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Running
| { | |
| "delta_value": [ | |
| "0-1", | |
| "1-0", | |
| "0-0", | |
| "(-inf, -10.5]", "(-10.5, -8.5]","(-8.5, -6.5]","(-6.5, -4.5]","(-4.5, -2.5]","(-2.5, -1.5]","(-1.5, -1.0]","(-1.0, -0.5]","(-0.5, 0.0]","(0.0, 0.5]","(0.5, 1.0]","(1.0, 1.5]","(1.5, 2.5]","(2.5, 4.5]","(4.5, 6.5]","(6.5, 8.5]","(8.5, 10.5]","(10.5, inf]" | |
| ], | |
| "activity": [ | |
| "IC50 (nM)", | |
| "Kd (nM)", | |
| "EC50 (nM)", | |
| "Ki (nM)" | |
| ], | |
| "toxicity": [ | |
| "toxcast-NVS_TR_rVMAT2", | |
| "toxcast-BSK_4H_SRB_down", | |
| "toxcast-Tanguay_ZF_120hpf_CFIN_up", | |
| "toxcast-OT_FXR_FXRSRC1_1440", | |
| "toxcast-ATG_GRE_CIS_up", | |
| "toxcast-TOX21_Aromatase_Inhibition", | |
| "toxcast-ATG_NRF2_ARE_CIS_dn", | |
| "toxcast-Tanguay_ZF_120hpf_PFIN_up", | |
| "toxcast-NVS_LGIC_h5HT3", | |
| "toxcast-APR_HepG2_NuclearSize_72h_dn", | |
| "toxcast-ATG_Sox_CIS_up", | |
| "toxcast-OT_NURR1_NURR1RXRa_0480", | |
| "toxcast-ATG_VDRE_CIS_up", | |
| "toxcast-OT_ER_ERaERa_1440", | |
| "toxcast-NVS_GPCR_hAdrb3", | |
| "toxcast-TOX21_NFkB_BLA_agonist_ch2", | |
| "toxcast-NCCT_QuantiLum_inhib_2_dn", | |
| "toxcast-Tanguay_ZF_120hpf_MORT_up", | |
| "toxcast-APR_HepG2_p53Act_72h_up", | |
| "toxcast-BSK_3C_VCAM1_down", | |
| "toxcast-ATG_RARg_TRANS_dn", | |
| "toxcast-ATG_ERRa_TRANS_dn", | |
| "toxcast-Tanguay_ZF_120hpf_TRUN_up", | |
| "toxcast-TOX21_PPARg_BLA_antagonist_viability", | |
| "toxcast-NVS_GPCR_rmAdra2B", | |
| "toxcast-NVS_GPCR_hAdoRA2a", | |
| "toxcast-TOX21_PPARd_BLA_antagonist_viability", | |
| "toxcast-BSK_hDFCGF_MIG_down", | |
| "toxcast-TOX21_HSE_BLA_agonist_ch2", | |
| "tox21-NR-AR-LBD", | |
| "toxcast-APR_HepG2_MitoticArrest_72h_up", | |
| "toxcast-ATG_RORE_CIS_dn", | |
| "toxcast-NVS_GPCR_hDRD4.4", | |
| "toxcast-NVS_GPCR_h5HT7", | |
| "toxcast-TOX21_VDR_BLA_agonist_ch2", | |
| "toxcast-BSK_LPS_TNFa_up", | |
| "toxcast-ATG_VDR_TRANS_up", | |
| "toxcast-BSK_CASM3C_SRB_down", | |
| "toxcast-Tanguay_ZF_120hpf_EYE_up", | |
| "toxcast-BSK_LPS_IL8_up", | |
| "toxcast-CLD_UGT1A1_48hr", | |
| "toxcast-TOX21_p53_BLA_p3_ch2", | |
| "toxcast-ATG_EGR_CIS_up", | |
| "toxcast-ATG_SREBP_CIS_up", | |
| "toxcast-TOX21_ERa_BLA_Antagonist_ch2", | |
| "toxcast-ATG_MRE_CIS_up", | |
| "toxcast-ATG_HNF6_CIS_dn", | |
| "toxcast-TOX21_p53_BLA_p2_ratio", | |
| "toxcast-BSK_SAg_MIG_down", | |
| "toxcast-ATG_NURR1_TRANS_dn", | |
| "toxcast-Tanguay_ZF_120hpf_PIG_up", | |
| "toxcast-NVS_ADME_hCYP19A1", | |
| "toxcast-APR_HepG2_OxidativeStress_72h_up", | |
| "toxcast-NVS_GPCR_rSST", | |
| "toxcast-APR_HepG2_MicrotubuleCSK_72h_up", | |
| "toxcast-NVS_NR_hER", | |
| "tox21-NR-ER-LBD", | |
| "toxcast-NVS_MP_rPBR", | |
| "toxcast-TOX21_p53_BLA_p5_ch2", | |
| "toxcast-TOX21_AR_BLA_Antagonist_ratio", | |
| "toxcast-TOX21_ARE_BLA_agonist_ratio", | |
| "toxcast-ATG_E_Box_CIS_dn", | |
| "toxcast-NVS_IC_hKhERGCh", | |
| "toxcast-ATG_M_06_TRANS_up", | |
| "toxcast-ATG_Xbp1_CIS_dn", | |
| "toxcast-ATG_HIF1a_CIS_dn", | |
| "toxcast-BSK_3C_TissueFactor_down", | |
| "toxcast-TOX21_p53_BLA_p5_viability", | |
| "toxcast-TOX21_NFkB_BLA_agonist_ratio", | |
