Datasets:

uuid
stringlengths
4
8
template_uuid
stringclasses
40 values
question
stringlengths
13
193
answer
stringlengths
29
2.2k
benchmark_query
stringlengths
133
622
execution_results
stringlengths
2
1.14M
query_type
stringclasses
2 values
sql_category
stringclasses
26 values
bio_category
stringclasses
14 values
Q4.1063
Q4
What drugs target the gene PDE9A?
The drugs that target PDE9A are Pentoxifylline and Dipyridamole.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PDE9A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4263', 'drugName': 'Pentoxifylline', 'newLinkedTargets_string': 'ADORA2B (ENSG00000170425), ADORA2A (ENSG00000128271), PDE5A (ENSG00000138735), PDE4A (ENSG00000065989), PDE3A (ENSG00000172572), PDE6H (ENSG00000139053), PDE6G (ENSG00000185527), PDE2A (ENSG00000186642), PDE7A (ENSG0000020526...
general
Select, Similarity Search, Order By
Genetic Target
Q4.1011
Q4
What drugs target the gene NRP1?
There are no approved drugs targeting NRP1, but the drug Vesencumab, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NRP1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1821', 'drugName': 'Vesencumab', 'newLinkedTargets_string': 'NRP1 (ENSG00000099250)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 1}]
general
Select, Similarity Search, Order By
Genetic Target
Q4.1433
Q4
What drugs target the gene TLR2?
There are no FDA approved drugs targeting the gene TLR2. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Tomaralimab and Vb-201.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TLR2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5402', 'drugName': 'Tomaralimab', 'newLinkedTargets_string': 'TLR2 (ENSG00000137462)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_5798', 'drugName': 'Vb-201', 'newLinkedTargets_string': 'TLR2 (ENSG00000137462), CD14 (ENSG00000170458)', 'drugIsApprove...
general
Select, Similarity Search, Order By
Genetic Target
Q4.131
Q4
What drugs target the gene CA12?
The drugs that target CA12 are Dichlorphenamide, Acetazolamide, Ethoxzolamide, Sulthiame, and Acetazolamide Sodium.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CA12 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_255', 'drugName': 'Dichlorphenamide', 'newLinkedTargets_string': 'CA1 (ENSG00000133742), CA12 (ENSG00000074410), CA2 (ENSG00000104267), CA4 (ENSG00000167434)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_6140', 'drugName': 'Acetazolamide Sodium', 'newL...
general
Select, Similarity Search, Order By
Genetic Target
Q4.1041
Q4
What drugs target the gene PDE10A?
The drugs that target PDE10A are Pentoxifylline and Dipyridamole.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PDE10A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4263', 'drugName': 'Pentoxifylline', 'newLinkedTargets_string': 'ADORA2B (ENSG00000170425), ADORA2A (ENSG00000128271), PDE5A (ENSG00000138735), PDE4A (ENSG00000065989), PDE3A (ENSG00000172572), PDE6H (ENSG00000139053), PDE6G (ENSG00000185527), PDE2A (ENSG00000186642), PDE7A (ENSG0000020526...
general
Select, Similarity Search, Order By
Genetic Target
Q4.333
Q4
What drugs target the gene CTSS?
There are no approved drugs targeting CTSS, but the drug Petesicatib, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CTSS %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1222', 'drugName': 'Petesicatib', 'newLinkedTargets_string': 'CTSS (ENSG00000163131)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
general
Select, Similarity Search, Order By
Genetic Target
Q4.325
Q4
What drugs target the gene CSNK1E?
The drugs that target CSNK1E are Umbralisib Tosylate and Umbralisib.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CSNK1E %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5649', 'drugName': 'Umbralisib', 'newLinkedTargets_string': 'CSNK1E (ENSG00000213923), PIK3CD (ENSG00000171608), ABL1 (ENSG00000097007)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3012', 'drugName': 'Umbralisib Tosylate', 'newLinkedTargets_string': '...
general
Select, Similarity Search, Order By
Genetic Target
Q4.1214
Q4
What drugs target the gene RBX1?
