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Q4.1447
Q4
What drugs target the gene TNFRSF17?
The drugs that target TNFRSF17 are Belantamab Mafodotin and Teclistamab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TNFRSF17 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1872', 'drugName': 'Belantamab Mafodotin', 'newLinkedTargets_string': 'TUBB4B (ENSG00000188229), TUBB1 (ENSG00000101162), TUBA3C (ENSG00000198033), TUBA4A (ENSG00000127824), TUBB3 (ENSG00000258947), TUBA1A (ENSG00000167552), TUBB4A (ENSG00000104833), TUBB8 (ENSG00000261456), TUBB (ENSG0000...
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Q4.130
Q4
What drugs target the gene CA1?
The drugs that target CA1 are Dichlorphenamide, Acetazolamide, Ethoxzolamide, Methazolamide, Methocarbamol, Sulthiame, and Acetazolamide Sodium.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CA1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_466', 'drugName': 'Acetazolamide', 'newLinkedTargets_string': 'CA12 (ENSG00000074410), CA2 (ENSG00000104267), CA4 (ENSG00000167434), CA1 (ENSG00000133742)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_469', 'drugName': 'Acetazolamide', 'newLinkedTarget...
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Q4.1178
Q4
What drugs target the gene PSMD12?
The drugs that target PSMD12 are Bortezomib, Carfilzomib, Ixazomib, and Ixazomib Citrate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PSMD12 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_559', 'drugName': 'Bortezomib', 'newLinkedTargets_string': 'PSMD1 (ENSG00000173692), PSMB2 (ENSG00000126067), PSMB1 (ENSG00000008018), PSMB5 (ENSG00000100804), PSMB8 (ENSG00000204264), PSMB9 (ENSG00000240065), PSMB6 (ENSG00000142507), PSMD14 (ENSG00000115233), PSMA1 (ENSG00000129084), PSMA...
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Q4.942
Q4
What drugs target the gene NDUFA4?
The drugs that target NDUFA4 are Metformin and Metformin Hydrochloride.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NDUFA4 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (ENSG00000165264), NDUFA4 (...
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Q4.1468
Q4
What drugs target the gene TOP1MT?
The drugs that target TOP1MT are Topotecan and Topotecan Hydrochloride.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TOP1MT %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5442', 'drugName': 'Topotecan Hydrochloride', 'newLinkedTargets_string': 'TOP1MT (ENSG00000184428)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1325', 'drugName': 'Topotecan', 'newLinkedTargets_string': 'TOP1MT (ENSG00000184428)', 'drugIsApproved': Tr...
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Q4.706
Q4
What drugs target the gene IL9?
There are no approved drugs targeting IL9, but the drug Enokizumab, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%IL9 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2346', 'drugName': 'Enokizumab', 'newLinkedTargets_string': 'IL9 (ENSG00000145839)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
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Q4.532
Q4
What drugs target the gene GPC3?
There are no approved drugs targeting GPC3, but the drug Codrituzumab, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%GPC3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4119', 'drugName': 'Codrituzumab', 'newLinkedTargets_string': 'GPC3 (ENSG00000147257)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
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Q4.246
Q4
What drugs target the gene CDK6?
The drugs that target CDK6 are Trilaciclib, Ribociclib Succinate, Palbociclib, Ribociclib, Trilaciclib Dihydrochloride, and Abemaciclib.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CDK6 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2093', 'drugName': 'Ribociclib Succinate', 'newLinkedTargets_string': 'CDK4 (ENSG00000135446), CDK6 (ENSG00000105810)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2461', 'drugName': 'Palbociclib', 'newLinkedTargets_string': 'CCND1 (ENSG00000110092), C...
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Q4.1046
Q4
What drugs target the gene PDE3A?
The drugs that target PDE3A are Anagrelide Hydrochloride, Theophylline Sodium Glycinate, Milrinone, Dyphylline, Theophylline Glycinate, Inamrinone, Cilostazol, Enoximone, Oxtriphylline, Milrinone Lactate, Pentoxifylline, Anagrelide, Inamrinone Lactate, Theophylline, Aminophylline, and Dipyridamole.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PDE3A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4546', 'drugName': 'Theophylline', 'newLinkedTargets_string': 'ADORA1 (ENSG00000163485), ADORA2B (ENSG00000170425), ADORA3 (ENSG00000282608), ADORA2A (ENSG00000128271), PDE3A (ENSG00000172572), PDE3B (ENSG00000152270), PDE4A (ENSG00000065989), PDE4D (ENSG00000113448), PDE4B (ENSG0000018458...
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Q4.1124
Q4
What drugs target the gene PRKAA1?
There are no approved drugs targeting PRKAA1, but the drug Acadesine, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PRKAA1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5888', 'drugName': 'Acadesine', 'newLinkedTargets_string': 'PRKAA2 (ENSG00000162409), PRKAB2 (ENSG00000131791), PRKAG1 (ENSG00000181929), PRKAG2 (ENSG00000106617), PRKAB1 (ENSG00000111725), PRKAA1 (ENSG00000132356), PRKAG3 (ENSG00000115592)', 'drugIsApproved': False, 'maxClinicalTrialPhase...
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Q4.844
Q4
What drugs target the gene MALT1?
The drugs that target MALT1 are Mepazine Acetate and Mepazine.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%MALT1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1830', 'drugName': 'Mepazine', 'newLinkedTargets_string': 'MALT1 (ENSG00000172175)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1820', 'drugName': 'Mepazine Acetate', 'newLinkedTargets_string': 'MALT1 (ENSG00000172175)', 'drugIsApproved': True, 'maxCl...
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Q4.1064
Q4
What drugs target the gene PDGFB?
There are no approved drugs targeting PDGFB, but the drug Pegpleranib Sodium, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PDGFB %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1062', 'drugName': 'Pegpleranib Sodium', 'newLinkedTargets_string': 'PDGFB (ENSG00000100311)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}]
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Q4.1480
Q4
What drugs target the gene TREM1?
There are no approved drugs targeting TREM1, but the drug Nangibotide, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TREM1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4000', 'drugName': 'Nangibotide', 'newLinkedTargets_string': 'TREM1 (ENSG00000124731)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
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Q4.233
Q4
What drugs target the gene CDK12?
There are no FDA approved drugs targeting the gene CDK12. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Roniciclib, Pha-793887, Azd-5438, and At-7519.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CDK12 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1429', 'drugName': 'Roniciclib', 'newLinkedTargets_string': 'CDK1 (ENSG00000170312), CDK4 (ENSG00000135446), CDK2 (ENSG00000123374), CDK5 (ENSG00000164885), CDK6 (ENSG00000105810), CDK7 (ENSG00000134058), CDK3 (ENSG00000250506), CDK16 (ENSG00000102225), CDK18 (ENSG00000117266), CDK8 (ENSG0...
