chembl_id
stringlengths
7
13
canonical_smiles
stringlengths
1
2.03k
CHEMBL20061
O=S(=O)(NCCCCCn1c(C2CCNCC2)nc2cc(Cl)c(Cl)cc21)c1ccccc1
CHEMBL20062
CCC(C)(C)/N=c1\c(O)c(O)\c1=N/Cc1c(C)cccc1Cl
CHEMBL21449
CCCn1c(=O)[nH]c(=O)c2[nH]c(C3CCCCC3)nc21
CHEMBL20147
COc1ccc(CCC(=O)OCCCc2c[nH]cn2)cc1I
CHEMBL20078
CCOc1nc2nc(C(=O)c3ccccc3)cn2c2c1CSCC2
CHEMBL20079
Brc1cccc(Br)c1N(CC1CC1)C1=NCCN1
CHEMBL20080
O=C1c2nc3n(c2C(=O)c2c1nc1n2CCC1)CCC3
CHEMBL20081
O=C1c2cc([N+](=O)[O-])cc3cc([N+](=O)[O-])cc(c23)C(=O)N1CCNCCO.O=S(=O)(O)O
CHEMBL20082
CCCc1c(SC)nc2nc(C(=O)c3ccccc3)cn2c1CC
CHEMBL20083
Cc1cc(Cl)cc(C[S+]([O-])c2nc3ccccc3[nH]2)c1N
CHEMBL19829
CCC(C)(C)/N=c1\c(O)c(O)\c1=N/Cc1ccc(F)cc1Cl
CHEMBL19920
NCCCCCC1CCCCC1
CHEMBL19921
Cc1cc(C)c(CC(=O)c2sccc2S(=O)(=O)Nc2onc(C)c2Cl)c(C)c1O
CHEMBL19844
CN1CCc2cc(O)c(O)cc2C1Cc1ccc(O)c(O)c1
CHEMBL19845
COC1CCN(S(=O)(=O)c2ccc(S(N)(=O)=O)c(Cl)c2)CC1
CHEMBL19846
C[C@H](NC(=O)[C@@H](S)Cc1ccccc1)C(=O)O
CHEMBL19847
CCCCCCC1(c2cc(O)c3c(c2)OC(C)(C)[C@@H]2CC=C(C)C[C@@H]32)CC1
CHEMBL19848
Nc1nc(O)c2ncn([C@@H]3O[C@H]4C[C@@H](C(=O)O)O[C@H]4[C@H]3O)c2n1
CHEMBL3310708
CC[C@H](C)[C@H](NC(C)=O)C(=O)N[C@H](C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(O)C(F)(F)C(=O)NCC(=O)OCc1ccccc1)[C@@H](C)OCc1ccccc1
CHEMBL20149
CC/N=C/C1=Cc2c(cc3c(c2OC)OCO3)C(c2cc(OC)c(OC)c(OC)c2)[C@@H]1C(=O)OC
CHEMBL4434946
O=C1CC2CCC(C1)N2CCc1ccc(F)cc1
CHEMBL4434947
CC(=O)N[C@@H](CC(C)C)C(=O)N[C@H](C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CSCc2cccc(c2)CSC[C@@H](C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@H](C(=O)N[C@@H](CO)C(=O)NCCOCCOCC(=O)N[C@@H](CCCCNC(=O)c2ccc(-c3c4ccc(=O)cc-4oc4cc(O)ccc34)c(C(=O)O)c2)C(N)=O)[C@@H](C)O)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccc(O)cc2)NC...