| "toxcast-CEETOX_H295R_OHPROG_dn", | |
| "toxcast-NVS_GPCR_rOpiate_NonSelectiveNa", | |
| "toxcast-BSK_3C_Vis_down", | |
| "toxcast-BSK_3C_Thrombomodulin_down", | |
| "skin_reaction", | |
| "toxcast-TOX21_AR_BLA_Antagonist_ch1", | |
| "toxcast-TOX21_NFkB_BLA_agonist_viability", | |
| "toxcast-NVS_ENZ_hElastase", | |
| "toxcast-NVS_GPCR_r5HT1_NonSelective", | |
| "toxcast-ATG_RXRa_TRANS_dn", | |
| "toxcast-APR_Hepat_MitoFxnI_24hr_dn", | |
| "toxcast-NVS_MP_hPBR", | |
| "toxcast-ATG_FXR_TRANS_up", | |
| "toxcast-BSK_CASM3C_SAA_up", | |
| "toxcast-BSK_CASM3C_HLADR_down", | |
| "toxcast-APR_HepG2_CellLoss_72h_dn", | |
| "toxcast-ATG_HIF1a_CIS_up", | |
| "toxcast-TOX21_MMP_viability", | |
| "toxcast-BSK_CASM3C_MIG_down", | |
| "toxcast-ATG_RARb_TRANS_dn", | |
| "toxcast-NCCT_HEK293T_CellTiterGLO", | |
| "toxcast-NVS_GPCR_g5HT4", | |
| "toxcast-TOX21_ERa_BLA_Agonist_ch2", | |
| "toxcast-TOX21_PPARg_BLA_Agonist_ch1", | |
| "toxcast-ATG_RORE_CIS_up", | |
| "toxcast-NVS_ENZ_oCOX2", | |
| "toxcast-NVS_NR_mERa", | |
| "toxcast-BSK_hDFCGF_PAI1_down", | |
| "toxcast-APR_HepG2_MicrotubuleCSK_72h_dn", | |
| "toxcast-ATG_E2F_CIS_dn", | |
| "toxcast-BSK_LPS_IL1a_up", | |
| "toxcast-ATG_RARa_TRANS_up", | |
| "toxcast-CLD_CYP1A2_24hr", | |
| "toxcast-ATG_GAL4_TRANS_dn", | |
| "toxcast-BSK_KF3CT_IP10_down", | |
| "toxcast-NVS_GPCR_hOpiate_D1", | |
| "toxcast-NVS_GPCR_rAdra2_NonSelective", | |
| "toxcast-ATG_RXRa_TRANS_up", | |
| "toxcast-CLD_GSTA2_48hr", | |
| "toxcast-ATG_HNF4a_TRANS_up", | |
| "toxcast-APR_HepG2_StressKinase_1h_up", | |
| "toxcast-BSK_KF3CT_uPA_down", | |
| "toxcast-TOX21_GR_BLA_Antagonist_viability", | |
| "toxcast-NVS_ENZ_hGSK3b", | |
| "toxcast-NVS_NR_rMR", | |
| "toxcast-CEETOX_H295R_PROG_up", | |
| "toxcast-ATG_PPARg_TRANS_up", | |
| "toxcast-BSK_KF3CT_MCP1_down", | |
| "toxcast-TOX21_HSE_BLA_agonist_viability", | |
| "toxcast-CLD_CYP1A1_6hr", | |
| "toxcast-NVS_GPCR_rAdrb_NonSelective", | |
| "toxcast-NVS_ADME_hCYP2C9", | |
| "toxcast-NVS_ADME_hCYP2A6", | |
| "toxcast-TOX21_VDR_BLA_antagonist_viability", | |
| "toxcast-OT_FXR_FXRSRC1_0480", | |
| "toxcast-BSK_3C_ICAM1_down", | |
| "toxcast-TOX21_PPARd_BLA_agonist_ratio", | |
| "toxcast-NVS_ENZ_hPTPN11", | |
| "toxcast-APR_HepG2_p53Act_24h_up", | |
| "toxcast-ATG_TA_CIS_up", | |
| "toxcast-ATG_THRa1_TRANS_dn", | |
| "toxcast-APR_Hepat_DNADamage_24hr_up", | |
| "toxcast-APR_HepG2_MitoticArrest_24h_up", | |
| "toxcast-BSK_KF3CT_TGFb1_down", | |
| "toxcast-TOX21_PPARg_BLA_Agonist_ch2", | |
| "toxcast-CLD_CYP1A1_48hr", | |
| "toxcast-ATG_THRa1_TRANS_up", | |
| "toxcast-TOX21_p53_BLA_p1_ratio", | |
| "toxcast-APR_Hepat_MitoFxnI_1hr_dn", | |
| "herg_central-hERG_at_1uM", | |
| "toxcast-APR_HepG2_CellCycleArrest_24h_dn", | |
| "toxcast-NVS_GPCR_hAdoRA1", | |
| "toxcast-TOX21_ERa_BLA_Agonist_ratio", | |
| "toxcast-OT_ER_ERbERb_0480", | |
| "toxcast-TOX21_AR_LUC_MDAKB2_Agonist", | |
| "toxcast-TOX21_GR_BLA_Antagonist_ratio", | |
| "toxcast-NVS_GPCR_hDRD2s", | |
| "toxcast-NVS_LGIC_rNNR_BungSens", | |
| "toxcast-BSK_KF3CT_SRB_down", | |
| "toxcast-NVS_GPCR_hDRD1", | |
| "toxcast-NVS_ENZ_hPTPN12", | |
