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Q4.1132
Q4
What drugs target the gene PRKAG2?
There are no approved drugs targeting PRKAG2, but the drug Acadesine, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PRKAG2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5888', 'drugName': 'Acadesine', 'newLinkedTargets_string': 'PRKAA2 (ENSG00000162409), PRKAB2 (ENSG00000131791), PRKAG1 (ENSG00000181929), PRKAG2 (ENSG00000106617), PRKAB1 (ENSG00000111725), PRKAA1 (ENSG00000132356), PRKAG3 (ENSG00000115592)', 'drugIsApproved': False, 'maxClinicalTrialPhase...
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Q4.1171
Q4
What drugs target the gene PSMC2?
The drugs that target PSMC2 are Bortezomib, Carfilzomib, Ixazomib, and Ixazomib Citrate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PSMC2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_559', 'drugName': 'Bortezomib', 'newLinkedTargets_string': 'PSMD1 (ENSG00000173692), PSMB2 (ENSG00000126067), PSMB1 (ENSG00000008018), PSMB5 (ENSG00000100804), PSMB8 (ENSG00000204264), PSMB9 (ENSG00000240065), PSMB6 (ENSG00000142507), PSMD14 (ENSG00000115233), PSMA1 (ENSG00000129084), PSMA...
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Q4.658
Q4
What drugs target the gene IFNGR2?
The drug that targets IFNGR2 is Interferon Gamma-1B.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%IFNGR2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3679', 'drugName': 'Interferon Gamma-1B', 'newLinkedTargets_string': 'IFNGR2 (ENSG00000159128), IFNGR1 (ENSG00000027697)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}]
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Q4.984
Q4
What drugs target the gene NLRP3?
There are no approved drugs targeting NLRP3, but the drug Dapansutrile, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NLRP3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1186', 'drugName': 'Dapansutrile', 'newLinkedTargets_string': 'NLRP3 (ENSG00000162711)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
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Q4.1032
Q4
What drugs target the gene P4HTM?
The drug that targets P4HTM is Roxadustat.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%P4HTM %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5393', 'drugName': 'Roxadustat', 'newLinkedTargets_string': 'EGLN2 (ENSG00000269858), P4HTM (ENSG00000178467), EGLN1 (ENSG00000135766), EGLN3 (ENSG00000129521)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2677', 'drugName': 'Daprodustat', 'newLinkedTa...
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Q4.241
Q4
What drugs target the gene CDK2?
There are no FDA approved drugs targeting the gene CDK2. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Dinaciclib, Zotiraciclib, Bms-387032, Roniciclib, Ag-24322, Pha-793887, Azd-5438, At-7519, Su-9516, Rg-547, Ucn-01, Rgb-286638, Alvocidib, Milciclib,...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CDK2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_46', 'drugName': 'Dinaciclib', 'newLinkedTargets_string': 'CDK5 (ENSG00000164885), CDK1 (ENSG00000170312), CDK9 (ENSG00000136807), CDK2 (ENSG00000123374)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_48', 'drugName': 'Dinaciclib', 'newLinkedTargets_st...
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Q4.1234
Q4
What drugs target the gene RPL13A?
The drug that targets RPL13A is Ataluren.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RPL13A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG00000083845), RPS7 (ENSG...
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Q4.363
Q4
What drugs target the gene DKK1?
There are no FDA approved drugs targeting the gene DKK1. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Bhq-880 and Dkn-01.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%DKK1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_643', 'drugName': 'Bhq-880', 'newLinkedTargets_string': 'DKK1 (ENSG00000107984)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_5287', 'drugName': 'Dkn-01', 'newLinkedTargets_string': 'DKK1 (ENSG00000107984)', 'drugIsApproved': False, 'maxClinicalTrialP...
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Q4.489
Q4
What drugs target the gene FZD8?
There are no FDA approved drugs targeting the gene FZD8. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Vantictumab and Ipafricept.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%FZD8 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5829', 'drugName': 'Vantictumab', 'newLinkedTargets_string': 'FZD2 (ENSG00000180340), FZD7 (ENSG00000155760), FZD1 (ENSG00000157240), FZD5 (ENSG00000163251), FZD8 (ENSG00000177283)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 1}, {'UUID': 'DrugGeneTargets_v2_5825', 'drugName': 'Vant...
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Q4.497
Q4
What drugs target the gene GABRA5?
The drugs that target GABRA5 are Meprobamate, Acamprosate Calcium, Enflurane, Methohexital, Metharbital, Butabarbital, Flurazepam Hydrochloride, Pentobarbital Sodium, Acamprosate, Primidone, Temazepam, Flunitrazepam, Ganaxolone, Diazepam, Methyprylon, Thiopental, Clonazepam, Topiramate, Remimazolam Besylate, Brexanolon...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%GABRA5 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1108', 'drugName': 'Temazepam', 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089), GABRA3 (ENSG00000011677), GABRP (ENSG00000094755)...
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Q4.369
Q4
What drugs target the gene DNPEP?
There are no approved drugs targeting DNPEP, but the drug Tosedostat, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%DNPEP %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_582', 'drugName': 'Tosedostat', 'newLinkedTargets_string': 'ANPEP (ENSG00000166825), NPEPPS (ENSG00000141279), RNPEP (ENSG00000176393), METAP1 (ENSG00000164024), LNPEP (ENSG00000113441), DNPEP (ENSG00000123992), ENPEP (ENSG00000138792), XPNPEP1 (ENSG00000108039), LAP3 (ENSG00000002549), ME...
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Q4.1096
Q4
What drugs target the gene PLK4?
There are no FDA approved drugs targeting the gene PLK4. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Cfi-400945 and Rg-1530.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PLK4 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_648', 'drugName': 'Cfi-400945', 'newLinkedTargets_string': 'PLK4 (ENSG00000142731)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_5521', 'drugName': 'Cfi-400945', 'newLinkedTargets_string': 'PLK4 (ENSG00000142731)', 'drugIsApproved': False, 'maxClinica...
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Q4.1328
Q4
What drugs target the gene S1PR4?
The drugs that target S1PR4 are Fingolimod Hydrochloride, Fingolimod, and Fingolimod Lauryl Sulfate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%S1PR4 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5906', 'drugName': 'Fingolimod Lauryl Sulfate', 'newLinkedTargets_string': 'S1PR5 (ENSG00000180739), S1PR2 (ENSG00000267534), S1PR4 (ENSG00000125910), S1PR3 (ENSG00000213694), S1PR1 (ENSG00000170989)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4765',...
