Datasets:

uuid
stringlengths
4
8
template_uuid
stringclasses
40 values
question
stringlengths
13
193
answer
stringlengths
29
2.2k
benchmark_query
stringlengths
133
622
execution_results
stringlengths
2
1.14M
query_type
stringclasses
2 values
sql_category
stringclasses
26 values
bio_category
stringclasses
14 values
Q17.492
Q17
What gene does the drug Onasemnogene Abeparvovec target?
The drug Onasemnogene Abeparvovec targets 2 genes: SMN1 and SMN2.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_3439', 'drugName': 'Onasemnogene Abeparvovec', 'tradeNames_string': '', 'drugSynonyms_string': 'AVXS-101, Onasemnogene abeparvovec, Zolgensma', 'linkedDiseasesDrug_string': 'Spinal Muscular Atrophy (EFO_0008525)', 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.445
Q17
What gene does the drug Cyclofenil target?
The drug Cyclofenil targets 2 genes: ESR2 and ESR1.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1475', 'drugName': 'Cyclofenil', 'tradeNames_string': 'Neoclym, Rehibin', 'drugSynonyms_string': 'Cyclofenil, F 6066, F-6066, ICI 48213, ICI-48213, NSC-86464, Sexovid', 'linkedDiseasesDrug_string': '', 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True, 'newLinked...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.274
Q17
What gene does the drug Capadenoson target?
The drug Capadenoson is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target the gene ADORA1.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_3660', 'drugName': 'Capadenoson', 'tradeNames_string': '', 'drugSynonyms_string': 'BAY 68-4986, BAY-68-4986, Bay-684986, Capadenoson', 'linkedDiseasesDrug_string': 'Angina Pectoris (EFO_0003913), Atrial Fibrillation (EFO_0000275)', 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'dru...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.187
Q17
What gene does the drug Mirdametinib target?
The drug Mirdametinib is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 2 genes: MAP2K2 and MAP2K1
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_179', 'drugName': 'Mirdametinib', 'tradeNames_string': '', 'drugSynonyms_string': 'Mirdametinib, PD-0325901, Pd 0325901, Pd 03525901, Pd 901, Pd-0325901', 'linkedDiseasesDrug_string': 'Cancer (MONDO_0004992), Neoplasm (EFO_0000616), Neurofibromatosis Type 1 (MONDO_0018975), Non-Small Cell ...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.950
Q17
What gene does the drug Tarenflurbil target?
The drug Tarenflurbil is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 6 genes: APH1A, APH1B, PSEN1, PSENEN, NCSTN and PSEN2
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2667', 'drugName': 'Tarenflurbil', 'tradeNames_string': 'Flurizan', 'drugSynonyms_string': 'E-7869, Flurbiprofen, (r)-, MPC-7869, R-flurbiprofen, Tarenflurbil', 'linkedDiseasesDrug_string': 'Alzheimer Disease (MONDO_0004975), Prostate Cancer (MONDO_0008315), Dementia (HP_0000726)', 'yearOf...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.247
Q17
What gene does the drug Prazosin Hydrochloride target?
The drug Prazosin Hydrochloride targets 3 genes: ADRA1D, ADRA1B and ADRA1A.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5265', 'drugName': 'Prazosin Hydrochloride', 'tradeNames_string': 'Alphavase 0.5, Alphavase 1, Alphavase 2, Alphavase 5, Hypovase, Hypovase b.d., Kentovace, Minipress, Minipress xl, Prazosin hydrochloride', 'drugSynonyms_string': 'CP-12,299-1, CP-12299-1, NSC-292810, Prazosin hcl, Prazosin...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1100
Q17
What gene does the drug Lerodalcibep target?
The drug Lerodalcibep is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target the gene PCSK9.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_6016', 'drugName': 'Lerodalcibep', 'tradeNames_string': '', 'drugSynonyms_string': 'Lerodalcibep', 'linkedDiseasesDrug_string': 'Familial Hypercholesterolemia (EFO_0004911), Homozygous Familial Hypercholesterolemia (MONDO_0018328), Cardiovascular Disease (EFO_0000319), Hypercholesterolemia...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1018
Q17
What gene does the drug Aclidinium Bromide target?
The drug Aclidinium Bromide targets the gene CHRM3.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_6136', 'drugName': 'Aclidinium Bromide', 'tradeNames_string': 'Eklira, Tudorza pressair', 'drugSynonyms_string': '14115700, Aclidinium bromide, Genuair, LAS 34273, LAS 34273 MICRONIZED, LAS W-330, LAS-34273, LAS-34273 MICRONIZED, LAS-W-330', 'linkedDiseasesDrug_string': 'Asthma (MONDO_0004...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.590
Q17
What gene does the drug Benzthiazide target?
The drug Benzthiazide targets the gene SLC12A3.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2994', 'drugName': 'Benzthiazide', 'tradeNames_string': 'Aquatag, Benzthiazide, Exna, Fovane, Urese', 'drugSynonyms_string': 'Benzothiazide, Benzthiazide, NSC-755902', 'linkedDiseasesDrug_string': '', 'yearOfFirstApproval': 1960, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True, 'newLink...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1629
Q17
What gene does the drug Gemfibrozil target?
The drug Gemfibrozil targets the gene PPARA.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_6015', 'drugName': 'Gemfibrozil', 'tradeNames_string': 'Emfib, Gemfibrozil, Lopid', 'drugSynonyms_string': 'CI-719, Gemfibrozil, NSC-757024', 'linkedDiseasesDrug_string': 'Cancer (MONDO_0004992), Alzheimer Disease (MONDO_0004975), Smoking Cessation (EFO_0004319), Hypertriglyceridemia (EFO_...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.535
Q17
What gene does the drug Norgestrel target?
The drug Norgestrel targets the gene PGR.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_6188', 'drugName': 'Norgestrel', 'tradeNames_string': 'Opill, Ovrette', 'drugSynonyms_string': 'Dl-norgestrel, FH-122A, NSC-757251, Norgestrel, Prefest, Previfem, SH-70850, SH-850, Sprintec, Tri-Previfem, Tri-Sprintec, WY-3707', 'linkedDiseasesDrug_string': 'Hemorrhage (MP_0001914), Endome...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.899
Q17
What gene does the drug Loperamide Hydrochloride target?
The drug Loperamide Hydrochloride targets the gene OPRM1.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_6052', 'drugName': 'Loperamide Hydrochloride', 'tradeNames_string': 'Arret, Diah-limit, Diaquitte, Diareze, Diarrhoea relief, Diasorb, Diocalm, Diocaps, Dioraleze, Entrocalm, Gppe pack, Imodium, Imodium Advanced, Imodium a-d, Imodium a-d ez chews, Imodium classic, Imodium ibs relief, Imodi...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1483
Q17
What gene does the drug Ono-2333Ms target?