The drugs that target RBX1 are Thalidomide, Lenalidomide, and Pomalidomide.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RBX1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_64', 'drugName': 'Thalidomide', 'newLinkedTargets_string': 'CRBN (ENSG00000113851), DDB1 (ENSG00000167986), CUL4A (ENSG00000139842), RBX1 (ENSG00000100387)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4886', 'drugName': 'Pomalidomide', 'newLinkedTarge...
general
Select, Similarity Search, Order By
Genetic Target
Q4.1471
Q4
What drugs target the gene TP53?
There are no FDA approved drugs targeting the gene TP53. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Cenersen Sodium, Eprenetapopt, Apg115, Teprasiran Sodium, Cenersen, Idasanutlin, Siremadlin, Teprasiran, Contusugene Ladenovec, and Navtemadlin.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TP53 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3191', 'drugName': 'Idasanutlin', 'newLinkedTargets_string': 'TP53 (ENSG00000141510), MDM2 (ENSG00000135679)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_4656', 'drugName': 'Teprasiran', 'newLinkedTargets_string': 'TP53 (ENSG00000141510)', 'drugIsApp...
general
Select, Similarity Search, Order By
Genetic Target
Q4.772
Q4
What drugs target the gene KCNK9?
The drugs that target KCNK9 are Enflurane, Sevoflurane, Desflurane, Halothane, Isoflurane, Doxapram, and Doxapram Hydrochloride.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%KCNK9 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5595', 'drugName': 'Isoflurane', 'newLinkedTargets_string': 'KCNK10 (ENSG00000100433), KCNK9 (ENSG00000169427), GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089...
general
Select, Similarity Search, Order By
Genetic Target
Q4.137
Q4
What drugs target the gene CA5A?
The drugs that target CA5A are Ethoxzolamide and Sulthiame.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CA5A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6095', 'drugName': 'Sulthiame', 'newLinkedTargets_string': 'CA2 (ENSG00000104267), CA7 (ENSG00000168748), CA1 (ENSG00000133742), CA3 (ENSG00000164879), CA6 (ENSG00000131686), CA12 (ENSG00000074410), CA14 (ENSG00000118298), CA9 (ENSG00000107159), CA4 (ENSG00000167434), CA13 (ENSG00000185015...
general
Select, Similarity Search, Order By
Genetic Target
Q4.711
Q4
What drugs target the gene INPP5D?
There are no approved drugs targeting INPP5D, but the drug Rosiptor, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%INPP5D %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2977', 'drugName': 'Rosiptor', 'newLinkedTargets_string': 'INPP5D (ENSG00000168918)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}]
general
Select, Similarity Search, Order By
Genetic Target
Q4.531
Q4
What drugs target the gene GPA33?
There are no FDA approved drugs targeting the gene GPA33. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Hua33, A33 131I, and Krn-330.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%GPA33 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2310', 'drugName': 'A33 131I', 'newLinkedTargets_string': 'GPA33 (ENSG00000143167)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_231', 'drugName': 'Hua33', 'newLinkedTargets_string': 'GPA33 (ENSG00000143167)', 'drugIsApproved': False, 'maxClinicalTria...
general
Select, Similarity Search, Order By
Genetic Target
Q4.749
Q4
What drugs target the gene KCND3?
The drugs that target KCND3 are Vernakalant, Dalfampridine, Guanidine, Amifampridine Phosphate, Guanidine Hydrochloride, and Amifampridine.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%KCND3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1734', 'drugName': 'Dalfampridine', 'newLinkedTargets_string': 'KCNQ1 (ENSG00000053918), KCND3 (ENSG00000171385), KCNH2 (ENSG00000055118), KCNA2 (ENSG00000177301), KCNA1 (ENSG00000111262), KCNQ2 (ENSG00000075043), KCNQ3 (ENSG00000184156), KCNA7 (ENSG00000104848), KCNQ5 (ENSG00000185760), K...
general
Select, Similarity Search, Order By
Genetic Target
Q4.437
Q4
What drugs target the gene F13A1?
The drug that targets F13A1 is Catridecacog.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%F13A1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_886', 'drugName': 'Catridecacog', 'newLinkedTargets_string': 'F13A1 (ENSG00000124491)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}]
general
Select, Similarity Search, Order By
Genetic Target
Q4.682
Q4
What drugs target the gene IL1A?