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Q4.30
Q4
What drugs target the gene ADORA2B?
The drugs that target ADORA2B are Theophylline Sodium Glycinate, Adenosine, Theophylline Glycinate, Oxtriphylline, Pentoxifylline, Theophylline, Caffeine, Aminophylline, Caffeine, and Citrated.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ADORA2B %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2664', 'drugName': 'Theophylline Glycinate', 'newLinkedTargets_string': 'ADORA1 (ENSG00000163485), ADORA2B (ENSG00000170425), ADORA3 (ENSG00000282608), ADORA2A (ENSG00000128271), PDE4A (ENSG00000065989), PDE4D (ENSG00000113448), PDE4B (ENSG00000184588), PDE4C (ENSG00000105650), PDE3A (ENSG...
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Q4.1033
Q4
What drugs target the gene PAH?
The drugs that target PAH are Sapropterin and Sapropterin Dihydrochloride.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PAH %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_636', 'drugName': 'Sapropterin', 'newLinkedTargets_string': 'PAH (ENSG00000171759)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4864', 'drugName': 'Sapropterin Dihydrochloride', 'newLinkedTargets_string': 'PAH (ENSG00000171759)', 'drugIsApproved': Tru...
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Q4.928
Q4
What drugs target the gene MYL7?
The drug that targets MYL7 is Mavacamten.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%MYL7 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1036', 'drugName': 'Mavacamten', 'newLinkedTargets_string': 'MYH7 (ENSG00000092054), MYH6 (ENSG00000197616), MYH7B (ENSG00000078814), MYL3 (ENSG00000160808), MYL2 (ENSG00000111245), MYL7 (ENSG00000106631), MYL4 (ENSG00000198336)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID...
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Q4.824
Q4
What drugs target the gene LIPF?
The drug that targets LIPF is Orlistat.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%LIPF %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1666', 'drugName': 'Orlistat', 'newLinkedTargets_string': 'LIPF (ENSG00000182333), PNLIP (ENSG00000175535)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1667', 'drugName': 'Orlistat', 'newLinkedTargets_string': 'LIPF (ENSG00000182333), PNLIP (ENSG00000...
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Q4.1437
Q4
What drugs target the gene TLR7?
The drugs that target TLR7 are Hydroxychloroquine, Imiquimod, and Hydroxychloroquine Sulfate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TLR7 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1394', 'drugName': 'Imiquimod', 'newLinkedTargets_string': 'TLR7 (ENSG00000196664)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3879', 'drugName': 'Hydroxychloroquine Sulfate', 'newLinkedTargets_string': 'TLR9 (ENSG00000239732), TLR7 (ENSG00000196664)...
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Q4.66
Q4
What drugs target the gene AOC1?
The drug that targets AOC1 is Proxibarbal.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%AOC1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_472', 'drugName': 'Proxibarbal', 'newLinkedTargets_string': 'AOC1 (ENSG00000002726), MAOA (ENSG00000189221)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_473', 'drugName': 'Proxibarbal', 'newLinkedTargets_string': 'AOC1 (ENSG00000002726), MAOA (ENSG000...
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Q4.1150
Q4
What drugs target the gene PSENEN?
There are no FDA approved drugs targeting the gene PSENEN. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Tarenflurbil, Rg-4733, Nirogacestat, Avagacestat, Begacestat, and Semagacestat.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PSENEN %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5562', 'drugName': 'Nirogacestat', 'newLinkedTargets_string': 'APH1A (ENSG00000117362), PSENEN (ENSG00000205155), APH1B (ENSG00000138613), PSEN1 (ENSG00000080815), NCSTN (ENSG00000162736), PSEN2 (ENSG00000143801)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTar...
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Q4.305
Q4
What drugs target the gene COL6A1?
The drugs that target COL6A1 are Collagenase Clostridium Histolyticum and Ocriplasmin.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%COL6A1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5818', 'drugName': 'Ocriplasmin', 'newLinkedTargets_string': 'FN1 (ENSG00000115414), COL1A2 (ENSG00000164692), COL1A1 (ENSG00000108821), COL2A1 (ENSG00000139219), COL3A1 (ENSG00000168542), COL4A1 (ENSG00000187498), COL5A1 (ENSG00000130635), COL6A1 (ENSG00000142156), COL11A1 (ENSG0000006071...
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Q4.464
Q4
What drugs target the gene FGFR1?
The drugs that target FGFR1 are Pazopanib Hydrochloride, Regorafenib, Infigratinib, Infigratinib Phosphate, Pemigatinib, Nintedanib Esylate, Pazopanib, Erdafitinib, Nintedanib, and Futibatinib.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%FGFR1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_391', 'drugName': 'Pazopanib Hydrochloride', 'newLinkedTargets_string': 'FGFR1 (ENSG00000077782), FGFR3 (ENSG00000068078), KIT (ENSG00000157404), CSF1R (ENSG00000182578), FLT1 (ENSG00000102755), FLT4 (ENSG00000037280), KDR (ENSG00000128052), ITK (ENSG00000113263), PDGFRB (ENSG00000113721),...
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Q4.1225
Q4
What drugs target the gene ROR1?
There are no approved drugs targeting ROR1, but the drug Cirmtuzumab, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ROR1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5735', 'drugName': 'Cirmtuzumab', 'newLinkedTargets_string': 'ROR1 (ENSG00000185483)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}]
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Q4.654
Q4
What drugs target the gene IFNAR2?
The drugs that target IFNAR2 are Interferon Alfa-N3, Interferon Beta-1A, Peginterferon Alfa-2B, Peginterferon Alfa-2A, Interferon Alfacon-1, Interferon Alfa-2B, Interferon Alfa-2A, Peginterferon Beta-1A, Interferon Beta-1B, and Ropeginterferon Alfa-2B.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%IFNAR2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_635', 'drugName': 'Interferon Beta-1A', 'newLinkedTargets_string': 'IFNAR1 (ENSG00000142166), IFNAR2 (ENSG00000159110)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5120', 'drugName': 'Interferon Beta-1B', 'newLinkedTargets_string': 'IFNAR1 (ENSG000001...
