chembl_id
stringlengths
7
13
canonical_smiles
stringlengths
1
2.03k
CHEMBL613
O=C(O)c1cnccn1
CHEMBL19797
c1ccc(CCCCCCCNCCc2ccccc2)cc1
CHEMBL19539
Oc1ccc2[nH]c3c(c2c1)CCCCCC3
CHEMBL19540
Cc1ccc(S(=O)(=O)N[C@H]2CC[C@H](O)[C@@H]2C/C=C\CCCC(=O)O)cc1
CHEMBL19541
CC(Cc1ccc2ccccc2c1)NCCCc1ccccc1
CHEMBL19542
C=C(C)[C@@H]1CC[C@]2(C(=O)N[C@@H](CCSC)C(=O)O)CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC[C@H](O)C(C)(C)[C@@H]5CC[C@]43C)[C@@H]12
CHEMBL19543
Clc1nc(-c2cccs2)c2ncn(Cc3ccccc3)c2n1
CHEMBL19628
c1ccc(CCCCNCc2ccccc2)cc1
CHEMBL19459
CCOC(=O)Cc1nc(-c2ccc(OC)cc2)oc1-c1ccco1
CHEMBL19561
C[C@H]1COc2c(N3CC(C)(N)C3)c(F)cc3c(=O)c(C(=O)O)cn1c23
CHEMBL19562
NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(CCC(=O)O)NC(=O)C(Cc1ccc(OP(=O)(O)O)cc1)c1cccc2ccccc12
CHEMBL3310707
CC[C@H](C)[C@H](NC(=O)[C@H](CCCCNC(=O)OCc1ccccc1)NC(C)=O)C(=O)N[C@H](C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(O)C(F)(F)C(=O)NCC(=O)OCc1ccccc1)[C@@H](C)OCc1ccccc1
CHEMBL19482
BrCCN(CCBr)c1ccccc1
CHEMBL19484
COc1cccc(N(C)C(=O)c2cc3cc(OC)ccc3n2C)c1
CHEMBL19485
N=C(Nc1ccc2ccc3cccnc3c2n1)c1ccccc1
CHEMBL19586
CC(C)c1ccc(C(c2ccc([N+](C)(C)C)cc2)c2ccc(C(C)C)cc(=O)c2O)c(O)c(=O)c1.[I-]
CHEMBL19888
CCOC(=O)/C=C/[C@H](CCC(N)=O)NC(=O)[C@@H](CC(=O)[C@@H](NC(=O)SC1CCCC1)C(C)C)Cc1ccc(C)cc1
CHEMBL19889
CSc1ccc(C(=O)c2c(SC)cc3n2CCC3C(=O)O)cc1
CHEMBL4434868
Cc1ccc(Sc2cc(Cl)cn3c([N+](=O)[O-])c(CS(=O)(=O)c4ccccc4)nc23)cc1
CHEMBL4434869
COc1cc(/C=N/OC/C=C/C=C(\C)CCC(O)c2cccs2)cc(OC)c1OC
CHEMBL4434870
CCCc1ccc(-c2ccc(N(C[C@@H](N)[C@@H](C)CC)C(=O)[C@@H]3C[C@H]3c3ccccn3)cc2)cc1.Cl
CHEMBL4434871
C=CC(=O)Nc1ccc(C(=O)Nc2cccc(Nc3n[nH]c4c3CN(C(=O)N[C@H](CN(C)C)c3ccccc3)C4(C)C)c2)cc1
CHEMBL4434872
O=C1CC2CCC(C1)N2CCc1ccc([N+](=O)[O-])cc1
CHEMBL4434873
CC/C=C\C(=O)Nc1cc(Nc2nc3c(c(-c4cn(C)c5ccc(F)cc45)n2)CS(=O)(=O)CC3)c(OC)cc1N(C)CCN(C)C
CHEMBL4434874
FC(F)(F)c1cc(Nc2ccccc2C(F)(F)F)c2cccc(C(F)(F)F)c2n1
CHEMBL4434875
COc1ccc([C@@H](O)[C@@H](C)Oc2ccc([C@@H]3CCN(c4ccc(OC)c(OC)c4)C3)cc2OC)cc1OC
CHEMBL4434876
Fc1ccc(C2CCN(CCCc3c[nH]c4ccc(F)cc34)CC2)c(-c2ccccc2)c1
CHEMBL4434877
CCOC(=O)c1ccccc1OS(=O)(=O)[N-]C(=O)Nc1nc(Br)cc(OC)n1.[Na+]