There are no FDA approved drugs targeting the gene IL1A. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Lutikizumab and Bermekimab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%IL1A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2597', 'drugName': 'Bermekimab', 'newLinkedTargets_string': 'IL1A (ENSG00000115008)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_573', 'drugName': 'Lutikizumab', 'newLinkedTargets_string': 'IL1A (ENSG00000115008), IL1B (ENSG00000125538)', 'drugIsAppr...
general
Select, Similarity Search, Order By
Genetic Target
Q4.1340
Q4
What drugs target the gene SCNN1A?
The drugs that target SCNN1A are Amiloride Hydrochloride, Amiloride, and Triamterene.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%SCNN1A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2590', 'drugName': 'Amiloride Hydrochloride', 'newLinkedTargets_string': 'SCNN1A (ENSG00000111319), SCNN1B (ENSG00000168447), SCNN1G (ENSG00000166828)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4230', 'drugName': 'Triamterene', 'newLinkedTargets_str...
general
Select, Similarity Search, Order By
Genetic Target
Q4.160
Q4
What drugs target the gene CACNG1?
The drugs that target CACNG1 are Gabapentin, Terodiline Hydrochloride, Phloroglucinol, Suloctidil, Pregabalin, Gabapentin Enacarbil, Bepridil Hydrochloride, Bepridil, and Terodiline.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CACNG1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_142', 'drugName': 'Gabapentin', 'newLinkedTargets_string': 'CACNA1H (ENSG00000196557), CACNA2D1 (ENSG00000153956), CACNA1C (ENSG00000151067), CACNA2D3 (ENSG00000157445), CACNA1S (ENSG00000081248), CACNA2D2 (ENSG00000007402), CACNA1D (ENSG00000157388), CACNA1A (ENSG00000141837), CACNA1B (EN...
general
Select, Similarity Search, Order By
Genetic Target
Q4.595
Q4
What drugs target the gene HLA-DRB5?
There are no approved drugs targeting HLA-DRB5, but the drug Apolizumab, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%HLA-DRB5 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_363', 'drugName': 'Apolizumab', 'newLinkedTargets_string': 'HLA-DRB3 (ENSG00000231679), HLA-DRB5 (ENSG00000198502), HLA-DRB1 (ENSG00000196126), HLA-DRB4 (ENSG00000231021)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
general
Select, Similarity Search, Order By
Genetic Target
Q4.1221
Q4
What drugs target the gene RNPEP?
There are no approved drugs targeting RNPEP, but the drug Tosedostat, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RNPEP %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_582', 'drugName': 'Tosedostat', 'newLinkedTargets_string': 'ANPEP (ENSG00000166825), NPEPPS (ENSG00000141279), RNPEP (ENSG00000176393), METAP1 (ENSG00000164024), LNPEP (ENSG00000113441), DNPEP (ENSG00000123992), ENPEP (ENSG00000138792), XPNPEP1 (ENSG00000108039), LAP3 (ENSG00000002549), ME...
general
Select, Similarity Search, Order By
Genetic Target
Q4.197
Q4
What drugs target the gene CCR9?
There are no FDA approved drugs targeting the gene CCR9. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Vercirnon and Mln3126.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CCR9 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1403', 'drugName': 'Vercirnon', 'newLinkedTargets_string': 'CCR9 (ENSG00000173585)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_2090', 'drugName': 'Mln3126', 'newLinkedTargets_string': 'CCR9 (ENSG00000173585)', 'drugIsApproved': False, 'maxClinicalTr...
general
Select, Similarity Search, Order By
Genetic Target
Q4.1272
Q4
What drugs target the gene RPLP0?
The drug that targets RPLP0 is Ataluren.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RPLP0 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG00000083845), RPS7 (ENSG...
general
Select, Similarity Search, Order By
Genetic Target
Q4.530
Q4
What drugs target the gene GP6?
There are no approved drugs targeting GP6, but the drug Glenzocimab, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%GP6 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5071', 'drugName': 'Glenzocimab', 'newLinkedTargets_string': 'GP6 (ENSG00000088053)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
general
Select, Similarity Search, Order By
Genetic Target
Q4.412
Q4
What drugs target the gene EPHA5?