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Q4.143
Q4
What drugs target the gene CACNA1B?
The drugs that target CACNA1B are Gabapentin, Levetiracetam, Terodiline Hydrochloride, Phloroglucinol, Suloctidil, Ziconotide, Pregabalin, Gabapentin Enacarbil, Bepridil Hydrochloride, Ziconotide Acetate, Bepridil, and Terodiline.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CACNA1B %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6292', 'drugName': 'Terodiline', 'newLinkedTargets_string': 'CHRM3 (ENSG00000133019), CHRM4 (ENSG00000180720), CHRM1 (ENSG00000168539), CHRM2 (ENSG00000181072), CHRM5 (ENSG00000184984), CACNA1H (ENSG00000196557), CACNA2D1 (ENSG00000153956), CACNA1C (ENSG00000151067), CACNA2D3 (ENSG00000157...
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Q4.579
Q4
What drugs target the gene HCRTR2?
The drugs that target HCRTR2 are Lemborexant, Daridorexant, Daridorexant Hydrochloride, and Suvorexant.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%HCRTR2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4413', 'drugName': 'Daridorexant', 'newLinkedTargets_string': 'HCRTR1 (ENSG00000121764), HCRTR2 (ENSG00000137252)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4411', 'drugName': 'Daridorexant', 'newLinkedTargets_string': 'HCRTR1 (ENSG00000121764), HCR...
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Q4.949
Q4
What drugs target the gene NDUFAB1?
The drugs that target NDUFAB1 are Metformin and Metformin Hydrochloride.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NDUFAB1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (ENSG00000165264), NDUFA4 (...
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Q4.563
Q4
What drugs target the gene GUCY1A1?
The drugs that target GUCY1A1 are Pentaerythritol Tetranitrate, Isosorbide Dinitrate, Nitroprusside, Nitroglycerin, Vericiguat, Isosorbide Mononitrate, Nitric Oxide, Sodium Nitroprusside, and Riociguat.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%GUCY1A1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2605', 'drugName': 'Vericiguat', 'newLinkedTargets_string': 'GUCY1B1 (ENSG00000061918), GUCY1B2 (ENSG00000123201), GUCY1A2 (ENSG00000152402), GUCY1A1 (ENSG00000164116)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1208', 'drugName': 'Nitroprusside', 'n...
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Genetic Target
Q4.726
Q4
What drugs target the gene ITGB6?
There are no FDA approved drugs targeting the gene ITGB6. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Stx-100 and Abituzumab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ITGB6 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1969', 'drugName': 'Abituzumab', 'newLinkedTargets_string': 'ITGAV (ENSG00000138448), ITGB6 (ENSG00000115221), ITGB5 (ENSG00000082781), ITGB3 (ENSG00000259207), ITGB1 (ENSG00000150093), ITGB8 (ENSG00000105855)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTarget...
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Genetic Target
Q4.277
Q4
What drugs target the gene CHRNG?
The drugs that target CHRNG are Pipecuronium, Decamethonium, Vecuronium, Rocuronium, Metocurine Iodide, Succinylcholine Chloride, Tubocurarine, Rocuronium Bromide, Cisatracurium, Cisatracurium Besylate, Mivacurium Chloride, Pancuronium, Gallamine, Vecuronium Bromide, Gallamine Triethiodide, Metocurine, Atracurium Besyl...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CHRNG %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2723', 'drugName': 'Succinylcholine Chloride', 'newLinkedTargets_string': 'CHRNA1 (ENSG00000138435), CHRNG (ENSG00000196811), CHRNB1 (ENSG00000170175), CHRND (ENSG00000135902), CHRNE (ENSG00000108556)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_922',...
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Genetic Target
Q4.611
Q4
What drugs target the gene HSPA1A?
There are no approved drugs targeting HSPA1A, but the drug Cd24Fc, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%HSPA1A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5250', 'drugName': 'Cd24Fc', 'newLinkedTargets_string': 'HSP90AA1 (ENSG00000080824), HSP90AB1 (ENSG00000096384), SIGLEC10 (ENSG00000142512), HMGB1 (ENSG00000189403), HSPA1A (ENSG00000204389), HSPA1B (ENSG00000204388)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGen...
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Genetic Target
Q4.1528
Q4
What drugs target the gene VIM?
There are no approved drugs targeting VIM, but the drug Pritumumab, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%VIM %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_551', 'drugName': 'Pritumumab', 'newLinkedTargets_string': 'VIM (ENSG00000026025)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 1}]
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Genetic Target
Q4.1269
Q4
What drugs target the gene RPL7A?
The drug that targets RPL7A is Ataluren.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RPL7A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG00000083845), RPS7 (ENSG...
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Genetic Target
Q4.777
Q4
What drugs target the gene KCNQ3?
The drugs that target KCNQ3 are Dalfampridine, Guanidine, Amifampridine Phosphate, Ezogabine, Guanidine Hydrochloride, and Amifampridine.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%KCNQ3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3665', 'drugName': 'Ezogabine', 'newLinkedTargets_string': 'KCNQ1 (ENSG00000053918), KCNQ2 (ENSG00000075043), KCNQ3 (ENSG00000184156), KCNQ5 (ENSG00000185760), KCNQ4 (ENSG00000117013)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5420', 'drugName': 'Am...
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Genetic Target
Q4.1142
Q4
What drugs target the gene PRKCZ?
The drug that targets PRKCZ is Midostaurin.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PRKCZ %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5666', 'drugName': 'Midostaurin', 'newLinkedTargets_string': 'KIT (ENSG00000157404), KDR (ENSG00000128052), PDGFRB (ENSG00000113721), PDGFRA (ENSG00000134853), FLT3 (ENSG00000122025), PRKD3 (ENSG00000115825), PRKCI (ENSG00000163558), PRKCA (ENSG00000154229), PRKCG (ENSG00000126583), PRKCD ...
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Genetic Target
Q4.1047
Q4
What drugs target the gene PDE3B?