CHEMBL4434948
N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H]1C/C=C\C[C@@H](NC(=O)[C@@H](N)Cc2ccc(O)cc2)C(=O)NCC(=O)N[C@@H](Cc2ccccc2)C(=O)NNC(=O)[C@H](Cc2ccccc2)NC(=O)CNC1=O.O=C(O)C(F)(F)F.O=C(O)C(F)(F)F
CHEMBL4434949
O=C(O)C1CCN(CCO/N=C/c2ccccc2-c2ccc(-c3ccccc3)cc2)C1
CHEMBL20151
COc1ccc2[nH]c([S+]([O-])Cc3cc(C)ccc3N)nc2c1
CHEMBL20240
CC(=N)N1CCC(Oc2ccc(N(Cc3ccc4ccc(C(=N)N)cc4c3)S(=O)(=O)CC(=O)O)cc2)CC1
CHEMBL20241
Brc1cccc(Br)c1N(Cc1ccccc1)C1=NCCN1
CHEMBL20168
Cc1cc2c(cc1CC(=O)c1sccc1S(=O)(=O)Nc1onc(C)c1C)OCO2
CHEMBL20169
O=C(O)Cc1nn(Cc2nc3cc(Br)ccc3s2)c(=O)c2ccccc12
CHEMBL20170
CN1CCC(NC2c3ccccc3Oc3ccccc32)CC1
CHEMBL1163504
CN1CCN(CCNC(=O)c2ccc3c(c2)/C(=C2/Nc4ccccc4C2=O)C(=O)N3)CC1.Cl
CHEMBL20173
CC(C)[C@H](NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@H](C(=O)N[C@@H](CC(=O)N(C)C)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](CC(C)(C)C)C(=O)O)C(C)C
CHEMBL20175
Cc1ccc(C(C)NC(=O)c2ccc(N)cc2)cc1
CHEMBL19922
CC(/N=c1\c(O)c(O)\c1=N/CCc1ccc(C#N)cc1)C(C)(C)C
CHEMBL19923
CC(=O)Nc1ccc(C(=O)NC(C)c2ccccc2)cc1
CHEMBL19924
CC(C)CN(C1=NCCN1)c1c(Br)cccc1Br
CHEMBL19925
Cc1nonc1/C=N/O
CHEMBL20016
CC[C@@H](C)[C@@H](NC(=O)[C@@H](C)N)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCSC)C(=O)O
CHEMBL20017
CC(C)Oc1cccc(N2CCNCC2)n1
CHEMBL3309346
C[C@@H](CC[C@H]1C(CO)=CC[C@H]2C(C)(C)CCC[C@@]21C)CC(=O)OCCCCCCN1CCCCC1
CHEMBL19849
Oc1nc2cc(C#CCN3CCC(Cc4ccc(F)cc4)CC3)c[nH]c-2n1
CHEMBL19945
Oc1nc2cc(C#CCN3CCC(CCc4ccc(F)cc4)CC3)ccc2[nH]1
CHEMBL19947
Cc1nnc2n1-c1ccc(C#CCN3C(=O)COc4ccccc43)cc1C(c1ccccc1F)=NC2
CHEMBL4434644
C#CCN(Cc1ccc(F)cc1F)CC(O)(Cn1cncn1)c1ccc(F)cc1F
CHEMBL4434645
O=C(NNS(=O)(=O)c1ccccc1)c1cccc(-c2ccccc2Cl)c1
CHEMBL4434646
COc1c(OCC(=O)O)cc2oc3cc4c(c(O)c3c(=O)c2c1CC=C(C)C)C=CC(C)(C)O4
CHEMBL4434647
O=C(Cn1cc(Cn2c3ccccc3c3ccccc32)nn1)c1cccc(F)c1
CHEMBL4434648
O=C(CO[N+](=O)[O-])N[C@@H](CC(=O)N1CCn2c(nnc2C(F)(F)F)C1)Cc1cc(F)c(F)cc1F
CHEMBL4434649