| "toxcast-NVS_GPCR_hNK2", | |
| "toxcast-APR_HepG2_OxidativeStress_24h_up", | |
| "toxcast-ATG_M_32_CIS_up", | |
| "toxcast-APR_HepG2_MitoMass_24h_up", | |
| "toxcast-TOX21_p53_BLA_p1_ch2", | |
| "toxcast-BSK_CASM3C_SAA_down", | |
| "toxcast-NVS_ENZ_hAurA", | |
| "toxcast-BSK_SAg_Eselectin_down", | |
| "toxcast-BSK_CASM3C_Proliferation_down", | |
| "toxcast-NVS_ENZ_hPDE4A1", | |
| "toxcast-APR_Hepat_NuclearSize_24hr_dn", | |
| "toxcast-BSK_CASM3C_MCSF_down", | |
| "toxcast-NVS_ENZ_hVEGFR2", | |
| "toxcast-CEETOX_H295R_ANDR_dn", | |
| "toxcast-NVS_GPCR_rabPAF", | |
| "toxcast-NVS_ENZ_hPI3Ka", | |
| "toxcast-ATG_AR_TRANS_up", | |
| "toxcast-ATG_NRF2_ARE_CIS_up", | |
| "toxcast-ATG_Pax6_CIS_up", | |
| "toxcast-APR_HepG2_MitoMass_24h_dn", | |
| "toxcast-ATG_HSE_CIS_dn", | |
| "clintox", | |
| "toxcast-ATG_CAR_TRANS_up", | |
| "toxcast-NVS_ENZ_rabI2C", | |
| "toxcast-NVS_GPCR_rNK3", | |
| "toxcast-TOX21_p53_BLA_p3_ch1", | |
| "toxcast-ATG_GLI_CIS_up", | |
| "toxcast-TOX21_ESRE_BLA_ch2", | |
| "toxcast-ATG_VDR_TRANS_dn", | |
| "toxcast-ATG_RORg_TRANS_dn", | |
| "tox21-SR-p53", | |
| "toxcast-BSK_CASM3C_MCSF_up", | |
| "toxcast-NVS_ENZ_hMMP2", | |
| "toxcast-APR_Hepat_DNATexture_48hr_up", | |
| "toxcast-ATG_SREBP_CIS_dn", | |
| "toxcast-BSK_LPS_MCSF_down", | |
| "toxcast-ATG_RORb_TRANS_dn", | |
| "toxcast-ATG_LXRa_TRANS_up", | |
| "toxcast-TOX21_p53_BLA_p4_ch1", | |
| "toxcast-APR_HepG2_MitoMass_72h_dn", | |
| "toxcast-OT_ERa_EREGFP_0120", | |
| "toxcast-TOX21_p53_BLA_p4_viability", | |
| "toxcast-ATG_FoxO_CIS_dn", | |
| "toxcast-BSK_3C_TissueFactor_up", | |
| "toxcast-APR_Hepat_DNADamage_48hr_up", | |
| "toxcast-ATG_M_32_TRANS_dn", | |
| "toxcast-TOX21_PPARd_BLA_agonist_ch1", | |
| "toxcast-TOX21_p53_BLA_p1_ch1", | |
| "toxcast-NVS_GPCR_rAdra1_NonSelective", | |
| "toxcast-ATG_STAT3_CIS_dn", | |
| "tox21-SR-ARE", | |
| "toxcast-TOX21_ESRE_BLA_viability", | |
| "toxcast-BSK_CASM3C_Proliferation_up", | |
| "toxcast-ATG_IR1_CIS_up", | |
| "toxcast-NVS_GPCR_gH2", | |
| "toxcast-BSK_CASM3C_VCAM1_down", | |
| "toxcast-TOX21_AR_BLA_Antagonist_viability", | |
| "toxcast-BSK_3C_HLADR_down", | |
| "toxcast-BSK_BE3C_MMP1_down", | |
| "toxcast-BSK_LPS_Eselectin_down", | |
| "toxcast-Tanguay_ZF_120hpf_JAW_up", | |
| "toxcast-BSK_BE3C_MIG_down", | |
| "toxcast-BSK_KF3CT_TIMP2_down", | |
| "herg_central-hERG_inhib", | |
| "toxcast-ATG_Oct_MLP_CIS_dn", | |
| "toxcast-TOX21_PPARg_BLA_antagonist_ratio", | |
| "toxcast-APR_Hepat_Steatosis_48hr_up", | |
| "toxcast-NVS_ENZ_hPDE10", | |
| "herg", | |
| "toxcast-ATG_TAL_CIS_up", | |
| "toxcast-NVS_GPCR_p5HT2C", | |
| "toxcast-ATG_PPARa_TRANS_up", | |
| "toxcast-NVS_NR_hTRa_Antagonist", | |
| "toxcast-TOX21_AhR_LUC_Agonist", | |
| "toxcast-TOX21_FXR_BLA_antagonist_viability", | |
| "toxcast-BSK_3C_SRB_down", | |
| "tox21-SR-MMP", | |
| "toxcast-APR_Hepat_MitoFxnI_48hr_dn", | |
| "toxcast-NVS_NR_hFXR_Agonist", | |
| "toxcast-NVS_NR_hPPARa", | |
| "toxcast-APR_HepG2_StressKinase_24h_up", | |
| "toxcast-TOX21_ERa_BLA_Antagonist_viability", | |
| "toxcast-NVS_ADME_hCYP3A4", | |
| "toxcast-CEETOX_H295R_DOC_up", | |