The drugs that target PDE3B are Anagrelide Hydrochloride, Theophylline Sodium Glycinate, Theophylline Glycinate, Enoximone, Oxtriphylline, Pentoxifylline, Anagrelide, Theophylline, Aminophylline, and Dipyridamole.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PDE3B %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5470', 'drugName': 'Aminophylline', 'newLinkedTargets_string': 'PDE4A (ENSG00000065989), PDE4D (ENSG00000113448), PDE4B (ENSG00000184588), PDE4C (ENSG00000105650), PDE3A (ENSG00000172572), PDE3B (ENSG00000152270), ADORA1 (ENSG00000163485), ADORA2B (ENSG00000170425), ADORA3 (ENSG00000282608...
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Genetic Target
Q4.1054
Q4
What drugs target the gene PDE6B?
The drugs that target PDE6B are Pentoxifylline and Dipyridamole.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PDE6B %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6107', 'drugName': 'Dipyridamole', 'newLinkedTargets_string': 'PDE5A (ENSG00000138735), PDE4A (ENSG00000065989), PDE3A (ENSG00000172572), PDE6H (ENSG00000139053), PDE6G (ENSG00000185527), PDE2A (ENSG00000186642), PDE7A (ENSG00000205268), PDE1A (ENSG00000115252), PDE9A (ENSG00000160191), PD...
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Genetic Target
Q4.1006
Q4
What drugs target the gene NR1H3?
There are no FDA approved drugs targeting the gene NR1H3. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Cs-8080, Bms-852927, Rovazolac, Lxr-623, Abequolixron, and Hyodeoxycholic_Acid.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NR1H3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_132', 'drugName': 'Rovazolac', 'newLinkedTargets_string': 'NR1H3 (ENSG00000025434), NR1H2 (ENSG00000131408)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_19', 'drugName': 'Cs-8080', 'newLinkedTargets_string': 'NR1H2 (ENSG00000131408), NR1H3 (ENSG00000...
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Genetic Target
Q4.45
Q4
What drugs target the gene AGTR1?
The drugs that target AGTR1 are Irbesartan, Azilsartan Kamedoxomil, Losartan Potassium, Olmesartan Medoxomil, Candesartan Cilexetil, Angiotensin Ii, Angiotensin Ii Acetate, Saralasin, Telmisartan, Valsartan, Saralasin Acetate, Azilsartan Medoxomil, Eprosartan Mesylate, Eprosartan, and Losartan.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%AGTR1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4486', 'drugName': 'Valsartan', 'newLinkedTargets_string': 'AGTR1 (ENSG00000144891)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2579', 'drugName': 'Candesartan Cilexetil', 'newLinkedTargets_string': 'AGTR1 (ENSG00000144891)', 'drugIsApproved': True, ...
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Genetic Target
Q4.1281
Q4
What drugs target the gene RPS16?
The drug that targets RPS16 is Ataluren.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RPS16 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG00000083845), RPS7 (ENSG...
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Genetic Target
Q4.272
Q4
What drugs target the gene CHRNB1?
The drugs that target CHRNB1 are Pipecuronium, Decamethonium, Vecuronium, Rocuronium, Metocurine Iodide, Succinylcholine Chloride, Tubocurarine, Rocuronium Bromide, Cisatracurium, Cisatracurium Besylate, Mivacurium Chloride, Pancuronium, Gallamine, Vecuronium Bromide, Gallamine Triethiodide, Metocurine, Atracurium Besy...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CHRNB1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2723', 'drugName': 'Succinylcholine Chloride', 'newLinkedTargets_string': 'CHRNA1 (ENSG00000138435), CHRNG (ENSG00000196811), CHRNB1 (ENSG00000170175), CHRND (ENSG00000135902), CHRNE (ENSG00000108556)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_922',...
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Genetic Target
Q4.1159
Q4
What drugs target the gene PSMB1?
The drugs that target PSMB1 are Bortezomib, Carfilzomib, Ixazomib, and Ixazomib Citrate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PSMB1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3334', 'drugName': 'Ixazomib', 'newLinkedTargets_string': 'PSMD1 (ENSG00000173692), PSMB2 (ENSG00000126067), PSMB1 (ENSG00000008018), PSMB5 (ENSG00000100804), PSMB8 (ENSG00000204264), PSMB9 (ENSG00000240065), PSMB6 (ENSG00000142507), PSMD14 (ENSG00000115233), PSMA1 (ENSG00000129084), PSMA2...
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Genetic Target
Q4.769
Q4
What drugs target the gene KCNK18?
The drugs that target KCNK18 are Enflurane, Sevoflurane, Desflurane, Halothane, and Isoflurane.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%KCNK18 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5599', 'drugName': 'Isoflurane', 'newLinkedTargets_string': 'KCNK10 (ENSG00000100433), KCNK9 (ENSG00000169427), GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089...
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Genetic Target
Q4.117
Q4
What drugs target the gene BMP10?
There are no approved drugs targeting BMP10, but the drug Dalantercept, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%BMP10 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_887', 'drugName': 'Dalantercept', 'newLinkedTargets_string': 'GDF2 (ENSG00000263761), BMP10 (ENSG00000163217)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_888', 'drugName': 'Dalantercept', 'newLinkedTargets_string': 'GDF2 (ENSG00000263761), BMP10 (EN...
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Genetic Target
Q4.311
Q4
What drugs target the gene CPS1?
The drug that targets CPS1 is Carglumic Acid.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CPS1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4749', 'drugName': 'Carglumic Acid', 'newLinkedTargets_string': 'CPS1 (ENSG00000021826)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}]
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Genetic Target
Q4.1000
Q4
What drugs target the gene NPR3?
There are no approved drugs targeting NPR3, but the drug Carperitide, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NPR3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2532', 'drugName': 'Carperitide', 'newLinkedTargets_string': 'NPR2 (ENSG00000159899), NPR1 (ENSG00000169418), NPR3 (ENSG00000113389)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}]
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Q4.793
Q4
What drugs target the gene KIR3DL2?
There are no approved drugs targeting KIR3DL2, but the drug Lacutamab, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%KIR3DL2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3590', 'drugName': 'Lacutamab', 'newLinkedTargets_string': 'KIR3DL2 (ENSG00000240403)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
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Genetic Target
Q4.617
Q4
What drugs target the gene HTR1D?