C=C(C)[C@@H]1CC[C@]2(C(=O)O)CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC[C@H](O)[C@@](C)(COC(=O)c6ccccc6C(F)(F)F)[C@@H]5CC[C@]43C)[C@@H]12
CHEMBL4434650
COc1cccc(CN2C(=O)[C@]3(CC(=O)Nc4c3nnn4[C@@H](C)c3ccc(Cl)cc3)c3cc(Cl)ccc32)c1
CHEMBL19948
CC(C)CC(=O)c1c(O)cc(O)cc1O
CHEMBL20244
O=C(O)C[C@]1(C(=O)O)C[C@@H]2C[C@@H](n3cnc4c(O)ncnc43)C[C@@H]2O1
CHEMBL20245
Cc1cccc(C[S+]([O-])c2nc3ccccc3[nH]2)c1N
CHEMBL20332
Nc1nc(O)c2ncn([C@@H]3C=C4C[C@](CC(=O)O)(C(=O)O)O[C@H]4[C@H]3O)c2n1
CHEMBL1163506
COS(=O)(=O)[O-].C[N+](C)(C)CCNC(=O)c1ccc2c(c1)/C(=C1/Nc3ccccc3C1=O)C(=O)N2
CHEMBL3310732
Cc1ccc(CN2CCOCC2)cc1NC(=O)c1ccc(Nc2nc(-c3ccc(OC(F)(F)F)cc3)c3ccsc3n2)cc1
CHEMBL20088
CC1=C(N2CC2)C(=O)c2nc3n(c2C1=O)CCC3N
CHEMBL20176
C=CCN(C1=NCCN1)c1c(Br)cccc1Br
CHEMBL4434708
O=Nc1c(NCCCc2ccccc2)[nH]c(=O)[nH]c1=O
CHEMBL4434709
CC(C)(C)[C@@H]1C=C(C(=O)N[C@@H](Cc2ccccc2)C(N)=O)[C@H](c2ccc(Cl)c(Cl)c2)N1S(=O)(=O)C(C)(C)C
CHEMBL4434710
Cc1c(N2CCN(C(=O)c3ccccc3)CC2)c(=O)n(C[C@H](N)c2ccccc2)c(=O)n1Cc1c(F)cccc1F
CHEMBL4434711
CNc1cc(Nc2cccn(-c3ccc(C(C)(C)O)cc3)c2=O)nn2c(C(=O)NC3CC3)cnc12
CHEMBL4434712
O=C(O)C(Cc1c[nH]c2ccccc12)N1C(=O)/C(=C/c2ccc3cc(OCc4ccc(Cl)cc4)ccc3c2)SC1=S
CHEMBL4434713
O=C(/C=C/c1cccc(OCCCCCCN2CCc3ccccc3C2)c1)c1ccccc1O
CHEMBL4434714
COc1ccc(N(Cc2ccccc2F)NC(=O)NCCCN2CCN(c3ccccc3OC)CC2)cc1
CHEMBL4434715
CN1C(=O)S/C(=C\c2cc(Oc3cccc(O)c3N)c(O)cc2Br)C1=O
CHEMBL4434716
Cn1cc(-c2ccnc(/C=C3/C(=O)N4[C@@H](C(=O)O)[C@](C)(COC(=O)Cc5ccc(O)c(O)c5)S(=O)(=O)[C@H]34)c2)cn1
CHEMBL4434717
COc1cc(-c2cncc(-c3ccc(N4C[C@H](C)N(C)[C@H](C)C4)cc3)c2C)cc(F)c1C(N)=O
CHEMBL4434718
CCc1nn(-c2nc(-c3ccc(Cl)cc3)cs2)c2c1Cc1ccccc1-2
CHEMBL4434719
COC[C@@H]1NC(=O)c2nccn2CCCCCCOC[C@@H](C(=O)N[C@@H](Cc2ccccc2)C(=O)[C@@]2(C)CO2)NC1=O
CHEMBL4434720
CS(=O)(=O)c1ccc2[nH]c(C(=O)N3CC(=O)N(Cc4ccccc4)[C@@H](Cc4ccccc4)C3)cc2c1
CHEMBL4434721
O=c1ccn(COCCOP(=O)([O-])CP(=O)([O-])[O-])c(=O)[nH]1.[Na+].[Na+].[Na+]
CHEMBL20177
CCc1cn(C2CC(F)C(CO)O2)c(=O)[nH]c1=O
CHEMBL20178
Cc1nnc2n1-c1sc(C#CCn3c(=O)c4ccccc4c4ccccc43)cc1C(c1ccccc1Cl)=NC2C
