Molecule name
stringlengths
12
12
SMILES
stringlengths
30
101
LogD
float64
-0.7
4.5
ASAP-0008674
CC(C)[C@H](NC1=NC=NC2=C1C=CN2)C1=CC=C2CCCS(=O)(=O)C2=C1
2.7
ASAP-0008668
CC(C)[C@H](NC1=NC=NC2=C1C=C(C1=CN(CC(=O)N(C)C)N=C1)N2)C1=CC=C2CCCS(=O)(=O)C2=C1
2.1
ASAP-0008641
CNC(=O)C1=CNC2=NC=NC(N[C@H](C3=CC=C4CCCS(=O)(=O)C4=C3)C(C)C)=C12
2.5
ASAP-0008637
CNC(=O)C1=CNC2=NC=NC(N[C@H](C3=CC=C4OCC(=O)NC4=C3)C(C)C)=C12
3.2
ASAP-0008651
CC(C)[C@H](NC1=NC=NC2=C1C=C(C1=C(C#N)N(C)N=C1)N2)C1=CC=C2CCCS(=O)(=O)C2=C1
3.6
ASAP-0008650
COCCNC(=O)C1=CNC2=NC=NC(N[C@H](C3=CC=C4CCCS(=O)(=O)C4=C3)C(C)C)=C12
2.8
ASAP-0008648
CC(C)(C)[C@H](NC1=NC=NC2=C1C=C(C1=CN(CC(N)=O)N=C1)N2)C1=CC=C2OCCOC2=N1
2.7
ASAP-0008647
CC(C)[C@H](NC1=NC=NC2=C1C(C(=O)NC1CC1)=CN2)C1=CC=C2CCCS(=O)(=O)C2=C1
3.1
ASAP-0008645
CN1N=CC(C2=CC3=C(N[C@H](C4=CC=C5OCCOC5=N4)C(C)(C)C)N=CN=C3N2)=C1C#N
2.7
ASAP-0008644
CC(C)[C@H](NC1=NC=NC2=C1C=C(C1=C(C#N)N(C)N=C1)N2)C1=CC=C2OCC(=O)NC2=N1
3.7
ASAP-0008646
CC(C)[C@H](NC1=NC=NC2=C1C=C(C1=CN(CC(N)=O)N=C1)N2)C1=CC=C2OCCOC2=N1
2.4
ASAP-0008621
CC(C)[C@H](NC1=NC=NC2=C1C=C(C1=CN(CC(N)=O)N=C1)N2)C1=CC=C2OCC(=O)NC2=C1
2.5
ASAP-0008565
CNC(=O)CN1C=C(C2=CC3=C(N[C@H](C4=CC=C5OCCOC5=C4)C(C)C)N=CN=C3N2)C=N1
2.9
ASAP-0008571
CNC(=O)C1=CC2=C(N[C@H](C3=CC=C4OCC(=O)NC4=C3)C(C)C)N=CN=C2N1
2.8
ASAP-0008576
CC(C)[C@H](NC1=NC=NC2=C1C=C(C1=C(C#N)N(C)N=C1)N2)C1=CC=C2OCC(=O)NC2=C1
4.1
ASAP-0008581
CC(C)(C)[C@H](NC1=NC=NC2=C1C=C(C1=CN(CC(N)=O)N=C1)N2)C1=CC=C2OCCOC2=C1
3.2
ASAP-0008482
CC(C)[C@H](NC1=NC=NC2=C1C=C(C1=CN(CCC(N)=O)N=C1)N2)C1=CC=C2OCCOC2=C1
3
ASAP-0008484
CN1N=CC(C2=CC3=C(N[C@H](C4=CC=C5OCCOC5=C4)C(C)(C)C)N=CN=C3N2)=C1C#N
2.9
ASAP-0008485
CC(C)[C@H](NC1=NC=NC2=C1C=C(C1=CN(CC(=O)N(C)C)N=C1)N2)C1=CC=C2OCCOC2=C1
2.3
ASAP-0008431
CC(C)[C@H](NC1=NC=NC2=C1C=CN2)C1=CC=C2OCC(=O)NC2=C1
2.2
ASAP-0008445
C[C@H](C(=O)O)[C@H](NC(=O)C1=NC=NC2=C1C=CN2)C1=CC=C(Br)C=C1
0.5
ASAP-0008450