The drugs that target HTR1D are Fenfluramine, Zimeldine, Rizatriptan Benzoate, Amisulpride, Sumatriptan Succinate, Eletriptan, Almotriptan, Dexfenfluramine, Ergotamine Tartrate, Almotriptan Malate, Frovatriptan, Ergotamine, Dexfenfluramine Hydrochloride, Fenfluramine Hydrochloride, Eletriptan Hydrobromide, Frovatriptan...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%HTR1D %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4362', 'drugName': 'Frovatriptan Succinate', 'newLinkedTargets_string': 'HTR1B (ENSG00000135312), HTR1D (ENSG00000179546)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_6077', 'drugName': 'Sumatriptan', 'newLinkedTargets_string': 'HTR1D (ENSG00000179546...
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Genetic Target
Q4.430
Q4
What drugs target the gene ESR1?
The drugs that target ESR1 are Estriol, Estradiol Cypionate, Toremifene, Allylestrenol, Bazedoxifene Acetate, Cyclofenil, Mestranol, Toremifene Citrate, Estrone Sulfuric Acid, Estropipate, Clomiphene, Ospemifene, Estrogens, Esterified, Estradiol Acetate, Estrone, Tamoxifen, Quinestrol, Diethylstilbestrol Diphosphate, ...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ESR1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5776', 'drugName': 'Ethinyl Estradiol', 'newLinkedTargets_string': 'ESR1 (ENSG00000091831)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3573', 'drugName': 'Estrone', 'newLinkedTargets_string': 'ESR1 (ENSG00000091831)', 'drugIsApproved': True, 'maxClin...
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Genetic Target
Q4.1274
Q4
What drugs target the gene RPS10?
The drug that targets RPS10 is Ataluren.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RPS10 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG00000083845), RPS7 (ENSG...
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Genetic Target
Q4.1357
Q4
What drugs target the gene SIRT1?
There are no FDA approved drugs targeting the gene SIRT1. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Ex-527 and Srt-2104.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%SIRT1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2060', 'drugName': 'Srt-2104', 'newLinkedTargets_string': 'SIRT1 (ENSG00000096717)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_2011', 'drugName': 'Ex-527', 'newLinkedTargets_string': 'SIRT1 (ENSG00000096717)', 'drugIsApproved': False, 'maxClinicalTr...
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Genetic Target
Q4.80
Q4
What drugs target the gene ATP1A1?
The drugs that target ATP1A1 are Acetyldigitoxin, Deslanoside, Digoxin, Lanatoside C, and Digitoxin.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ATP1A1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2499', 'drugName': 'Digoxin', 'newLinkedTargets_string': 'ATP1A1 (ENSG00000163399), ATP1B2 (ENSG00000129244), ATP1B1 (ENSG00000143153), ATP1A2 (ENSG00000018625), ATP1B3 (ENSG00000069849), ATP1A3 (ENSG00000105409), ATP1A4 (ENSG00000132681), FXYD2 (ENSG00000137731)', 'drugIsApproved': True, ...
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Genetic Target
Q4.989
Q4
What drugs target the gene NOTCH1?
There are no approved drugs targeting NOTCH1, but the drug Brontictuzumab, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NOTCH1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3524', 'drugName': 'Brontictuzumab', 'newLinkedTargets_string': 'NOTCH1 (ENSG00000148400)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 1}]
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Q4.1418
Q4
What drugs target the gene TEK?
The drugs that target TEK are Regorafenib and Vandetanib.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TEK %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1934', 'drugName': 'Vandetanib', 'newLinkedTargets_string': 'TEK (ENSG00000120156), ERBB2 (ENSG00000141736), EGFR (ENSG00000146648), ERBB4 (ENSG00000178568), ERBB3 (ENSG00000065361), EPHA2 (ENSG00000142627), EPHB2 (ENSG00000133216), EPHA5 (ENSG00000145242), EPHA4 (ENSG00000116106), EPHA8 (...
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Genetic Target
Q4.963
Q4
What drugs target the gene NDUFB8?
The drugs that target NDUFB8 are Metformin and Metformin Hydrochloride.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NDUFB8 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (ENSG00000165264), NDUFA4 (...
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Genetic Target
Q4.1084
Q4
What drugs target the gene PIM1?
There are no FDA approved drugs targeting the gene PIM1. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Sgi-1776, Azd-1208, and Lgh-447.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PIM1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_295', 'drugName': 'Sgi-1776', 'newLinkedTargets_string': 'PIM1 (ENSG00000137193), PIM2 (ENSG00000102096), PIM3 (ENSG00000198355)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 1}, {'UUID': 'DrugGeneTargets_v2_3068', 'drugName': 'Azd-1208', 'newLinkedTargets_string': 'PIM1 (ENSG0000013...
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Genetic Target
Q4.318
Q4
What drugs target the gene CRIPTO?
There are no approved drugs targeting CRIPTO, but the drug Biib-015, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CRIPTO %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5970', 'drugName': 'Biib-015', 'newLinkedTargets_string': 'CRIPTO (ENSG00000241186)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 1}]
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Genetic Target
Q4.279
Q4
What drugs target the gene CLDN18?
There are no approved drugs targeting CLDN18, but the drug Zolbetuximab, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CLDN18 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3305', 'drugName': 'Zolbetuximab', 'newLinkedTargets_string': 'CLDN18 (ENSG00000066405)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}]
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Genetic Target
Q4.16
Q4
What drugs target the gene ACVRL1?
There are no FDA approved drugs targeting the gene ACVRL1. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Ascrinvacumab and Panulisib.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ACVRL1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_526', 'drugName': 'Ascrinvacumab', 'newLinkedTargets_string': 'ACVRL1 (ENSG00000139567)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_2427', 'drugName': 'Panulisib', 'newLinkedTargets_string': 'ACVRL1 (ENSG00000139567), MTOR (ENSG00000198793), PIK3R1 ...
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Genetic Target
Q4.582
Q4
What drugs target the gene HDAC11?
The drugs that target HDAC11 are Belinostat, Panobinostat, Panobinostat Lactate, and Romidepsin.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%HDAC11 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6063', 'drugName': 'Romidepsin', 'newLinkedTargets_string': 'HDAC1 (ENSG00000116478), HDAC3 (ENSG00000171720), HDAC6 (ENSG00000094631), HDAC2 (ENSG00000196591), HDAC5 (ENSG00000108840), HDAC7 (ENSG00000061273), HDAC8 (ENSG00000147099), HDAC11 (ENSG00000163517), HDAC4 (ENSG00000068024), HDA...
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Genetic Target
Q4.376
Q4
What drugs target the gene DRD4?