| "toxcast-BSK_CASM3C_uPAR_up", | |
| "toxcast-BSK_BE3C_IP10_down", | |
| "toxcast-OT_AR_ARSRC1_0480", | |
| "toxcast-CEETOX_H295R_11DCORT_dn", | |
| "toxcast-Tanguay_ZF_120hpf_AXIS_up", | |
| "toxcast-NVS_GPCR_gLTD4", | |
| "toxcast-ATG_CRE_CIS_up", | |
| "toxcast-TOX21_p53_BLA_p5_ch1", | |
| "tox21-NR-AR", | |
| "toxcast-ATG_TAL_CIS_dn", | |
| "toxcast-TOX21_p53_BLA_p2_ch1", | |
| "toxcast-ATG_PXRE_CIS_up", | |
| "toxcast-NVS_ENZ_oCOX1", | |
| "toxcast-ATG_BRE_CIS_up", | |
| "toxcast-ATG_PPRE_CIS_up", | |
| "toxcast-NVS_GPCR_rTRH", | |
| "toxcast-ATG_C_EBP_CIS_up", | |
| "toxcast-NVS_GPCR_rV1", | |
| "toxcast-BSK_KF3CT_IP10_up", | |
| "toxcast-ATG_RORg_TRANS_up", | |
| "toxcast-NCCT_TPO_GUA_dn", | |
| "toxcast-ATG_Myb_CIS_up", | |
| "toxcast-ATG_Myc_CIS_dn", | |
| "toxcast-TOX21_PPARg_BLA_Antagonist_ch1", | |
| "toxcast-NVS_ENZ_rAChE", | |
| "tox21-SR-HSE", | |
| "toxcast-ATG_LXRb_TRANS_up", | |
| "toxcast-BSK_hDFCGF_MMP1_up", | |
| "toxcast-NVS_LGIC_rGABAR_NonSelective", | |
| "toxcast-TOX21_FXR_BLA_antagonist_ratio", | |
| "toxcast-ATG_RARa_TRANS_dn", | |
| "toxcast-BSK_SAg_IL8_down", | |
| "toxcast-NVS_ENZ_hBACE", | |
| "toxcast-CEETOX_H295R_ESTRONE_dn", | |
| "ames", | |
| "toxcast-APR_HepG2_MicrotubuleCSK_24h_up", | |
| "toxcast-ATG_FoxA2_CIS_dn", | |
| "toxcast-NVS_TR_hNET", | |
| "toxcast-ATG_AP_1_CIS_dn", | |
| "toxcast-ATG_CMV_CIS_up", | |
| "toxcast-ATG_p53_CIS_up", | |
| "toxcast-ATG_PPRE_CIS_dn", | |
| "toxcast-BSK_LPS_SRB_down", | |
| "toxcast-TOX21_p53_BLA_p4_ratio", | |
| "toxcast-BSK_3C_MCP1_down", | |
| "toxcast-Tanguay_ZF_120hpf_CIRC_up", | |
| "toxcast-BSK_3C_Thrombomodulin_up", | |
| "toxcast-BSK_CASM3C_LDLR_up", | |
| "toxcast-NVS_IC_rCaDHPRCh_L", | |
| "toxcast-TOX21_p53_BLA_p2_viability", | |
| "toxcast-Tanguay_ZF_120hpf_OTIC_up", | |
| "toxcast-TOX21_GR_BLA_Agonist_ch1", | |
| "toxcast-CEETOX_H295R_TESTO_dn", | |
| "toxcast-NVS_ENZ_hMMP7", | |
| "toxcast-BSK_KF3CT_MMP9_down", | |
| "toxcast-TOX21_HSE_BLA_agonist_ratio", | |
| "toxcast-BSK_LPS_MCP1_down", | |
| "toxcast-BSK_LPS_VCAM1_down", | |
| "toxcast-TOX21_TR_LUC_GH3_Agonist", | |
| "toxcast-NVS_GPCR_hAdra2C", | |
| "toxcast-NVS_GPCR_hAdra2A", | |
| "toxcast-NVS_ENZ_hMMP9", | |
| "toxcast-TOX21_ERa_BLA_Antagonist_ch1", | |
| "toxcast-ATG_AR_TRANS_dn", | |
| "toxcast-BSK_4H_Pselectin_down", | |
| "toxcast-BSK_hDFCGF_CollagenIII_down", | |
| "toxcast-BSK_hDFCGF_TIMP1_down", | |
| "toxcast-ATG_RXRb_TRANS_up", | |
| "toxcast-TOX21_GR_BLA_Antagonist_ch2", | |
| "toxcast-BSK_LPS_PGE2_down", | |
| "toxcast-ATG_p53_CIS_dn", | |
| "toxcast-BSK_CASM3C_uPAR_down", | |
| "toxcast-NVS_IC_rCaBTZCHL", | |
| "toxcast-TOX21_AutoFluor_HEK293_Cell_blue", | |
| "toxcast-BSK_BE3C_MMP1_up", | |
| "toxcast-TOX21_ARE_BLA_agonist_viability", | |
| "toxcast-ATG_RARb_TRANS_up", | |
| "toxcast-TOX21_ESRE_BLA_ratio", | |
| "toxcast-ATG_E_Box_CIS_up", | |
| "toxcast-TOX21_AR_LUC_MDAKB2_Antagonist2", | |
| "toxcast-NVS_ENZ_rMAOBP", | |
| "toxcast-NCCT_TPO_AUR_dn", | |
| "toxcast-APR_HepG2_StressKinase_72h_up", | |
| "toxcast-TOX21_p53_BLA_p2_ch2", | |
| "toxcast-ATG_TGFb_CIS_dn", | |
| "toxcast-TOX21_PPARd_BLA_Antagonist_ch1", | |