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Q4.33
Q4
What drugs target the gene ADRA1B?
The drugs that target ADRA1B are Methoxamine, Oxymetazoline, Naphazoline Hydrochloride, Oxymetazoline Hydrochloride, Tetrahydrozoline, Trimipramine Maleate, Terazosin, Moxisylyte, Dipivefrin, Epinephrine, Carvedilol Phosphate, Doxazosin Mesylate, Tamsulosin, Methoxamine Hydrochloride, Alfuzosin Hydrochloride, Terazosin...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ADRA1B %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2489', 'drugName': 'Isoxsuprine Hydrochloride', 'newLinkedTargets_string': 'ADRB2 (ENSG00000169252), ADRA1A (ENSG00000120907), ADRA1D (ENSG00000171873), ADRA1B (ENSG00000170214)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3132', 'drugName': 'Ergotami...
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Q4.687
Q4
What drugs target the gene IL1RL2?
The drug that targets IL1RL2 is Spesolimab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%IL1RL2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2421', 'drugName': 'Spesolimab', 'newLinkedTargets_string': 'IL1RL2 (ENSG00000115598), IL1RAP (ENSG00000196083)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_102', 'drugName': 'Imsidolimab', 'newLinkedTargets_string': 'IL1RL2 (ENSG00000115598), IL1RAP ...
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Q4.493
Q4
What drugs target the gene GABRA1?
The drugs that target GABRA1 are Meprobamate, Acamprosate Calcium, Enflurane, Methohexital, Metharbital, Butabarbital, Flurazepam Hydrochloride, Pentobarbital Sodium, Acamprosate, Primidone, Temazepam, Flunitrazepam, Ganaxolone, Diazepam, Methyprylon, Thiopental, Clonazepam, Topiramate, Remimazolam Besylate, Brexanolon...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%GABRA1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1496', 'drugName': 'Clonazepam', 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089), GABRA3 (ENSG00000011677), GABRP (ENSG00000094755...
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Q4.1004
Q4
What drugs target the gene NQO1?
There are no approved drugs targeting NQO1, but the drug Vatiquinone, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NQO1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2788', 'drugName': 'Vatiquinone', 'newLinkedTargets_string': 'NQO1 (ENSG00000181019)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}]
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Q4.945
Q4
What drugs target the gene NDUFA6?
The drugs that target NDUFA6 are Metformin and Metformin Hydrochloride.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NDUFA6 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (ENSG00000165264), NDUFA4 (...
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Q4.886
Q4
What drugs target the gene MGLL?
There are no approved drugs targeting MGLL, but the drug Elcubragistat, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%MGLL %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4556', 'drugName': 'Elcubragistat', 'newLinkedTargets_string': 'MGLL (ENSG00000074416)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
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Q4.621
Q4
What drugs target the gene HTR2B?
The drugs that target HTR2B are Methylergonovine, Zimeldine, Amisulpride, Methylergonovine Maleate, Clothiapine, Methysergide Maleate, Dexfenfluramine, Methysergide, Dexfenfluramine Hydrochloride, Minaprine Hydrochloride, Minaprine, and Zimeldine Hydrochloride.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%HTR2B %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5327', 'drugName': 'Minaprine', 'newLinkedTargets_string': 'MAOA (ENSG00000189221), DRD2 (ENSG00000149295), DRD1 (ENSG00000184845), HTR2B (ENSG00000135914), HTR2A (ENSG00000102468), HTR2C (ENSG00000147246), CHRM1 (ENSG00000168539), ACHE (ENSG00000087085)', 'drugIsApproved': True, 'maxClini...
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Q4.797
Q4
What drugs target the gene KLKB1?
The drugs that target KLKB1 are Berotralstat, Human C1-Esterase Inhibitor, Ecallantide, Lanadelumab, Aprotinin, and Berotralstat Hydrochloride.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%KLKB1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4053', 'drugName': 'Aprotinin', 'newLinkedTargets_string': 'PLG (ENSG00000122194), KLKB1 (ENSG00000164344)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4296', 'drugName': 'Berotralstat Hydrochloride', 'newLinkedTargets_string': 'KLKB1 (ENSG00000164344...
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Q4.955
Q4
What drugs target the gene NDUFB10?
The drugs that target NDUFB10 are Metformin and Metformin Hydrochloride.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NDUFB10 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (ENSG00000165264), NDUFA4 (...
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Q4.537
Q4
What drugs target the gene GPRC5D?
There are no approved drugs targeting GPRC5D, but the drug Talquetamab, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%GPRC5D %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5924', 'drugName': 'Talquetamab', 'newLinkedTargets_string': 'GPRC5D (ENSG00000111291), CD3E (ENSG00000198851), CD3G (ENSG00000160654), CD3D (ENSG00000167286)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_5925', 'drugName': 'Talquetamab', 'newLinkedTa...
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Q4.1367
Q4
What drugs target the gene SLC22A8?
The drug that targets SLC22A8 is Probenecid.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%SLC22A8 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1876', 'drugName': 'Probenecid', 'newLinkedTargets_string': 'SLC22A8 (ENSG00000149452), SLC22A6 (ENSG00000197901), SLC22A11 (ENSG00000168065)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1877', 'drugName': 'Probenecid', 'newLinkedTargets_string': 'SLC...
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Q4.529
Q4
What drugs target the gene GP1BA?
There are no approved drugs targeting GP1BA, but the drug Anfibatide, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%GP1BA %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4499', 'drugName': 'Anfibatide', 'newLinkedTargets_string': 'GP1BA (ENSG00000185245)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
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Q4.165
Q4
What drugs target the gene CACNG6?
The drugs that target CACNG6 are Gabapentin, Terodiline Hydrochloride, Phloroglucinol, Suloctidil, Pregabalin, Gabapentin Enacarbil, Bepridil Hydrochloride, Bepridil, and Terodiline.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CACNG6 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_142', 'drugName': 'Gabapentin', 'newLinkedTargets_string': 'CACNA1H (ENSG00000196557), CACNA2D1 (ENSG00000153956), CACNA1C (ENSG00000151067), CACNA2D3 (ENSG00000157445), CACNA1S (ENSG00000081248), CACNA2D2 (ENSG00000007402), CACNA1D (ENSG00000157388), CACNA1A (ENSG00000141837), CACNA1B (EN...