The drugs that target DRD4 are Promazine Hydrochloride, Haloperidol Decanoate, Loxapine Succinate, Bromocriptine, Levomepromazine, Pramipexole, Droperidol, Ropinirole, Olanzapine Pamoate, Ropinirole Hydrochloride, Rotigotine, Amoxapine, Clothiapine, Olanzapine, Chlorpromazine Hydrochloride, Chlorpromazine, Pimozide, Ap...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%DRD4 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5162', 'drugName': 'Haloperidol Lactate', 'newLinkedTargets_string': 'HTR2A (ENSG00000102468), DRD2 (ENSG00000149295), DRD3 (ENSG00000151577), DRD4 (ENSG00000069696)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3300', 'drugName': 'Apomorphine Hydrochl...
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Genetic Target
Q4.177
Q4
What drugs target the gene CASP2?
There are no approved drugs targeting CASP2, but the drug Emricasan, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CASP2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_45', 'drugName': 'Emricasan', 'newLinkedTargets_string': 'CASP4 (ENSG00000196954), CASP9 (ENSG00000132906), CASP3 (ENSG00000164305), CASP5 (ENSG00000137757), CASP6 (ENSG00000138794), CASP7 (ENSG00000165806), CASP8 (ENSG00000064012), CASP1 (ENSG00000137752), CASP2 (ENSG00000106144), CASP10 ...
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Genetic Target
Q4.1209
Q4
What drugs target the gene RAMP2?
The drugs that target RAMP2 are Pramlintide and Pramlintide Acetate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RAMP2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_359', 'drugName': 'Pramlintide', 'newLinkedTargets_string': 'CALCR (ENSG00000004948), RAMP1 (ENSG00000132329), RAMP2 (ENSG00000131477), RAMP3 (ENSG00000122679)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2395', 'drugName': 'Pramlintide Acetate', 'new...
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Genetic Target
Q4.1520
Q4
What drugs target the gene UMPS?
The drug that targets UMPS is Azaribine.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%UMPS %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5699', 'drugName': 'Azaribine', 'newLinkedTargets_string': 'UMPS (ENSG00000114491)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}]
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Genetic Target
Q4.741
Q4
What drugs target the gene KCNB1?
The drugs that target KCNB1 are Dalfampridine, Guanidine, Amifampridine Phosphate, Guanidine Hydrochloride, and Amifampridine.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%KCNB1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5118', 'drugName': 'Guanidine Hydrochloride', 'newLinkedTargets_string': 'KCNQ1 (ENSG00000053918), KCND3 (ENSG00000171385), KCNH2 (ENSG00000055118), KCNA2 (ENSG00000177301), KCNA1 (ENSG00000111262), KCNQ2 (ENSG00000075043), KCNQ3 (ENSG00000184156), KCNA7 (ENSG00000104848), KCNQ5 (ENSG00000...
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Q4.291
Q4
What drugs target the gene COL24A1?
The drugs that target COL24A1 are Collagenase Clostridium Histolyticum and Ocriplasmin.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%COL24A1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5818', 'drugName': 'Ocriplasmin', 'newLinkedTargets_string': 'FN1 (ENSG00000115414), COL1A2 (ENSG00000164692), COL1A1 (ENSG00000108821), COL2A1 (ENSG00000139219), COL3A1 (ENSG00000168542), COL4A1 (ENSG00000187498), COL5A1 (ENSG00000130635), COL6A1 (ENSG00000142156), COL11A1 (ENSG0000006071...
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Q4.1307
Q4
What drugs target the gene RPS6KB2?
There are no FDA approved drugs targeting the gene RPS6KB2. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Xl-418, Msc-2363318A, Tas0612, and Ly-2780301.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RPS6KB2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2168', 'drugName': 'Xl-418', 'newLinkedTargets_string': 'AKT2 (ENSG00000105221), AKT3 (ENSG00000117020), AKT1 (ENSG00000142208), RPS6KB2 (ENSG00000175634), RPS6KB1 (ENSG00000108443)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 1}, {'UUID': 'DrugGeneTargets_v2_3348', 'drugName': 'Tas...
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Q4.874
Q4
What drugs target the gene MCAM?
There are no approved drugs targeting MCAM, but the drug Abx-Ma1, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%MCAM %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5969', 'drugName': 'Abx-Ma1', 'newLinkedTargets_string': 'MCAM (ENSG00000076706)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 1}]
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Q4.564
Q4
What drugs target the gene GUCY1A2?
The drugs that target GUCY1A2 are Pentaerythritol Tetranitrate, Isosorbide Dinitrate, Nitroprusside, Nitroglycerin, Vericiguat, Isosorbide Mononitrate, Nitric Oxide, Sodium Nitroprusside, and Riociguat.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%GUCY1A2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2605', 'drugName': 'Vericiguat', 'newLinkedTargets_string': 'GUCY1B1 (ENSG00000061918), GUCY1B2 (ENSG00000123201), GUCY1A2 (ENSG00000152402), GUCY1A1 (ENSG00000164116)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1208', 'drugName': 'Nitroprusside', 'n...
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Q4.205
Q4
What drugs target the gene CD274?
The drugs that target CD274 are Durvalumab, Atezolizumab, and Avelumab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CD274 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3138', 'drugName': 'Avelumab', 'newLinkedTargets_string': 'CD274 (ENSG00000120217)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_449', 'drugName': 'Atezolizumab', 'newLinkedTargets_string': 'CD274 (ENSG00000120217)', 'drugIsApproved': True, 'maxClinica...
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Q4.1485
Q4
What drugs target the gene TRPV1?
The drugs that target TRPV1 are Acetaminophen and Capsaicin.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TRPV1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_147', 'drugName': 'Acetaminophen', 'newLinkedTargets_string': 'PTGS2 (ENSG00000073756), PTGS1 (ENSG00000095303), TRPV1 (ENSG00000196689), FAAH (ENSG00000117480)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_146', 'drugName': 'Acetaminophen', 'newLinked...
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Q4.1238
Q4
What drugs target the gene RPL18?
The drug that targets RPL18 is Ataluren.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RPL18 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG00000083845), RPS7 (ENSG...
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Q4.516
Q4
What drugs target the gene GGCX?