The drug that targets EPHA5 is Vandetanib.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%EPHA5 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1936', 'drugName': 'Vandetanib', 'newLinkedTargets_string': 'TEK (ENSG00000120156), ERBB2 (ENSG00000141736), EGFR (ENSG00000146648), ERBB4 (ENSG00000178568), ERBB3 (ENSG00000065361), EPHA2 (ENSG00000142627), EPHB2 (ENSG00000133216), EPHA5 (ENSG00000145242), EPHA4 (ENSG00000116106), EPHA8 (...
general
Select, Similarity Search, Order By
Genetic Target
Q4.98
Q4
What drugs target the gene AVPR2?
The drugs that target AVPR2 are Desmopressin, Lypressin, Conivaptan, Desmopressin Acetate, Vasopressin, Conivaptan Hydrochloride, Tolvaptan, Argipressin Tannate, Vasopressin Tannate, and Terlipressin.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%AVPR2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2993', 'drugName': 'Desmopressin Acetate', 'newLinkedTargets_string': 'AVPR2 (ENSG00000126895), AVPR1A (ENSG00000166148), AVPR1B (ENSG00000198049)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3359', 'drugName': 'Conivaptan Hydrochloride', 'newLinkedTa...
general
Select, Similarity Search, Order By
Genetic Target
Q4.1484
Q4
What drugs target the gene TRPM8?
The drug that targets TRPM8 is Menthol.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TRPM8 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5721', 'drugName': 'Menthol', 'newLinkedTargets_string': 'TRPA1 (ENSG00000104321), TRPM8 (ENSG00000144481)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5722', 'drugName': 'Menthol', 'newLinkedTargets_string': 'TRPA1 (ENSG00000104321), TRPM8 (ENSG00000...
general
Select, Similarity Search, Order By
Genetic Target
Q4.158
Q4
What drugs target the gene CACNB3?
The drugs that target CACNB3 are Gabapentin, Terodiline Hydrochloride, Phloroglucinol, Suloctidil, Pregabalin, Gabapentin Enacarbil, Bepridil Hydrochloride, Bepridil, and Terodiline.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CACNB3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_142', 'drugName': 'Gabapentin', 'newLinkedTargets_string': 'CACNA1H (ENSG00000196557), CACNA2D1 (ENSG00000153956), CACNA1C (ENSG00000151067), CACNA2D3 (ENSG00000157445), CACNA1S (ENSG00000081248), CACNA2D2 (ENSG00000007402), CACNA1D (ENSG00000157388), CACNA1A (ENSG00000141837), CACNA1B (EN...
general
Select, Similarity Search, Order By
Genetic Target
Q4.421
Q4
What drugs target the gene EPHX2?
There are no FDA approved drugs targeting the gene EPHX2. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Ar9281 and Gsk2256294.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%EPHX2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2804', 'drugName': 'Gsk2256294', 'newLinkedTargets_string': 'EPHX2 (ENSG00000120915)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_572', 'drugName': 'Ar9281', 'newLinkedTargets_string': 'EPHX2 (ENSG00000120915)', 'drugIsApproved': False, 'maxClinicalT...
general
Select, Similarity Search, Order By
Genetic Target
Q4.995
Q4
What drugs target the gene NPEPL1?
There are no approved drugs targeting NPEPL1, but the drug Tosedostat, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NPEPL1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_582', 'drugName': 'Tosedostat', 'newLinkedTargets_string': 'ANPEP (ENSG00000166825), NPEPPS (ENSG00000141279), RNPEP (ENSG00000176393), METAP1 (ENSG00000164024), LNPEP (ENSG00000113441), DNPEP (ENSG00000123992), ENPEP (ENSG00000138792), XPNPEP1 (ENSG00000108039), LAP3 (ENSG00000002549), ME...
general
Select, Similarity Search, Order By
Genetic Target
Q4.479
Q4
What drugs target the gene FOLR1?