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Q4.1477
Q4
What drugs target the gene TRAF3IP2?
There are no approved drugs targeting TRAF3IP2, but the drug Iguratimod, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TRAF3IP2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5945', 'drugName': 'Iguratimod', 'newLinkedTargets_string': 'MIF (ENSG00000240972), TRAF3IP2 (ENSG00000056972), PTGS2 (ENSG00000073756)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_5946', 'drugName': 'Iguratimod', 'newLinkedTargets_string': 'MIF (ENS...
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Q4.1525
Q4
What drugs target the gene VEGFA?
The drugs that target VEGFA are Faricimab, Bevacizumab, Aflibercept, Brolucizumab, Ranibizumab, and Pegaptanib Sodium.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%VEGFA %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_997', 'drugName': 'Aflibercept', 'newLinkedTargets_string': 'VEGFA (ENSG00000112715), PGF (ENSG00000119630)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4833', 'drugName': 'Pegaptanib Sodium', 'newLinkedTargets_string': 'VEGFA (ENSG00000112715)', 'dru...
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Q4.1368
Q4
What drugs target the gene SLC29A1?
The drug that targets SLC29A1 is Dipyridamole.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%SLC29A1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6106', 'drugName': 'Dipyridamole', 'newLinkedTargets_string': 'PDE5A (ENSG00000138735), PDE4A (ENSG00000065989), PDE3A (ENSG00000172572), PDE6H (ENSG00000139053), PDE6G (ENSG00000185527), PDE2A (ENSG00000186642), PDE7A (ENSG00000205268), PDE1A (ENSG00000115252), PDE9A (ENSG00000160191), PD...
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Genetic Target
Q4.1104
Q4
What drugs target the gene POLD3?
The drugs that target POLD3 are Gemcitabine Hydrochloride, Gemcitabine, Clofarabine, Fludarabine Phosphate, and Cytarabine.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%POLD3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4', 'drugName': 'Gemcitabine Hydrochloride', 'newLinkedTargets_string': 'POLA1 (ENSG00000101868), POLD4 (ENSG00000175482), POLD3 (ENSG00000077514), POLD1 (ENSG00000062822), POLD2 (ENSG00000106628), POLE (ENSG00000177084), POLA2 (ENSG00000014138), PRIM1 (ENSG00000198056), PRIM2 (ENSG0000014...
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Genetic Target
Q4.727
Q4
What drugs target the gene ITGB7?
The drugs that target ITGB7 are Natalizumab and Vedolizumab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ITGB7 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5015', 'drugName': 'Natalizumab', 'newLinkedTargets_string': 'ITGA4 (ENSG00000115232), ITGB7 (ENSG00000139626), ITGB1 (ENSG00000150093)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5088', 'drugName': 'Vedolizumab', 'newLinkedTargets_string': 'ITGA4 (E...
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Genetic Target
Q4.601
Q4
What drugs target the gene HRAS?
There are no approved drugs targeting HRAS, but the drug Salirasib, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%HRAS %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3775', 'drugName': 'Salirasib', 'newLinkedTargets_string': 'HRAS (ENSG00000174775), NRAS (ENSG00000213281), KRAS (ENSG00000133703)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
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Genetic Target
Q4.677
Q4
What drugs target the gene IL17F?
The drug that targets IL17F is Bimekizumab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%IL17F %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_305', 'drugName': 'Bimekizumab', 'newLinkedTargets_string': 'IL17F (ENSG00000112116), IL17A (ENSG00000112115)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_306', 'drugName': 'Bimekizumab', 'newLinkedTargets_string': 'IL17F (ENSG00000112116), IL17A (ENS...
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Genetic Target
Q4.346
Q4
What drugs target the gene CYP19A1?
The drugs that target CYP19A1 are Exemestane, Testolactone, Aminoglutethimide, Anastrozole, and Letrozole.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CYP19A1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_923', 'drugName': 'Exemestane', 'newLinkedTargets_string': 'CYP19A1 (ENSG00000137869)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2073', 'drugName': 'Testolactone', 'newLinkedTargets_string': 'CYP19A1 (ENSG00000137869)', 'drugIsApproved': True, 'maxC...
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Genetic Target
Q4.1217
Q4
What drugs target the gene RET?
The drugs that target RET are Sorafenib, Regorafenib, Selpercatinib, Alectinib Hydrochloride, Sorafenib Tosylate, Vandetanib, Pralsetinib, Sunitinib, Sunitinib Malate, and Alectinib.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RET %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1549', 'drugName': 'Sorafenib Tosylate', 'newLinkedTargets_string': 'FLT3 (ENSG00000122025), RAF1 (ENSG00000132155), PDGFRB (ENSG00000113721), BRAF (ENSG00000157764), RET (ENSG00000165731), FLT1 (ENSG00000102755), FLT4 (ENSG00000037280), KDR (ENSG00000128052), KIT (ENSG00000157404)', 'drug...
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Genetic Target
Q4.857
Q4
What drugs target the gene MAPK1?
There are no FDA approved drugs targeting the gene MAPK1. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Ravoxertinib, Ulixertinib, Temuterkib, Asn007, Ko-947, and Mk-8353.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%MAPK1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4297', 'drugName': 'Temuterkib', 'newLinkedTargets_string': 'MAPK3 (ENSG00000102882), MAPK1 (ENSG00000100030)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_1863', 'drugName': 'Ulixertinib', 'newLinkedTargets_string': 'MAPK3 (ENSG00000102882), MAPK1 (E...
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Genetic Target
Q4.194
Q4
What drugs target the gene CCR2?
There are no FDA approved drugs targeting the gene CCR2. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Ilacirnon, Bms-813160, Mk-0812, Bms-741672, Pf-4136309, Pf-04634817, Cenicriviroc, Jnj-41443532, Plozalizumab, and Azd2423.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CCR2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3740', 'drugName': 'Cenicriviroc', 'newLinkedTargets_string': 'CCR2 (ENSG00000121807), CCR5 (ENSG00000160791)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_3741', 'drugName': 'Cenicriviroc', 'newLinkedTargets_string': 'CCR2 (ENSG00000121807), CCR5 (EN...
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Genetic Target
Q4.698
Q4
What drugs target the gene IL3RA?
The drug that targets IL3RA is Tagraxofusp.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%IL3RA %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6264', 'drugName': 'Tagraxofusp', 'newLinkedTargets_string': 'EEF2 (ENSG00000167658), IL3RA (ENSG00000185291)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_6265', 'drugName': 'Tagraxofusp', 'newLinkedTargets_string': 'EEF2 (ENSG00000167658), IL3RA (ENS...