The drug Ono-2333Ms is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target the gene CRHR1.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2958', 'drugName': 'Ono-2333Ms', 'tradeNames_string': '', 'drugSynonyms_string': 'Ono-2333ms', 'linkedDiseasesDrug_string': 'Major Depressive Disorder (MONDO_0002009)', 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False, 'newLinkedTargets_string': 'CRHR1 (ENSG000...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1109
Q17
What gene does the drug Dorzolamide target?
The drug Dorzolamide targets the gene CA2.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_333', 'drugName': 'Dorzolamide', 'tradeNames_string': 'Dorzant, Trusopt', 'drugSynonyms_string': 'Dorzolamide, Dorzolamide, trans-(-)-, MK-507, Trusopt', 'linkedDiseasesDrug_string': 'Open-Angle Glaucoma (EFO_0004190), Ocular Hypertension (EFO_1001069), Wet Macular Degeneration (EFO_000468...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.421
Q17
What gene does the drug Ranitidine target?
The drug Ranitidine targets the gene HRH2.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1617', 'drugName': 'Ranitidine Hydrochloride', 'tradeNames_string': 'Azantac, Dumoran, Gavilast, Gavilast-p, Histac, Raciran 150, Raciran 300, Ranicalm, Raniplex, Ranitic, Ranitidine hydrochloride, Ranitil, Rantec, Ranzac, Vivatak, Zaedoc 150, Zaedoc 300, Zantac, Zantac 150, Zantac 25, Zan...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.277
Q17
What gene does the drug Doxepin target?
The drug Doxepin targets the gene SLC6A2.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2495', 'drugName': 'Doxepin Hydrochloride', 'tradeNames_string': 'Adapin, Doxepin hydrochloride, Quitaxon, Silenor, Sinequan, Xepin, Zonalon', 'drugSynonyms_string': 'Doxepin hcl, Doxepin hydrochloride, NSC-108160, P-3693A', 'linkedDiseasesDrug_string': 'Unipolar Depression (EFO_0003761), ...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1174
Q17
What gene does the drug Obeticholic Acid target?
The drug Obeticholic Acid targets the gene NR1H4.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_3863', 'drugName': 'Obeticholic Acid', 'tradeNames_string': 'Ocaliva', 'drugSynonyms_string': '6-ecdca, 6-ethylchenodeoxycholic acid, DSP-1747, INT-747, Obeticholic acid', 'linkedDiseasesDrug_string': "Familial Adenomatous Polyposis (Orphanet_733), Hepatitis, Alcoholic (EFO_1001345), Diarr...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1487
Q17
What gene does the drug Balsalazide target?
The drug Balsalazide targets 4 genes: PTGS2, PPARG, ALOX5 and PTGS1.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1298', 'drugName': 'Balsalazide Disodium', 'tradeNames_string': 'Balsalazide disodium, Colazal, Colazide, Giazo', 'drugSynonyms_string': 'BX-661A, BX661A, Balsalazide disodium, Balsalazide disodium anhydrous, Balsalazide disodium dihydrate, Balsalazide disodium salt dihydrate, Balsalazide ...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1456
Q17
What gene does the drug Milciclib target?
The drug Milciclib is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 4 genes: NTRK1, CDK4, CDK2 and CDK1
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5842', 'drugName': 'Milciclib', 'tradeNames_string': '', 'drugSynonyms_string': 'Milciclib, PHA 848125, PHA-848125, Pha-848125', 'linkedDiseasesDrug_string': 'Neoplasm (EFO_0000616), Hepatocellular Carcinoma (EFO_0000182), Thymic Carcinoma (EFO_1000576), Thymoma (EFO_1000581)', 'yearOfFirs...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.253
Q17
What gene does the drug Terfenadine target?
The drug Terfenadine targets the gene HRH1.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2637', 'drugName': 'Terfenadine', 'tradeNames_string': 'Antihistamine, Histafen, Histafen 120, Seldane, Terfenor, Terfenor fte, Terfex, Terfinax 120, Terfinax 60, Triludan, Triludan fte', 'drugSynonyms_string': 'NSC-665802, NSC-758627, RMI 9918, RMI-9918, Terfenadine', 'linkedDiseasesDrug_...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.419
Q17
What gene does the drug Prednisone target?
The drug Prednisone targets the gene NR3C1.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2255', 'drugName': 'Prednisone', 'tradeNames_string': 'Cortan, Cortancyl, Decortisyl, Delta-dome, Deltasone, Fernisone, Liquid pred, Lodotra, Meticorten, Orasone, Paracort, Prednicen-m, Prednisone, Prednisone intensol, Rayos, Servisone, Sterapred', 'drugSynonyms_string': '3en3hg4wsw, Decor...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1590
Q17
What gene does the drug Dipyrone target?
The drug Dipyrone targets 2 genes: PTGS2 and PTGS1.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2814', 'drugName': 'Dipyrone', 'tradeNames_string': 'Diprofarn, Novaldin', 'drugSynonyms_string': 'Dipyrone', 'linkedDiseasesDrug_string': 'Sepsis (HP_0100806), Migraine Disorder (MONDO_0005277), Pain (EFO_0003843), Fever (HP_0001945), Chronic Pain (HP_0012532), Gastroenteritis (EFO_100146...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1895
Q17
What gene does the drug Fosaprepitant Dimeglumine target?
The drug Fosaprepitant Dimeglumine targets the gene TACR1.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5495', 'drugName': 'Fosaprepitant Dimeglumine', 'tradeNames_string': 'Emend, Fosaprepitant dimeglumine', 'drugSynonyms_string': 'Fosaprepitant (as dimeglumine), Fosaprepitant dimeglumine, Fosaprepitant meglumine, MK-0517', 'linkedDiseasesDrug_string': 'Cancer (MONDO_0004992), Chemotherapy-...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.582
Q17
What gene does the drug Pf-03715455 target?
The drug Pf-03715455 is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target the gene MAPK14.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5605', 'drugName': 'Pf-03715455', 'tradeNames_string': '', 'drugSynonyms_string': 'PF-03715455, Pf-03715455, Pf-3715455', 'linkedDiseasesDrug_string': 'Asthma (MONDO_0004979), Chronic Obstructive Pulmonary Disease (EFO_0000341)', 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugI...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.314
Q17
What gene does the drug Orphenadrine target?
The drug Orphenadrine targets 19 genes: SLC6A2, SCN9A, SCN7A, SCN10A, GRIN3B, SCN4A, SCN8A, GRIN3A, SCN2A, SCN3A, GRIN2B, GRIN2A, SCN5A, GRIN1, SCN1A, SCN11A, HRH1, GRIN2D and GRIN2C.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_4306', 'drugName': 'Orphenadrine Hydrochloride', 'tradeNames_string': 'Biorphen, Disipal', 'drugSynonyms_string': 'Mephenamin, NSC-82357, Orphenadrine (chloride), Orphenadrine Chloride, Orphenadrine hcl, Orphenadrine hydrochloride', 'linkedDiseasesDrug_string': 'Parkinson Disease (MONDO_00...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1962
Q17
What gene does the drug Icotinib target?