CHEMBL4434878
CN1CCN(C(=O)c2cccc(Nc3nnc(-c4cc(C#N)cs4)o3)c2)CC1
CHEMBL4434879
C=CC(=O)Nc1cccc(Nc2nc(Nc3ccc(OCCSC(=S)NCc4ccc(OC)cc4)cc3)ncc2F)c1
CHEMBL4434880
Cc1ccccc1NCc1ccc(CNc2ccccc2C)nc1
CHEMBL4434881
Cc1c(NC(=O)c2cccn(-c3ccc(F)cc3)c2=O)ccc(Oc2ccncc2)c1C
CHEMBL4434882
Oc1c(C(NCc2ccccc2)c2ccncc2)ccc2cccnc12
CHEMBL4434883
C/C(=C\CO)CC/C=C(\C)C(=O)O[C@@H]1O[C@H](CO)[C@@H](O)[C@H](O)[C@H]1O
CHEMBL4434884
Cl.NCc1cc(=O)c2ccc(N3CCN(C(=O)c4ccccc4)CC3)cc2o1
CHEMBL4434885
CCc1ccc2nc(N3CCC(NCC4(C)COC4)CC3)c(-c3nc(C)no3)cc2c1
CHEMBL19890
Nc1nc(O)c2ncn(CCSCP(=O)(O)O)c2n1
CHEMBL19891
COC(=O)[C@H](c1ccc(O)cc1)[C@H]1CCCCN1C
CHEMBL19630
C=C(OCC)c1nc(Cl)nc2c1ncn2Cc1ccccc1
CHEMBL19631
Cc1c2ccnc(NCCCN)c2cc2c1[nH]c1ccc(OCc3ccccc3)cc12
CHEMBL19632
COP(=O)(CC1OC(C)(C)C(C)(C)O1)OC
CHEMBL19633
COc1ccc(Cc2cnc(N)nc2N)cc1OC
CHEMBL19563
CC(=O)[C@H](O)[C@H](CC1CCCCC1)NC(=O)[C@H](CC(C)C)NC(=O)CCC(C)C
CHEMBL19564
CC(=O)Nc1ccc(-c2cn3nc(S(N)(=O)=O)sc3n2)cc1
CHEMBL19651
CN(C)c1ccc(C(=O)Nc2ccccc2)cc1
CHEMBL19653
COc1ccc2c(c1)[C@H](N1CCN(C(=O)C3CC3)CC1)CC2
CHEMBL19654
CC(C)COc1cccc(N2CCN(C)CC2)n1
CHEMBL19587
COc1ccc2[nH]c(C(=O)N(C)c3ccccc3)cc2c1
CHEMBL19588
N[C@@H](CO)Cc1c[nH]cn1
CHEMBL19589
O=C(c1ccccc1)C1CCN(CCc2ccccc2)CC1
CHEMBL19291
CCOC(=O)[C@H](O)[C@H](CC1CCCCC1)NC(=O)[C@H](NC(=O)Cc1ccccc1)C(C)C
CHEMBL19292
CC(C)(CCCOc1ccc(Cc2ccccc2)cc1)C(=O)O
CHEMBL19293
Nc1ncc(Cc2ccc(Br)cc2)c(N)n1
CHEMBL20047
COc1ccc(NS(=O)(=O)c2ccc(N)cc2)c2[nH]cc(Cl)c12
CHEMBL20048
O=C(NC1c2ccccc2Oc2ccccc21)OCc1ccccc1
CHEMBL19341
COc1ccc2c(Cc3ccc(CN4CCCC4)c(OC)c3)c(-c3ccc(OCCN4CCCC4)cc3)sc2c1
CHEMBL19342
Oc1nc2ccc(C#CCN3CCC(O)(Cc4ccc(F)cc4)CC3)cc2s1
CHEMBL19343
CN(C(=O)c1cc2cc(O)ccc2n1C)c1cccc(C(F)(F)F)c1
CHEMBL19344
Oc1ccc(CC2NCCc3cc(O)c(O)cc32)cc1
CHEMBL19655
CCC(=O)c1c(O)cc(O)c(C(=O)CC)c1O
CHEMBL19657
Cn1c2c(c3cc(O)ccc31)CCCCC2
CHEMBL19363
NC[C@H](O)c1ccccc1
CHEMBL19364
CNC(C)(C)C(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N[C@H](Cc1c[nH]c2ccccc12)NC(=O)C1CCCCN1
CHEMBL19365
CC(=N)N1CC[C@H](Oc2ccc([C@@H](Cc3ccc4ccc(C(=N)N)cc4c3)C(=O)O)cc2)C1
CHEMBL19294
O=C(O)C[C@@H]1CN[C@H](C(=O)O)C1
CHEMBL19296
CC(C)N(C)C(=O)N1C[C@H](N)[C@H](C(=O)O)C1
