmol), 1-(3-dimethylaminopropyl)-3-ethyl carbodiimide hydrochloride (8.0 mg, 0.042 mmol) and 2-methylbutylamine (0.34 mmol) were mixed in DMF (0.7 ml) and the reaction left at room temperature for 18 ...
CCC(C)CNC(=O)c1ccc(-c2cc(-c3nnc(C)o3)ccc2C)cc1
null
Cc1nnc(-c2ccc(C)c(-c3ccc(C(=O)O)cc3)c2)o1
CCC(C)CN
null
[CH3:1][C:2]1[CH:7]=[CH:6][C:5]([C:8]2[O:9][C:10]([CH3:13])=[N:11][N:12]=2)=[CH:4][C:3]=1[C:14]1[CH:19]=[CH:18][C:17]([C:20]([OH:22])=O)=[CH:16][CH:15]=1.C1C=CC2N(O)N=NC=2C=1.Cl.CN(C)CCCN=C=NCC.[CH3:45][CH:46]([CH2:49][CH3:50])[CH2:47][NH2:48]>CN(C=O)C>[CH3:1][C:2]1[CH:7]=[CH:6][C:5]([C:8]2[O:9][C:10]([CH3:13])=[N:11][...
18
CN(C)C=O
null
null
null
null
null
392,293
715,344
null
null
null
null
ord_dataset-c8a367b56b4f406b878f51867b157d19
2006-01-01T00:06:00
true
15.2 ml (101 mmol) of 1-morpholino-1-cyclopentene is carefully added in drops to a solution of 20.0 g (101 mmol) of 3-bromophenylisocyanate in 100 ml of chloroform. The batch is refluxed for 15 minutes and concentrated by evaporation in a vacuum. Column chromatography on silica gel with hexane-ethyl acetate yielded 25....
O=C1CCCC1C(=O)Nc1cccc(Br)c1
null
C1=C(N2CCOCC2)CCC1
O=C=Nc1cccc(Br)c1
CCOC(C)=O
O1CCN([C:7]2[CH2:11][CH2:10][CH2:9][CH:8]=2)CC1.[Br:12][C:13]1[CH:14]=[C:15]([N:19]=[C:20]=[O:21])[CH:16]=[CH:17][CH:18]=1.CCCCCC.C(OCC)(=[O:30])C>C(Cl)(Cl)Cl>[Br:12][C:13]1[CH:14]=[C:15]([NH:19][C:20]([CH:7]2[CH2:8][CH2:9][CH2:10][C:11]2=[O:30])=[O:21])[CH:16]=[CH:17][CH:18]=1
null
ClC(Cl)Cl
CCCCCC
null
null
null
null
218,565
1,084,872
null
null
null
null
ord_dataset-afd812677c134591a99f46ce28de2524
2011-01-01T00:08:00
true
Step 2 Trifluoroacetic acid (0.56 mL, 7.3 mmol) was added to a solution of tert-butyl 2-[4-(2-oxopropoxy)phenyl]ethylcarbamate (216 mg, 0.74 mmol) in CH2Cl2 (4 mL). The reaction mixture was stirred for 3 hr at ambient temperature, and then reaction mixture was stripped of volatiles in vacuo. The residue (143 mg) was us...
CC(=O)COc1ccc(CCN)cc1
null
CC(=O)COc1ccc(CCNC(=O)OC(C)(C)C)cc1
null
null
FC(F)(F)C(O)=O.[O:8]=[C:9]([CH3:28])[CH2:10][O:11][C:12]1[CH:17]=[CH:16][C:15]([CH2:18][CH2:19][NH:20]C(=O)OC(C)(C)C)=[CH:14][CH:13]=1>C(Cl)Cl>[NH2:20][CH2:19][CH2:18][C:15]1[CH:16]=[CH:17][C:12]([O:11][CH2:10][C:9]([CH3:28])=[O:8])=[CH:13][CH:14]=1
3
ClCCl
O=C(O)C(F)(F)F
null
25
null
null
297,973
1,103,208
O=S(=O)(O)O
null
null
null
ord_dataset-375a420ee9b042918ddca20f02df37d3
2011-01-01T00:11:00
true
Nitric acid (10 mL) was slowly added to sulfuric acid (10 mL) at 0° C., and the mixture was stirred at the same temperature for 10 min. To this solution was slowly added 1-benzothiophene 1,1-dioxide (3.99 g) at 0° C., and the mixture was further stirred at the same temperature for 30 min. The reaction mixture was poure...
O=[N+]([O-])c1ccc2c(c1)S(=O)(=O)C=C2
null
O=[N+]([O-])O
O=S1(=O)C=Cc2ccccc21
null
[N+:1]([O-:4])(O)=[O:2].[S:5]1(=[O:15])(=[O:14])[C:9]2[CH:10]=[CH:11][CH:12]=[CH:13][C:8]=2[CH:7]=[CH:6]1>S(=O)(=O)(O)O>[N+:1]([C:11]1[CH:12]=[CH:13][C:8]2[CH:7]=[CH:6][S:5](=[O:15])(=[O:14])[C:9]=2[CH:10]=1)([O-:4])=[O:2]
0.17
null
null
null
0
null
84
717,569
495,402
[H-]
[Na+]
null
null
ord_dataset-9df8b3ec9c8742b3802e0efaac6f6ef3
2001-01-01T00:03:00
true
2.0 g (4.15 mmol) of 4-{[6-(quinolin-8-yl-sulphonylamino)-1-methyl-2-oxo-1,2-dihydroquinoxalin-3-yl]-methyl}-benzonitrile are dissolved in 150 ml tetrahydrofuran and after the addition of 0.2 g (4.15 mmol) of sodium hydride (50% in oil) stirred for 2 hours at ambient temperature. After the addition of 0.47 ml (4.15 mmo...
COC(=O)CN(c1ccc2c(c1)nc(Cc1ccc(C#N)cc1)c(=O)n2C)S(=O)(=O)c1cccc2cccnc12
null
Cn1c(=O)c(Cc2ccc(C#N)cc2)nc2cc(NS(=O)(=O)c3cccc4cccnc34)ccc21
CCOC(=O)CBr
null
[N:1]1[C:10]2[C:5](=[CH:6][CH:7]=[CH:8][C:9]=2[S:11]([NH:14][C:15]2[CH:16]=[C:17]3[C:22](=[CH:23][CH:24]=2)[N:21]([CH3:25])[C:20](=[O:26])[C:19]([CH2:27][C:28]2[CH:35]=[CH:34][C:31]([C:32]#[N:33])=[CH:30][CH:29]=2)=[N:18]3)(=[O:13])=[O:12])[CH:4]=[CH:3][CH:2]=1.[H-].[Na+].Br[CH2:39][C:40]([O:42][CH2:43]C)=[O:41]>O1CCCC...
2
C1CCOC1
null
null
25
null
null
533,328
500,355
COc1ccc(C(C)=O)cc1
COc1ccc([C@H](C)O)cc1
null
null
ord_dataset-18e9ed24dbd44e98b33bdc22aa7580a8
2001-01-01T00:04:00
true
As shown here, the biochemical conversion reaction of immobilized soy bean protein for the substrate (±)-1-(4-methoxyphenyl)ethanol (200 mg) requires 5 days by going through bioconversion to 4-methoxyacetophenone accompanying sterically selective oxidation of (S)-1-(4-methoxyphenyl)ethanol to obtain 96 mg of (R)-1-(4-m...
COc1ccc([C@@H](C)O)cc1
null
COc1ccc(C(C)O)cc1
null
null
[CH3:1][O:2][C:3]1[CH:8]=[CH:7][C:6]([CH:9]([OH:11])[CH3:10])=[CH:5][CH:4]=1.CC(C1C=CC(OC)=CC=1)=O.COC1C=CC([C@@H](O)C)=CC=1>>[CH3:1][O:2][C:3]1[CH:8]=[CH:7][C:6]([C@H:9]([OH:11])[CH3:10])=[CH:5][CH:4]=1
120
null
null
null
null
null
48
244,776
673,054
[I-]
[Na+]
null
null
ord_dataset-e90cd41afe844e49875435eb99903799
2005-01-01T00:05:00
true
3,4-dimethoxyphenylsulfonyl chloride (2.3 mmol) was dissolved in acetone (60 mL), and then NaI (3.4 g, 23 mmol) and fluoroacetic anhydride (1.45 mL, 6.9 mmol) were added and the mixture was stirred at room temperature for one hour. The reaction solution was concentrated, water was added, extraction was performed with e...
COc1ccc(SSc2ccc(OC)c(OC)c2)cc1OC
null
O=C(CF)OC(=O)CF
COc1ccc(S(=O)(=O)Cl)cc1OC
null
[CH3:1][O:2][C:3]1[CH:4]=[C:5]([S:11](Cl)(=O)=O)[CH:6]=[CH:7][C:8]=1[O:9][CH3:10].[Na+].[I-].FC[C:19]([O:21][C:22](=O)[CH2:23]F)=O>CC(C)=O>[CH3:1][O:2][C:3]1[CH:4]=[C:5]([S:11][S:11][C:5]2[CH:6]=[CH:23][C:22]([O:21][CH3:19])=[C:3]([O:2][CH3:1])[CH:4]=2)[CH:6]=[CH:7][C:8]=1[O:9][CH3:10]
1
CC(C)=O
null
null
25
null
null
73,269
967,286
null
null
null
null
ord_dataset-03ba810b7f464a06b5d8787af2e8b64e
2010-01-01T00:06:00
true
3,5 difluorophenylacetonitrile (5 g) was dissolved in THF (100 mL) and a solution of BH3 in THF (200 mL of 1 M) was added dropwise. The mixture was refluxed overnight, cooled in an ice bath, and the reaction quenched with methanol (20 mL). The solvent was removed by rotary evaporation and the residue partitioned betwee...
NCCc1cc(F)cc(F)c1
null
N#CCc1cc(F)cc(F)c1
null
null
[F:1][C:2]1[CH:3]=[C:4]([CH2:9][C:10]#[N:11])[CH:5]=[C:6]([F:8])[CH:7]=1>C1COCC1>[F:1][C:2]1[CH:3]=[C:4]([CH2:9][CH2:10][NH2:11])[CH:5]=[C:6]([F:8])[CH:7]=1
null
C1CCOC1
null
null
null
null
null
759,184
115,117
null
null
null
null
ord_dataset-d182ca8cf3f34de69c7a38343db8c930
1984-01-01T00:03:00
true
Using the method of Example 15, 1-(p-chlorophenyl)-3-azabicyclo[3.1.0]hexane (Example 1) is reacted with acetyl chloride to give 3-acetyl-1-(p-chlorophenyl)-3-azabicyclo[3.1.0]hexane and then is converted to 1-(p-chlorophenyl)-3-ethyl-3-azabicyclo[3.1.0]hexane which is obtained as a brown oil.
CC(=O)N1CC2CC2(c2ccc(Cl)cc2)C1
null
Clc1ccc(C23CNCC2C3)cc1
CC(=O)Cl
null
[Cl:1][C:2]1[CH:7]=[CH:6][C:5]([C:8]23[CH2:13][CH:12]2[CH2:11][NH:10][CH2:9]3)=[CH:4][CH:3]=1.[C:14](Cl)(=[O:16])[CH3:15]>>[C:14]([N:10]1[CH2:11][CH:12]2[C:8]([C:5]3[CH:4]=[CH:3][C:2]([Cl:1])=[CH:7][CH:6]=3)([CH2:13]2)[CH2:9]1)(=[O:16])[CH3:15]
null
null
null
null
null
null
null
884,588
588,339
null
null
null
null
ord_dataset-7a74d48eeefd45aba53e7258f3ae067a
2003-01-01T00:04:00
true
Using 6-(dimethylamino)-hexylamine and N-[2-(3-Cyano-1H-indol-5-yl)-ethyl]-4-[2-chloro-pyrimidin-4-yl]-benzamide (reference example 1az) as substrates. MS (ion spray) m/z 510 (M+H)+.