The drug Icotinib is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target the gene EGFR.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5477', 'drugName': 'Icotinib', 'tradeNames_string': '', 'drugSynonyms_string': 'BPI-2009H, Bpi-2009, Icotinib', 'linkedDiseasesDrug_string': 'Pancreatic Carcinoma (EFO_0002618), Psoriasis (EFO_0000676), Lung Adenocarcinoma (EFO_0000571), Breast Cancer (MONDO_0007254), Lung Cancer (MONDO_00...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.387
Q17
What gene does the drug Pirenzepine target?
The drug Pirenzepine targets the gene CHRM1.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5044', 'drugName': 'Pirenzepine', 'tradeNames_string': 'Gastri p, Gastrozepin', 'drugSynonyms_string': 'ACI-91, Pirenzepine', 'linkedDiseasesDrug_string': 'Peptic Ulcer (HP_0004398), Gastroesophageal Reflux Disease (EFO_0003948)', 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drug...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.541
Q17
What gene does the drug Procaine Hydrochloride target?
The drug Procaine Hydrochloride targets 10 genes: SCN1A, SCN9A, SCN7A, SCN8A, SCN11A, SCN10A, SCN2A, SCN5A, SCN4A and SCN3A.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2951', 'drugName': 'Procaine Hydrochloride', 'tradeNames_string': 'Novocain, Pasconeural n, Procaine hydrochloride', 'drugSynonyms_string': 'Anestil, Enpro, Jenacaine, Medaject, NSC-757280, Naucaine, Neocaine, Omnicain, Planocaine, Procaine hcl, Procaine hydrochloride, Procaini hydrochlori...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.431
Q17
What gene does the drug Remifentanil Hydrochloride target?
The drug Remifentanil Hydrochloride targets the gene OPRM1.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_577', 'drugName': 'Remifentanil Hydrochloride', 'tradeNames_string': 'Ultiva', 'drugSynonyms_string': 'GI 87084B, GI-87084B, Remifentanil hcl, Remifentanil hydrochloride', 'linkedDiseasesDrug_string': '', 'yearOfFirstApproval': 1996, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True, 'new...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.657
Q17
What gene does the drug Anileridine Phosphate target?
The drug Anileridine Phosphate targets 2 genes: OPRK1 and OPRM1.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_4938', 'drugName': 'Anileridine Phosphate', 'tradeNames_string': 'Leritine', 'drugSynonyms_string': 'Anileridine phosphate, Leritine phosphate', 'linkedDiseasesDrug_string': '', 'yearOfFirstApproval': 1982, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True, 'newLinkedTargets_string': 'OPR...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1642
Q17
What gene does the drug Decamethonium Bromide target?
The drug Decamethonium Bromide targets 5 genes: CHRNB1, CHRNA1, CHRND, CHRNE and CHRNG.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5170', 'drugName': 'Decamethonium Bromide', 'tradeNames_string': 'Syncurine', 'drugSynonyms_string': 'Decamethonium Bromide, Decamethonium bromide, Decamethonium diiodide, Decamethonium iodide, NSC-23004', 'linkedDiseasesDrug_string': '', 'yearOfFirstApproval': 1982, 'maxClinicalTrialPhase...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1318
Q17
What gene does the drug Amoxapine target?
The drug Amoxapine targets 7 genes: SLC6A2, DRD4, DRD1, SLC6A4, DRD2, DRD5 and DRD3.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2376', 'drugName': 'Amoxapine', 'tradeNames_string': 'Amoxapine, Asendin, Asendis, Defanyl', 'drugSynonyms_string': 'Amoxapine, CL 67,772, CL 67772, CL-67,772, CL-67772, NSC-759559', 'linkedDiseasesDrug_string': 'Unipolar Depression (EFO_0003761)', 'yearOfFirstApproval': 1980, 'maxClinical...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1358
Q17
What gene does the drug Nomifensine Maleate target?
The drug Nomifensine Maleate targets 3 genes: SLC6A4, SLC6A2 and SLC6A3.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2665', 'drugName': 'Nomifensine Maleate', 'tradeNames_string': 'Merital', 'drugSynonyms_string': 'HOE 984, HOE-984, Hostalival, NSC-289114, Nomifensine hydrogen maleate, Nomifensine maleate, Psicronizer', 'linkedDiseasesDrug_string': '', 'yearOfFirstApproval': 1984, 'maxClinicalTrialPhase'...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.414
Q17
What gene does the drug Ubrogepant target?
The drug Ubrogepant targets the gene CALCRL.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_528', 'drugName': 'Ubrogepant', 'tradeNames_string': 'Ubrelvy', 'drugSynonyms_string': 'MK-1602, Ubrogepant, Ubrogepant anhydrous', 'linkedDiseasesDrug_string': 'Migraine Disorder (MONDO_0005277)', 'yearOfFirstApproval': 2019, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True, 'newLinkedT...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1615
Q17
What gene does the drug Diphemanil Methylsulfate target?
The drug Diphemanil Methylsulfate targets 2 genes: CHRM1 and CHRM3.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1327', 'drugName': 'Diphemanil Methylsulfate', 'tradeNames_string': 'Prantal', 'drugSynonyms_string': 'Diphemanil methylsulfate, Diphemanil methylsulphate, Diphemanil metilsulfate, NSC-41725', 'linkedDiseasesDrug_string': '', 'yearOfFirstApproval': 1982, 'maxClinicalTrialPhase': 4, 'drugIs...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.687
Q17
What gene does the drug Bi-671800 target?
The drug Bi-671800 is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target the gene PTGDR2.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5746', 'drugName': 'Bi-671800', 'tradeNames_string': '', 'drugSynonyms_string': 'Actimis, BI 671800, BI671800, Bi 671800, Bi-671800', 'linkedDiseasesDrug_string': 'Asthma (MONDO_0004979)', 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False, 'newLinkedTargets_stri...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.621
Q17
What gene does the drug Begacestat target?
The drug Begacestat is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 6 genes: APH1A, APH1B, PSEN1, PSENEN, NCSTN and PSEN2
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_6270', 'drugName': 'Begacestat', 'tradeNames_string': '', 'drugSynonyms_string': 'Begacestat, GSI-953', 'linkedDiseasesDrug_string': 'Alzheimer Disease (MONDO_0004975)', 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drugIsApproved': False, 'newLinkedTargets_string': 'APH1A (ENSG00...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.923
Q17
What gene does the drug Vedolizumab target?