| "toxcast-TOX21_ERa_BLA_Agonist_ch1", | |
| "toxcast-ATG_PPARa_TRANS_dn", | |
| "toxcast-ATG_M_19_CIS_dn", | |
| "toxcast-Tanguay_ZF_120hpf_ActivityScore", | |
| "toxcast-BSK_LPS_TNFa_down", | |
| "toxcast-ATG_M_32_TRANS_up", | |
| "toxcast-BSK_BE3C_TGFb1_down", | |
| "toxcast-NVS_ENZ_hAChE", | |
| "toxcast-ATG_Ets_CIS_dn", | |
| "toxcast-TOX21_ELG1_LUC_Agonist", | |
| "toxcast-ATG_Ets_CIS_up", | |
| "toxcast-BSK_LPS_PGE2_up", | |
| "toxcast-TOX21_p53_BLA_p1_viability", | |
| "toxcast-APR_HepG2_CellLoss_24h_dn", | |
| "toxcast-CLD_CYP1A1_24hr", | |
| "toxcast-ATG_NFI_CIS_up", | |
| "toxcast-CLD_CYP3A4_6hr", | |
| "toxcast-ATG_NF_kB_CIS_dn", | |
| "toxcast-BSK_hDFCGF_EGFR_up", | |
| "toxcast-APR_Hepat_Apoptosis_24hr_up", | |
| "toxcast-ATG_ERE_CIS_dn", | |
| "toxcast-ATG_ISRE_CIS_up", | |
| "toxcast-NVS_GPCR_bAdoR_NonSelective", | |
| "toxcast-NVS_NR_cAR", | |
| "toxcast-APR_Hepat_CellLoss_24hr_dn", | |
| "toxcast-TOX21_PPARd_BLA_agonist_ch2", | |
| "toxcast-ATG_E2F_CIS_up", | |
| "toxcast-Tanguay_ZF_120hpf_SNOU_up", | |
| "toxcast-CLD_CYP3A4_24hr", | |
| "toxcast-NVS_GPCR_h5HT6", | |
| "toxcast-ATG_GATA_CIS_up", | |
| "toxcast-ATG_TCF_b_cat_CIS_dn", | |
| "toxcast-TOX21_GR_BLA_Agonist_ratio", | |
| "toxcast-BSK_SAg_SRB_down", | |
| "toxcast-ACEA_T47D_80hr_Positive", | |
| "toxcast-NVS_ENZ_hCASP5", | |
| "toxcast-Tanguay_ZF_120hpf_SWIM_up", | |
| "toxcast-ATG_PXR_TRANS_dn", | |
| "toxcast-NVS_GPCR_rOpiate_NonSelective", | |
| "toxcast-NVS_ADME_hCYP4F12", | |
| "toxcast-ATG_ERa_TRANS_up", | |
| "toxcast-ATG_FoxA2_CIS_up", | |
| "toxcast-BSK_3C_uPAR_down", | |
| "tox21-NR-PPAR-gamma", | |
| "toxcast-NVS_ENZ_rMAOBC", | |
| "toxcast-ATG_AP_2_CIS_dn", | |
| "toxcast-ATG_TA_CIS_dn", | |
| "toxcast-BSK_BE3C_tPA_down", | |
| "toxcast-NVS_NR_hPXR", | |
| "toxcast-NVS_TR_hSERT", | |
| "toxcast-TOX21_HSE_BLA_agonist_ch1", | |
| "toxcast-OT_ER_ERaERa_0480", | |
| "toxcast-ATG_CMV_CIS_dn", | |
| "toxcast-ATG_ERRg_TRANS_dn", | |
| "toxcast-NVS_GPCR_hAdrb1", | |
| "toxcast-BSK_hDFCGF_SRB_down", | |
| "toxcast-Tanguay_ZF_120hpf_BRAI_up", | |
| "toxcast-TOX21_p53_BLA_p3_ratio", | |
| "toxcast-ATG_NFI_CIS_dn", | |
| "toxcast-BSK_SAg_MCP1_down", | |
| "toxcast-BSK_SAg_CD38_down", | |
| "toxcast-NVS_ENZ_rMAOAP", | |
| "toxcast-TOX21_ESRE_BLA_ch1", | |
| "toxcast-NVS_ENZ_rMAOAC", | |
| "toxcast-ATG_Ahr_CIS_up", | |
| "toxcast-ATG_LXRa_TRANS_dn", | |
| "toxcast-ATG_GR_TRANS_dn", | |
| "toxcast-NVS_GPCR_h5HT5A", | |
| "toxcast-NVS_ADME_hCYP2D6", | |
| "toxcast-TOX21_AutoFluor_HEK293_Media_blue", | |
| "toxcast-BSK_BE3C_SRB_down", | |
| "toxcast-CLD_CYP2B6_48hr", | |
| "toxcast-NVS_TR_hDAT", | |
| "toxcast-BSK_BE3C_IL1a_down", | |
| "tox21-SR-ATAD5", | |
| "toxcast-NVS_ENZ_hMMP3", | |
| "toxcast-NVS_TR_hAdoT", | |
| "toxcast-BSK_CASM3C_TissueFactor_down", | |
| "toxcast-APR_HepG2_NuclearSize_24h_dn", | |
| "toxcast-TOX21_VDR_BLA_Agonist_viability", | |
| "toxcast-APR_HepG2_MitoMembPot_24h_dn", | |
| "toxcast-BSK_4H_Pselectin_up", | |
| "toxcast-ATG_NF_kB_CIS_up", | |
| "toxcast-CEETOX_H295R_ESTRADIOL_dn", | |
| "toxcast-NVS_NR_hCAR_Antagonist", | |