CN(C)CCCCCCNc1nccc(-c2ccc(C(=O)NCCc3ccc4[nH]cc(C#N)c4c3)cc2)n1
null
CN(C)CCCCCCN
N#Cc1c[nH]c2ccc(CCNC(=O)c3ccc(-c4ccnc(Cl)n4)cc3)cc12
null
[CH3:1][N:2]([CH3:10])[CH2:3][CH2:4][CH2:5][CH2:6][CH2:7][CH2:8][NH2:9].[C:11]([C:13]1[C:21]2[C:16](=[CH:17][CH:18]=[C:19]([CH2:22][CH2:23][NH:24][C:25](=[O:39])[C:26]3[CH:31]=[CH:30][C:29]([C:32]4[CH:37]=[CH:36][N:35]=[C:34](Cl)[N:33]=4)=[CH:28][CH:27]=3)[CH:20]=2)[NH:15][CH:14]=1)#[N:12]>>[C:11]([C:13]1[C:21]2[C:16](...
null
null
null
null
null
null
null
274,597
50,110
null
null
null
null
ord_dataset-e5870fef54544989915ccced8dd8d849
1979-01-01T00:01:00
true
Analogously to Example 10, 5-amino-N-(2-hydroxy-1,1-dimethylethyl)-2,4,6-triiodoisophthalamic acid is reacted with hexanedioic acid dichloride in dimethylacetamide, and the reaction mixture is worked up. The thus-obtained product melts at 280°-281° C., with decomposition.
CC(C)(CO)NC(=O)c1c(I)c(NC(=O)CCCCC(=O)Nc2c(I)c(C(=O)O)c(I)c(C(=O)NC(C)(C)CO)c2I)c(I)c(C(=O)O)c1I
null
O=C(Cl)CCCCC(=O)Cl
CC(C)(CO)NC(=O)c1c(I)c(N)c(I)c(C(=O)O)c1I
null
[NH2:1][C:2]1[C:3]([I:21])=[C:4]([C:13]([NH:15][C:16]([CH3:20])([CH3:19])[CH2:17][OH:18])=[O:14])[C:5]([I:12])=[C:6]([C:10]=1[I:11])[C:7]([OH:9])=[O:8].[C:22](Cl)(=[O:30])[CH2:23][CH2:24][CH2:25][CH2:26][C:27](Cl)=[O:28]>CC(N(C)C)=O>[C:22]([NH:1][C:2]1[C:3]([I:21])=[C:4]([C:13]([NH:15][C:16]([CH3:19])([CH3:20])[CH2:17]...
null
CC(=O)N(C)C
null
null
null
null
null
606,606
1,413,310
null
null
null
null
ord_dataset-f8e6e6a2d2bf4135b9e346456c81700f
2014-01-01T00:04:00
true
According to the method of 1-7 of Example 1, a target compound was prepared from 2-fluoro-N-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)-3-(methylamino)benzamide and 2,2,2-trichloroethoxycarbonylchloride.
CN(C(=O)OCC(Cl)(Cl)Cl)c1cccc(C(=O)Nc2c(I)cc(C(F)(C(F)(F)F)C(F)(F)C(F)(F)F)cc2C(F)(F)F)c1F
null
CNc1cccc(C(=O)Nc2c(I)cc(C(F)(C(F)(F)F)C(F)(F)C(F)(F)F)cc2C(F)(F)F)c1F
O=C(Cl)OCC(Cl)(Cl)Cl
null
[F:1][C:2]1[C:34]([NH:35][CH3:36])=[CH:33][CH:32]=[CH:31][C:3]=1[C:4]([NH:6][C:7]1[C:12]([C:13]([F:16])([F:15])[F:14])=[CH:11][C:10]([C:17]([F:29])([C:22]([F:28])([F:27])[C:23]([F:26])([F:25])[F:24])[C:18]([F:21])([F:20])[F:19])=[CH:9][C:8]=1[I:30])=[O:5].[Cl:37][C:38]([Cl:45])([Cl:44])[CH2:39][O:40][C:41](Cl)=[O:42]>>...
null
null
null
null
null
null
null
20,395
1,745,766
null
null
null
null
ord_dataset-60a3e71da3174666a50a61dcfa611a9f
2016-01-01T00:07:00
true
4,6-Dichloro-N-(3-fluoro-5-methoxyphenyl)pyrimidine-5-carboxamide (800 mg, 1.42 mmol) was dissolved in dioxane (5 ml) and cooled in an ice bath. Ammonia solution (1 ml, 7N in MeOH) was added dropwise and the mixture was stirred at 0° C. for 6 h and overnight at room temperature. After evaporation of the solvent under r...
COc1cc(F)cc(NC(=O)c2c(N)ncnc2Cl)c1
null
COc1cc(F)cc(NC(=O)c2c(Cl)ncnc2Cl)c1
N
null
[Cl:1][C:2]1[C:7]([C:8]([NH:10][C:11]2[CH:16]=[C:15]([O:17][CH3:18])[CH:14]=[C:13]([F:19])[CH:12]=2)=[O:9])=[C:6](Cl)[N:5]=[CH:4][N:3]=1.[NH3:21]>O1CCOCC1>[NH2:21][C:6]1[C:7]([C:8]([NH:10][C:11]2[CH:16]=[C:15]([O:17][CH3:18])[CH:14]=[C:13]([F:19])[CH:12]=2)=[O:9])=[C:2]([Cl:1])[N:3]=[CH:4][N:5]=1
8
C1COCCO1
null
null
0
null
null
477,885
1,488,149
CCCC[N+](CCCC)(CCCC)CCCC
[F-]
null
null
ord_dataset-c3c1091f873b4f40827973a6f1f9b685
2014-01-01T00:09:00
true
To a solution of 8-{[4-({[tert-butyl(dimethyl)silyl]oxy}methyl)-2-methoxyphenyl]amino}-N-(2,6-diethylphenyl)-1-methyl-4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline-3-carboxamide (300 mg, 0.48 mmol) in 6 ml of dry THF, 800 μl of commercial TBAF solution in THF were added. The mixture was stirred at room temperature for 1 h ...
CCc1cccc(CC)c1NC(=O)c1nn(C)c2c1CCc1cnc(Nc3ccc(CO)cc3OC)nc1-2
null
CCc1cccc(CC)c1NC(=O)c1nn(C)c2c1CCc1cnc(Nc3ccc(CO[Si](C)(C)C(C)(C)C)cc3OC)nc1-2
null
null
[Si]([O:8][CH2:9][C:10]1[CH:15]=[CH:14][C:13]([NH:16][C:17]2[N:26]=[CH:25][C:24]3[CH2:23][CH2:22][C:21]4[C:27]([C:31]([NH:33][C:34]5[C:39]([CH2:40][CH3:41])=[CH:38][CH:37]=[CH:36][C:35]=5[CH2:42][CH3:43])=[O:32])=[N:28][N:29]([CH3:30])[C:20]=4[C:19]=3[N:18]=2)=[C:12]([O:44][CH3:45])[CH:11]=1)(C(C)(C)C)(C)C>C1COCC1.CCCC...
1
C1CCOC1
null
null
25
null
85
864,645
704,612
CC(=O)OI1(OC(C)=O)(OC(C)=O)OC(=O)c2ccccc21
null
null
null
ord_dataset-c408dfed796e4354b61e312e67f7143f
2006-01-01T00:04:00
true
A solution of (R)-2-Cyclohexylmethyl-N-{(S)-1-[hydroxy-(5-trifluoromethyl-1,2,4-oxadiazol-3-yl)-methyl]-propyl}-4-morpholin-4-yl-4-oxo-butyramide (324 mg, 0.661 mmol) in methylene chloride (10 ml) was treated with Dess Martin periodinane (308 mg, 0.726 mmol) and stirred at room temperature for 90 minutes. The reaction ...
CC[C@H](NC(=O)[C@@H](CC(=O)N1CCOCC1)CC1CCCCC1)C(=O)c1noc(C(F)(F)F)n1
null
CC[C@H](NC(=O)[C@@H](CC(=O)N1CCOCC1)CC1CCCCC1)C(O)c1noc(C(F)(F)F)n1
null
null
[CH:1]1([CH2:7][C@H:8]([CH2:26][C:27]([N:29]2[CH2:34][CH2:33][O:32][CH2:31][CH2:30]2)=[O:28])[C:9]([NH:11][C@H:12]([CH:15]([OH:25])[C:16]2[N:20]=[C:19]([C:21]([F:24])([F:23])[F:22])[O:18][N:17]=2)[CH2:13][CH3:14])=[O:10])[CH2:6][CH2:5][CH2:4][CH2:3][CH2:2]1.CC(OI1(OC(C)=O)(OC(C)=O)OC(=O)C2C=CC=CC1=2)=O>C(Cl)Cl>[CH:1]1(...
1.5
ClCCl
null
null
25
null
null
240,518
1,249,175
Cl
null
null
null
ord_dataset-c544c0c663f54dbea4ddb52ddde7934e
2013-01-01T00:01:00
true
The title compound was prepared as described in Example 1d from 6-chloro-N-{3-[8-(2,6-difluorophenyl)-2-(methylsulfonyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methylphenyl}-3-pyridinecarboxamide and (1H-imidazol-2-ylmethyl)amine dihydrochloride: LC-MS m/z 599 (M+H)+, 1.92 min (ret time).
Cc1ccc(NC(=O)c2ccc(Cl)nc2)cc1-c1nc(NCc2ncc[nH]2)nc2c1ccc(=O)n2-c1c(F)cccc1F
null
Cc1ccc(NC(=O)c2ccc(Cl)nc2)cc1-c1nc(S(C)(=O)=O)nc2c1ccc(=O)n2-c1c(F)cccc1F
NCc1ncc[nH]1
null
[Cl:1][C:2]1[N:7]=[CH:6][C:5]([C:8]([NH:10][C:11]2[CH:16]=[CH:15][C:14]([CH3:17])=[C:13]([C:18]3[C:19]4[CH:31]=[CH:30][C:29](=[O:32])[N:28]([C:33]5[C:38]([F:39])=[CH:37][CH:36]=[CH:35][C:34]=5[F:40])[C:20]=4[N:21]=[C:22](S(C)(=O)=O)[N:23]=3)[CH:12]=2)=[O:9])=[CH:4][CH:3]=1.Cl.Cl.[NH:43]1[CH:47]=[CH:46][N:45]=[C:44]1[CH...
null
null
null
null
null
null
null
305,482
497,277
Cl
null
null
null
ord_dataset-9df8b3ec9c8742b3802e0efaac6f6ef3
2001-01-01T00:03:00
true
Following General Procedure A and using N-(3,5-difluorophenylacetyl)-L-alanine (from Example B2 above) and methyl (S)-2-amino-3-(thiazol-4-yl)propionate hydrochloride (General Procedure H with methanol and HCl on methyl (S)-2-amino-3-(thiazol-4-yl)propyl acid (Synthetech)), the title compound was prepared as a solid (m...
COC(=O)[C@H](Cc1cscn1)NC(=O)[C@H](C)NC(=O)Cc1cc(F)cc(F)c1
null
C[C@H](NC(=O)Cc1cc(F)cc(F)c1)C(=O)O
COC(=O)[C@@H](N)Cc1cscn1
null
[F:1][C:2]1[CH:3]=[C:4]([CH2:9][C:10]([NH:12][C@H:13]([C:15]([OH:17])=O)[CH3:14])=[O:11])[CH:5]=[C:6]([F:8])[CH:7]=1.Cl.[NH2:19][C@@H:20]([CH2:25][C:26]1[N:27]=[CH:28][S:29][CH:30]=1)[C:21]([O:23][CH3:24])=[O:22]>CO.C(Cl)Cl>[F:8][C:6]1[CH:5]=[C:4]([CH2:9][C:10]([NH:12][C@H:13]([C:15]([NH:19][C@@H:20]([CH2:25][C:26]2[N:...
null
CO
ClCCl
null
null
null
null
392,773
1,632,215
null
null
null
null
ord_dataset-f0794d5ded7a4d3fab45cc3d7a89ee3d
2015-01-01T00:09:00
true
Using N-((2S)-1-((2-(4-(benzyloxy)-3,5-difluorophenyl)-1,3-benzoxazol-6-yl)oxy)propan-2-yl)acetamide and iodoethane, and in the same manner as in Example 5, the title compound was obtained.