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Genetic Target
Q4.341
Q4
What drugs target the gene CXCR4?
The drug that targets CXCR4 is Plerixafor.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CXCR4 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5536', 'drugName': 'Plerixafor', 'newLinkedTargets_string': 'CXCR4 (ENSG00000121966)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5036', 'drugName': 'Mavorixafor', 'newLinkedTargets_string': 'CXCR4 (ENSG00000121966)', 'drugIsApproved': False, 'maxClin...
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Genetic Target
Q4.503
Q4
What drugs target the gene GABRE?
The drugs that target GABRE are Meprobamate, Acamprosate Calcium, Enflurane, Methohexital, Metharbital, Butabarbital, Flurazepam Hydrochloride, Pentobarbital Sodium, Acamprosate, Primidone, Temazepam, Flunitrazepam, Ganaxolone, Diazepam, Methyprylon, Thiopental, Clonazepam, Topiramate, Remimazolam Besylate, Brexanolone...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%GABRE %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1494', 'drugName': 'Thiopental', 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089), GABRA3 (ENSG00000011677), GABRP (ENSG00000094755...
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Q4.64
Q4
What drugs target the gene ANO1?
The drug that targets ANO1 is Crofelemer.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ANO1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2220', 'drugName': 'Crofelemer', 'newLinkedTargets_string': 'CFTR (ENSG00000001626), ANO1 (ENSG00000131620)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2221', 'drugName': 'Crofelemer', 'newLinkedTargets_string': 'CFTR (ENSG00000001626), ANO1 (ENSG000...
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Q4.709
Q4
What drugs target the gene IMPDH2?
The drugs that target IMPDH2 are Mycophenolate Mofetil, Mycophenolic Acid, Mycophenolate Sodium, Mycophenolate Mofetil Hydrochloride, and Thioguanine.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%IMPDH2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_290', 'drugName': 'Mycophenolate Mofetil', 'newLinkedTargets_string': 'IMPDH1 (ENSG00000106348), IMPDH2 (ENSG00000178035)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5258', 'drugName': 'Thioguanine', 'newLinkedTargets_string': 'IMPDH1 (ENSG0000010634...
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Q4.1302
Q4
What drugs target the gene RPS6KA1?
There are no approved drugs targeting RPS6KA1, but the drug Tas0612, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RPS6KA1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3347', 'drugName': 'Tas0612', 'newLinkedTargets_string': 'RPS6KB2 (ENSG00000175634), RPS6KB1 (ENSG00000108443), AKT2 (ENSG00000105221), AKT3 (ENSG00000117020), AKT1 (ENSG00000142208), RPS6KA3 (ENSG00000177189), RPS6KA2 (ENSG00000071242), RPS6KA6 (ENSG00000072133), RPS6KA1 (ENSG00000117676)...
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Q4.926
Q4
What drugs target the gene MYL3?
The drug that targets MYL3 is Mavacamten.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%MYL3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1036', 'drugName': 'Mavacamten', 'newLinkedTargets_string': 'MYH7 (ENSG00000092054), MYH6 (ENSG00000197616), MYH7B (ENSG00000078814), MYL3 (ENSG00000160808), MYL2 (ENSG00000111245), MYL7 (ENSG00000106631), MYL4 (ENSG00000198336)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID...
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Q4.938
Q4
What drugs target the gene NDUFA12?
The drugs that target NDUFA12 are Metformin and Metformin Hydrochloride.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NDUFA12 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (ENSG00000165264), NDUFA4 (...
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Q4.1185
Q4
What drugs target the gene PSMD7?
The drugs that target PSMD7 are Bortezomib, Carfilzomib, Ixazomib, and Ixazomib Citrate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PSMD7 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_559', 'drugName': 'Bortezomib', 'newLinkedTargets_string': 'PSMD1 (ENSG00000173692), PSMB2 (ENSG00000126067), PSMB1 (ENSG00000008018), PSMB5 (ENSG00000100804), PSMB8 (ENSG00000204264), PSMB9 (ENSG00000240065), PSMB6 (ENSG00000142507), PSMD14 (ENSG00000115233), PSMA1 (ENSG00000129084), PSMA...
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Q4.276
Q4
What drugs target the gene CHRNE?
The drugs that target CHRNE are Pipecuronium, Decamethonium, Vecuronium, Rocuronium, Metocurine Iodide, Succinylcholine Chloride, Tubocurarine, Rocuronium Bromide, Cisatracurium, Cisatracurium Besylate, Mivacurium Chloride, Pancuronium, Gallamine, Vecuronium Bromide, Gallamine Triethiodide, Metocurine, Atracurium Besyl...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CHRNE %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2723', 'drugName': 'Succinylcholine Chloride', 'newLinkedTargets_string': 'CHRNA1 (ENSG00000138435), CHRNG (ENSG00000196811), CHRNB1 (ENSG00000170175), CHRND (ENSG00000135902), CHRNE (ENSG00000108556)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_922',...
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Q4.541
Q4
What drugs target the gene GRIA3?
The drugs that target GRIA3 are Topiramate and Perampanel.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%GRIA3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2165', 'drugName': 'Perampanel', 'newLinkedTargets_string': 'GRIA4 (ENSG00000152578), GRIA3 (ENSG00000125675), GRIA2 (ENSG00000120251), GRIA1 (ENSG00000155511)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1593', 'drugName': 'Topiramate', 'newLinkedTar...
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Q4.863
Q4
What drugs target the gene MAPK9?
There are no FDA approved drugs targeting the gene MAPK9. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Tanzisertib, Cc-401, and Bentamapimod.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%MAPK9 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2634', 'drugName': 'Cc-401', 'newLinkedTargets_string': 'MAPK9 (ENSG00000050748), MAPK8 (ENSG00000107643), MAPK10 (ENSG00000109339)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_2632', 'drugName': 'Cc-401', 'newLinkedTargets_string': 'MAPK9 (ENSG00000...
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Q4.750
Q4
What drugs target the gene KCNF1?
The drugs that target KCNF1 are Dalfampridine, Guanidine, Amifampridine Phosphate, Guanidine Hydrochloride, and Amifampridine.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%KCNF1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5118', 'drugName': 'Guanidine Hydrochloride', 'newLinkedTargets_string': 'KCNQ1 (ENSG00000053918), KCND3 (ENSG00000171385), KCNH2 (ENSG00000055118), KCNA2 (ENSG00000177301), KCNA1 (ENSG00000111262), KCNQ2 (ENSG00000075043), KCNQ3 (ENSG00000184156), KCNA7 (ENSG00000104848), KCNQ5 (ENSG00000...