The drug that targets GGCX is Anisindione.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%GGCX %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1072', 'drugName': 'Anisindione', 'newLinkedTargets_string': 'GGCX (ENSG00000115486)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}]
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Q4.415
Q4
What drugs target the gene EPHA8?
The drug that targets EPHA8 is Vandetanib.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%EPHA8 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1936', 'drugName': 'Vandetanib', 'newLinkedTargets_string': 'TEK (ENSG00000120156), ERBB2 (ENSG00000141736), EGFR (ENSG00000146648), ERBB4 (ENSG00000178568), ERBB3 (ENSG00000065361), EPHA2 (ENSG00000142627), EPHB2 (ENSG00000133216), EPHA5 (ENSG00000145242), EPHA4 (ENSG00000116106), EPHA8 (...
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Q4.1408
Q4
What drugs target the gene SV2C?
There are no approved drugs targeting SV2C, but the drug Padsevonil, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%SV2C %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2155', 'drugName': 'Padsevonil', 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089), GABRA3 (ENSG00000011677), GABRP (ENSG00000094755...
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Q4.909
Q4
What drugs target the gene MT-ND2?
The drugs that target MT-ND2 are Metformin and Metformin Hydrochloride.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%MT-ND2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (ENSG00000165264), NDUFA4 (...
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Genetic Target
Q4.1042
Q4
What drugs target the gene PDE1A?
The drugs that target PDE1A are Pentoxifylline and Dipyridamole.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PDE1A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6107', 'drugName': 'Dipyridamole', 'newLinkedTargets_string': 'PDE5A (ENSG00000138735), PDE4A (ENSG00000065989), PDE3A (ENSG00000172572), PDE6H (ENSG00000139053), PDE6G (ENSG00000185527), PDE2A (ENSG00000186642), PDE7A (ENSG00000205268), PDE1A (ENSG00000115252), PDE9A (ENSG00000160191), PD...
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Q4.186
Q4
What drugs target the gene CCDC6?
The drugs that target CCDC6 are Selpercatinib and Pralsetinib.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CCDC6 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_898', 'drugName': 'Selpercatinib', 'newLinkedTargets_string': 'RET (ENSG00000165731), CCDC6 (ENSG00000108091), KIF5B (ENSG00000170759)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2688', 'drugName': 'Pralsetinib', 'newLinkedTargets_string': 'RET (ENSG...
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Q4.1189
Q4
What drugs target the gene PTGDR2?
There are no FDA approved drugs targeting the gene PTGDR2. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Vidupiprant, Qav680, Am-211, Donitriptan, Rg7185, Am-461, Fevipiprant, Setipiprant, Azd1981, Oc000459, Arry-502, Mk-7246, Adc3680, Bi-671800, Ramat...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PTGDR2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3585', 'drugName': 'Setipiprant', 'newLinkedTargets_string': 'PTGDR2 (ENSG00000183134)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_3282', 'drugName': 'Fevipiprant', 'newLinkedTargets_string': 'PTGDR2 (ENSG00000183134)', 'drugIsApproved': False, 'max...
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Genetic Target
Q4.849
Q4
What drugs target the gene MAP3K1?
There are no approved drugs targeting MAP3K1, but the drug E-6201, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%MAP3K1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3601', 'drugName': 'E-6201', 'newLinkedTargets_string': 'MAP2K1 (ENSG00000169032), MAP3K1 (ENSG00000095015)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_3602', 'drugName': 'E-6201', 'newLinkedTargets_string': 'MAP2K1 (ENSG00000169032), MAP3K1 (ENSG00...
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Genetic Target
Q4.57
Q4
What drugs target the gene ALOX12?
The drug that targets ALOX12 is Benoxaprofen.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ALOX12 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5509', 'drugName': 'Benoxaprofen', 'newLinkedTargets_string': 'ALOX12 (ENSG00000108839)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}]
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Q4.991
Q4
What drugs target the gene NOTCH3?
There are no approved drugs targeting NOTCH3, but the drug Tarextumab, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NOTCH3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4401', 'drugName': 'Tarextumab', 'newLinkedTargets_string': 'NOTCH2 (ENSG00000134250), NOTCH3 (ENSG00000074181)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 1}, {'UUID': 'DrugGeneTargets_v2_4402', 'drugName': 'Tarextumab', 'newLinkedTargets_string': 'NOTCH2 (ENSG00000134250), NOTCH3...
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Q4.485
Q4
What drugs target the gene FZD1?
There are no approved drugs targeting FZD1, but the drug Vantictumab, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%FZD1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5828', 'drugName': 'Vantictumab', 'newLinkedTargets_string': 'FZD2 (ENSG00000180340), FZD7 (ENSG00000155760), FZD1 (ENSG00000157240), FZD5 (ENSG00000163251), FZD8 (ENSG00000177283)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 1}, {'UUID': 'DrugGeneTargets_v2_5825', 'drugName': 'Vant...
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Q4.384
Q4
What drugs target the gene E2F7?
There are no FDA approved drugs targeting the gene E2F7. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Edifoligide and Edifoligide Sodium.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%E2F7 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4614', 'drugName': 'Edifoligide Sodium', 'newLinkedTargets_string': 'E2F1 (ENSG00000101412), E2F2 (ENSG00000007968), E2F3 (ENSG00000112242), E2F4 (ENSG00000205250), E2F5 (ENSG00000133740), E2F6 (ENSG00000169016), E2F7 (ENSG00000165891), E2F8 (ENSG00000129173)', 'drugIsApproved': False, 'ma...
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Q4.44
Q4
What drugs target the gene AGT?
There are no approved drugs targeting AGT, but the drug Gsk-2586881, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%AGT %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5371', 'drugName': 'Gsk-2586881', 'newLinkedTargets_string': 'AGT (ENSG00000135744)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
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Q4.1524
Q4
What drugs target the gene VDR?
The drugs that target VDR are Ergocalciferol, Calcifediol, Cholecalciferol, Paricalcitol, Calcitriol, Doxercalciferol, Alfacalcidol, Calcipotriene, and Dihydrotachysterol.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%VDR %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4241', 'drugName': 'Doxercalciferol', 'newLinkedTargets_string': 'VDR (ENSG00000111424)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4543', 'drugName': 'Alfacalcidol', 'newLinkedTargets_string': 'VDR (ENSG00000111424)', 'drugIsApproved': True, 'maxCli...
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Q4.640
Q4
What drugs target the gene IFNA1?