CCOc1c(F)cc(-c2nc3ccc(OC[C@H](C)NC(C)=O)cc3o2)cc1F
null
CC(=O)N[C@@H](C)COc1ccc2nc(-c3cc(F)c(OCc4ccccc4)c(F)c3)oc2c1
null
null
[CH2:1]([O:8][C:9]1[C:14]([F:15])=[CH:13][C:12]([C:16]2[O:17][C:18]3[CH:24]=[C:23]([O:25][CH2:26][C@@H:27]([NH:29][C:30](=[O:32])[CH3:31])[CH3:28])[CH:22]=[CH:21][C:19]=3[N:20]=2)=[CH:11][C:10]=1[F:33])[C:2]1C=CC=CC=1.ICC>>[CH2:1]([O:8][C:9]1[C:10]([F:33])=[CH:11][C:12]([C:16]2[O:17][C:18]3[CH:24]=[C:23]([O:25][CH2:26]...
null
CCI
null
null
null
null
null
563,762
387,896
O=[Pt]
null
null
null
ord_dataset-44d518e567bd4c039d77233023f78bb2
1998-01-01T00:01:00
true
The title compound was prepared by hydrogenation of 5,11-dihydro-3,4-dimethyl-11-ethyl-5-methyl-8-(phenylethynyl)-6H-dipyrido[3,2-b:2',3'-e][1,4]diazepin-6-one over platinum oxide, as described in Example 42b. The product crystallized from ether/petroleum ether, m.p. 187°-188° C.
CCN1c2ncc(CCc3ccccc3)cc2C(=O)N(C)c2c1ncc(C)c2C
null
CCN1c2ncc(C#Cc3ccccc3)cc2C(=O)N(C)c2c1ncc(C)c2C
null
null
[CH3:1][C:2]1[CH:12]=[N:11][C:10]2[N:9]([CH2:13][CH3:14])[C:8]3[N:15]=[CH:16][C:17]([C:19]#[C:20][C:21]4[CH:26]=[CH:25][CH:24]=[CH:23][CH:22]=4)=[CH:18][C:7]=3[C:6](=[O:27])[N:5]([CH3:28])[C:4]=2[C:3]=1[CH3:29]>[Pt]=O>[CH3:1][C:2]1[CH:12]=[N:11][C:10]2[N:9]([CH2:13][CH3:14])[C:8]3[N:15]=[CH:16][C:17]([CH2:19][CH2:20][C...
null
null
null
null
null
null
null
755,460
1,015,220
null
null
null
null
ord_dataset-f024e9664ab64906a71a2ff6004cb3d0
2010-01-01T00:12:00
true
This was prepared analogously from 2-{1-[1-(3-bromo-phenyl)-1H-benzoimidazol-5-yl]-ethyl}-isoindole-1,3-dione and 5-pyrimidineboronic acid.
CC(c1ccc2c(c1)ncn2-c1cccc(-c2cncnc2)c1)N1C(=O)c2ccccc2C1=O
null
CC(c1ccc2c(c1)ncn2-c1cccc(Br)c1)N1C(=O)c2ccccc2C1=O
OB(O)c1cncnc1
null
Br[C:2]1[CH:3]=[C:4]([N:8]2[C:12]3[CH:13]=[CH:14][C:15]([CH:17]([N:19]4[C:27](=[O:28])[C:26]5[C:21](=[CH:22][CH:23]=[CH:24][CH:25]=5)[C:20]4=[O:29])[CH3:18])=[CH:16][C:11]=3[N:10]=[CH:9]2)[CH:5]=[CH:6][CH:7]=1.[N:30]1[CH:35]=[C:34](B(O)O)[CH:33]=[N:32][CH:31]=1>>[N:30]1[CH:35]=[C:34]([C:2]2[CH:3]=[C:4]([N:8]3[C:12]4[CH...
null
null
null
null
null
null
null
404,815
2,616
O=C([O-])[O-]
[Na+]
null
null
ord_dataset-a0bc986c3cf848c2a1ea93b297d1ad89
1976-01-01T00:02:00
true
A stirred mixture of 8.0 g of (4.6-dichloro-2-pyrimidinylthio)acetic acid ethyl ester, 2.8 g of aniline and 3.2 g of sodium carbonate in 100 ml. of ethanol was heated under reflux for 5 hr. The reaction mixture was filtered and water was added to the filtrate to start precipitation. The crude product was recrystallized...
CCOC(=O)CSc1nc(Cl)cc(Nc2ccccc2)n1
null
Nc1ccccc1
CCOC(=O)CSc1nc(Cl)cc(Cl)n1
null
[CH2:1]([O:3][C:4](=[O:15])[CH2:5][S:6][C:7]1[N:12]=[C:11]([Cl:13])[CH:10]=[C:9](Cl)[N:8]=1)[CH3:2].[NH2:16][C:17]1[CH:22]=[CH:21][CH:20]=[CH:19][CH:18]=1.C(=O)([O-])[O-].[Na+].[Na+]>C(O)C>[CH2:1]([O:3][C:4](=[O:15])[CH2:5][S:6][C:7]1[N:8]=[C:9]([NH:16][C:17]2[CH:22]=[CH:21][CH:20]=[CH:19][CH:18]=2)[CH:10]=[C:11]([Cl:1...
null
CCO
null
null
null
69.1
null
12,353
899,471
c1ccc([PH](c2ccccc2)(c2ccccc2)[Pd-4]([PH](c2ccccc2)(c2ccccc2)c2ccccc2)([PH](c2ccccc2)(c2ccccc2)c2ccccc2)[PH](c2ccccc2)(c2ccccc2)c2ccccc2)cc1
[Cs+]
[F-]
null
ord_dataset-de6bce51790e4004a27e1a8f2bcc7ded
2009-01-01T00:08:00
true
According to the procedure described for example 26b the use of 1-bromo-3-methanesulfonyl-benzene (1.07 g, 4.55 mmol), (E)-3-cyclohexyl-2-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-prop-2-en-1-ol (1.57 g, 5.92 mmol), caesium fluoride (2.07 g, 13.7 mmol) and tetrakis(triphenylphosphino)palladium(0) (525 mg, 455 μmol...
CS(=O)(=O)c1cccc(/C(=C\C2CCCCC2)CO)c1
null
CS(=O)(=O)c1cccc(Br)c1
CC1(C)OB(/C(=C\C2CCCCC2)CO)OC1(C)C
null
Br[C:2]1[CH:7]=[CH:6][CH:5]=[C:4]([S:8]([CH3:11])(=[O:10])=[O:9])[CH:3]=1.[CH:12]1(/[CH:18]=[C:19](\B2OC(C)(C)C(C)(C)O2)/[CH2:20][OH:21])[CH2:17][CH2:16][CH2:15][CH2:14][CH2:13]1.[F-].[Cs+]>O1CCOCC1.C1(P([Pd-4](P(C2C=CC=CC=2)(C2C=CC=CC=2)C2C=CC=CC=2)(P(C2C=CC=CC=2)(C2C=CC=CC=2)C2C=CC=CC=2)P(C2C=CC=CC=2)(C2C=CC=CC=2)C2C...
null
C1COCCO1
null
null
null
51.7
null
30,740
89,761
[Na+]
[OH-]
null
null
ord_dataset-aeb5378e6e67443e8a4f5c7a5ec3de51
1981-01-01T00:12:00
true
To an ice cold solution of 1.60 g (0.04 mol) of NaOH in 45 ml of water is added 9.64 g (0.04 mol) of 5-cyano-1-(2,6-dimethylphenyl)uracil, obtained as in Example 1. After dissolution, 50 ml of ice cold dichloromethane is added, followed by a solution of 9.36 g (0.04 mol) of 1,1,2,2-tetrachloroethanesulphenyl chloride (...
Cc1cccc(C)c1-n1cc(C#N)c(=O)n(SC(Cl)(Cl)C(Cl)Cl)c1=O
null
Cc1cccc(C)c1-n1cc(C#N)c(=O)[nH]c1=O
ClSC(Cl)(Cl)C(Cl)Cl
null
[OH-].[Na+].[C:3]([C:5]1[C:6](=[O:20])[NH:7][C:8](=[O:19])[N:9]([C:11]2[C:16]([CH3:17])=[CH:15][CH:14]=[CH:13][C:12]=2[CH3:18])[CH:10]=1)#[N:4].[Cl:21][C:22]([Cl:28])([S:26]Cl)[CH:23]([Cl:25])[Cl:24].ClCCl>O>[C:3]([C:5]1[C:6](=[O:20])[N:7]([S:26][C:22]([Cl:28])([Cl:21])[CH:23]([Cl:25])[Cl:24])[C:8](=[O:19])[N:9]([C:11]...
0.5
ClCCl
O
null
25
null
null
627,780
25,292
CCN1C(=CC#CC2N(CC)c3nc4ccccc4nc3[NH+]2CC)N(CC)c2nc3ccccc3nc21
[O-][Cl+3]([O-])([O-])[O-]
null
null
ord_dataset-fcf7c02bbb814fe696760b5fbfee16bb
1977-01-01T00:05:00
true
Phosphoryl chloride (1.0 ml) is added to a stirred suspension of 1,3-Bis(1-methyl-2-(1H)-quinolylidene)acetone (0.68 g, 0.002 mol) in pyridine (10 ml). The mixture is stirred for 5 min., then the solid is collected and washed with a little pyridine, then with ether. The dye is converted to its perchlorate salt by solut...
CN1C(=CC#Cc2ccc3ccccc3[n+]2C)C=Cc2ccccc21
null
CN1C(=CC(=O)C=C2C=Cc3ccccc3N2C)C=Cc2ccccc21
null
null
P(Cl)(Cl)(Cl)=O.[CH3:6][N:7]1[C:16]2[C:11](=[CH:12][CH:13]=[CH:14][CH:15]=2)[CH:10]=[CH:9][C:8]1=[CH:17][C:18]([CH:20]=[C:21]1[CH:30]=[CH:29][C:28]2[C:23](=[CH:24][CH:25]=[CH:26][CH:27]=2)[N:22]1[CH3:31])=O.[Cl:32]([O-:36])(=[O:35])(=[O:34])=[O:33].C([NH+]1C2=NC3C(N=C2N(CC)C1C#CC=C1N(CC)C2=NC4C(N=C2N1CC)=CC=CC=4)=CC=CC...
0.08
O=P(Cl)(Cl)Cl
c1ccncc1
CC#N
null
35
null
130,467
560,636
null
null
null
null
ord_dataset-7c28974b7fcf4c9c86d5f2a42ba328a2
2002-01-01T00:09:00
true
The title compound was prepared from N-[5-((1R)-2-Amino-1-hydroxy-ethyl)-2-hydroxy-phenyl]-methanesulfonamide and Reference Example 14, 1-[4-(4-oxo-piperidin-1-yl)-benzenesulfonyl]-pyrrolidine-2-carboxylic acid isopropyl ester, according to the procedure of Example 1 as an off-white solid; mp 52-58° C.; 1H NMR (300 MHz...
CC(C)OC(=O)C1CCCN1S(=O)(=O)c1ccc(N2CCC(NCC(O)c3ccc(O)c(NS(C)(=O)=O)c3)CC2)cc1
null
CS(=O)(=O)Nc1cc([C@@H](O)CN)ccc1O
CC(C)OC(=O)C1CCCN1S(=O)(=O)c1ccc(N2CCC(=O)CC2)cc1
null
[NH2:1][CH2:2][C@@H:3]([C:5]1[CH:6]=[CH:7][C:8]([OH:16])=[C:9]([NH:11][S:12]([CH3:15])(=[O:14])=[O:13])[CH:10]=1)[OH:4].[CH:17]([O:20][C:21]([CH:23]1[CH2:27][CH2:26][CH2:25][N:24]1[S:28]([C:31]1[CH:36]=[CH:35][C:34]([N:37]2[CH2:42][CH2:41][C:40](=O)[CH2:39][CH2:38]2)=[CH:33][CH:32]=1)(=[O:30])=[O:29])=[O:22])([CH3:19])...
null
null
null
null
null
null
null
109,351
1,756,725
null
null
null
null
ord_dataset-97eb2ab57fec4160922caae33b54d956
2016-01-01T00:08:00
true
4-(chlorosulfonyl)benzoic acid (500 mg, 2.27 mmol) was treated with 6-methoxy-1,2,3,4-tetrahydroquinoline (1.0 g, 6.13 mmol) using method A to give 4-(6-methoxy-3,4-dihydroquinolin-1(2H)-ylsulfonyl)benzoic acid as an off-white solid. Yield: 358 mg (46%). 1H-NMR: 8.04 (d, J=8.5 Hz, 2H), 7.64 (d, J=8.5 Hz, 2H), 7.52 (d, ...