| "toxcast-BSK_LPS_CD40_down", | |
| "toxcast-NHEERL_ZF_144hpf_TERATOSCORE_up", | |
| "toxcast-NVS_ENZ_hMMP1", | |
| "toxcast-NVS_TR_rNET", | |
| "toxcast-NVS_IC_rNaCh_site2", | |
| "toxcast-ATG_NURR1_TRANS_up", | |
| "toxcast-APR_Hepat_Apoptosis_48hr_up", | |
| "toxcast-TOX21_ARE_BLA_Agonist_ch2", | |
| "toxcast-OT_ER_ERbERb_1440", | |
| "toxcast-ATG_Ahr_CIS_dn", | |
| "toxcast-ATG_TCF_b_cat_CIS_up", | |
| "toxcast-ATG_DR4_LXR_CIS_dn", | |
| "toxcast-BSK_SAg_PBMCCytotoxicity_up", | |
| "toxcast-NVS_TR_rSERT", | |
| "toxcast-TOX21_MMP_ratio_down", | |
| "toxcast-ATG_Sox_CIS_dn", | |
| "toxcast-TOX21_NFkB_BLA_agonist_ch1", | |
| "toxcast-NVS_NR_hGR", | |
| "toxcast-NVS_GPCR_hLTB4_BLT1", | |
| "toxcast-BSK_4H_uPAR_down", | |
| "toxcast-ATG_IR1_CIS_dn", | |
| "toxcast-OT_NURR1_NURR1RXRa_1440", | |
| "toxcast-BSK_3C_Proliferation_down", | |
| "toxcast-NVS_ENZ_hAMPKa1", | |
| "toxcast-ATG_GRE_CIS_dn", | |
| "toxcast-BSK_hDFCGF_VCAM1_down", | |
| "toxcast-BSK_SAg_IL8_up", | |
| "toxcast-ATG_XTT_Cytotoxicity_up", | |
| "toxcast-CEETOX_H295R_ESTRONE_up", | |
| "toxcast-ATG_DR5_CIS_dn", | |
| "toxcast-BSK_hDFCGF_Proliferation_down", | |
| "toxcast-TOX21_p53_BLA_p3_viability", | |
| "toxcast-BSK_3C_IL8_down", | |
| "toxcast-BSK_LPS_IL8_down", | |
| "toxcast-NVS_ENZ_hSIRT2", | |
| "toxcast-TOX21_ERa_LUC_BG1_Agonist", | |
| "toxcast-BSK_BE3C_HLADR_down", | |
| "toxcast-NVS_GPCR_hH1", | |
| "toxcast-ATG_RARg_TRANS_up", | |
| "toxcast-Tanguay_ZF_120hpf_PE_up", | |
| "toxcast-NVS_ENZ_hPTPRC", | |
| "toxcast-NVS_GPCR_hM1", | |
| "toxcast-ATG_VDRE_CIS_dn", | |
| "toxcast-NVS_NR_hPR", | |
| "toxcast-BSK_4H_VCAM1_down", | |
| "toxcast-CLD_CYP2B6_6hr", | |
| "toxcast-Tanguay_ZF_120hpf_YSE_up", | |
| "toxcast-CEETOX_H295R_ESTRADIOL_up", | |
| "toxcast-ATG_M_32_CIS_dn", | |
| "toxcast-BSK_BE3C_uPAR_down", | |
| "toxcast-TOX21_AR_BLA_Agonist_ratio", | |
| "carcinogens_lagunin", | |
| "toxcast-ATG_NRF1_CIS_dn", | |
| "toxcast-ATG_HSE_CIS_up", | |
| "toxcast-BSK_KF3CT_ICAM1_down", | |
| "toxcast-BSK_LPS_Eselectin_up", | |
| "toxcast-ATG_Oct_MLP_CIS_up", | |
| "toxcast-ATG_GATA_CIS_dn", | |
| "toxcast-APR_HepG2_MitoMembPot_72h_dn", | |
| "tox21-NR-Aromatase", | |
| "toxcast-NVS_TR_gDAT", | |
| "toxcast-BSK_CASM3C_MCP1_down", | |
| "toxcast-BSK_SAg_PBMCCytotoxicity_down", | |
| "toxcast-NVS_GPCR_hTXA2", | |
| "toxcast-ATG_PBREM_CIS_up", | |
| "toxcast-Tanguay_ZF_120hpf_TR_up", | |
| "toxcast-ACEA_T47D_80hr_Negative", | |
| "toxcast-NVS_GPCR_hM4", | |
| "toxcast-ATG_GLI_CIS_dn", | |
| "toxcast-NVS_ENZ_hDUSP3", | |
| "toxcast-TOX21_AR_BLA_Antagonist_ch2", | |
| "toxcast-BSK_CASM3C_MCP1_up", | |
| "toxcast-ATG_NRF1_CIS_up", | |
| "toxcast-NVS_GPCR_rAdra1B", | |
| "toxcast-TOX21_VDR_BLA_antagonist_ratio", | |
| "toxcast-BSK_BE3C_PAI1_down", | |
| "toxcast-BSK_LPS_TissueFactor_down", | |
| "toxcast-NVS_ENZ_hTrkA", | |
| "herg_central-hERG_at_10uM", | |
| "toxcast-BSK_LPS_TissueFactor_up", | |
| "toxcast-Tanguay_ZF_120hpf_SOMI_up", | |
| "toxcast-NVS_GPCR_hAdrb2", | |
| "toxcast-BSK_hDFCGF_MCSF_down", | |
| "toxcast-NVS_ADME_hCYP2C19", | |
| "toxcast-OT_ER_ERaERb_1440", | |
| "toxcast-CLD_SULT2A_48hr", | |