CC(C)[C@H](NC1=NC=NC2=C1C=C(C1=CN(CC(N)=O)N=C1)N2)C1=CC=C2OCCOC2=C1
2.9
ASAP-0008449
CC(C)[C@H](NC1=NC=NC2=C1C=C(C1=CN(CC(N)=O)N=C1)N2)C1=CC=C2OCCOC2=C1
2.9
ASAP-0008430
CC(C)[C@H](NC1=NC=NC2=C1C=CN2)C1=CC=C2OCC(=O)NC2=C1
1.8
ASAP-0008444
CCNC(=O)C1=CC2=C(N[C@H](C3=CC=C4OCCOC4=C3)C(C)C)N=CN=C2N1
3
ASAP-0008418
CC(C)[C@H](NC1=NC=NC2=C1C=C(C1=C(C#N)N(C)N=C1)N2)C1=CC=C2OCCOC2=N1
3.4
ASAP-0008399
CC(C)[C@H](NC1=NC=NC2=C1C(C(N)=O)=CN2)C1=CC=C2OCCOC2=C1
3.2
ASAP-0008406
CNC(=O)C1=CNC2=NC=NC(N[C@H](C3=CC=C4OCCOC4=C3)C(C)C)=C12
3.6
ASAP-0008340
COC1=CC=C([C@H](CC2=NN=NN2)NC(=O)C2=NC=NC3=C2C=CN3)C=C1
-0.1
ASAP-0008348
CNC(=O)C1=CC2=C(N[C@H](C3=CC=C4OCCOC4=C3)C(C)C)N=CN=C2N1
2.76
ASAP-0008327
CC(C)[C@H](NC1=NC=NC2=C1C=CN2)C1=CC=C2CCCS(=O)(=O)C2=C1
2.5
ASAP-0008288
CC(C)[C@H](NC1=NC=NC2=C1C=C(C1=CN(CC(N)=O)N=C1)N2)C1=CC=C2OCCOC2=C1
0.9
ASAP-0008279
CC(C)[C@H](NC1=NC=NC2=C1C=CN2)C1=CC=C2OCCOC2=C1
3
ASAP-0008270
CC(C)[C@H](NC1=NC=NC2=C1C=CN2)C1=CC=C2OCCOC2=N1
2.8
ASAP-0008275
CC(C)[C@H](NC1=NC=NC2=C1C=C(C1=C(C#N)N(C)N=C1)N2)C1=CC=C2OCCOC2=C1
3
ASAP-0000775
C[C@H]1CN(C2=CN=CC3=CC=CC=C23)C(=O)[C@@]12CN(CC(=O)NCC1=NN(C)C=C1)C(=O)C1=CC=C(Cl)C=C12
1.8
ASAP-0000774
C[C@H]1CN(C2=CN=CC3=CC=CC=C23)C(=O)[C@@]12CN(CC(=O)NCC1=CC=NN1C)C(=O)C1=CC=C(Cl)C=C12
2
ASAP-0000738
CNC(=O)CN1C[C@]2(C(=O)N(C3=CN=CC4=CC=CC=C34)C[C@H]2CC2CC2)C2=CC(Cl)=CC=C2C1=O
2.3
ASAP-0000733
CNC(=O)CN1C[C@@]2(C(=O)N(C3=CN=CC4=CC=CC=C34)C[C@@H]2C)C2=CC(Cl)=CC=C2C1=O
1.94
ASAP-0000627
O=C(NC1=C2NC=C(C(=O)N[C@H]3C4=CC=CC=C4C[C@H]3C(=O)O)C2=CC=C1)NC1CC1
-0.05
ASAP-0000591
COC1=CC=C([C@H](CC(=O)O)NC(=O)C2=NC=NC3=C2C=CN3)C=C1
-0.38
ASAP-0000528
CNC(=O)CN1C[C@]2(CCN(C3=CN=CC4=CC=C(OC[C@H](O)CN(C)C)C=C34)C2=O)C2=CC(Cl)=CC=C2C1=O
0.19
ASAP-0000541
CNC(=O)CN1C[C@@]2(C(=O)N(C3=CN=CC4=CC=CC=C34)C[C@@H]2C)C2=CC=CC=C2C1=O
0.7
ASAP-0000502
COC1=CC=C2C(=C1)CCN(C1=NC=NC3=C1C=CN3)[C@H]2C(C)C
4.33
ASAP-0000450