COc1ccc2c(c1)CCCN2S(=O)(=O)c1ccc(C(=O)O)cc1
null
O=C(O)c1ccc(S(=O)(=O)Cl)cc1
COc1ccc2c(c1)CCCN2
null
Cl[S:2]([C:5]1[CH:13]=[CH:12][C:8]([C:9]([OH:11])=[O:10])=[CH:7][CH:6]=1)(=[O:4])=[O:3].[CH3:14][O:15][C:16]1[CH:17]=[C:18]2[C:23](=[CH:24][CH:25]=1)[NH:22][CH2:21][CH2:20][CH2:19]2>>[CH3:14][O:15][C:16]1[CH:17]=[C:18]2[C:23](=[CH:24][CH:25]=1)[N:22]([S:2]([C:5]1[CH:13]=[CH:12][C:8]([C:9]([OH:11])=[O:10])=[CH:7][CH:6]=...
null
null
null
null
null
null
null
204,582
1,228,110
[I-]
[Zn+2]
null
null
ord_dataset-cde802cdb7434a5f82a22981ccaefc4e
2012-01-01T00:11:00
true
To a mixture of 0.83 g of 4-[5-[3,5-bis(trifluoromethyl)phenyl]-5-trifluoromethyl-4,5-dihydroisoxazole-3-yl]benzaldehyde and 0.36 g of trimethylsilylcyanide, 0.01 g of zinc iodide was added while stirring the mixture at 0° C. The resultant mixture was stirred at 60° C. for 10 minutes, and then left to be cooled down to...
N#CC(N)c1ccc(C2=NOC(c3cc(C(F)(F)F)cc(C(F)(F)F)c3)(C(F)(F)F)C2)cc1
null
C[Si](C)(C)C#N
O=Cc1ccc(C2=NOC(c3cc(C(F)(F)F)cc(C(F)(F)F)c3)(C(F)(F)F)C2)cc1
N
[F:1][C:2]([F:31])([F:30])[C:3]1[CH:4]=[C:5]([C:13]2([C:26]([F:29])([F:28])[F:27])[O:17][N:16]=[C:15]([C:18]3[CH:25]=[CH:24][C:21]([CH:22]=O)=[CH:20][CH:19]=3)[CH2:14]2)[CH:6]=[C:7]([C:9]([F:12])([F:11])[F:10])[CH:8]=1.C[Si]([C:36]#[N:37])(C)C.[NH3:38].CO>[I-].[Zn+2].[I-]>[NH2:38][CH:22]([C:21]1[CH:24]=[CH:25][C:18]([C...
null
CO
null
null
0
null
null
29,434
764,662
CN
null
null
null
ord_dataset-7a8649d55889427e85b208ae89475895
2007-01-01T00:04:00
true
A mixture of 2-{cis-4-[(4-methyl-1-tetrahydro-2H-pyran-2-yl-1H-indazol-5-yl)oxy]cyclohexyl}-1H-isoindole-1,3(2H)-dione (95.5 mg, 0.208 mmol) and a 30% methylamine-ethanol solution (5.0 ml) was stirred with heating under reflux for 2 hours. The reaction solution was allowed to cool, and then was concentrated under reduc...
Cc1c(O[C@H]2CC[C@@H](N)CC2)ccc2c1cnn2C1CCCCO1
null
Cc1c(O[C@H]2CC[C@@H](N3C(=O)c4ccccc4C3=O)CC2)ccc2c1cnn2C1CCCCO1
null
null
[CH3:1][C:2]1[C:10]([O:11][C@@H:12]2[CH2:17][CH2:16][C@H:15]([N:18]3C(=O)C4C(=CC=CC=4)C3=O)[CH2:14][CH2:13]2)=[CH:9][CH:8]=[C:7]2[C:3]=1[CH:4]=[N:5][N:6]2[CH:29]1[CH2:34][CH2:33][CH2:32][CH2:31][O:30]1.CN.C(O)C>>[CH3:1][C:2]1[C:10]([O:11][C@@H:12]2[CH2:13][CH2:14][C@H:15]([NH2:18])[CH2:16][CH2:17]2)=[CH:9][CH:8]=[C:7]2...
null
CCO
null
null
null
null
null
350,390
449,628
[H-]
[Na+]
null
null
ord_dataset-a4f0b79f6b9847168861270b79f84afa
1999-01-01T00:11:00
true
A mixture of 1-[[1-(3,4-dimethoxyphenyl)cyclopropyl]methyl]-1,3-dihydro-2H-imidazol-2-one (1.9 g) in DMF (20 ml) was stirred at RT. Sodium hydride (60%) (0.28 g) was added portionwise over 15 minutes. The mixture was stirred for 30 minutes. A solution of bromomethylbenzene (1.45 g) in DMF (5 ml) was added dropwise over...
COc1ccc(C2(Cn3ccn(Cc4ccccc4)c3=O)CC2)cc1OC
null
BrCc1ccccc1
COc1ccc(C2(Cn3cc[nH]c3=O)CC2)cc1OC
null
[CH3:1][O:2][C:3]1[CH:4]=[C:5]([C:11]2([CH2:14][N:15]3[CH:19]=[CH:18][NH:17][C:16]3=[O:20])[CH2:13][CH2:12]2)[CH:6]=[CH:7][C:8]=1[O:9][CH3:10].[H-].[Na+].Br[CH2:24][C:25]1[CH:30]=[CH:29][CH:28]=[CH:27][CH:26]=1>CN(C=O)C>[CH3:1][O:2][C:3]1[CH:4]=[C:5]([C:11]2([CH2:14][N:15]3[CH:19]=[CH:18][N:17]([CH2:24][C:25]4[CH:30]=[...
null
CN(C)C=O
null
null
25
null
51.5
512,871
1,465,539
[Na+]
[OH-]
null
null
ord_dataset-fd1fa959d6264608b0b7fcda16741bfd
2014-01-01T00:08:00
true
A solution of 1.5 g (3.59 mmol) of 4-{2-[4-(3-carboxyphenyl)piperazin-1-yl]ethyl}piperidine-1-carboxylic acid tert-butyl ester in 20 mL of dry tetrahydrofuran is cooled to −10° C. under argon. An addition of 11 mL of a 1M solution of boranetetrahydrofuran complex in tetrahydrofuran is performed at −10° C. Stirring is m...
CC(C)(C)OC(=O)N1CCC(CCN2CCN(c3cccc(CO)c3)CC2)CC1
null
CC(C)(C)OC(=O)N1CCC(CCN2CCN(c3cccc(C(=O)O)c3)CC2)CC1
null
null
[C:1]([O:5][C:6]([N:8]1[CH2:13][CH2:12][CH:11]([CH2:14][CH2:15][N:16]2[CH2:21][CH2:20][N:19]([C:22]3[CH:27]=[CH:26][CH:25]=[C:24]([C:28](O)=[O:29])[CH:23]=3)[CH2:18][CH2:17]2)[CH2:10][CH2:9]1)=[O:7])([CH3:4])([CH3:3])[CH3:2].[OH-].[Na+]>O1CCCC1>[C:1]([O:5][C:6]([N:8]1[CH2:13][CH2:12][CH:11]([CH2:14][CH2:15][N:16]2[CH2:...
null
C1CCOC1
null
null
25
69
null
728,187
216,123
Br
null
null
null
ord_dataset-67ed03c283094854909157b1038e38e3
1990-01-01T00:10:00
true
1.21 g (7.6 mmol) of bromine in 5 ml of glacial acetic acid are added to a solution of 1.2 g (7.5 mmol) of 5-acetylbenzimidazole and 1.35 g of 48% strength aqueous HBr (=8 mmol of HB) in 15 ml of glacial acetic acid at room temperature. The mixture is stirred at 40° C. for 30 minutes and cooled and the product which ha...
O=C(CBr)c1ccc2nc[nH]c2c1
null
CC(=O)c1ccc2nc[nH]c2c1
BrBr
null
[Br:1]Br.[C:3]([C:6]1[CH:14]=[CH:13][C:9]2[N:10]=[CH:11][NH:12][C:8]=2[CH:7]=1)(=[O:5])[CH3:4].[BrH:15]>C(O)(=O)C>[BrH:1].[Br:15][CH2:4][C:3]([C:6]1[CH:14]=[CH:13][C:9]2[N:10]=[CH:11][NH:12][C:8]=2[CH:7]=1)=[O:5]
0.5
CC(=O)O
null
null
40
null
null
260,182
275,000
c1ccc(P(c2ccccc2)c2ccccc2)cc1
null
null
null
ord_dataset-02ee2261663048188cf6d85d2cc96e3f
1993-01-01T00:09:00
true
3-Ethenylbenzyl alcohol (5.26 g) was dissolved in carbon tetrachloride (100 ml) and triphenylphosphine (10.2 g) added. The solution was refluxed overnight and then left to cool. A white precipitate formed which was filtered through celite. The filtrate was evaporated in vacuo to yield a crude product. The residue was p...
C=Cc1cccc(CCl)c1
null
C=Cc1cccc(CO)c1
ClC(Cl)(Cl)Cl
null
[CH:1]([C:3]1[CH:4]=[C:5]([CH:8]=[CH:9][CH:10]=1)[CH2:6]O)=[CH2:2].C1(P(C2C=CC=CC=2)C2C=CC=CC=2)C=CC=CC=1.C(Cl)(Cl)(Cl)[Cl:31]>>[CH:1]([C:3]1[CH:4]=[C:5]([CH:8]=[CH:9][CH:10]=1)[CH2:6][Cl:31])=[CH2:2]
null
null
null
null
null
null
null
722,732
531,825
null
null
null
null
ord_dataset-7774db17e619477ea20ee621abe71257
2002-01-01T00:01:00
true
To a solution of the diamine of Step A (3.28 g) in dry chloroform (48 mL) was added dropwise under nitrogen at 0° C. triethylamine (3.62 mL). Thiophosgene (1.49 mL) was then added dropwise via syringe and the mixture was stirred in the cold for another 15 minutes. Stirring was continued at room temperature for 1.5 hour...
Cc1cccc(Cl)c1N1CCCN(C2CCC2)C1=S
null
Cc1cccc(Cl)c1NCCCNC1CCC1
S=C(Cl)Cl
null
[Cl:1][C:2]1[C:7]([NH:8][CH2:9][CH2:10][CH2:11][NH:12][CH:13]2[CH2:16][CH2:15][CH2:14]2)=[C:6]([CH3:17])[CH:5]=[CH:4][CH:3]=1.C(N(CC)CC)C.[C:25](Cl)(Cl)=[S:26].O>C(Cl)(Cl)Cl>[Cl:1][C:2]1[C:7]([N:8]2[CH2:9][CH2:10][CH2:11][N:12]([CH:13]3[CH2:16][CH2:15][CH2:14]3)[C:25]2=[S:26])=[C:6]([CH3:17])[CH:5]=[CH:4][CH:3]=1
0.25
ClC(Cl)Cl
CCN(CC)CC
O
null
null
81
594,519
515,028
null
null
null
null
ord_dataset-41760195182e4bb4bc779bd722456071
2001-01-01T00:08:00
true
The title compound was prepared according to the procedure described in step 2 of Example 1 from 2-[(ethoxycarbonyl)amino]-4fluorobenzonitrile (step 1) and 2-bromoacetophenone.
CCOC(=O)n1c(C(=O)c2ccccc2)c(N)c2ccc(F)cc21
null
CCOC(=O)Nc1cc(F)ccc1C#N
O=C(CBr)c1ccccc1
null
[CH2:1]([O:3][C:4]([NH:6][C:7]1[CH:14]=[C:13]([F:15])[CH:12]=[CH:11][C:8]=1[C:9]#[N:10])=[O:5])[CH3:2].Br[CH2:17][C:18]([C:20]1[CH:25]=[CH:24][CH:23]=[CH:22][CH:21]=1)=[O:19]>>[NH2:10][C:9]1[C:8]2[C:7](=[CH:14][C:13]([F:15])=[CH:12][CH:11]=2)[N:6]([C:4]([O:3][CH2:1][CH3:2])=[O:5])[C:17]=1[C:18](=[O:19])[C:20]1[CH:25]=[...
null
null
null
null
null
null
null
343,996
79,849
C[O-]
[Na+]
null
null
ord_dataset-2d589ad46f82417ab9ddc07f7655411c
1981-01-01T00:04:00
true
To a solution of 1.42 g. sodium methoxide in 250 ml. methanol is added 8.0 g. of 4-[2-(1-naphthyloxy)ethylamino]benzoic acid. After one-half hour, the mixture is concentrated under vacuum to a solid which is washed with methanol and then CH2Cl2. This solid is immediately dried in a vacuum oven to minimize absorption of...