| "toxcast-ATG_Xbp1_CIS_up", | |
| "toxcast-OT_ER_ERaERb_0480", | |
| "toxcast-CLD_UGT1A1_24hr", | |
| "toxcast-NVS_ENZ_hPTPN13", | |
| "tox21-NR-ER", | |
| "toxcast-TOX21_PPARd_BLA_Agonist_viability", | |
| "toxcast-ATG_PPARd_TRANS_up", | |
| "toxcast-CLD_ABCB1_48hr", | |
| "toxcast-ATG_PBREM_CIS_dn", | |
| "toxcast-BSK_CASM3C_IL6_up", | |
| "toxcast-ATG_GR_TRANS_up", | |
| "toxcast-NVS_GPCR_gMPeripheral_NonSelective", | |
| "toxcast-NVS_GPCR_hM2", | |
| "toxcast-ATG_DR4_LXR_CIS_up", | |
| "toxcast-APR_HepG2_MitoMembPot_1h_dn", | |
| "toxcast-NVS_ENZ_hSIRT1", | |
| "toxcast-ATG_FoxO_CIS_up", | |
| "toxcast-NVS_LGIC_hNNR_NBungSens", | |
| "toxcast-BSK_4H_Eotaxin3_down", | |
| "toxcast-ATG_CRE_CIS_dn", | |
| "toxcast-CLD_CYP1A2_48hr", | |
| "toxcast-ATG_Myc_CIS_up", | |
| "toxcast-ATG_TGFb_CIS_up", | |
| "toxcast-NVS_GPCR_hAT1", | |
| "toxcast-NVS_ENZ_hCK1D", | |
| "toxcast-TOX21_FXR_BLA_agonist_ratio", | |
| "toxcast-BSK_BE3C_uPA_down", | |
| "toxcast-APR_Hepat_Steatosis_24hr_up", | |
| "toxcast-ATG_PXR_TRANS_up", | |
| "toxcast-APR_HepG2_MitoMass_72h_up", | |
| "toxcast-NVS_ENZ_hFGFR1", | |
| "toxcast-ATG_M_19_TRANS_up", | |
| "toxcast-TOX21_FXR_BLA_agonist_ch2", | |
| "toxcast-ATG_Sp1_CIS_dn", | |
| "toxcast-BSK_KF3CT_IL1a_down", | |
| "toxcast-BSK_hDFCGF_MMP1_down", | |
| "toxcast-TOX21_PPARg_BLA_Agonist_ratio", | |
| "toxcast-NVS_GPCR_gLTB4", | |
| "toxcast-TOX21_TR_LUC_GH3_Antagonist", | |
| "dili", | |
| "toxcast-TOX21_PPARd_BLA_antagonist_ratio", | |
| "toxcast-NVS_GPCR_hOpiate_mu", | |
| "toxcast-BSK_CASM3C_Thrombomodulin_down", | |
| "toxcast-ATG_LXRb_TRANS_dn", | |
| "toxcast-APR_Hepat_NuclearSize_48hr_dn", | |
| "toxcast-TOX21_ERa_LUC_BG1_Antagonist", | |
| "toxcast-ATG_M_61_TRANS_up", | |
| "toxcast-TOX21_AutoFluor_HEPG2_Media_green", | |
| "toxcast-APR_HepG2_CellCycleArrest_72h_dn", | |
| "toxcast-BSK_3C_Eselectin_down", | |
| "toxcast-BSK_SAg_Eselectin_up", | |
| "toxcast-OT_AR_ARSRC1_0960", | |
| "toxcast-BSK_CASM3C_IL6_down", | |
| "toxcast-TOX21_AutoFluor_HEPG2_Cell_blue", | |
| "toxcast-TOX21_p53_BLA_p5_ratio", | |
| "toxcast-TOX21_AR_BLA_Agonist_ch1", | |
| "toxcast-BSK_BE3C_uPAR_up", | |
| "toxcast-NVS_ADME_hCYP1A2", | |
| "toxcast-NVS_ADME_rCYP2C12", | |
| "toxcast-APR_HepG2_CellCycleArrest_24h_up", | |
| "toxcast-ATG_C_EBP_CIS_dn", | |
| "toxcast-NVS_GPCR_rNK1", | |
| "toxcast-NVS_NR_bER", | |
| "toxcast-NVS_NR_hRAR_Antagonist", | |
| "toxcast-ATG_HNF4a_TRANS_dn", | |
| "toxcast-CEETOX_H295R_OHPREG_up", | |
| "toxcast-BSK_hDFCGF_IP10_down", | |
| "toxcast-ATG_Sp1_CIS_up", | |
| "toxcast-NVS_NR_bPR", | |
| "toxcast-CEETOX_H295R_DOC_dn", | |
| "toxcast-NVS_ENZ_hES", | |
| "toxcast-BSK_CASM3C_VCAM1_up", | |
| "toxcast-ATG_ERE_CIS_up", | |
| "toxcast-CLD_SULT2A_24hr", | |
| "toxcast-BSK_4H_uPAR_up", | |
| "tox21-NR-AhR", | |
| "toxcast-BSK_4H_MCP1_down", | |
| "toxcast-TOX21_ERa_BLA_Antagonist_ratio", | |
| "toxcast-TOX21_AutoFluor_HEPG2_Cell_green", | |
| "toxcast-NVS_GPCR_r5HT_NonSelective", | |
| "toxcast-NVS_NR_hFXR_Antagonist", | |
| "toxcast-ATG_RXRb_TRANS_dn", | |
| "toxcast-NVS_LGIC_bGABARa1", | |