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Q4.200
Q4
What drugs target the gene CD2?
The drug that targets CD2 is Alefacept.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CD2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4052', 'drugName': 'Alefacept', 'newLinkedTargets_string': 'CD2 (ENSG00000116824)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1616', 'drugName': 'Siplizumab', 'newLinkedTargets_string': 'CD2 (ENSG00000116824)', 'drugIsApproved': False, 'maxClinicalTr...
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Q4.453
Q4
What drugs target the gene FCGR3A?
There are no approved drugs targeting FCGR3A, but the drug Imgatuzumab, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%FCGR3A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1400', 'drugName': 'Imgatuzumab', 'newLinkedTargets_string': 'FCGR3A (ENSG00000203747), EGFR (ENSG00000146648)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_1401', 'drugName': 'Imgatuzumab', 'newLinkedTargets_string': 'FCGR3A (ENSG00000203747), EGFR (...
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Genetic Target
Q4.970
Q4
What drugs target the gene NDUFS4?
The drugs that target NDUFS4 are Metformin and Metformin Hydrochloride.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NDUFS4 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (ENSG00000165264), NDUFA4 (...
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Genetic Target
Q4.546
Q4
What drugs target the gene GRIK4?
The drug that targets GRIK4 is Topiramate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%GRIK4 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1594', 'drugName': 'Topiramate', 'newLinkedTargets_string': 'GRIK1 (ENSG00000171189), GRIK5 (ENSG00000105737), GRIK4 (ENSG00000149403), GRIK2 (ENSG00000164418), GRIK3 (ENSG00000163873), CA4 (ENSG00000167434), SCN1A (ENSG00000144285), SCN5A (ENSG00000183873), SCN4A (ENSG00000007314), SCN7A ...
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Q4.1293
Q4
What drugs target the gene RPS27A?
The drug that targets RPS27A is Ataluren.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RPS27A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG00000083845), RPS7 (ENSG...
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Q4.273
Q4
What drugs target the gene CHRNB2?
The drugs that target CHRNB2 are Varenicline Tartrate, Nicotine, Varenicline, and Nicotine Polacrilex.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CHRNB2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2697', 'drugName': 'Varenicline', 'newLinkedTargets_string': 'CHRNB2 (ENSG00000160716), CHRNA4 (ENSG00000101204)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2698', 'drugName': 'Varenicline', 'newLinkedTargets_string': 'CHRNB2 (ENSG00000160716), CHRNA...
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Genetic Target
Q4.1169
Q4
What drugs target the gene PSMB9?
The drugs that target PSMB9 are Bortezomib, Carfilzomib, Ixazomib, and Ixazomib Citrate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PSMB9 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3334', 'drugName': 'Ixazomib', 'newLinkedTargets_string': 'PSMD1 (ENSG00000173692), PSMB2 (ENSG00000126067), PSMB1 (ENSG00000008018), PSMB5 (ENSG00000100804), PSMB8 (ENSG00000204264), PSMB9 (ENSG00000240065), PSMB6 (ENSG00000142507), PSMD14 (ENSG00000115233), PSMA1 (ENSG00000129084), PSMA2...
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Genetic Target
Q4.220
Q4
What drugs target the gene CD52?
The drug that targets CD52 is Alemtuzumab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CD52 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1142', 'drugName': 'Alemtuzumab', 'newLinkedTargets_string': 'CD52 (ENSG00000169442)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}]
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Q4.1015
Q4
What drugs target the gene NTRK3?
The drugs that target NTRK3 are Larotrectinib, Entrectinib, Cenegermin, and Larotrectinib Sulfate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NTRK3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_894', 'drugName': 'Larotrectinib', 'newLinkedTargets_string': 'NTRK1 (ENSG00000198400), NTRK2 (ENSG00000148053), NTRK3 (ENSG00000140538)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3786', 'drugName': 'Cenegermin', 'newLinkedTargets_string': 'NTRK1 (E...
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Genetic Target
Q4.1241
Q4
What drugs target the gene RPL21?
The drug that targets RPL21 is Ataluren.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RPL21 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG00000083845), RPS7 (ENSG...
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Genetic Target
Q4.427
Q4
What drugs target the gene ERBB4?
The drugs that target ERBB4 are Afatinib, Vandetanib, Neratinib, Afatinib Dimaleate, Dacomitinib, and Neratinib Maleate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ERBB4 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1044', 'drugName': 'Afatinib', 'newLinkedTargets_string': 'ERBB4 (ENSG00000178568), EGFR (ENSG00000146648), ERBB2 (ENSG00000141736)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1996', 'drugName': 'Neratinib', 'newLinkedTargets_string': 'EGFR (ENSG0000...
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Genetic Target
Q4.352
Q4
What drugs target the gene CYP46A1?
There are no approved drugs targeting CYP46A1, but the drug Soticlestat, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CYP46A1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5773', 'drugName': 'Soticlestat', 'newLinkedTargets_string': 'CYP46A1 (ENSG00000036530)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}]
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Genetic Target
Q4.1401
Q4
What drugs target the gene SSTR5?
The drugs that target SSTR5 are Lanreotide, Lutetium Dotatate, Octreotide Acetate, Pasireotide Diaspartate, Lanreotide Acetate, Lutetium Dotatate Lu-177, Pasireotide, Octreotide, and Pasireotide Pamoate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%SSTR5 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6122', 'drugName': 'Pasireotide Pamoate', 'newLinkedTargets_string': 'SSTR3 (ENSG00000278195), SSTR5 (ENSG00000162009), SSTR2 (ENSG00000180616), SSTR1 (ENSG00000139874)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2626', 'drugName': 'Lanreotide Acetat...
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Genetic Target
Q4.1267
Q4
What drugs target the gene RPL6?
The drug that targets RPL6 is Ataluren.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RPL6 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG00000083845), RPS7 (ENSG...
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Genetic Target
Q4.466
Q4
What drugs target the gene FGFR3?
The drugs that target FGFR3 are Pazopanib Hydrochloride, Infigratinib, Infigratinib Phosphate, Pemigatinib, Nintedanib Esylate, Masitinib, Pazopanib, Erdafitinib, Nintedanib, and Futibatinib.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%FGFR3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5658', 'drugName': 'Pazopanib', 'newLinkedTargets_string': 'FLT1 (ENSG00000102755), FLT4 (ENSG00000037280), KDR (ENSG00000128052), ITK (ENSG00000113263), PDGFRB (ENSG00000113721), PDGFRA (ENSG00000134853), FGFR3 (ENSG00000068078), KIT (ENSG00000157404), CSF1R (ENSG00000182578), LCK (ENSG00...