CC(C)[C@H](NC1=NC=NC2=C1C=CN2)C1=CC=C2OCCOC2=C1
3.2
ASAP-0000453
CC(C)[C@H](CO)NC1=NC=NC2=C1C=CN2
1.69
ASAP-0000272
CNC(=O)CN1C[C@@]2(C(=O)N(C3=CN=CC4=CC=CC=C34)C[C@@H]2C)C2=C(C=CC(F)=C2)C1=O
1.07
ASAP-0000175
C=CC(=O)NC1=CC=CC(N(CC2=CC=CC(Cl)=C2)C(=O)CC2=CN=CC3=CC=CC=C23)=C1
3.8
ASAP-0000136
O=C(O)C[C@H](NC(=O)C1=NC=NC2=C1C=CN2)C1=CC=C(Br)C=C1
0.22
ASAP-0000132
O=C(NC1=CC=CC=C1)NC1=CC=C(C(=O)NC2C3=C(CC2C(=O)O)C(O)=CC=C3)C=C1
0.12
ASAP-0023299
NCC1=CC(Cl)=CC(C(=O)NC2=CC=C3CNCC3=C2)=C1
2
ASAP-0000688
COC(=O)NC1=NC2=CC=C(C(=O)C3=CC=CC=C3)C=C2N1
2.9
ASAP-0031558
CC(C)[C@H]1C2=C(CCN1C(=O)CC1=CN=CC3=CC=CC=C13)SC=C2
3.6
ASAP-0031372
CC(C)C1(C)CCN(C(=O)CC2=CN=CC3=CC=CC=C23)CC1
3.7
ASAP-0031411
O=C(CC1=CN=CC2=CC=CC=C12)N1CCC2=C(C=CS2)C12CCC2
3.4
ASAP-0031442
CC1(CC(F)(F)F)CCN(C(=O)CC2=CN=CC3=CC=CC=C23)CC1
3
ASAP-0031187
CCC1=CC=C([C@H]2C[C@H](C)CCN2C(=O)CC2=CN=CC3=CC=CC=C23)O1
4.3
ASAP-0031242
O=C(CC1=CN=CC2=CC=CC=C12)N1CCC2=C(C1)N=CS2
1.6
ASAP-0031213
CC1=CN=CC(CC(=O)N2CCC3=C(C=CS3)C2)=C1
2.2
ASAP-0031146
CC(C)C1(F)CCN(C(=O)CC2=CN=CC3=CC=CC=C23)CC1
2.8
ASAP-0030055
COCC1CCN(C(=O)CC2=CN=CC3=CC=CC=C23)CC1
1.5
ASAP-0029987
O=C1C2=CC=C(Cl)C=C2[C@@]2(CN1CC1=NNC=C1)C(=O)N(C1=CN=CC3=CC=CC=C13)C[C@@H]2CNC1=NN=C(C(F)(F)F)O1
3.2
ASAP-0029984
O=C1C2=CC=C(Cl)C=C2[C@@]2(CN1CC1=NNC=C1)C(=O)N(C1=CN=CC3=CC=CC=C13)C[C@@H]2CNC1=NN=CS1
1.8
ASAP-0029947
O=C(CC1=CN=CC2=CC=CC=C12)N1CCC(C(F)(F)F)CC1
2.2
ASAP-0029694
CC1=NC=CC(CN2C[C@@]3(C(=O)N(C4=CN=CC5=CC=CC=C45)C[C@@H]3CNC3=NN=CO3)C3=CC(Cl)=CC=C3C2=O)=N1
1.4
ASAP-0029657
CCC1CCN(C(=O)CC2=CN=CC3=CC=CC=C23)CC1
2.8
ASAP-0029741
CC1=NC=CC(CN2C[C@@]3(C(=O)N(C4=CN=CC5=CC=CC=C45)C[C@@H]3CNC3=NN=C(C(F)(F)F)O3)C3=CC(Cl)=CC=C3C2=O)=N1
3
ASAP-0029738
C[C@@H]1CCN(C(=O)CC2=CN=CC3=CC=CC=C23)[C@H](C)C1
2.6
ASAP-0029707
CC1(C)CCN(C(=O)CC2=CN=CC3=CC=CC=C23)CC1
2.6
ASAP-0029604
CC(C)C1CCN(C(=O)CC2=CN=CC3=CC=CC=C23)CC1
3.2
ASAP-0029643