The drug Vedolizumab targets 2 genes: ITGB7 and ITGA4.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5088', 'drugName': 'Vedolizumab', 'tradeNames_string': 'Entyvio', 'drugSynonyms_string': 'LDP-02, LDP02, MLN-0002, MLN-02, MLN0002, MLN02, Vedolizumab', 'linkedDiseasesDrug_string': "Hiv Infection (EFO_0000764), Infection (EFO_0000544), Crohn'S Disease (EFO_0000384), Ulcerative Colitis (EF...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1199
Q17
What gene does the drug Tesamorelin target?
The drug Tesamorelin targets the gene GHRHR.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2825', 'drugName': 'Tesamorelin', 'tradeNames_string': '', 'drugSynonyms_string': 'TH-9507, TH9507, Tesamorelin', 'linkedDiseasesDrug_string': 'Hiv Infection (EFO_0000764), Cognitive Impairment (HP_0100543), Hiv-Associated Lipodystrophy Syndrome (EFO_1001348), Chronic Obstructive Pulmonary...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.839
Q17
What gene does the drug Sitagliptin target?
The drug Sitagliptin targets the gene DPP4.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2411', 'drugName': 'Sitagliptin Phosphate', 'tradeNames_string': 'Janumet Xr, Januvia', 'drugSynonyms_string': 'Glactiv, MK-0431, MK0431, ONO-5435, Sitagliptin monophosphate, Sitagliptin monophosphate anhydrous, Sitagliptin monophosphate monohydrate, Sitagliptin phosphate, Sitagliptin phos...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1771
Q17
What gene does the drug Ribociclib target?
The drug Ribociclib targets 2 genes: CDK4 and CDK6.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_3488', 'drugName': 'Ribociclib', 'tradeNames_string': '', 'drugSynonyms_string': 'LEE-011, LEE-011A, LEE011, LEE011A, Lee-011, NVP-LEE011, Ribociclib', 'linkedDiseasesDrug_string': 'Ovarian Carcinoma (EFO_0001075), Cancer (MONDO_0004992), Teratoma (MONDO_0002601), Neuroblastoma (EFO_000062...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.953
Q17
What gene does the drug Interferon Alfa-N3 target?
The drug Interferon Alfa-N3 targets 2 genes: IFNAR1 and IFNAR2.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_404', 'drugName': 'Interferon Alfa-N3', 'tradeNames_string': 'Alferon ldo, Alferon n gel, Alferon n injection', 'drugSynonyms_string': '.alpha.-interferons, Alferon, Alferon n, Interferon alfa-n3, Interferon alpha-n3, Leukocyte interferon', 'linkedDiseasesDrug_string': 'Severe Acute Respir...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.185
Q17
What gene does the drug Argipressin Tannate target?
The drug Argipressin Tannate targets 3 genes: AVPR2, AVPR1A and AVPR1B.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5273', 'drugName': 'Argipressin Tannate', 'tradeNames_string': 'Pitressin tannate (synthetic)', 'drugSynonyms_string': 'Argipressin, Argipressin tannate, CI-107', 'linkedDiseasesDrug_string': '', 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True, 'newLinkedTarget...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1072
Q17
What gene does the drug Butamben Picrate target?
The drug Butamben Picrate targets 2 genes: TRPV4 and TRPA1.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_268', 'drugName': 'Butamben Picrate', 'tradeNames_string': '', 'drugSynonyms_string': 'ABBOTT-34842, Butamben picrate', 'linkedDiseasesDrug_string': '', 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True, 'newLinkedTargets_string': 'TRPV4 (ENSG00000111199), TRPA1 ...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.711
Q17
What gene does the drug Chloroprocaine target?
The drug Chloroprocaine targets 10 genes: SCN1A, SCN9A, SCN7A, SCN8A, SCN11A, SCN10A, SCN2A, SCN5A, SCN4A and SCN3A.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1606', 'drugName': 'Chloroprocaine', 'tradeNames_string': '', 'drugSynonyms_string': '2-chloroprocaine, Chloroprocaine', 'linkedDiseasesDrug_string': 'Cataract (MONDO_0005129), Pregnancy (EFO_0002950), Pain (EFO_0003843)', 'yearOfFirstApproval': 1955, 'maxClinicalTrialPhase': 4, 'drugIsApp...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.173
Q17
What gene does the drug 9-Aminocamptothecin target?
The drug 9-Aminocamptothecin is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target the gene TOP1.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_121', 'drugName': '9-Aminocamptothecin', 'tradeNames_string': '', 'drugSynonyms_string': '9-amino-20(s)-camptothecin, 9-aminocamptothecin, Aminocamptothecin, NSC-603071', 'linkedDiseasesDrug_string': 'Cancer (MONDO_0004992), Lung Cancer (MONDO_0008903), Kidney Cancer (MONDO_0002367), Lymph...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.296
Q17
What gene does the drug Benoxinate target?
The drug Benoxinate targets 10 genes: SCN1A, SCN9A, SCN7A, SCN8A, SCN11A, SCN10A, SCN2A, SCN5A, SCN4A and SCN3A.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1754', 'drugName': 'Benoxinate', 'tradeNames_string': '', 'drugSynonyms_string': 'Benoxinate, Conjucain, Dorsacain, Monofree oxybuprocaine, Oxybucaine, Oxybuprocaine', 'linkedDiseasesDrug_string': 'Pruritus (HP_0000989)', 'yearOfFirstApproval': 1982, 'maxClinicalTrialPhase': 4, 'drugIsAppr...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.554
Q17
What gene does the drug Carteolol Hydrochloride target?
The drug Carteolol Hydrochloride targets 3 genes: ADRB3, ADRB2 and ADRB1.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1755', 'drugName': 'Carteolol Hydrochloride', 'tradeNames_string': 'Carteolol hydrochloride, Cartrol, Ocupress, Teoptic', 'drugSynonyms_string': 'ABBOTT-43326, Carteolol hcl, Carteolol hydrochloride, NSC-300906, OPC-1085', 'linkedDiseasesDrug_string': 'Open-Angle Glaucoma (EFO_0004190)', '...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.763
Q17
What gene does the drug Denosumab target?
The drug Denosumab targets the gene TNFSF11.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1723', 'drugName': 'Denosumab', 'tradeNames_string': 'Prolia, Prolia, Ranmark Xgeva, Prolia, xgeva, Xgeva', 'drugSynonyms_string': 'AMG 162, AMG-162, Denosumab, Denosumab biosimilar (ql-1206), Denosumab biosimilar tk-006, QL-1206, QL1206, Ql1206, TK-006, TK006', 'linkedDiseasesDrug_string'...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.304
Q17
What gene does the drug Daunorubicin Hydrochloride target?
The drug Daunorubicin Hydrochloride targets the gene TOP2A.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1919', 'drugName': 'Daunorubicin Hydrochloride', 'tradeNames_string': 'Cerubidine, Daunorubicin hydrochloride, Daunoxome', 'drugSynonyms_string': 'Daunorubicin (as hydrochloride), Daunorubicin hcl, Daunorubicin hydrochloride, FI 6339 HYDROCHLORIDE, FI 6339 [AS THE BASE], FI-6339, FI-6339 H...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1878
Q17
What gene does the drug Desvenlafaxine Succinate target?