CHEMBL19297
CCOC(=O)COc1ccc(C(c2ccc(C(C)C)cc(=O)c2O)c2ccc(C(C)C)cc(=O)c2O)cc1
CHEMBL19387
c1ccc(CCCCn2nnc(-c3ccc(OCCCCc4nnn[nH]4)cc3)n2)cc1
CHEMBL19388
O=C(O)CC[n+]1ccc(/C=C/c2cccc3ccccc23)cc1.[Br-]
CHEMBL19704
O=C1c2cc(Cl)c(Cl)cc2C(=O)N1CCCCCn1c(C2CCNCC2)nc2cc(Cl)c(Cl)cc21
CHEMBL19706
CC(NC(=O)c1ccc(CN(C)C)cc1)c1ccccc1
CHEMBL19707
C=Cc1nc(Cl)c2ncn(Cc3ccccc3)c2n1
CHEMBL19708
O=C(O)CCC/C=C\C[C@@H]1[C@H](O)CC[C@H]1NS(=O)(=O)c1ccc(F)cc1
CHEMBL19709
NC(=O)NC(=O)CBr
CHEMBL19438
Cc1cnc(NCCc2ccccc2)c(=O)n1CC(=O)NCc1cnc(N)nc1
CHEMBL19439
N=C(N)SCCc1c[nH]cn1
CHEMBL19440
C=C(C)[C@@H]1CC[C@]2(C(=O)N[C@H](C(=O)O)C(C)C)CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC[C@H](O)C(C)(C)[C@@H]5CC[C@]43C)[C@@H]12
CHEMBL19441
CC(C)C(=O)NC[C@@H]1C[C@H]1c1cccc2c1OC(C(C)C)N2
CHEMBL19442
COc1ccc2cccc(N3CCN(C(=O)C4CC4)CC3)c2c1
CHEMBL19366
CCn1cc(C(=O)O)c(=O)c2c(N)c(F)c(N3C[C@H](N)[C@H]3C)c(F)c21
CHEMBL19461
CC(=O)N1CCN(C(=O)/C=C/c2ccc(Sc3ccc4c(c3)OCO4)c(Cl)c2)CC1
CHEMBL19462
Cc1cccc(N(CCCl)CCCl)c1
CHEMBL19463
CCOC(=O)/C=C/[C@H](CCC(N)=O)NC(=O)[C@@H](CC(=O)[C@H](Cc1ccccc1)NC(=O)SC1CCCC1)Cc1ccc(F)cc1
CHEMBL19464
O=C(O)C(=O)CC(=O)c1cccc(Cc2ccccc2)c1
CHEMBL19391
C(#Cc1ncc2ncn(Cc3ccccc3)c2n1)c1ccccc1
CHEMBL19392
O=C1NC(=O)C(c2cc(Cl)ccc2S(=O)(=O)NCCCCc2ccccc2)N1
CHEMBL19393
C[C@@H](N)Cc1ccccc1
CHEMBL19486
OCC[n+]1ccc(/C=C/c2cccc3ccccc23)cc1.[Br-]
CHEMBL19488
NC[C@H](O)C1CCCCCCC1
CHEMBL19489
O=C(O)[C@@H]1CN[C@H](C(=O)O)C1
CHEMBL19490
Cc1cc(CC(=O)O)n(C)c1C(=O)c1ccc(Cl)cc1
CHEMBL19710
CCNC(=O)N1CCN([C@H]2CCc3ccc(OC)cc32)CC1
CHEMBL19798
COc1cccc(S(=O)(=O)Nc2cccn(CC(=O)NCc3nc(C(=N)N)cs3)c2=O)c1
CHEMBL19799
CCC(C)(C)/N=c1\c(O)c(O)\c1=N/Cc1c(C)cc(C)cc1Cl
CHEMBL19800
CCCC(=O)[C@H](O)[C@H](CC1CCCCC1)NC(=O)[C@H](CC(C)C)NC(=O)CCC(C)C
CHEMBL19544
CN(CCCCCc1ccccc1)CCc1ccccc1
CHEMBL19545
CC(C)[C@H](NC(=O)OCc1ccccc1)C(=O)NC(Cc1ccc(OCc2ccccc2)cc1)C(=O)C(F)(F)C(=O)N[C@@H](C(=O)OC(C)(C)C)C(C)C
CHEMBL19546
CN1CCCC1CNC[C@H](O[C@@H]1O[C@H](CN)[C@@H](O)[C@H]1O)[C@@H]1C[C@@H](O)[C@H](n2ccc(=O)[nH]c2=O)O1.O=C(O)C(F)(F)F
CHEMBL19547
Clc1nc2c(-c3ccccc3)ncnc2n1Cc1ccccc1
CHEMBL19548
Cc1cnc(NCCc2ccccc2)c(=O)n1CC(=O)NC[C@@H]1CNC(N)=N[C@@H]1C