O=C([O-])c1ccc(NCCOc2cccc3ccccc23)cc1
null
O=C(O)c1ccc(NCCOc2cccc3ccccc23)cc1
null
null
C[O-].[Na+:3].[C:4]1([O:14][CH2:15][CH2:16][NH:17][C:18]2[CH:26]=[CH:25][C:21]([C:22]([OH:24])=[O:23])=[CH:20][CH:19]=2)[C:13]2[C:8](=[CH:9][CH:10]=[CH:11][CH:12]=2)[CH:7]=[CH:6][CH:5]=1>CO>[C:4]1([O:14][CH2:15][CH2:16][NH:17][C:18]2[CH:19]=[CH:20][C:21]([C:22]([O-:24])=[O:23])=[CH:25][CH:26]=2)[C:13]2[C:8](=[CH:9][CH:...
null
CO
null
null
null
null
null
350,802
1,392,605
CC(C)OC(=O)N=NC(=O)OC(C)C
c1ccc(P(c2ccccc2)c2ccccc2)cc1
null
null
ord_dataset-12dc3bd21bcf44d09e5b4249afe15161
2014-01-01T00:02:00
true
A mixture of 2-(1-methyl-1H-pyrazol-5-yl)ethanol (1.00 g), 4-hydroxybenzotrifluoride (2.57 g), 1.9 M diisopropyl azodicarboxylate (6.26 mL, toluene solution), triphenylphosphine (3.12 g) and tetrahydrofuran (50 mL) was stirred at a room temperature for 2 days. Thereafter, water was added to the reaction solution, and t...
Cn1nccc1CCOc1ccc(C(F)(F)F)cc1
null
Cn1nccc1CCO
Oc1ccc(C(F)(F)F)cc1
null
[CH3:1][N:2]1[C:6]([CH2:7][CH2:8][OH:9])=[CH:5][CH:4]=[N:3]1.O[C:11]1[CH:16]=[CH:15][C:14]([C:17]([F:20])([F:19])[F:18])=[CH:13][CH:12]=1.N(C(OC(C)C)=O)=NC(OC(C)C)=O.C1(P(C2C=CC=CC=2)C2C=CC=CC=2)C=CC=CC=1>O.O1CCCC1>[CH3:1][N:2]1[C:6]([CH2:7][CH2:8][O:9][C:11]2[CH:16]=[CH:15][C:14]([C:17]([F:20])([F:19])[F:18])=[CH:13][...
48
C1CCOC1
O
null
25
54.6
null
166,508
72,553
null
null
null
null
ord_dataset-520610070b3c4780a03b44c7fcecc28f
1980-01-01T00:10:00
true
A solution of 4.75 g. of N-trifluoroacetyl-4-(4-tetradecenylamino)benzoyl chloride and 1.2 g. of triethylamine in 200 ml. of warm ether is treated with 1.55 g. alanine ethyl ester and refluxed for 24 hours. The hot solution is filtered, the residue is washed with hot ether, and the combined filtrate and washings are ev...
CCCCCCCCCC=CCCCNc1ccc(C(=O)N[C@@H](C)C(=O)O)cc1
null
CCOC(=O)[C@H](C)N
CCCCCCCCCC=CCCCN(C(=O)C(F)(F)F)c1ccc(C(=O)Cl)cc1
null
FC(F)(F)C([N:5]([CH2:15][CH2:16][CH2:17][CH:18]=[CH:19][CH2:20][CH2:21][CH2:22][CH2:23][CH2:24][CH2:25][CH2:26][CH2:27][CH3:28])[C:6]1[CH:14]=[CH:13][C:9]([C:10](Cl)=[O:11])=[CH:8][CH:7]=1)=O.C(N(CC)CC)C.C([O:40][C:41](=[O:45])[C@H:42]([CH3:44])[NH2:43])C>CCOCC>[CH2:15]([NH:5][C:6]1[CH:7]=[CH:8][C:9]([C:10]([NH:43][C@H...
null
CCN(CC)CC
CCOCC
null
null
null
null
154,482
1,387,562
null
null
null
null
ord_dataset-31641fb65b34430fa7435229b949b604
2014-01-01T00:01:00
true
2-{6-[8-(2-Methoxy-5-trifluoromethyl-phenyl)-[1,2,4]-triazolo[1,5-a]pyridin-2-ylamino]-3,4-dihydro-1H-isoquinolin-2-yl}-N,N-dimethyl-acetamide was prepared from [8-(2-methoxy-5-trifluoromethyl-phenyl)-[1,2,4]-triazolo[1,5-a]pyridin-2-yl]-(1,2,3,4-tetrahydro-isoquinolin-6-yl)-amine (0.150 g, 0.341 mmol) and 2-chloro-N,N...
COc1ccc(C(F)(F)F)cc1-c1cccn2nc(Nc3ccc4c(c3)CCN(CC(=O)N(C)C)C4)nc12
null
COc1ccc(C(F)(F)F)cc1-c1cccn2nc(Nc3ccc4c(c3)CCNC4)nc12
CN(C)C(=O)CCl
null
[CH3:1][O:2][C:3]1[CH:8]=[CH:7][C:6]([C:9]([F:12])([F:11])[F:10])=[CH:5][C:4]=1[C:13]1[C:14]2[N:15]([N:19]=[C:20]([NH:22][C:23]3[CH:24]=[C:25]4[C:30](=[CH:31][CH:32]=3)[CH2:29][NH:28][CH2:27][CH2:26]4)[N:21]=2)[CH:16]=[CH:17][CH:18]=1.Cl[CH2:34][C:35]([N:37]([CH3:39])[CH3:38])=[O:36]>>[CH3:1][O:2][C:3]1[CH:8]=[CH:7][C:...
null
null
null
null
null
null
null
390,321
595,376
null
null
null
null
ord_dataset-278fb6af8a994ac69e4d95e6e6eff756
2003-01-01T00:05:00
true
To a solution of 2-chloro-5-nitropyridine (30 mmol, 5.0 g) in absolute ethanol was added a solution of hydrazine hydrate (320 mmol, 15.8 g) in ethanol using syringe pump. At the end of the addition, the reaction was refrigerated. The named product precipitated from the reaction medium, was collected by filtration, and ...
NNc1ccc([N+](=O)[O-])cn1
null
NN
O=[N+]([O-])c1ccc(Cl)nc1
null
Cl[C:2]1[CH:7]=[CH:6][C:5]([N+:8]([O-:10])=[O:9])=[CH:4][N:3]=1.O.[NH2:12][NH2:13]>C(O)C>[N+:8]([C:5]1[CH:6]=[CH:7][C:2]([NH:12][NH2:13])=[N:3][CH:4]=1)([O-:10])=[O:9]
null
CCO
O
null
null
null
null
210,529
1,395,602
Cl
[Li+]
[OH-]
null
ord_dataset-12dc3bd21bcf44d09e5b4249afe15161
2014-01-01T00:02:00
true
To a mixture of EtOH (0.2 mL) and H2O (0.1 mL) was suspended ethyl 5-hydroxy-4-[1-hydroxyimino-3-[3-propyl-6-(trifluoromethyl)-benzothiophen-2-yl]propyl]-2-methylphenoxyacetate (7.5 mg, 0.0143 mmol) obtained above. After the addition of lithium hydroxide monohydrate (1.8 mg, 0.0429 mmol), the mixture was heated for 1 h...
CCCc1c(CCC(=NO)c2cc(C)c(OCC(=O)O)cc2O)sc2cc(C(F)(F)F)ccc12
null
CCCc1c(CCC(=NO)c2cc(C)c(OCC(=O)OCC)cc2O)sc2cc(C(F)(F)F)ccc12
null
null
CCO.[OH:4][C:5]1[C:6]([C:19](=[N:38][OH:39])[CH2:20][CH2:21][C:22]2[S:23][C:24]3[CH:33]=[C:32]([C:34]([F:37])([F:36])[F:35])[CH:31]=[CH:30][C:25]=3[C:26]=2[CH2:27][CH2:28][CH3:29])=[CH:7][C:8]([CH3:18])=[C:9]([CH:17]=1)[O:10][CH2:11][C:12]([O:14]CC)=[O:13].O.[OH-].[Li+].Cl>O>[OH:4][C:5]1[C:6]([C:19](=[N:38][OH:39])[CH2...
null
O
CCO
null
25
null
112.9
187,619
1,511,149
null
null
null
null
ord_dataset-1a1aa5d1c3224edca0aec6e3398da985
2014-01-01T00:11:00
true
tert-Butyl 4-(quinolin-8-yl)piperazine-1-carboxylate (2.4 g, 7.66 mmol) was dissolved in methanol (50 ml) and SOCl2 was added to the solution dropwise at 0° C. The resulting solution was refluxed for 1 day and evaporated under reduced pressure. EtOAc (50 ml) was added to the residue and stirred for 2 hours to produce l...
Cl
c1cnc2c(N3CCNCC3)cccc2c1
O=S(Cl)Cl
CC(C)(C)OC(=O)N1CCN(c2cccc3cccnc23)CC1
null
[N:1]1[C:10]2[C:5](=[CH:6][CH:7]=[CH:8][C:9]=2[N:11]2[CH2:16][CH2:15][N:14](C(OC(C)(C)C)=O)[CH2:13][CH2:12]2)[CH:4]=[CH:3][CH:2]=1.O=S(Cl)[Cl:26]>CO>[ClH:26].[N:11]1([C:9]2[CH:8]=[CH:7][CH:6]=[C:5]3[C:10]=2[N:1]=[CH:2][CH:3]=[CH:4]3)[CH2:16][CH2:15][NH:14][CH2:13][CH2:12]1
2
CO
null
null
null
null
null
164,256
1,581,679
Cl
null
null
null
ord_dataset-380e279f82154dba9e08ab51b3bdd08a
2015-01-01T00:05:00
true
Prepared from 5-(4-Methyl-5-trifluoromethyl-isoxazol-3-yl)-thiophene-2-carboxylic acid and 4-N-Boc-2-(R)-methyl-piperazine by the method described in Example 2 Method B. The reaction mixture was evaporated to a solid, triturated and filtered with the aid of water, then washed with a 1 N aqueous hydrochloric acid soluti...
Cc1c(-c2ccc(C(=O)N3CCNC[C@H]3C)s2)noc1C(F)(F)F
null
Cc1c(-c2ccc(C(=O)O)s2)noc1C(F)(F)F
C[C@@H]1CN(C(=O)OC(C)(C)C)CCN1
null
[CH3:1][C:2]1[C:3]([C:11]2[S:15][C:14]([C:16]([OH:18])=O)=[CH:13][CH:12]=2)=[N:4][O:5][C:6]=1[C:7]([F:10])([F:9])[F:8].C([N:26]1[CH2:31][CH2:30][NH:29][C@H:28]([CH3:32])[CH2:27]1)(OC(C)(C)C)=O.[ClH:33]>O1CCOCC1>[ClH:33].[CH3:32][C@@H:28]1[CH2:27][NH:26][CH2:31][CH2:30][N:29]1[C:16]([C:14]1[S:15][C:11]([C:3]2[C:2]([CH3:...
2
C1COCCO1
null
null
null
86
null
464,205
761,382
null
null
null
null
ord_dataset-2e58cb8db2bf482bbea23283b7e04488
2007-01-01T00:03:00
true
1-(2-Amino-4,5-dimethoxy-phenyl)-2-(3,4-dichloro-phenyl)-ethanone (5.52 g, 16.24 mmol) was dissolved in dichloromethane (20 ml), distilled water was then added (2 ml) and the resulting solution was cooled at −5° C. under nitrogen. Bromoacetylbromide (1.63 ml, 18.68 mmol) was dissolved in dichloromethane (10 ml) and add...
COc1cc(NC(=O)CBr)c(C(=O)Cc2ccc(Cl)c(Cl)c2)cc1OC
null
COc1cc(N)c(C(=O)Cc2ccc(Cl)c(Cl)c2)cc1OC
O=C(Br)CBr
null
[NH2:1][C:2]1[CH:7]=[C:6]([O:8][CH3:9])[C:5]([O:10][CH3:11])=[CH:4][C:3]=1[C:12](=[O:22])[CH2:13][C:14]1[CH:19]=[CH:18][C:17]([Cl:20])=[C:16]([Cl:21])[CH:15]=1.[Br:23][CH2:24][C:25](Br)=[O:26]>ClCCl>[Br:23][CH2:24][C:25]([NH:1][C:2]1[CH:7]=[C:6]([O:8][CH3:9])[C:5]([O:10][CH3:11])=[CH:4][C:3]=1[C:12](=[O:22])[CH2:13][C:...