The drug Desvenlafaxine Succinate targets 2 genes: SLC6A4 and SLC6A2.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_735', 'drugName': 'Desvenlafaxine Succinate', 'tradeNames_string': 'Desvenlafaxine succinate, Pristiq', 'drugSynonyms_string': 'DVS-233, Desvenlafaxine succinate, Desvenlafaxine succinate anhydrous, Desvenlafaxine succinate hydrate, Desvenlafaxine succinate monohydrate, Dvs anhydrous, O-de...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1093
Q17
What gene does the drug Pseudoephedrine Hydrochloride target?
The drug Pseudoephedrine Hydrochloride targets the gene SLC6A2.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_151', 'drugName': 'Pseudoephedrine Hydrochloride', 'tradeNames_string': 'Actifed, Contac, Dimotane plus, Dimotane plus l.a., Galpseud, Galpseud plus, Novafed, Otrivine mu-cron, Pseudoephedrine hydrochloride, Pseudophed, Sinutab, Sudafed, Sudafed 12 hour, Sudafed 12 hr decongest, Sudafed 24...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1747
Q17
What gene does the drug Brompheniramine Maleate target?
The drug Brompheniramine Maleate targets the gene HRH1.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1014', 'drugName': 'Brompheniramine Maleate', 'tradeNames_string': 'Brompheniramine maleate, Dimegan, Dimetane, Dimetane-ten, Dimotane, Dimotane l.a.', 'drugSynonyms_string': '(+)-Brompheniramine Maleate, Brompheniramine fumarate, Brompheniramine maleate, NSC-758652, Parabromdylamine malea...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1652
Q17
What gene does the drug Bitolterol Mesylate target?
The drug Bitolterol Mesylate targets the gene ADRB2.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_3535', 'drugName': 'Bitolterol Mesylate', 'tradeNames_string': 'Tomalate, Tornalate', 'drugSynonyms_string': 'Bitolterol mesilate, Bitolterol mesylate, Bitolterol methanesulfonate, WIN 32,784, WIN-32784', 'linkedDiseasesDrug_string': '', 'yearOfFirstApproval': 1984, 'maxClinicalTrialPhase'...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.914
Q17
What gene does the drug Phensuximide target?
The drug Phensuximide targets 3 genes: CACNA1G, CACNA1I and CACNA1H.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1498', 'drugName': 'Phensuximide', 'tradeNames_string': 'Milontin', 'drugSynonyms_string': '1-methyl-3-phenylsuccinimide, Epimid, Lifene, Milonton, Mirontin, N-methyl-3-phenylpyrrolidinedione, NSC-760079, PM-334, Phensuximid, Phensuximide, Racemic phensuximide, Succitimal', 'linkedDiseases...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1932
Q17
What gene does the drug Histamine target?
The drug Histamine targets the gene HRH1.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2616', 'drugName': 'Histamine', 'tradeNames_string': '', 'drugSynonyms_string': '.beta.-aminoethylglyoxaline, Ergamine, Ergotidine, Histamine, NSC-33792', 'linkedDiseasesDrug_string': 'Asthma (MONDO_0004979), Non-Hodgkins Lymphoma (EFO_0005952), Pterygium (EFO_0000678), Leukemia (EFO_00005...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.275
Q17
What gene does the drug Dalcetrapib target?
The drug Dalcetrapib is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target the gene CETP.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_4061', 'drugName': 'Dalcetrapib', 'tradeNames_string': '', 'drugSynonyms_string': 'Dalcetrapib, JTT-705, RO-4607381, RO4607381', 'linkedDiseasesDrug_string': 'Abnormal Circulating Lipid Concentration (HP_0003119), Hyperlipidemia (MONDO_0021187), Coronary Artery Disease (EFO_0001645), Perip...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1147
Q17
What gene does the drug Codeine Phosphate target?
The drug Codeine Phosphate targets 3 genes: OPRK1, OPRM1 and OPRD1.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_4198', 'drugName': 'Dihydrocodeine Bitartrate', 'tradeNames_string': '', 'drugSynonyms_string': 'Codeine, dihydro-, tartrate (1:1), DF 118, DF-118, Dihydrocodeine bitartrate, Dihydrocodeine bitartrate cii, Dihydrocodeine hydrogen tartrate, Dihydrocodeine phosphate, Dihydrocodeine tartrate,...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1589
Q17
What gene does the drug Basimglurant target?
The drug Basimglurant is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target the gene GRM5.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_784', 'drugName': 'Basimglurant', 'tradeNames_string': '', 'drugSynonyms_string': 'Basimglurant, NOE-101, RG-7090, RO-4917523, RO4917523, Rg7090', 'linkedDiseasesDrug_string': 'Fragile X Syndrome (MONDO_0010383), Major Depressive Disorder (MONDO_0002009), Tuberous Sclerosis (MONDO_0001734)...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.700
Q17
What gene does the drug Aprepitant target?
The drug Aprepitant targets the gene TACR1.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1299', 'drugName': 'Aprepitant', 'tradeNames_string': 'Aprepitant, Cinvanti, Emend', 'drugSynonyms_string': 'Aprepitant, L-754,030, MK-0869, MK-869, NSC-748825', 'linkedDiseasesDrug_string': 'Cancer (MONDO_0004992), Multiple Myeloma (EFO_0001378), Nausea (HP_0002018), Chemotherapy-Induced ...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1765
Q17
What gene does the drug Tiotropium Bromide target?
The drug Tiotropium Bromide targets the gene CHRM3.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_4878', 'drugName': 'Tiotropium Bromide', 'tradeNames_string': 'Spiriva, Spiriva respimat', 'drugSynonyms_string': 'BA 679 BR, BA-679 BR, BA-679-BR, BA-679BR, Tiotropium bromide, Tiotropium bromide anhydrous, Tiotropium bromide hydrate, Tiotropium bromide monohydrate', 'linkedDiseasesDrug_s...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.488
Q17
What gene does the drug Diphenylpyraline target?
The drug Diphenylpyraline targets the gene HRH1.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_6116', 'drugName': 'Diphenylpyraline', 'tradeNames_string': '', 'drugSynonyms_string': 'Diphenylpyraline', 'linkedDiseasesDrug_string': 'Allergic Disease (MONDO_0005271)', 'yearOfFirstApproval': 1982, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True, 'newLinkedTargets_string': 'HRH1 (ENS...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.428
Q17
What gene does the drug Siponimod Fumarate target?
The drug Siponimod Fumarate targets the gene S1PR1.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_4451', 'drugName': 'Siponimod Fumarate', 'tradeNames_string': 'Mayzent', 'drugSynonyms_string': 'NVP-BAF312-AEA, Siponimod fumarate, Siponimod fumaric acid, Siponimod hemifumarate, Siponimod hemifumaric acid', 'linkedDiseasesDrug_string': 'Multiple Sclerosis (MONDO_0005301), Relapsing-Remi...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.377
Q17
What gene does the drug Exemestane target?