| "toxcast-TOX21_p53_BLA_p4_ch2", | |
| "toxcast-BSK_hDFCGF_IL8_down", | |
| "toxcast-ATG_ISRE_CIS_dn", | |
| "toxcast-CLD_CYP3A4_48hr", | |
| "toxcast-BSK_4H_VEGFRII_down", | |
| "toxcast-ATG_AP_1_CIS_up", | |
| "toxcast-NVS_NR_rAR", | |
| "toxcast-BSK_3C_MIG_down", | |
| "toxcast-TOX21_FXR_BLA_Antagonist_ch2", | |
| "toxcast-APR_Hepat_DNATexture_24hr_up", | |
| "toxcast-BSK_SAg_Proliferation_down", | |
| "toxcast-ATG_CAR_TRANS_dn", | |
| "toxcast-CEETOX_H295R_OHPROG_up", | |
| "toxcast-APR_HepG2_MicrotubuleCSK_24h_dn", | |
| "toxcast-CLD_CYP2B6_24hr", | |
| "toxcast-BSK_CASM3C_IL8_down", | |
| "toxcast-TOX21_MMP_ratio_up", | |
| "toxcast-NVS_GPCR_h5HT2A", | |
| "toxcast-NVS_GPCR_bDR_NonSelective", | |
| "toxcast-NVS_ENZ_hMMP13", | |
| "toxcast-TOX21_AR_LUC_MDAKB2_Antagonist", | |
| "toxcast-TOX21_GR_BLA_Agonist_ch2", | |
| "toxcast-ATG_M_19_TRANS_dn", | |
| "toxcast-CEETOX_H295R_CORTISOL_dn", | |
| "toxcast-OT_AR_ARELUC_AG_1440", | |
| "toxcast-TOX21_VDR_BLA_Antagonist_ch1", | |
| "toxcast-ATG_Myb_CIS_dn", | |
| "toxcast-ATG_BRE_CIS_dn", | |
| "ld50_zhu", | |
| "toxcast-NVS_NR_hAR", | |
| "toxcast-ATG_ERRg_TRANS_up", | |
| "toxcast-NCCT_QuantiLum_inhib_dn", | |
| "toxcast-ATG_STAT3_CIS_up", | |
| "toxcast-TOX21_ARE_BLA_Agonist_ch1", | |
| "toxcast-CLD_CYP1A2_6hr", | |
| "toxcast-BSK_KF3CT_MCP1_up", | |
| "toxcast-NVS_GPCR_hM3", | |
| "toxcast-NVS_OR_gSIGMA_NonSelective", | |
| "toxcast-ATG_DR5_CIS_up", | |
| "toxcast-NVS_ADME_hCYP1A1", | |
| "toxcast-BSK_SAg_CD69_down", | |
| "toxcast-APR_HepG2_NuclearSize_72h_up", | |
| "toxcast-CLD_ABCG2_48hr", | |
| "toxcast-NVS_GPCR_gOpiateK", | |
| "toxcast-ATG_AP_2_CIS_up", | |
| "toxcast-NVS_ENZ_hPTPN9", | |
| "toxcast-APR_Hepat_CellLoss_48hr_dn", | |
| "toxcast-OT_ERa_EREGFP_0480", | |
| "toxcast-NVS_NR_hRARa_Agonist", | |
| "toxcast-BSK_CASM3C_Thrombomodulin_up", | |
| "toxcast-NVS_ENZ_hPTEN", | |
| "toxcast-NVS_ADME_hCYP2B6", | |
| "toxcast-TOX21_VDR_BLA_agonist_ratio", | |
| "toxcast-NVS_ENZ_hPDE5", | |
| "toxcast-NVS_NR_hPPARg", | |
| "toxcast-NVS_ENZ_rCNOS", | |
| "toxcast-BSK_LPS_IL1a_down", | |
| "toxcast-BSK_CASM3C_LDLR_down", | |
| "toxcast-ATG_HNF6_CIS_up", | |
| "toxcast-TOX21_AutoFluor_HEPG2_Media_blue", | |
| "toxcast-BSK_hDFCGF_EGFR_down", | |
| "toxcast-TOX21_AR_BLA_Agonist_ch2", | |
| "toxcast-TOX21_FXR_BLA_Antagonist_ch1", | |
| "toxcast-ATG_PXRE_CIS_dn", | |
| "toxcast-BSK_SAg_CD40_down" | |
| ], | |
| "metabolism": [ | |
| "cyp3a4_substrate_carbonmangels", | |
| "cyp3a4_veith", | |
| "cyp2c19_veith", | |
| "cyp2c9_substrate_carbonmangels", | |
| "cyp2d6_substrate_carbonmangels", | |
| "cyp1a2_veith", | |
| "cyp2c9_veith", | |
| "cyp2d6_veith" | |
| ], | |
| "absorption": [ | |
| "lipophilicity_astrazeneca", | |
| "pgp_broccatelli", | |
| "bioavailability_ma", | |
| "hia_hou", | |
| "pampa_ncats", | |
| "caco2_wang", | |
| "hydrationfreeenergy_freesolv", | |
| "solubility_aqsoldb" | |
| ], | |
| "excretion": [ | |
| "half_life_obach", | |
| "clearance_microsome_az", | |
| "clearance_hepatocyte_az" | |
| ], | |
| "distribution": [ | |
| "bbb_martins", | |
| "ppbr_az", | |
| "vdss_lombardo" | |
| ] | |
| } |