CHEMBL20179
CCC(C)(C)/N=c1\c(O)c(O)\c1=N/Cc1c(C)cccc1C
CHEMBL3310764
Clc1ccc(CNC2CCCn3nc(COc4ccccc4)cc32)cc1
CHEMBL20018
CC(C)(C)/N=c1\c(O)c(O)\c1=N/Cc1ccccc1F
CHEMBL20019
Cc1nnc2n1-c1sc(C#CCC34CCCc5cccc(c53)NC4=O)cc1C(c1ccccc1Cl)=NC2
CHEMBL19740
Cc1cnc(NCC(F)(F)c2ccc(F)cc2)c(=O)n1CC(=O)NCc1cnc(N)cn1
CHEMBL3309347
C[C@@H](CC[C@H]1C(CO)=CC[C@H]2C(C)(C)CCC[C@@]21C)CC(=O)OCCN1CCOCC1
CHEMBL19949
CC[N+](C)(CCCCCC(=O)N1CCC(CCC2CCN(C(=O)CCCCC[N+](C)(CC)Cc3ccccc3OC)CC2)CC1)Cc1ccccc1OC.[I-].[I-]
CHEMBL19950
CC(=O)c1cc(C)cc(C)c1NC(=O)c1sccc1S(=O)(=O)Nc1onc(C)c1Cl
CHEMBL20038
CC(C)C(=O)c1c(O)cc(O)cc1O
CHEMBL20040
c1ccc(CNC2c3ccccc3Oc3ccccc32)nc1
CHEMBL20041
CC(C)(C)/N=c1\c(O)c(O)\c1=N/Cc1ccc(Cl)cc1
CHEMBL20333
CCCCCC/N=C/C1=Cc2cc3c(cc2C(c2cc(OC)c(OC)c(OC)c2)[C@@H]1C(=O)OC)OCO3
CHEMBL20335
CCCN(C1=NCCN1)c1c(Br)cccc1Br
CHEMBL20063
Clc1cc2nc(C3CCNCC3)n(CCCCCn3c(C4CCNCC4)nc4cc(Cl)c(Cl)cc43)c2cc1Cl
CHEMBL20346
CSc1nc2nc(C(=O)c3ccccc3)cn2c2c1CSCC2
CHEMBL4434782
Cc1cc(Cl)ccc1OCC(=O)N/N=C/c1cccc(F)c1
CHEMBL4434783
CCc1nc(Nc2ccc(CO)cc2)nc(-c2cccc(Cl)c2)n1
CHEMBL4434784
Cc1cc(C)cc(C(=O)NOCc2ccc(/C=C/C(=O)NO)cc2)c1
CHEMBL4434785
COc1cc2c(cc1Oc1c3c(cc(OC)c1OC)CCN(C)C3)C(=O)N(C)CC2
CHEMBL4434786
C/C=C1/CN2CCC1C(=O)c1[nH]c3c(OC)cccc3c1C2.O=S(=O)(O)O
CHEMBL4434787
CN1CCCC1c1cncc(-c2cn(C[C@H]3O[C@@H]4O[C@@H]5[C@@H](Cn6cc(-c7cncc(C8CCCN8C)c7)nn6)O[C@H](O[C@@H]6[C@@H](Cn7cc(-c8cncc(C9CCCN9C)c8)nn7)O[C@H](O[C@@H]7[C@@H](Cn8cc(-c9cncc(C%10CCCN%10C)c9)nn8)O[C@H](O[C@@H]8[C@@H](Cn9cc(-c%10cncc(C%11CCCN%11C)c%10)nn9)O[C@H](O[C@@H]9[C@@H](Cn%10cc(-c%11cncc(C%12CCCN%12C)c%11)nn%10)O[C@H](...
CHEMBL4434788
CC(C)(O)Cn1/c(=N/C(=O)c2ccnc(-c3ccccc3)c2)[nH]c2ccccc21
CHEMBL4434789
O=C(N/N=C/c1cc[n+](Cc2ccccc2)c2ccccc12)c1ccc2ccc3ccc(C(=O)N/N=C/c4cc[n+](Cc5ccccc5)c5ccccc45)nc3c2n1.[Br-].[Br-]
CHEMBL20348
CCCN(C)CCCCCc1ccccc1
CHEMBL20349
CCOc1nc2nc(C(=O)c3ccccc3)cn2c2c1CCCCC2
CHEMBL3310765
COc1ccc(CNC2CCCn3nc(COc4ccccc4)cc32)cc1