The drug Exemestane targets the gene CYP19A1.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_923', 'drugName': 'Exemestane', 'tradeNames_string': 'Aromasin, Exemestane', 'drugSynonyms_string': 'Exemestane, FCE-24304, FCE24304, NSC-758907, PNU-155971', 'linkedDiseasesDrug_string': 'Breast Neoplasm (EFO_0003869), Cancer (MONDO_0004992), Prostate Cancer (MONDO_0008315), Breast Cancer...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1008
Q17
What gene does the drug Panobinostat Lactate target?
The drug Panobinostat Lactate targets 11 genes: HDAC4, HDAC3, HDAC2, HDAC1, HDAC5, HDAC7, HDAC8, HDAC9, HDAC11, HDAC6 and HDAC10.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5237', 'drugName': 'Panobinostat Lactate', 'tradeNames_string': 'Farydak', 'drugSynonyms_string': 'Panobinostat lactate, Panobinostat lactate anhydrous', 'linkedDiseasesDrug_string': 'Multiple Myeloma (EFO_0001378)', 'yearOfFirstApproval': 2015, 'maxClinicalTrialPhase': 4, 'drugIsApproved'...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1003
Q17
What gene does the drug Flavoxate target?
The drug Flavoxate targets 8 genes: PDE7B, PDE7A, PDE8A, PDE4D, PDE4B, PDE4A, PDE4C and PDE8B.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_766', 'drugName': 'Flavoxate', 'tradeNames_string': '', 'drugSynonyms_string': 'Bladuril, Flavoxate', 'linkedDiseasesDrug_string': 'Polyuria (HP_0000103), Prostatitis (EFO_0003830), Urinary Tract Infection (EFO_0003103), Urethritis (EFO_0003878), Urinary Incontinence (HP_0000020), Dysuria ...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1940
Q17
What gene does the drug Vernakalant target?
The drug Vernakalant targets 6 genes: KCND3, KCNJ3, KCNJ5, SCN5A, KCNA5 and KCNH2.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_716', 'drugName': 'Vernakalant', 'tradeNames_string': '', 'drugSynonyms_string': 'Vernakalant', 'linkedDiseasesDrug_string': 'Cardiac Arrhythmia (EFO_0004269), Atrial Flutter (EFO_0003911), Atrial Fibrillation (EFO_0000275)', 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApp...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.714
Q17
What gene does the drug Interferon Gamma-1B target?
The drug Interferon Gamma-1B targets 2 genes: IFNGR1 and IFNGR2.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_3679', 'drugName': 'Interferon Gamma-1B', 'tradeNames_string': 'Actimmune, Immukin', 'drugSynonyms_string': 'Ifn-.gamma., Ifn-.gamma.1b, Imifn, Immune ifn, Interferon .gamma.-1b, Interferon gama-1b, Interferon gamma, Interferon gamma-1b, Interferon gamma-1b, recombinant, Interferon gamma-1...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1335
Q17
What gene does the drug Ticlopidine Hydrochloride target?
The drug Ticlopidine Hydrochloride targets the gene P2RY12.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1201', 'drugName': 'Ticlopidine Hydrochloride', 'tradeNames_string': 'Ticlid, Ticlopidine hydrochloride, Tiklid', 'drugSynonyms_string': '4-C-32, 53-32C, Ipaton, NSC-759165, Ticlopidine hcl, Ticlopidine hydrochloride', 'linkedDiseasesDrug_string': 'Thrombotic Disease (MONDO_0000831), Strok...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1156
Q17
What gene does the drug Abt-102 target?
The drug Abt-102 is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target the gene TRPV1.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_3254', 'drugName': 'Abt-102', 'tradeNames_string': '', 'drugSynonyms_string': 'ABT-102, Abt-102', 'linkedDiseasesDrug_string': '', 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drugIsApproved': False, 'newLinkedTargets_string': 'TRPV1 (ENSG00000196689)', 'numberLinkedTargets': 1}]
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.338
Q17
What gene does the drug Tazemetostat target?
The drug Tazemetostat targets the gene EZH2.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1211', 'drugName': 'Tazemetostat', 'tradeNames_string': '', 'drugSynonyms_string': 'E-7438, E7438, EPZ-6438, EPZ6438, Tazemetostat', 'linkedDiseasesDrug_string': 'Multiple Myeloma (EFO_0001378), Non-Hodgkins Lymphoma (EFO_0005952), Follicular Lymphoma (MONDO_0018906), Small Cell Lung Carci...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1343
Q17
What gene does the drug Ocriplasmin target?
The drug Ocriplasmin targets 38 genes: LAMA1, LAMA3, LAMB4, COL2A1, LAMA4, LAMC1, COL28A1, COL6A2, COL18A1, COL11A2, COL4A1, COL6A6, COL15A1, COL4A5, LAMC3, LAMB3, COL5A3, COL6A3, COL4A3, COL24A1, COL4A6, COL4A4, COL1A1, LAMB1, LAMC2, COL4A2, COL6A5, COL27A1, COL11A1, FN1, COL1A2, COL3A1, COL5A1, LAMA2, LAMA5, COL6A1, ...
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5818', 'drugName': 'Ocriplasmin', 'tradeNames_string': '', 'drugSynonyms_string': 'Jetrea, MICROPLASMIN, Microplasmin (synthetic human), Ocriplasmin, Plasmin, micro- (synthetic human), Recombinant human microplasmin', 'linkedDiseasesDrug_string': 'Uveitis (EFO_1001231), Macular Degeneratio...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1593
Q17
What gene does the drug Masupirdine target?
The drug Masupirdine is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target the gene HTR6.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_4255', 'drugName': 'Masupirdine', 'tradeNames_string': '', 'drugSynonyms_string': 'Masupirdine, SUVN-502, Suvn-502', 'linkedDiseasesDrug_string': 'Alzheimer Disease (MONDO_0004975)', 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False, 'newLinkedTargets_string': '...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1993
Q17
What gene does the drug Dopamine Hydrochloride target?
The drug Dopamine Hydrochloride targets the gene ADRB1.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_4778', 'drugName': 'Dopamine Hydrochloride', 'tradeNames_string': 'Dopamin-Natterman, Dopamine hydrochloride, Dopmin, Dynatra, Intropin, Sabax Dopamin, Selectajet', 'drugSynonyms_string': 'ASL-279, Cardiosteril, Dopamine hcl, Dopamine hydrochloride, Dopamini hydrochloridum, Inotropin, NSC-...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.598
Q17
What gene does the drug Alisertib target?