0.25
ClCCl
null
null
-5
70.1
null
195,649
1,469,717
null
null
null
null
ord_dataset-fd1fa959d6264608b0b7fcda16741bfd
2014-01-01T00:08:00
true
The compound prepared in Example 126 (1.00 g) was suspended in tetrahydrofuran (20 mL) and dimethylamine (2 M) (7.66 mL) added and the reaction mixture stirred at room temperature for 3 hours. The reaction mixture was partitioned between saturated aqueous sodium bicarbonate and ethyl acetate. The organics were washed w...
CCOC(=O)c1sc(-c2ccccc2)nc1CN(C)C
null
CCOC(=O)c1sc(-c2ccccc2)nc1CBr
CNC
null
Br[CH2:2][C:3]1[N:4]=[C:5]([C:13]2[CH:18]=[CH:17][CH:16]=[CH:15][CH:14]=2)[S:6][C:7]=1[C:8]([O:10][CH2:11][CH3:12])=[O:9].[CH3:19][NH:20][CH3:21]>O1CCCC1>[CH3:19][N:20]([CH2:2][C:3]1[N:4]=[C:5]([C:13]2[CH:18]=[CH:17][CH:16]=[CH:15][CH:14]=2)[S:6][C:7]=1[C:8]([O:10][CH2:11][CH3:12])=[O:9])[CH3:21]
3
C1CCOC1
null
null
25
null
null
498,286
419,882
C[O-]
Cc1ccc(S(=O)(=O)O)cc1
[Na+]
null
ord_dataset-94e21e9990034c729ea727e7d2ab0eb0
1998-01-01T00:12:00
true
21.1 g (114 mmol) of 4-bromobenzaldehyde and 20 ml (182 mmol) of trimethyl orthoformate (both Fluka, Buchs, Switzerland) are dissolved in 35 ml of methanol, and 0.65 g (3.4 mmol) of p-toluenesulfonic acid monohydrate is added at room temperature (exothermic reaction). The reaction mixture is stirred at room temperature...
COC(OC)c1ccc(Br)cc1
null
COC(OC)OC
O=Cc1ccc(Br)cc1
null
[Br:1][C:2]1[CH:9]=[CH:8][C:5](C=O)=[CH:4][CH:3]=1.[CH:10](OC)([O:13][CH3:14])[O:11][CH3:12].O.C1(C)C=CC(S(O)(=O)=O)=CC=1.C[O-].[Na+]>CO>[CH3:12][O:11][CH:10]([O:13][CH3:14])[C:5]1[CH:8]=[CH:9][C:2]([Br:1])=[CH:3][CH:4]=1
20
CO
O
null
25
null
null
831,299
1,605,142
[Fe]
[Cl-]
[NH4+]
null
ord_dataset-9cecb3a8d3b9494191b28dcefea66af2
2015-01-01T00:07:00
true
Iron (2.41 g, 42.3 mmol) and ammonium chloride (2.58 g, 48.4 mmol) are added to a solution of 5-nitro-1-(tetrahydro-2H-pyran-4-yl)-1H-pyrazolo[3,4-b]pyridine (3 g, 12 mmol) in ethanol/THF/H2O (4:2:1, 35 mL). The mixture is heated at 100° C. for 2 h. The iron is removed by filtration through pad of Celite® and the filtr...
Nc1cnc2c(cnn2C2CCOCC2)c1
null
O=[N+]([O-])c1cnc2c(cnn2C2CCOCC2)c1
null
null
[Cl-].[NH4+].[N+:3]([C:6]1[CH:7]=[C:8]2[CH:14]=[N:13][N:12]([CH:15]3[CH2:20][CH2:19][O:18][CH2:17][CH2:16]3)[C:9]2=[N:10][CH:11]=1)([O-])=O>C(O)C.C1COCC1.O.[Fe]>[O:18]1[CH2:17][CH2:16][CH:15]([N:12]2[C:9]3=[N:10][CH:11]=[C:6]([NH2:3])[CH:7]=[C:8]3[CH:14]=[N:13]2)[CH2:20][CH2:19]1
null
O
C1CCOC1
CCO
100
null
108.8
729,905
4,309
null
null
null
null
ord_dataset-a5669edbeffe43bf8514c1bfede8f882
1976-01-01T00:04:00
true
69 g of bromine were added to a mixture of 69.2 g of 4-ethoxycarbonyl-4-thiazoline-2-one in 500 ml of chloroform and the mixture was refluxed for 20 hours. The mixture was distilled to dryness under reduced pressure and after the addition of isopropyl ether, the mixture was vacuum filtered to obtain 75.2 g of 5-bromo-4...
CCOC(=O)c1[nH]c(=O)sc1Br
null
CCOC(=O)c1csc(=O)[nH]1
BrBr
null
[Br:1]Br.[CH2:3]([O:5][C:6]([C:8]1[NH:9][C:10](=[O:13])[S:11][CH:12]=1)=[O:7])[CH3:4]>C(Cl)(Cl)Cl>[Br:1][C:12]1[S:11][C:10](=[O:13])[NH:9][C:8]=1[C:6]([O:5][CH2:3][CH3:4])=[O:7]
null
ClC(Cl)Cl
null
null
null
null
74.7
642,869
1,141,391
Cn1c(=O)c2c(-c3cc(F)ccc3Br)c(CN)c(N3CCOCC3)nc2n(C)c1=O
null
null
null
ord_dataset-68715347640045adb1b09e6a04722b0e
2012-01-01T00:03:00
true
The title compound was prepared from Compound 47a (Example and 1,2-diphenylethanamine, according to procedure described in the synthesis of Compound 47. MS [m+H] calc'd C30H28BrFN5O2 588; found 588.
Cn1c(=O)c2c(-c3cc(F)ccc3Br)c(CN)c(NC(Cc3ccccc3)c3ccccc3)nc2n(C)c1=O
null
Cn1c(=O)c2c(-c3cc(F)ccc3Br)c(C#N)c(Cl)nc2n(C)c1=O
NC(Cc1ccccc1)c1ccccc1
null
[Br:1][C:2]1[CH:7]=[CH:6][C:5]([F:8])=[CH:4][C:3]=1[C:9]1[C:18]2[C:17](=[O:19])[N:16]([CH3:20])[C:15](=[O:21])[N:14]([CH3:22])[C:13]=2[N:12]=[C:11](Cl)[C:10]=1[C:24]#[N:25].[C:26]1([CH:32]([NH2:40])[CH2:33][C:34]2[CH:39]=[CH:38][CH:37]=[CH:36][CH:35]=2)[CH:31]=[CH:30][CH:29]=[CH:28][CH:27]=1.NCC1C(N2CCOCC2)=NC2N(C)C(=O...
null
null
null
null
null
null
null
208,370
885,939
[H-]
[Na+]
null
null
ord_dataset-d728a2f811c0424cbcdb5a84d02b93ae
2009-01-01T00:06:00
true
To a cooled (0° C.) suspension of NaH (45 mg, 1.1 mmol, 60% w/w in mineral oil) in DMF (0.5 ml) is added a solution of 2-Methyl-3-{4-[2-(3-methyl-2-oxo-imidazolidin-4-yl)-ethoxy]-phenyl}-2-phenoxy-propionic acid ethyl ester (320 mg, 0.75 mmol) in DMF (1.5 ml). After 5 minutes, the reaction mixture is removed from the c...
CCOC(=O)C(C)(Cc1ccc(OCCC2CN(Cc3ccc(C(=O)c4ccccc4)cc3)C(=O)N2C)cc1)Oc1ccccc1
null
CCOC(=O)C(C)(Cc1ccc(OCCC2CNC(=O)N2C)cc1)Oc1ccccc1
O=C(c1ccccc1)c1ccc(CBr)cc1
null
[H-].[Na+].[CH2:3]([O:5][C:6](=[O:33])[C:7]([CH3:32])([O:25][C:26]1[CH:31]=[CH:30][CH:29]=[CH:28][CH:27]=1)[CH2:8][C:9]1[CH:14]=[CH:13][C:12]([O:15][CH2:16][CH2:17][CH:18]2[CH2:22][NH:21][C:20](=[O:23])[N:19]2[CH3:24])=[CH:11][CH:10]=1)[CH3:4].Br[CH2:35][C:36]1[CH:49]=[CH:48][C:39]([C:40]([C:42]2[CH:47]=[CH:46][CH:45]=...
0.08
CN(C)C=O
null
null
25
null
10.9
550,139
35,539
O=C([O-])[O-]
[K+]
null
null
ord_dataset-c8db783fb93842e89cdcd41afa59a141
1978-01-01T00:01:00
true
A mixture of 7.6 g of the product of Step A, 9.5 g of diethyl chlorothiophosphate and 7 g of potassium carbonate in 50 ml of acetone was stirred overnight at room temperature and the mixture was then filtered. The filtrate was concentrated by evaporation under reduced pressure and was chromatographed over silica. Eluti...
CCOP(=S)(OCC)Oc1nsc(SC)n1
null
CCOP(=S)(Cl)OCC
CSc1nc(O)ns1
null
[OH:1][C:2]1[N:6]=[C:5]([S:7][CH3:8])[S:4][N:3]=1.[P:9](Cl)([O:14][CH2:15][CH3:16])([O:11][CH2:12][CH3:13])=[S:10].C(=O)([O-])[O-].[K+].[K+]>CC(C)=O>[CH2:12]([O:11][P:9]([O:1][C:2]1[N:6]=[C:5]([S:7][CH3:8])[S:4][N:3]=1)([O:14][CH2:15][CH3:16])=[S:10])[CH3:13]
8
CC(C)=O
null
null
25
null
null
410,107
1,375,730
[Pt]
null
null
null
ord_dataset-d23f2f15886d4c22b7d7ba5f0e203e81
2013-01-01T00:12:00
true
4-Bromo-3-methyl-2-nitrophenol (10 g, 43.1 mmol) was dissolved in methanol (254 ml), purged with nitrogen and loaded with Pt/C (1.013 g, 10.13 mmol). The reaction was stirred under 60 psi of hydrogen for 5 hours. When complete, the reaction was filtered carefully on Celite™. The top was covered by more Celite™, flushed...
Cc1c(Br)ccc(O)c1N
null
[H][H]
Cc1c(Br)ccc(O)c1[N+](=O)[O-]
null
[Br:1][C:2]1[CH:7]=[CH:6][C:5]([OH:8])=[C:4]([N+:9]([O-])=O)[C:3]=1[CH3:12].[H][H]>CO.[Pt]>[NH2:9][C:4]1[C:3]([CH3:12])=[C:2]([Br:1])[CH:7]=[CH:6][C:5]=1[OH:8]
null
CO
null
null
null
98.8
null
393,786
1,749,047
CN(C)C(On1nnc2cccnc21)=[N+](C)C
F[P-](F)(F)(F)(F)F
null
null
ord_dataset-60a3e71da3174666a50a61dcfa611a9f
2016-01-01T00:07:00
true
66 mg (0.228 mmol) of the compound of Example 6A and 74 mg (0.228 mmol) of the compound of Example 32A were dissolved in 1.5 ml of anhydrous DMF, and 104 mg (0.273 mmol) of HATU and 48 μl (0.273 mmol) of N,N-diisopropylethylamine were added in succession. The reaction mixture was stirred at RT for 4 h and then separate...
Cc1ccc(NC(=O)c2cc(S(C)(=O)=O)cc(S(F)(F)(F)(F)F)c2)cc1-n1ccn2nc(-c3cccnc3)cc12
null
Cc1ccc(N)cc1-n1ccn2nc(-c3cccnc3)cc12
CS(=O)(=O)c1cc(C(=O)O)cc(S(F)(F)(F)(F)F)c1
null
[CH3:1][C:2]1[CH:8]=[CH:7][C:5]([NH2:6])=[CH:4][C:3]=1[N:9]1[C:16]2[N:12]([N:13]=[C:14]([C:17]3[CH:18]=[N:19][CH:20]=[CH:21][CH:22]=3)[CH:15]=2)[CH:11]=[CH:10]1.[CH3:23][S:24]([C:27]1[CH:28]=[C:29]([CH:33]=[C:34]([S:36]([F:41])([F:40])([F:39])([F:38])[F:37])[CH:35]=1)[C:30](O)=[O:31])(=[O:26])=[O:25].CN(C(ON1N=NC2C=CC=...