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Genetic Target
Q4.1060
Q4
What drugs target the gene PDE7B?
The drugs that target PDE7B are Flavoxate, Flavoxate Hydrochloride, Pentoxifylline, and Dipyridamole.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PDE7B %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_766', 'drugName': 'Flavoxate', 'newLinkedTargets_string': 'PDE8B (ENSG00000113231), PDE8A (ENSG00000073417), PDE7A (ENSG00000205268), PDE7B (ENSG00000171408), PDE4A (ENSG00000065989), PDE4D (ENSG00000113448), PDE4B (ENSG00000184588), PDE4C (ENSG00000105650)', 'drugIsApproved': True, 'maxCl...
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Genetic Target
Q4.1353
Q4
What drugs target the gene SI?
There are no FDA approved drugs targeting the gene SI. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Celgosivir and Voglibose.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%SI %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4560', 'drugName': 'Voglibose', 'newLinkedTargets_string': 'MGAM (ENSG00000257335), GAA (ENSG00000171298), SI (ENSG00000090402), MGAM2 (ENSG00000257743)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_3655', 'drugName': 'Celgosivir', 'newLinkedTargets_s...
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Genetic Target
Q4.866
Q4
What drugs target the gene MAPT?
There are no FDA approved drugs targeting the gene MAPT. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Zagotenemab, Gosuranemab, Bepranemab, Semorinemab, Posdinemab, and Tilavonemab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%MAPT %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5139', 'drugName': 'Posdinemab', 'newLinkedTargets_string': 'MAPT (ENSG00000186868)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_5485', 'drugName': 'Tilavonemab', 'newLinkedTargets_string': 'MAPT (ENSG00000186868)', 'drugIsApproved': False, 'maxClini...
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Genetic Target
Q4.614
Q4
What drugs target the gene HSPB1?
There are no FDA approved drugs targeting the gene HSPB1. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Apatorsen and Apatorsen Sodium.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%HSPB1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1706', 'drugName': 'Apatorsen', 'newLinkedTargets_string': 'HSPB1 (ENSG00000106211)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_3133', 'drugName': 'Apatorsen Sodium', 'newLinkedTargets_string': 'HSPB1 (ENSG00000106211)', 'drugIsApproved': False, 'ma...
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Genetic Target
Q4.383
Q4
What drugs target the gene E2F6?
There are no FDA approved drugs targeting the gene E2F6. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Edifoligide and Edifoligide Sodium.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%E2F6 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4614', 'drugName': 'Edifoligide Sodium', 'newLinkedTargets_string': 'E2F1 (ENSG00000101412), E2F2 (ENSG00000007968), E2F3 (ENSG00000112242), E2F4 (ENSG00000205250), E2F5 (ENSG00000133740), E2F6 (ENSG00000169016), E2F7 (ENSG00000165891), E2F8 (ENSG00000129173)', 'drugIsApproved': False, 'ma...
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Q4.647
Q4
What drugs target the gene IFNA21?
There are no FDA approved drugs targeting the gene IFNA21. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Rontalizumab and Sifalimumab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%IFNA21 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5087', 'drugName': 'Sifalimumab', 'newLinkedTargets_string': 'IFNA6 (ENSG00000120235), IFNA8 (ENSG00000120242), IFNA5 (ENSG00000147873), IFNA10 (ENSG00000186803), IFNA2 (ENSG00000188379), IFNA1 (ENSG00000197919), IFNA13 (ENSG00000233816), IFNA7 (ENSG00000214042), IFNA21 (ENSG00000137080), ...
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Genetic Target
Q4.1165
Q4
What drugs target the gene PSMB5?
The drugs that target PSMB5 are Bortezomib, Carfilzomib, Ixazomib, and Ixazomib Citrate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PSMB5 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3334', 'drugName': 'Ixazomib', 'newLinkedTargets_string': 'PSMD1 (ENSG00000173692), PSMB2 (ENSG00000126067), PSMB1 (ENSG00000008018), PSMB5 (ENSG00000100804), PSMB8 (ENSG00000204264), PSMB9 (ENSG00000240065), PSMB6 (ENSG00000142507), PSMD14 (ENSG00000115233), PSMA1 (ENSG00000129084), PSMA2...
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Q4.1040
Q4
What drugs target the gene PDCD1LG2?
There are no approved drugs targeting PDCD1LG2, but the drug Rhigm12B7, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PDCD1LG2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5506', 'drugName': 'Rhigm12B7', 'newLinkedTargets_string': 'PDCD1LG2 (ENSG00000197646)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 1}]
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Q4.764
Q4
What drugs target the gene KCNJ2?
The drugs that target KCNJ2 are Dronedarone Hydrochloride and Dronedarone.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%KCNJ2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3873', 'drugName': 'Dronedarone Hydrochloride', 'newLinkedTargets_string': 'CACNA1C (ENSG00000151067), CACNA1S (ENSG00000081248), CACNA1D (ENSG00000157388), CACNA1F (ENSG00000102001), HCN4 (ENSG00000138622), SCN1A (ENSG00000144285), SCN5A (ENSG00000183873), SCN4A (ENSG00000007314), SCN7A (...
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Q4.818
Q4
What drugs target the gene LGALS1?
There are no approved drugs targeting LGALS1, but the drug Davanat, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%LGALS1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6359', 'drugName': 'Davanat', 'newLinkedTargets_string': 'LGALS3 (ENSG00000131981), LGALS1 (ENSG00000100097)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_6360', 'drugName': 'Davanat', 'newLinkedTargets_string': 'LGALS3 (ENSG00000131981), LGALS1 (ENSG...
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Q4.1108
Q4
What drugs target the gene POLE3?
The drugs that target POLE3 are Gemcitabine Hydrochloride, Gemcitabine, Clofarabine, Fludarabine Phosphate, and Cytarabine.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%POLE3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4', 'drugName': 'Gemcitabine Hydrochloride', 'newLinkedTargets_string': 'POLA1 (ENSG00000101868), POLD4 (ENSG00000175482), POLD3 (ENSG00000077514), POLD1 (ENSG00000062822), POLD2 (ENSG00000106628), POLE (ENSG00000177084), POLA2 (ENSG00000014138), PRIM1 (ENSG00000198056), PRIM2 (ENSG0000014...
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Q4.1039
Q4
What drugs target the gene PDCD1?