The drug Alisertib is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target the gene AURKA.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1576', 'drugName': 'Alisertib', 'tradeNames_string': '', 'drugSynonyms_string': 'Alisertib, MLN 8237, MLN-8237, MLN8237, Mln-8237', 'linkedDiseasesDrug_string': 'Ovarian Carcinoma (EFO_0001075), Cancer (MONDO_0004992), Multiple Myeloma (EFO_0001378), Neuroblastoma (EFO_0000621), Burkitts L...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.16
Q17
What gene does the drug Afatinib target?
The drug Afatinib targets 3 genes: ERBB2, ERBB4 and EGFR.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2560', 'drugName': 'Afatinib Dimaleate', 'tradeNames_string': 'Gilotrif', 'drugSynonyms_string': 'Afatinib dimaleate, Afatinib maleate, BIBW-2992 MA2, BIBW-2992-MA2, BIBW-2992MA2, BIBW2992 MA2, BIBW2992-MA2', 'linkedDiseasesDrug_string': 'Multiple Myeloma (EFO_0001378), Non-Small Cell Lung...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1855
Q17
What gene does the drug Ozanimod Hydrochloride target?
The drug Ozanimod Hydrochloride targets the gene S1PR1.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5399', 'drugName': 'Ozanimod Hydrochloride', 'tradeNames_string': 'Zeposia', 'drugSynonyms_string': 'Ozanimod hydrochloride, RPC-1063 HCL, RPC1063 HCL', 'linkedDiseasesDrug_string': 'Multiple Sclerosis (MONDO_0005301)', 'yearOfFirstApproval': 2020, 'maxClinicalTrialPhase': 4, 'drugIsApprov...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1634
Q17
What gene does the drug Parecoxib Sodium target?
The drug Parecoxib Sodium targets the gene PTGS2.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2672', 'drugName': 'Parecoxib Sodium', 'tradeNames_string': 'Dynastat', 'drugSynonyms_string': 'Parecoxib sodium, Parecoxib sodium salt, SC-69124A', 'linkedDiseasesDrug_string': 'Pain (EFO_0003843), Osteoarthritis (MONDO_0005178)', 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'dru...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1686
Q17
What gene does the drug Inotuzumab target?
The drug Inotuzumab targets the gene CD22.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_6318', 'drugName': 'Inotuzumab Ozogamicin', 'tradeNames_string': 'Besponsa', 'drugSynonyms_string': 'CMC-544, Inotuzumab ozogamicin, PF-05208773, WAY-207294, WAY-207294 CMC-544', 'linkedDiseasesDrug_string': 'Non-Hodgkins Lymphoma (EFO_0005952), Follicular Lymphoma (MONDO_0018906), Neoplas...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.600
Q17
What gene does the drug Perhexiline Maleate target?
The drug Perhexiline Maleate targets 3 genes: CPT2, CPT1B and MTOR.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1724', 'drugName': 'Perhexiline Maleate', 'tradeNames_string': 'Pexid, Pexsig', 'drugSynonyms_string': 'NSC-758409, Perhexiline maleate, Perhexilinum', 'linkedDiseasesDrug_string': '', 'yearOfFirstApproval': 1974, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True, 'newLinkedTargets_string...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.924
Q17
What gene does the drug Tebentafusp target?
The drug Tebentafusp targets the gene PMEL.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5977', 'drugName': 'Tebentafusp', 'tradeNames_string': 'Kimmtrak', 'drugSynonyms_string': 'IMCGP-100, IMCGP100, IMCgp 100, IMMTAC IMCGP100, Imcgp100, ImmTAC IMCgpgp 100, Kimmtrak, Tebentafusp, Tebentafusp tebn, Tebentafusp-tebn', 'linkedDiseasesDrug_string': 'Melanoma (EFO_0000756), Uveal ...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.471
Q17
What gene does the drug Pitavastatin Sodium target?
The drug Pitavastatin Sodium targets the gene HMGCR.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1489', 'drugName': 'Pitavastatin Sodium', 'tradeNames_string': 'Nikita', 'drugSynonyms_string': 'Pitavastatin sodium', 'linkedDiseasesDrug_string': 'Abnormal Circulating Lipid Concentration (HP_0003119), Familial Hypercholesterolemia (EFO_0004911), Hyperlipidemia (MONDO_0021187), Hyperchol...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.202
Q17
What gene does the drug Icatibant target?
The drug Icatibant targets the gene BDKRB2.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_226', 'drugName': 'Icatibant Acetate', 'tradeNames_string': 'Firazyr', 'drugSynonyms_string': 'HOE 140, HOE-140, Icatibant acetate', 'linkedDiseasesDrug_string': 'Angioedema (EFO_0005532), Hereditary Angioedema (MONDO_0019623), Inflammation (MP_0001845), Covid-19 (MONDO_0100096)', 'yearOfF...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1206
Q17
What gene does the drug Methylprednisolone Hemisuccinate target?
The drug Methylprednisolone Hemisuccinate targets the gene NR3C1.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_670', 'drugName': 'Methylprednisolone Hemisuccinate', 'tradeNames_string': '', 'drugSynonyms_string': 'Methylprednisolone hemisuccinate, Methylprednisolone succinate', 'linkedDiseasesDrug_string': 'Multiple Myeloma (EFO_0001378), Non-Hodgkins Lymphoma (EFO_0005952), Chronic Lymphocytic Leu...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1056
Q17
What gene does the drug Mk-0893 target?
The drug Mk-0893 is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target the gene GCGR.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_4471', 'drugName': 'Mk-0893', 'tradeNames_string': '', 'drugSynonyms_string': 'MK-0893, Mk-0893, Mk0893', 'linkedDiseasesDrug_string': 'Type 2 Diabetes Mellitus (MONDO_0005148)', 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False, 'newLinkedTargets_string': 'GCGR...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1195
Q17
What gene does the drug Eltrombopag target?
The drug Eltrombopag targets the gene MPL.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2769', 'drugName': 'Eltrombopag Olamine', 'tradeNames_string': 'Promacta, Promacta kit', 'drugSynonyms_string': 'Eltrombopag (as olamine), Eltrombopag compd with 2-aminoethanol (1:2), Eltrombopag olamine, SB-497115-GR', 'linkedDiseasesDrug_string': 'Thrombocytopenia (HP_0001873), Autoimmun...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1300
Q17
What gene does the drug Gilteritinib Fumarate target?
The drug Gilteritinib Fumarate targets 2 genes: AXL and FLT3.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_3307', 'drugName': 'Gilteritinib Fumarate', 'tradeNames_string': 'Xospata', 'drugSynonyms_string': 'ASP-2215 HEMIFUMARATE, ASP2215 hemifumarate, Gilteritinib fumarate, Gilteritinib hemifumarate', 'linkedDiseasesDrug_string': 'Acute Myeloid Leukemia (EFO_0000222), Myeloid Leukemia (MONDO_00...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1276
Q17
What gene does the drug Lumacaftor target?