4
CCN(C(C)C)C(C)C
CN(C)C=O
null
25
null
null
637,694
1,222,283
null
null
null
null
ord_dataset-cde802cdb7434a5f82a22981ccaefc4e
2012-01-01T00:11:00
true
To a solution of 6-(3-nitrophenoxy)[1,2,4]triazolo[1,5-a]pyridin-2-amine (3.49 g, 12.9 mmol) in N,N-dimethylacetamide (20 mL) was added with stirring under ice-cooling cyclopropanecarbonyl chloride (2.46 mL, 27.0 mmol), and the mixture was stirred at room temperature for 15 hr. Water (40 mL) was added to the reaction m...
O=C(Nc1nc2ccc(Oc3cccc([N+](=O)[O-])c3)cn2n1)C1CC1
null
O=C(Cl)C1CC1
Nc1nc2ccc(Oc3cccc([N+](=O)[O-])c3)cn2n1
null
[N+:1]([C:4]1[CH:5]=[C:6]([CH:18]=[CH:19][CH:20]=1)[O:7][C:8]1[CH:9]=[CH:10][C:11]2[N:12]([N:14]=[C:15]([NH2:17])[N:16]=2)[CH:13]=1)([O-:3])=[O:2].[CH:21]1([C:24](Cl)=[O:25])[CH2:23][CH2:22]1.O>CN(C)C(=O)C>[N+:1]([C:4]1[CH:5]=[C:6]([CH:18]=[CH:19][CH:20]=1)[O:7][C:8]1[CH:9]=[CH:10][C:11]2[N:12]([N:14]=[C:15]([NH:17][C:...
null
CC(=O)N(C)C
O
null
null
null
88.2
828,787
318,202
O=C([O-])[O-]
[K+]
null
null
ord_dataset-eb32c2b9cbdf4fc39ce6c9fe0fa11430
1995-01-01T00:10:00
true
Isovanillin (50 g, 0.328 mol) is placed in a 1 liter round bottom flask which is equipped with a stir bar and reflux condensor and is charged with 500 ml of dimethylformamide. Potassium carbonate (45.3 g, 0.328 mol) is added to the reaction mixture which is heated to 80° C. At this temperature exo-2-bromonorbornane (12...
COc1ccc(C=O)c(OC2CC3CCC2C3)c1
null
BrC1CC2CCC1C2
CN(C)C=O
COc1ccc(C=O)cc1O
[O:1]=[CH:2][C:3]1[CH:11]=[CH:10][C:7]([O:8][CH3:9])=[C:5](O)[CH:4]=1.CN(C)[CH:14]=[O:15].C(=O)([O-])[O-].[K+].[K+].[CH2:23]1[CH:27]2C[CH:29](Br)[CH:25]([CH2:26]2)[CH2:24]1>O>[CH:27]12[CH2:26][CH:25]([CH2:24][CH2:23]1)[CH2:29][CH:14]2[O:15][C:4]1[CH:5]=[C:7]([O:8][CH3:9])[CH:10]=[CH:11][C:3]=1[CH:2]=[O:1]
null
O
null
null
80
null
null
356,102
879,957
Cl
null
null
null
ord_dataset-3592bd645cd143ee8274cd0d834ae581
2009-01-01T00:05:00
true
Trans-3-[4-aminocyclohexylcarbonylamino]-N-(4-chlorophenyl)benzofuran-2-carboxamide hydrochloride (150 mg) obtained in Example 225 is suspended in acetonitrile/methanol (5/1, 6 ml), and thereto is added triethylamine (93 μl), and the mixture is stirred at room temperature for several minutes. The reaction solution is c...
O=C(Nc1ccc(Cl)cc1)c1oc2ccccc2c1NC(=O)[C@H]1CC[C@H](NCCO)CC1
null
OCCI
N[C@H]1CC[C@H](C(=O)Nc2c(C(=O)Nc3ccc(Cl)cc3)oc3ccccc23)CC1
null
Cl.[NH2:2][C@H:3]1[CH2:8][CH2:7][C@H:6]([C:9]([NH:11][C:12]2[C:16]3[CH:17]=[CH:18][CH:19]=[CH:20][C:15]=3[O:14][C:13]=2[C:21]([NH:23][C:24]2[CH:29]=[CH:28][C:27]([Cl:30])=[CH:26][CH:25]=2)=[O:22])=[O:10])[CH2:5][CH2:4]1.C(N(CC)CC)C.I[CH2:39][CH2:40][OH:41]>C(Cl)(Cl)Cl.CO>[OH:41][CH2:40][CH2:39][NH:2][C@H:3]1[CH2:8][CH2...
null
CO
CCN(CC)CC
ClC(Cl)Cl
25
null
null
101,191
1,394,935
null
null
null
null
ord_dataset-12dc3bd21bcf44d09e5b4249afe15161
2014-01-01T00:02:00
true
The title compound was synthesized in analogy to Example 1 using 5-(4-chlorophenyl)-6-(2,2,2-trifluoroethoxy)-3-pyridinecarboxylic acid (CAN 1018782-82-5) and 4-(t-butyl-dimethyl-silanyloxymethyl)-piperidin-1-ylamine trifluoroacetate (1:1) as starting materials; the silyl protecting group was lost during reaction and w...
O=C(NN1CCC(CCO)CC1)c1cnc(OCC(F)(F)F)c(-c2ccc(Cl)cc2)c1
null
O=C(O)C(F)(F)F
O=C(O)c1cnc(OCC(F)(F)F)c(-c2ccc(Cl)cc2)c1
CC(C)(C)[SiH2]OC(C)(C)C1CCN(N)CC1
[Cl:1][C:2]1[CH:7]=[CH:6][C:5]([C:8]2[CH:9]=[C:10]([C:20]([OH:22])=O)[CH:11]=[N:12][C:13]=2[O:14][CH2:15][C:16]([F:19])([F:18])[F:17])=[CH:4][CH:3]=1.F[C:24](F)(F)[C:25]([OH:27])=O.C([SiH2]OC(C)(C)[CH:37]1[CH2:42][CH2:41][N:40]([NH2:43])[CH2:39][CH2:38]1)(C)(C)C>>[Cl:1][C:2]1[CH:7]=[CH:6][C:5]([C:8]2[CH:9]=[C:10]([C:20...
null
null
null
null
null
null
null
694,949
1,500,354
null
null
null
null
ord_dataset-366bdd9ee72d474cbe6f3f9e54dd96d2
2014-01-01T00:10:00
true
The mixture of 2,4,6-trichloroquinoline (300 mg, 1.29 mmol), 7-bromo-2,3,4,5-tetrahydro-1H-2-benzazepine (291 mg, 1.29 mmol) and n-butanol (3 mL) was heated with stirring in a 10 mL microwave process vial for 1 hour at 160° C. under microwave irradiation. The mixture was cooled to room temperature and diluted with ethy...
Clc1ccc2nc(N3CCCc4cc(Br)ccc4C3)cc(Cl)c2c1
null
Clc1ccc2nc(Cl)cc(Cl)c2c1
Brc1ccc2c(c1)CCCNC2
null
Cl[C:2]1[CH:11]=[C:10]([Cl:12])[C:9]2[C:4](=[CH:5][CH:6]=[C:7]([Cl:13])[CH:8]=2)[N:3]=1.[Br:14][C:15]1[CH:16]=[CH:17][C:18]2[CH2:24][NH:23][CH2:22][CH2:21][CH2:20][C:19]=2[CH:25]=1.C(O)CCC>C(OCC)(=O)C>[Br:14][C:15]1[CH:16]=[CH:17][C:18]2[CH2:24][N:23]([C:2]3[CH:11]=[C:10]([Cl:12])[C:9]4[C:4](=[CH:5][CH:6]=[C:7]([Cl:13]...
1
CCCCO
CCOC(C)=O
null
160
40.8
null
373,927
930,185
null
null
null
null
ord_dataset-d8a5dc784dde4465894ec7c69d2e3ba6
2010-01-01T00:01:00
true
To a stirred and cooled suspension of N-tert-butyl-3-[6-methyl-4-(4-trifluoromethylphenyl)-[2,4′]bipyridinyl-2′-yl]-benzenesulfonamide (example 287) (0.239 g, 0.455 mmol) in dichloromethane (1.5 mL) was added TFA (10 mL) and the reaction mixture was allowed to stir at room temperature for 16 h. The mixture was evaporat...
Cc1cc(-c2ccc(C(F)(F)F)cc2)cc(-c2ccnc(-c3cccc(S(N)(=O)=O)c3)c2)n1
null
Cc1cc(-c2ccc(C(F)(F)F)cc2)cc(-c2ccnc(-c3cccc(S(=O)(=O)NC(C)(C)C)c3)c2)n1
null
null
C([NH:5][S:6]([C:9]1[CH:14]=[CH:13][CH:12]=[C:11]([C:15]2[CH:20]=[C:19]([C:21]3[CH:26]=[C:25]([C:27]4[CH:32]=[CH:31][C:30]([C:33]([F:36])([F:35])[F:34])=[CH:29][CH:28]=4)[CH:24]=[C:23]([CH3:37])[N:22]=3)[CH:18]=[CH:17][N:16]=2)[CH:10]=1)(=[O:8])=[O:7])(C)(C)C.C(O)(C(F)(F)F)=O>ClCCl>[CH3:37][C:23]1[N:22]=[C:21]([C:19]2[...
null
ClCCl
O=C(O)C(F)(F)F
null
null
93.6
null
779,260
1,377,807
Cl
[BH4-]
[Na+]
null
ord_dataset-d23f2f15886d4c22b7d7ba5f0e203e81
2013-01-01T00:12:00
true
Sodium borohydride (63.58 mg; 1.68 mmol; 0.07 eq) is suspended in DME (6.5 mL) at room temperature. Borane-methyl sulfide complex (39.61 mL; 2 M; 79.22 mmol; 3.3 eq) is added dropwise. After 30 min stirring at room temperature, a solution of 4-(4-methoxy-2-nitrobenzylidene)tetrahydro-2H-thiopyran (6.37 g; 24.01 mmol; 1...
COc1ccc(CC2CCSCC2)c(N)c1
null
COc1ccc(C=C2CCSCC2)c([N+](=O)[O-])c1
null
null
[BH4-].[Na+].[CH3:3][O:4][C:5]1[CH:17]=[CH:16][C:8]([CH:9]=[C:10]2[CH2:15][CH2:14][S:13][CH2:12][CH2:11]2)=[C:7]([N+:18]([O-])=O)[CH:6]=1.Cl>COCCOC.CO>[CH3:3][O:4][C:5]1[CH:17]=[CH:16][C:8]([CH2:9][CH:10]2[CH2:15][CH2:14][S:13][CH2:12][CH2:11]2)=[C:7]([CH:6]=1)[NH2:18]
0.5
CO
COCCOC
null
25
null
41.9
637,305
1,132,803
[Cu]Br
O=N[O-]
[Na+]
null
ord_dataset-aaeaab5f3720492494c1cbbdd0ed2820
2012-01-01T00:02:00
true
A mixture of ethyl 5-amino-2-methylbenzoate (1.50 g, 8.3 mmol) in 48% HBr (12 mL) and water (24 mL) was cooled with an ice-bath for 15 min. Sodium nitrite (0.59 g, 8.6 mmol) was then added dropwise as a solution in water (2 mL), and the resulting mixture stirred for 5 min. After this time, the mixture was added to an i...
CCOC(=O)c1cc(Br)ccc1C
null
CCOC(=O)c1cc(N)ccc1C
Br
null
N[C:2]1[CH:3]=[CH:4][C:5]([CH3:13])=[C:6]([CH:12]=1)[C:7]([O:9][CH2:10][CH3:11])=[O:8].N([O-])=O.[Na+].[BrH:18]>O.C(OCC)C.[Cu]Br>[Br:18][C:2]1[CH:3]=[CH:4][C:5]([CH3:13])=[C:6]([CH:12]=1)[C:7]([O:9][CH2:10][CH3:11])=[O:8]
0.08
CCOCC
O
null
70
69
null
15,380
590,662
Cl
null
null
null
ord_dataset-7a74d48eeefd45aba53e7258f3ae067a
2003-01-01T00:04:00
true
Dissolve 2-phenylpropionic acid (30 g) in 2B ethanol (100 mL and add anhydrous HCl (10 g). Allow to sit for 48-72 hours, evaporate the solvent in vacuo and purify by distillation to give ethyl 2-phenylpropionate (31 g); bp 100 C at 6 mm.