The drugs that target PDCD1 are Nivolumab, Cemiplimab, Pembrolizumab, and Dostarlimab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PDCD1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4032', 'drugName': 'Cemiplimab', 'newLinkedTargets_string': 'PDCD1 (ENSG00000188389)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1668', 'drugName': 'Nivolumab', 'newLinkedTargets_string': 'PDCD1 (ENSG00000188389)', 'drugIsApproved': True, 'maxClinica...
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Genetic Target
Q4.1067
Q4
What drugs target the gene PDK1?
The drug that targets PDK1 is Sodium Dichloroacetate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PDK1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2764', 'drugName': 'Sodium Dichloroacetate', 'newLinkedTargets_string': 'PDK2 (ENSG00000005882), PDK3 (ENSG00000067992), PDK4 (ENSG00000004799), PDK1 (ENSG00000152256)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}]
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Genetic Target
Q4.1149
Q4
What drugs target the gene PSEN2?
There are no FDA approved drugs targeting the gene PSEN2. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Tarenflurbil, Rg-4733, Nirogacestat, Avagacestat, Begacestat, and Semagacestat.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PSEN2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5562', 'drugName': 'Nirogacestat', 'newLinkedTargets_string': 'APH1A (ENSG00000117362), PSENEN (ENSG00000205155), APH1B (ENSG00000138613), PSEN1 (ENSG00000080815), NCSTN (ENSG00000162736), PSEN2 (ENSG00000143801)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTar...
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Q4.1193
Q4
What drugs target the gene PTGER3?
The drugs that target PTGER3 are Misoprostol and Dinoprostone.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PTGER3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4965', 'drugName': 'Dinoprostone', 'newLinkedTargets_string': 'PTGER1 (ENSG00000160951), PTGER4 (ENSG00000171522), PTGER2 (ENSG00000125384), PTGER3 (ENSG00000050628)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4262', 'drugName': 'Misoprostol', 'newLi...
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Genetic Target
Q4.1505
Q4
What drugs target the gene TUBB4A?
The drugs that target TUBB4A are Polatuzumab Vedotin, Cabazitaxel, Vinflunine, Brentuximab Vedotin, Docetaxel, Belantamab Mafodotin, Paclitaxel, Vinorelbine, Ixabepilone, Enfortumab Vedotin, Eribulin Mesylate, Vincristine Sulfate, Tisotumab Vedotin, Vinblastine, Colchicine, Vincristine, Eribulin, Trastuzumab Emtansine,...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TUBB4A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1084', 'drugName': 'Brentuximab Vedotin', 'newLinkedTargets_string': 'TNFRSF8 (ENSG00000120949), TUBB4B (ENSG00000188229), TUBB1 (ENSG00000101162), TUBA3C (ENSG00000198033), TUBA4A (ENSG00000127824), TUBB3 (ENSG00000258947), TUBA1A (ENSG00000167552), TUBB4A (ENSG00000104833), TUBB8 (ENSG00...
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Genetic Target
Q4.238
Q4
What drugs target the gene CDK17?
There are no FDA approved drugs targeting the gene CDK17. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Roniciclib, Pha-793887, Azd-5438, and At-7519.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CDK17 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1429', 'drugName': 'Roniciclib', 'newLinkedTargets_string': 'CDK1 (ENSG00000170312), CDK4 (ENSG00000135446), CDK2 (ENSG00000123374), CDK5 (ENSG00000164885), CDK6 (ENSG00000105810), CDK7 (ENSG00000134058), CDK3 (ENSG00000250506), CDK16 (ENSG00000102225), CDK18 (ENSG00000117266), CDK8 (ENSG0...
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Genetic Target
Q4.1362
Q4
What drugs target the gene SLC12A3?
The drugs that target SLC12A3 are Methyclothiazide, Hydrochlorothiazide, Hydroflumethiazide, Bendroflumethiazide, Indapamide, Cyclothiazide, Polythiazide, Benzthiazide, Trichlormethiazide, Chlorothiazide, Metolazone, Chlorthalidone, Chlorothiazide Sodium, and Quinethazone.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%SLC12A3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2403', 'drugName': 'Indapamide', 'newLinkedTargets_string': 'SLC12A3 (ENSG00000070915)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_926', 'drugName': 'Methyclothiazide', 'newLinkedTargets_string': 'SLC12A3 (ENSG00000070915)', 'drugIsApproved': True, '...
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Q4.992
Q4
What drugs target the gene NOX1?
There are no approved drugs targeting NOX1, but the drug Setanaxib, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NOX1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5524', 'drugName': 'Setanaxib', 'newLinkedTargets_string': 'NOX4 (ENSG00000086991), NOX1 (ENSG00000007952)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_5525', 'drugName': 'Setanaxib', 'newLinkedTargets_string': 'NOX4 (ENSG00000086991), NOX1 (ENSG0000...
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Genetic Target
Q4.1482
Q4
What drugs target the gene TRHR?
The drug that targets TRHR is Protirelin.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TRHR %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4776', 'drugName': 'Protirelin', 'newLinkedTargets_string': 'TRHR (ENSG00000174417)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5311', 'drugName': 'Rovatirelin', 'newLinkedTargets_string': 'TRHR (ENSG00000174417)', 'drugIsApproved': False, 'maxClinic...
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Q4.600
Q4
What drugs target the gene HPSE?
There are no approved drugs targeting HPSE, but the drug Muparfostat, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%HPSE %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5103', 'drugName': 'Muparfostat', 'newLinkedTargets_string': 'HPSE (ENSG00000173083), FGF1 (ENSG00000113578), FGF2 (ENSG00000138685), VEGFA (ENSG00000112715)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_5102', 'drugName': 'Muparfostat', 'newLinkedTar...
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Q4.500
Q4
What drugs target the gene GABRB2?
The drugs that target GABRB2 are Meprobamate, Acamprosate Calcium, Enflurane, Methohexital, Metharbital, Butabarbital, Flurazepam Hydrochloride, Pentobarbital Sodium, Acamprosate, Primidone, Temazepam, Flunitrazepam, Ganaxolone, Diazepam, Methyprylon, Thiopental, Clonazepam, Topiramate, Remimazolam Besylate, Brexanolon...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%GABRB2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1108', 'drugName': 'Temazepam', 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089), GABRA3 (ENSG00000011677), GABRP (ENSG00000094755)...
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Q4.210
Q4
What drugs target the gene CD38?
The drugs that target CD38 are Isatuximab and Daratumumab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CD38 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_169', 'drugName': 'Isatuximab', 'newLinkedTargets_string': 'CD38 (ENSG00000004468)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4167', 'drugName': 'Daratumumab', 'newLinkedTargets_string': 'CD38 (ENSG00000004468)', 'drugIsApproved': True, 'maxClinical...