The drug Lumacaftor targets the gene CFTR.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1147', 'drugName': 'Lumacaftor', 'tradeNames_string': '', 'drugSynonyms_string': 'Lumacaftor, VRT 826809, VRT-826809, VX 809, VX-809', 'linkedDiseasesDrug_string': 'Liver Disease (EFO_0001421), Cystic Fibrosis (MONDO_0009061)', 'yearOfFirstApproval': 2015, 'maxClinicalTrialPhase': 4, 'drug...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1814
Q17
What gene does the drug Vorsetuzumab Mafodotin target?
The drug Vorsetuzumab Mafodotin is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target the gene CD70.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_4780', 'drugName': 'Vorsetuzumab Mafodotin', 'tradeNames_string': 'Sgn-75', 'drugSynonyms_string': 'SGN-75, Vorsetuzumab mafodotin', 'linkedDiseasesDrug_string': 'Renal Cell Carcinoma (EFO_0000681)', 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drugIsApproved': False, 'newLinkedT...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1402
Q17
What gene does the drug Potassium Oxybate target?
The drug Potassium Oxybate targets 2 genes: GABBR2 and GABBR1.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2573', 'drugName': 'Potassium Oxybate', 'tradeNames_string': '', 'drugSynonyms_string': 'Oxybate potassium, Potassium oxybate', 'linkedDiseasesDrug_string': '', 'yearOfFirstApproval': 2020, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True, 'newLinkedTargets_string': 'GABBR1 (ENSG00000204...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1807
Q17
What gene does the drug Isopropamide target?
The drug Isopropamide targets 2 genes: CHRM1 and CHRM3.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_3463', 'drugName': 'Isopropamide', 'tradeNames_string': '', 'drugSynonyms_string': 'Isopropamide, Isopropamide cation, Isopropamide ion', 'linkedDiseasesDrug_string': 'Gastrointestinal Disease (EFO_0010282)', 'yearOfFirstApproval': 1957, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True, ...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.661
Q17
What gene does the drug Budesonide target?
The drug Budesonide targets the gene NR3C1.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_3329', 'drugName': 'Budesonide', 'tradeNames_string': 'Aircort, Budeflam aquanase, Budelin novolizer, Budenofalk, Budesonide, Cortiment, Duoresp spiromax, Entocort, Entocort cr, Entocort ec, Ortikos, Preferid, Pulmaxan, Pulmicort, Pulmicort flexhaler, Pulmicort l.s., Pulmicort respules, Rh...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.560
Q17
What gene does the drug Pl-3994 target?
The drug Pl-3994 is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target the gene NPR1.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_478', 'drugName': 'Pl-3994', 'tradeNames_string': '', 'drugSynonyms_string': 'Pl-3994', 'linkedDiseasesDrug_string': 'Heart Failure (EFO_0003144), Asthma (MONDO_0004979)', 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False, 'newLinkedTargets_string': 'NPR1 (ENSG0...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.44
Q17
What gene does the drug Phenylephrine Hydrochloride target?
The drug Phenylephrine Hydrochloride targets 3 genes: ADRA1D, ADRA1B and ADRA1A.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_3941', 'drugName': 'Phenylephrine Hydrochloride', 'tradeNames_string': 'Afrin 4 hour nasal spray, Biomydrin, Biorphen, Fenilfar, Fenox, Mydfrin, Nazex, Neo-synephrine, Neosynephrine, Nostril, Nurofen sinus pain relief, Phenylephrine hydrochloride, Prefrin, Vazculep', 'drugSynonyms_string':...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.278
Q17
What gene does the drug Avanafil target?
The drug Avanafil targets the gene PDE5A.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5497', 'drugName': 'Avanafil', 'tradeNames_string': 'Spedra, Stendra', 'drugSynonyms_string': 'Avanafil, TA-1790', 'linkedDiseasesDrug_string': 'Kidney Disease (EFO_0003086), Erectile Dysfunction (EFO_0004234)', 'yearOfFirstApproval': 2011, 'maxClinicalTrialPhase': 4, 'drugIsApproved': Tru...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.1096
Q17
What gene does the drug Navafenterol target?
The drug Navafenterol is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 2 genes: CHRM3 and ADRB2
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_6388', 'drugName': 'Navafenterol', 'tradeNames_string': '', 'drugSynonyms_string': 'AZD-8871, AZD8871, Azd 8871, Azd-8871, Azd8871, LAS-191351, LAS191351, Navafenterol', 'linkedDiseasesDrug_string': 'Chronic Obstructive Pulmonary Disease (EFO_0000341)', 'yearOfFirstApproval': 0, 'maxClinic...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.104
Q17
What gene does the drug Bempedoic Acid target?
The drug Bempedoic Acid targets the gene ACLY.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5953', 'drugName': 'Bempedoic Acid', 'tradeNames_string': 'Nexletol', 'drugSynonyms_string': 'Bempedoic acid, ESP-55016, ETC-1002, ETC1002', 'linkedDiseasesDrug_string': 'Hyperlipidemia (MONDO_0021187), Coronary Artery Disease (EFO_0001645), Familial Hypercholesterolemia (EFO_0004911), Car...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.856
Q17
What gene does the drug Pyrovalerone target?
The drug Pyrovalerone targets 2 genes: SLC6A2 and SLC6A3.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_225', 'drugName': 'Pyrovalerone', 'tradeNames_string': '', 'drugSynonyms_string': 'J8.659B, Pyrovalerone', 'linkedDiseasesDrug_string': '', 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True, 'newLinkedTargets_string': 'SLC6A3 (ENSG00000142319), SLC6A2 (ENSG000001...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.985
Q17
What gene does the drug Alectinib target?
The drug Alectinib targets 3 genes: EML4, ALK and RET.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1251', 'drugName': 'Alectinib Hydrochloride', 'tradeNames_string': 'Alecensa', 'drugSynonyms_string': 'Alectinib hydrochloride', 'linkedDiseasesDrug_string': 'Non-Small Cell Lung Carcinoma (EFO_0003060)', 'yearOfFirstApproval': 2015, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True, 'new...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status
Q17.948
Q17
What gene does the drug Linerixibat target?
The drug Linerixibat is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target the gene SLC10A2.
SELECT DISTINCT UUID, drugName, tradeNames_string, drugSynonyms_string, linkedDiseasesDrug_string, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved, newLinkedTargets_string, numberLinkedTargets FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1185', 'drugName': 'Linerixibat', 'tradeNames_string': '', 'drugSynonyms_string': 'GSK2330672, Gsk-2330672, Gsk2330672, Linerixibat', 'linkedDiseasesDrug_string': 'Type 2 Diabetes Mellitus (MONDO_0005148), Pruritus (HP_0000989), Cholestasis (MONDO_0001751), Intrahepatic Cholestasis (MONDO_...
general
Distinct, Similarity Search, Order By
Genetic Target, Approval Status