CCOC(=O)C(C)c1ccccc1
null
CC(C(=O)O)c1ccccc1
CCO
null
[C:1]1([CH:7]([CH3:11])[C:8]([OH:10])=[O:9])[CH:6]=[CH:5][CH:4]=[CH:3][CH:2]=1.Cl.[CH2:13](O)[CH3:14]>>[C:1]1([CH:7]([CH3:11])[C:8]([O:10][CH2:13][CH3:14])=[O:9])[CH:6]=[CH:5][CH:4]=[CH:3][CH:2]=1
60
null
null
null
null
null
null
446,250
1,025,106
O=C([O-])[O-]
[K+]
null
null
ord_dataset-136cfada6ce247b4919085a57363459e
2011-01-01T00:01:00
true
A mixture of 2,4-difluoro-1-nitrobenzene (50 g, 314 mmol), 4-methyl-1H-imidazole (25.7 g, 314 mmol) and potassium carbonate (100 g, 725 mmol) in dichloromethane (600 mL) was stirred at room temperature for 4 days. The mixture was washed with water then dried over magnesium sulfate. Solvent was removed under reduced pre...
Cc1cn(-c2cc(F)ccc2[N+](=O)[O-])cn1
null
Cc1c[nH]cn1
O=[N+]([O-])c1ccc(F)cc1F
null
F[C:2]1[CH:7]=[C:6]([F:8])[CH:5]=[CH:4][C:3]=1[N+:9]([O-:11])=[O:10].[CH3:12][C:13]1[N:14]=[CH:15][NH:16][CH:17]=1.C(=O)([O-])[O-].[K+].[K+]>ClCCl>[F:8][C:6]1[CH:5]=[CH:4][C:3]([N+:9]([O-:11])=[O:10])=[C:2]([N:16]2[CH:17]=[C:13]([CH3:12])[N:14]=[CH:15]2)[CH:7]=1
96
ClCCl
null
null
25
null
50.4
256,324
431,994
null
null
null
null
ord_dataset-8cbb58558c904b2b85fa7a1b084a0de9
1999-01-01T00:06:00
true
2-Amino-4-chloro-6-hydroxy-5-nitropyrimidine (4 g), 3-methylbutylamine (1.8 g) and triethylamine (6 ml) were heated at reflux for 5 h then left stirring overnight at room temperature in ethanol. The precipitate was filtered and washed with water and air dried to yield the title compound as a yellow solid.
CC(C)CCNc1nc(N)nc(O)c1[N+](=O)[O-]
null
CC(C)CCN
Nc1nc(O)c([N+](=O)[O-])c(Cl)n1
null
[NH2:1][C:2]1[N:7]=[C:6](Cl)[C:5]([N+:9]([O-:11])=[O:10])=[C:4]([OH:12])[N:3]=1.[CH3:13][CH:14]([CH3:18])[CH2:15][CH2:16][NH2:17].C(N(CC)CC)C>C(O)C>[NH2:1][C:2]1[N:7]=[C:6]([NH:17][CH2:16][CH2:15][CH:14]([CH3:18])[CH3:13])[C:5]([N+:9]([O-:11])=[O:10])=[C:4]([OH:12])[N:3]=1
null
CCO
CCN(CC)CC
null
null
null
null
516,145
683,395
null
null
null
null
ord_dataset-359b8fc87f4244be89d6f02bc5036eac
2005-01-01T00:09:00
true
A mixture of the title compound of Example 89 (30 mg, 0.06 mmol) and N,N-dimethylmethyleneiminium iodide (57 mg, 0.23 mmol) in anhydrous dichloromethane was stirred at room temperature overnight. The reaction mixture was purified by solid phase extraction using a Varian Bond Elut SCX cartridge (methanol for washing, me...
CCCOc1ccc(S(=O)(=O)N2CCN(C)CC2)cc1-c1[nH]c2c(c1CN(C)C)c(=O)n(C)c(=O)n2CCC
null
CCCOc1ccc(S(=O)(=O)N2CCN(C)CC2)cc1-c1cc2c(=O)n(C)c(=O)n(CCC)c2[nH]1
null
null
[CH3:1][N:2]1[C:7](=[O:8])[C:6]2[CH:9]=[C:10]([C:12]3[CH:17]=[C:16]([S:18]([N:21]4[CH2:26][CH2:25][N:24]([CH3:27])[CH2:23][CH2:22]4)(=[O:20])=[O:19])[CH:15]=[CH:14][C:13]=3[O:28][CH2:29][CH2:30][CH3:31])[NH:11][C:5]=2[N:4]([CH2:32][CH2:33][CH3:34])[C:3]1=[O:35]>ClCCl>[CH3:1][N:2]([CH2:7][C:9]1[C:6]2[C:7](=[O:8])[N:2]([...
8
ClCCl
null
null
25
null
190.2
140,088
1,591,795
c1ccc([P](c2ccccc2)(c2ccccc2)[Pd]([P](c2ccccc2)(c2ccccc2)c2ccccc2)([P](c2ccccc2)(c2ccccc2)c2ccccc2)[P](c2ccccc2)(c2ccccc2)c2ccccc2)cc1
O=C([O-])[O-]
[Na+]
null
ord_dataset-e8c6a25568b64529b960953990e6921f
2015-01-01T00:06:00
true
A mixture of 6.5 g (14 mmol) of 2-(4-(10-bromoanthracen-9-yl)naphthalene-1-yl)thiophene, 7.53 g (16 mmol) of 2-(10,10-dimethyl-10H-indeno[1,2-b]triphenylen-12-yl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane, 0.16 g (0.14 mmol) of tetrakis(triphenylphosphine)palladium, 11 ml of 2M Na2CO3, 30 ml of EtOH and 65 ml toluene was...
CC1(C)C=C(c2c3ccccc3c(-c3ccc(-c4cccs4)c4ccccc34)c3ccccc23)C=C2C=c3cc4c5ccccc5c5ccccc5c4cc3=C21
null
CC1(C)C=C(B2OC(C)(C)C(C)(C)O2)C=C2C=c3cc4c5ccccc5c5ccccc5c4cc3=C21
Brc1c2ccccc2c(-c2ccc(-c3cccs3)c3ccccc23)c2ccccc12
null
Br[C:2]1[C:15]2[C:10](=[CH:11][CH:12]=[CH:13][CH:14]=2)[C:9]([C:16]2[C:25]3[C:20](=[CH:21][CH:22]=[CH:23][CH:24]=3)[C:19]([C:26]3[S:27][CH:28]=[CH:29][CH:30]=3)=[CH:18][CH:17]=2)=[C:8]2[C:3]=1[CH:4]=[CH:5][CH:6]=[CH:7]2.[CH3:31][C:32]1([CH3:66])[C:56]2[C:36]([CH:37]=[C:38]3[CH:55]=[C:54]4[C:41]([C:42]5[C:47]([C:48]6[C:...
null
CO
Cc1ccccc1
CCO
90
null
62.7
364,106
1,735,814
[Al+3]
[Cl-]
null
null
ord_dataset-eacfee6d16d8455a93348409f1b37be4
2016-01-01T00:06:00
true
To 11-(2-ethylhexyl)-11H-benzo[a]carbazole (10.0 g, 30.6 mmol) in CH2Cl2 (150 mL) are added 4-fluorobenzoyl chloride (5.03 g, 31.7 mmol) and AlCl3 (4.58 g, 34.3 mmol) at 0° C. After stirring for 0.5 hour, the reaction mixture is stirred for 2 hours at room temperature. The reaction mixture is poured into ice-water, and...
CCCCC(CC)Cn1c2ccccc2c2cc(C(=O)c3ccc(F)cc3)c3ccccc3c21
null
CCCCC(CC)Cn1c2ccccc2c2ccc3ccccc3c21
O=C(Cl)c1ccc(F)cc1
null
[CH2:1]([CH:3]([CH2:22][CH2:23][CH2:24][CH3:25])[CH2:4][N:5]1[C:17]2[C:12](=[CH:13][CH:14]=[C:15]3[CH:21]=[CH:20][CH:19]=[CH:18][C:16]3=2)[C:11]2[C:6]1=[CH:7][CH:8]=[CH:9][CH:10]=2)[CH3:2].[F:26][C:27]1[CH:35]=[CH:34][C:30]([C:31](Cl)=[O:32])=[CH:29][CH:28]=1.[Al+3].[Cl-].[Cl-].[Cl-]>C(Cl)Cl>[CH2:1]([CH:3]([CH2:22][CH2...
0.5
ClCCl
null
null
0
null
null
522,456
1,281,159
null
null
null
null
ord_dataset-d5c54236ecd94d61aaa071461bcfc426
2013-01-01T00:04:00
true
Using the same method as in Example 19-(ii), 3-thiopheneboronic acid was reacted with the 2-[((2-[(3-bromobenzyl)amino]-2-oxoethoxy)acetyl)amino]-5-chlorobenzoic acid methyl ester to give 5-chloro-2-([(2-oxo-2-([3-(thiophene-3-yl)benzyl]amino)ethoxy)acetyl]amino)benzoic acid.methyl ester (yield: 77%).
O=C(COCC(=O)Nc1ccc(Cl)cc1C(=O)O)NCc1cccc(-c2ccsc2)c1
null
OB(O)c1ccsc1
COC(=O)c1cc(Cl)ccc1NC(=O)COCC(=O)NCc1cccc(Br)c1
null
[S:1]1[CH:5]=[CH:4][C:3](B(O)O)=[CH:2]1.C[O:10][C:11](=[O:36])[C:12]1[CH:17]=[C:16]([Cl:18])[CH:15]=[CH:14][C:13]=1[NH:19][C:20](=[O:35])[CH2:21][O:22][CH2:23][C:24]([NH:26][CH2:27][C:28]1[CH:33]=[CH:32][CH:31]=[C:30](Br)[CH:29]=1)=[O:25]>>[Cl:18][C:16]1[CH:15]=[CH:14][C:13]([NH:19][C:20](=[O:35])[CH2:21][O:22][CH2:23]...
null
null
null
null
null
null
null
796,545
1,597,439
null
null
null
null
ord_dataset-e8c6a25568b64529b960953990e6921f
2015-01-01T00:06:00
true
To a mixture of 1-(3-fluorophenyl)-N-methoxy-N-methyl-1H-indole-2-carboxamide (0.52 g, 1.7 mmol) in tetrahydrofuran (10 mL) was added 3.0 M methylmagnesium bromide in ether (4.6 mL, 0.014 mol). The reaction was stirred at room temperature overnight. The reaction was quenched with saturated NH4Cl solution and extracted ...
CC(=O)c1cc2ccccc2n1-c1cccc(F)c1
null
CON(C)C(=O)c1cc2ccccc2n1-c1cccc(F)c1
C[Mg]Br
null
[F:1][C:2]1[CH:3]=[C:4]([N:8]2[C:16]3[C:11](=[CH:12][CH:13]=[CH:14][CH:15]=3)[CH:10]=[C:9]2[C:17](N(OC)C)=[O:18])[CH:5]=[CH:6][CH:7]=1.[CH3:23][Mg]Br.CCOCC>O1CCCC1>[F:1][C:2]1[CH:3]=[C:4]([N:8]2[C:16]3[C:11](=[CH:12][CH:13]=[CH:14][CH:15]=3)[CH:10]=[C:9]2[C:17](=[O:18])[CH3:23])[CH:5]=[CH:6][CH:7]=1
8
C1CCOC1
CCOCC
null
25
91
null
1,022
1,198,953
CC(C)(C)[O-]
[K+]
null
null
ord_dataset-fb72428f30234761b4216139dc228d0c
2012-01-01T00:09:00
true
A solution of 5-fluoro-1H-indole (16.9 mmol) and potassium tert-butoxide (33.8 mmol) in DMF (76 mL) is stirred at rt under N2 for 2 h. 0.15 M NH2Cl. in ether (169.2 mL) is added drop-wise for 15 minutes at rt. The reaction mixture is stirred at rt for 2 h, then quenched with 10% Na2S2O3 aqueous solution and extracted w...
Nn1ccc2cc(F)ccc21
null
Fc1ccc2[nH]ccc2c1
NCl
null
[F:1][C:2]1[CH:3]=[C:4]2[C:8](=[CH:9][CH:10]=1)[NH:7][CH:6]=[CH:5]2.CC(C)([O-])C.[K+].[NH2:17]Cl>CN(C=O)C.CCOCC>[F:1][C:2]1[CH:3]=[C:4]2[C:8](=[CH:9][CH:10]=1)[N:7]([NH2:17])[CH:6]=[CH:5]2
2
CN(C)C=O
CCOCC
null
25
null
30