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Q4.1081
Q4
What drugs target the gene PIK3R3?
There are no FDA approved drugs targeting the gene PIK3R3. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Bgt-226, Pictilisib, Zstk-474, Azd-6482, Gsk-1059615, Paxalisib, Sf-1126, Sonolisib, Samotolisib, Panulisib, Voxtalisib, Wx-037, Pf-04691502, Bupar...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PIK3R3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5563', 'drugName': 'Dactolisib', 'newLinkedTargets_string': 'PIK3R1 (ENSG00000145675), PIK3CB (ENSG00000051382), PIK3CG (ENSG00000105851), PIK3CA (ENSG00000121879), PIK3R2 (ENSG00000105647), PIK3CD (ENSG00000171608), PIK3R5 (ENSG00000141506), PIK3R3 (ENSG00000117461), MTOR (ENSG00000198793...
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Q4.413
Q4
What drugs target the gene EPHA6?
The drug that targets EPHA6 is Vandetanib.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%EPHA6 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1936', 'drugName': 'Vandetanib', 'newLinkedTargets_string': 'TEK (ENSG00000120156), ERBB2 (ENSG00000141736), EGFR (ENSG00000146648), ERBB4 (ENSG00000178568), ERBB3 (ENSG00000065361), EPHA2 (ENSG00000142627), EPHB2 (ENSG00000133216), EPHA5 (ENSG00000145242), EPHA4 (ENSG00000116106), EPHA8 (...
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Q4.1305
Q4
What drugs target the gene RPS6KA6?
There are no approved drugs targeting RPS6KA6, but the drug Tas0612, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RPS6KA6 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3347', 'drugName': 'Tas0612', 'newLinkedTargets_string': 'RPS6KB2 (ENSG00000175634), RPS6KB1 (ENSG00000108443), AKT2 (ENSG00000105221), AKT3 (ENSG00000117020), AKT1 (ENSG00000142208), RPS6KA3 (ENSG00000177189), RPS6KA2 (ENSG00000071242), RPS6KA6 (ENSG00000072133), RPS6KA1 (ENSG00000117676)...
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Q4.59
Q4
What drugs target the gene ALOX5AP?
There are no FDA approved drugs targeting the gene ALOX5AP. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Fiboflapon Sodium, Fiboflapon, and Veliflapon.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ALOX5AP %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_160', 'drugName': 'Fiboflapon Sodium', 'newLinkedTargets_string': 'ALOX5AP (ENSG00000132965)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_2102', 'drugName': 'Fiboflapon', 'newLinkedTargets_string': 'ALOX5AP (ENSG00000132965)', 'drugIsApproved': False...
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Q4.852
Q4
What drugs target the gene MAP3K12?
There are no approved drugs targeting MAP3K12, but the drug Cep-1347, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%MAP3K12 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6091', 'drugName': 'Cep-1347', 'newLinkedTargets_string': 'MAP3K13 (ENSG00000073803), MAP3K12 (ENSG00000139625), MAP3K10 (ENSG00000130758), MAP3K9 (ENSG00000006432), MAP3K11 (ENSG00000173327)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_6088', 'drugN...
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Q4.1333
Q4
What drugs target the gene SCN2A?
The drugs that target SCN2A are Propoxycaine, Orphenadrine, Indecainide, Quinidine Polygalacturonate, Fosphenytoin Sodium, Prilocaine Hydrochloride, Zonisamide, Mexiletine, Hexylcaine Hydrochloride, Fosphenytoin, Phenazopyridine Hydrochloride, Primidone, Phenytoin Sodium, Propafenone, Topiramate, Chloroprocaine, Etidoc...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%SCN2A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_485', 'drugName': 'Mexiletine', 'newLinkedTargets_string': 'SCN1A (ENSG00000144285), SCN5A (ENSG00000183873), SCN4A (ENSG00000007314), SCN7A (ENSG00000136546), SCN2A (ENSG00000136531), SCN9A (ENSG00000169432), SCN3A (ENSG00000153253), SCN11A (ENSG00000168356), SCN8A (ENSG00000196876), SCN1...
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Q4.429
Q4
What drugs target the gene ERVW-1?
There are no approved drugs targeting ERVW-1, but the drug Temelimab, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ERVW-1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1980', 'drugName': 'Temelimab', 'newLinkedTargets_string': 'ERVW-1 (ENSG00000242950)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
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Q4.1506
Q4
What drugs target the gene TUBB4B?
The drugs that target TUBB4B are Polatuzumab Vedotin, Cabazitaxel, Vinflunine, Brentuximab Vedotin, Docetaxel, Belantamab Mafodotin, Paclitaxel, Vinorelbine, Ixabepilone, Enfortumab Vedotin, Eribulin Mesylate, Vincristine Sulfate, Tisotumab Vedotin, Vinblastine, Colchicine, Vincristine, Eribulin, Trastuzumab Emtansine,...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TUBB4B %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1084', 'drugName': 'Brentuximab Vedotin', 'newLinkedTargets_string': 'TNFRSF8 (ENSG00000120949), TUBB4B (ENSG00000188229), TUBB1 (ENSG00000101162), TUBA3C (ENSG00000198033), TUBA4A (ENSG00000127824), TUBB3 (ENSG00000258947), TUBA1A (ENSG00000167552), TUBB4A (ENSG00000104833), TUBB8 (ENSG00...
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Q4.1220
Q4
What drugs target the gene RIPK1?
There are no approved drugs targeting RIPK1, but the drug Gsk2982772, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RIPK1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4958', 'drugName': 'Gsk2982772', 'newLinkedTargets_string': 'RIPK1 (ENSG00000137275)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
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Q4.1052
Q4
What drugs target the gene PDE5A?
The drugs that target PDE5A are Tadalafil, Vardenafil, Sildenafil Citrate, Pentoxifylline, Vardenafil Hydrochloride, Avanafil, Sildenafil, and Dipyridamole.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PDE5A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4264', 'drugName': 'Pentoxifylline', 'newLinkedTargets_string': 'ADORA2B (ENSG00000170425), ADORA2A (ENSG00000128271), PDE5A (ENSG00000138735), PDE4A (ENSG00000065989), PDE3A (ENSG00000172572), PDE6H (ENSG00000139053), PDE6G (ENSG00000185527), PDE2A (ENSG00000186642), PDE7A (ENSG0000020526...
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Q4.1240
Q4
What drugs target the gene RPL19?
The drug that targets RPL19 is Ataluren.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RPL19 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG00000083845), RPS7 (ENSG...
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