CC1=NC=CC(CN2C[C@@]3(C(=O)N(C4=CN=CC5=CC=CC=C45)C[C@@H]3CNC3=NN=C(C)O3)C3=CC(Cl)=CC=C3C2=O)=N1
1.6
ASAP-0029634
C[C@H]1C[C@@H](C)N(C(=O)CC2=CN=CC3=CC=CC=C23)[C@@H](C)C1
3.1
ASAP-0029560
CC1=NC=CC(CN2C[C@@]3(C(=O)N(C4=CN=CC5=CC=CC=C45)C[C@@H]3CNC3=NN=CS3)C3=CC(Cl)=CC=C3C2=O)=N1
1.7
ASAP-0029539
O=C(CC1=CN=CC2=CC=CC=C12)N1CCC(C(F)F)CC1
1.9
ASAP-0029423
CC(F)(F)C1CCN(C(=O)CC2=CN=CC3=CC=CC=C23)CC1
2.2
ASAP-0029287
CC(C)CC1(C)CCN(C(=O)CC2=CN=CC3=CC=CC=C23)CC1
3.9
ASAP-0028999
O=C(CC1=CN=CC2=CC=CC=C12)N(CC1=CC=CC(Cl)=C1)C1=CC=C2N=CNC2=C1
1.8
ASAP-0028832
COC1=CC=C(N(CC2=CC=CC(Cl)=C2)C(=O)CC2=CN=CC=C2C)C=C1
3.9
ASAP-0028820
C[C@H]1C2=C(CCN1C(=O)CC1=CN=CC3=CC=CC=C13)SC=C2
2.9
ASAP-0028829
C[C@H]1CCN(C(=O)CC2=CN=CC3=CC=CC=C23)C1
1.7
ASAP-0028830
C[C@H]1CCN1C(=O)CC1=CN=CC2=CC=CC=C12
1.3
ASAP-0028818
CC1=NC2=CC=C(N(CC3=CC=CC(Cl)=C3)C(=O)CC3=CN=CC4=CC=CC=C34)C=C2N1
3.9
ASAP-0028833
O=C(CC1=CN=CC2=CC=CC=C12)N1CCCN2N=CC=C2C1
1
ASAP-0028823
O=C(CC1=CN=CC2=CC=CC=C12)N1CCC2=C(Cl)C=CC=C2C1
3.7
ASAP-0028815
O=C(CC1=CN=CC2=CC=CC=C12)N1CCN2N=CC=C2C1
1.2
ASAP-0028819
C[C@H]1C2=C(CCN1C(=O)CC1=CN=CC3=CC=CC=C13)SC=C2
2.9
ASAP-0028810
O=C(CC1=CN=CC2=CC=CC=C12)N1CCC1
0.9
ASAP-0028872
C[C@H]1CCN(C(=O)CC2=CN=CC3=CC=CC=C23)CCO1
1.1
ASAP-0028866
CC1CN(C(=O)CC2=CN=CC3=CC=CC=C23)C1
1.3
ASAP-0028843
O=C(CC1=CN=CC2=CC=CC=C12)N1CCCOCC1
0.8
ASAP-0028890
CN(C)C(=O)CC1=CN=CC2=CC=CC=C12
0.9
ASAP-0028889
C[C@H]1CCOCCN1C(=O)CC1=CN=CC2=CC=CC=C12
1.1
ASAP-0028881
C[C@H]1CN(C(=O)CC2=CN=CC3=CC=CC=C23)CCCO1
1.1
ASAP-0028867
O=C(CC1=CN=CC2=CC=CC=C12)N1CCCCC1
1.8
ASAP-0028856
CC1CCN(C(=O)CC2=CN=CC3=CC=CC=C23)CC1
2.2
ASAP-0028855
CN1C=NC2=C1CCN(C(=O)CC1=CN=CC3=CC=CC=C13)C2
0.9
ASAP-0028844
CC1=NC2=C(CCN(C(=O)CC3=CN=CC4=CC=CC=C34)C2)N1C
0.9
ASAP-0028841
O=C(CC1=CN=CC2=CC=CC=C12)N1CCCC1
1.2
ASAP-0028838
CC[C@H]1C2=C(CCN1C(=O)CC1=CN=CC3=CC=CC=C13)SC=C2
3.3
ASAP-0028837
CC[C@H]1C2=C(CCN1C(=O)CC1=CN=CC3=CC=CC=C13)SC=C2
3.3