There are no FDA approved drugs targeting the gene IFNA1. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Faralimomab, Rontalizumab, and Sifalimumab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%IFNA1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4431', 'drugName': 'Rontalizumab', 'newLinkedTargets_string': 'IFNA6 (ENSG00000120235), IFNA8 (ENSG00000120242), IFNA5 (ENSG00000147873), IFNA10 (ENSG00000186803), IFNA2 (ENSG00000188379), IFNA1 (ENSG00000197919), IFNA13 (ENSG00000233816), IFNA7 (ENSG00000214042), IFNA21 (ENSG00000137080),...
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Q4.1202
Q4
What drugs target the gene PTK2B?
There are no FDA approved drugs targeting the gene PTK2B. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Conteltinib and Defactinib.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PTK2B %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3098', 'drugName': 'Defactinib', 'newLinkedTargets_string': 'PTK2B (ENSG00000120899), PTK2 (ENSG00000169398)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_3099', 'drugName': 'Defactinib', 'newLinkedTargets_string': 'PTK2B (ENSG00000120899), PTK2 (ENSG...
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Q4.1438
Q4
What drugs target the gene TLR8?
There are no FDA approved drugs targeting the gene TLR8. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Enpatoran, Selgantolimod, Resiquimod, Motolimod, Telratolimod, and Bazlitoran.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TLR8 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4151', 'drugName': 'Resiquimod', 'newLinkedTargets_string': 'TLR7 (ENSG00000196664), TLR8 (ENSG00000101916)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_4761', 'drugName': 'Motolimod', 'newLinkedTargets_string': 'TLR8 (ENSG00000101916)', 'drugIsAppro...
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Q4.103
Q4
What drugs target the gene BCL2A1?
There are no FDA approved drugs targeting the gene BCL2A1. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Obatoclax and Obatoclax Mesylate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%BCL2A1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2965', 'drugName': 'Obatoclax Mesylate', 'newLinkedTargets_string': 'BCL2 (ENSG00000171791), BCL2L1 (ENSG00000171552), MCL1 (ENSG00000143384), BCL2L2-PABPN1 (ENSG00000258643), BCL2L2 (ENSG00000129473), BCL2A1 (ENSG00000140379), BCL2L10 (ENSG00000137875)', 'drugIsApproved': False, 'maxClini...
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Q4.921
Q4
What drugs target the gene MUC5AC?
There are no FDA approved drugs targeting the gene MUC5AC. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Ensituximab, Yttrium Y 90 Clivatuzumab Tetraxetan, and Clivatuzumab Tetraxetan.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%MUC5AC %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6036', 'drugName': 'Yttrium Y 90 Clivatuzumab Tetraxetan', 'newLinkedTargets_string': 'MUC5AC (ENSG00000215182)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_6285', 'drugName': 'Clivatuzumab Tetraxetan', 'newLinkedTargets_string': 'MUC5AC (ENSG0000021...
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Q4.580
Q4
What drugs target the gene HDAC1?
The drugs that target HDAC1 are Belinostat, Vorinostat, Panobinostat, Panobinostat Lactate, and Romidepsin.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%HDAC1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2373', 'drugName': 'Vorinostat', 'newLinkedTargets_string': 'HDAC1 (ENSG00000116478), HDAC2 (ENSG00000196591), HDAC3 (ENSG00000171720), HDAC6 (ENSG00000094631)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2372', 'drugName': 'Vorinostat', 'newLinkedTar...
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Q4.109
Q4
What drugs target the gene BDKRB1?
There are no FDA approved drugs targeting the gene BDKRB1. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Bi113823, Mk0686, and Safotibant.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%BDKRB1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6374', 'drugName': 'Safotibant', 'newLinkedTargets_string': 'BDKRB1 (ENSG00000100739)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_5481', 'drugName': 'Mk0686', 'newLinkedTargets_string': 'BDKRB1 (ENSG00000100739)', 'drugIsApproved': False, 'maxClinic...
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Q4.356
Q4
What drugs target the gene DDC?
The drugs that target DDC are Benserazide and Carbidopa.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%DDC %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2020', 'drugName': 'Benserazide', 'newLinkedTargets_string': 'DDC (ENSG00000132437)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3213', 'drugName': 'Carbidopa', 'newLinkedTargets_string': 'DDC (ENSG00000132437)', 'drugIsApproved': True, 'maxClinicalTr...
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Q4.1229
Q4
What drugs target the gene RPL10?
The drug that targets RPL10 is Ataluren.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RPL10 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG00000083845), RPS7 (ENSG...
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Q4.222
Q4
What drugs target the gene CD70?
There are no FDA approved drugs targeting the gene CD70. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Mdx-1411, Cusatuzumab, Vorsetuzumab, and Vorsetuzumab Mafodotin.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CD70 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1493', 'drugName': 'Cusatuzumab', 'newLinkedTargets_string': 'CD70 (ENSG00000125726)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_1402', 'drugName': 'Mdx-1411', 'newLinkedTargets_string': 'CD70 (ENSG00000125726)', 'drugIsApproved': False, 'maxClinica...
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Q4.407
Q4
What drugs target the gene EPHA1?
The drug that targets EPHA1 is Vandetanib.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%EPHA1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1936', 'drugName': 'Vandetanib', 'newLinkedTargets_string': 'TEK (ENSG00000120156), ERBB2 (ENSG00000141736), EGFR (ENSG00000146648), ERBB4 (ENSG00000178568), ERBB3 (ENSG00000065361), EPHA2 (ENSG00000142627), EPHB2 (ENSG00000133216), EPHA5 (ENSG00000145242), EPHA4 (ENSG00000116106), EPHA8 (...
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Q4.798
Q4
What drugs target the gene KLRC1?
There are no approved drugs targeting KLRC1, but the drug Monalizumab, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%KLRC1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1573', 'drugName': 'Monalizumab', 'newLinkedTargets_string': 'KLRC1 (ENSG00000134545)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}]
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Q4.1253
Q4
What drugs target the gene RPL31?
The drug that targets RPL31 is Ataluren.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RPL31 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG00000083845), RPS7 (ENSG...
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Q4.1252
Q4
What drugs target the gene RPL30?
The drug that targets RPL30 is Ataluren.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RPL30 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG00000083845), RPS7 (ENSG...
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