There are no FDA approved drugs targeting the gene FOLR1. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Vintafolide, Farletuzumab, Mirvetuximab, and Mirvetuximab Soravtansine.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%FOLR1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5727', 'drugName': 'Mirvetuximab Soravtansine', 'newLinkedTargets_string': 'FOLR1 (ENSG00000110195), TUBB4B (ENSG00000188229), TUBB1 (ENSG00000101162), TUBA3C (ENSG00000198033), TUBA4A (ENSG00000127824), TUBB3 (ENSG00000258947), TUBA1A (ENSG00000167552), TUBB4A (ENSG00000104833), TUBB8 (EN...
general
Select, Similarity Search, Order By
Genetic Target
Q4.1201
Q4
What drugs target the gene PTK2?
There are no FDA approved drugs targeting the gene PTK2. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Bi-853520, Pf-00562271, Conteltinib , Defactinib, Cep-37440, Vs-4718, and Gsk-2256098.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PTK2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3099', 'drugName': 'Defactinib', 'newLinkedTargets_string': 'PTK2B (ENSG00000120899), PTK2 (ENSG00000169398)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_6171', 'drugName': 'Gsk-2256098', 'newLinkedTargets_string': 'PTK2 (ENSG00000169398)', 'drugIsAp...
general
Select, Similarity Search, Order By
Genetic Target
Q4.668
Q4
What drugs target the gene IL11RA?
The drug that targets IL11RA is Oprelvekin.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%IL11RA %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2215', 'drugName': 'Oprelvekin', 'newLinkedTargets_string': 'IL11RA (ENSG00000137070)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}]
general
Select, Similarity Search, Order By
Genetic Target
Q4.1236
Q4
What drugs target the gene RPL15?
The drug that targets RPL15 is Ataluren.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RPL15 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG00000083845), RPS7 (ENSG...
general
Select, Similarity Search, Order By
Genetic Target
Q4.449
Q4
What drugs target the gene FAU?
The drug that targets FAU is Ataluren.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%FAU %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG00000083845), RPS7 (ENSG...
general
Select, Similarity Search, Order By
Genetic Target
Q4.180
Q4
What drugs target the gene CASP5?
There are no approved drugs targeting CASP5, but the drug Emricasan, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CASP5 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_45', 'drugName': 'Emricasan', 'newLinkedTargets_string': 'CASP4 (ENSG00000196954), CASP9 (ENSG00000132906), CASP3 (ENSG00000164305), CASP5 (ENSG00000137757), CASP6 (ENSG00000138794), CASP7 (ENSG00000165806), CASP8 (ENSG00000064012), CASP1 (ENSG00000137752), CASP2 (ENSG00000106144), CASP10 ...
general
Select, Similarity Search, Order By
Genetic Target
Q4.392
Q4
What drugs target the gene EGFL7?
There are no approved drugs targeting EGFL7, but the drug Parsatuzumab, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%EGFL7 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5915', 'drugName': 'Parsatuzumab', 'newLinkedTargets_string': 'EGFL7 (ENSG00000172889)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
general
Select, Similarity Search, Order By
Genetic Target
Q4.1322
Q4
What drugs target the gene RXRG?
The drugs that target RXRG are Etretinate, Alitretinoin, Bexarotene, and Acitretin.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RXRG %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5080', 'drugName': 'Acitretin', 'newLinkedTargets_string': 'RXRB (ENSG00000204231), RARG (ENSG00000172819), RXRG (ENSG00000143171), RARB (ENSG00000077092), RARA (ENSG00000131759), RXRA (ENSG00000186350)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_701...
general
Select, Similarity Search, Order By
Genetic Target
Q4.935
Q4
What drugs target the gene NDUFA1?
The drugs that target NDUFA1 are Metformin and Metformin Hydrochloride.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NDUFA1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (ENSG00000165264), NDUFA4 (...
general
Select, Similarity Search, Order By
Genetic Target
Q4.1388
Q4
What drugs target the gene SOD1?
There are no approved drugs targeting SOD1, but the drug Tofersen, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%SOD1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_651', 'drugName': 'Tofersen', 'newLinkedTargets_string': 'SOD1 (ENSG00000142168)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}]
general
Select, Similarity Search, Order By
Genetic Target
Q4.625
Q4
What drugs target the gene HTR3C?
The drugs that target HTR3C are Zimeldine, Amisulpride, Clothiapine, Dexfenfluramine, Tropisetron, Dexfenfluramine Hydrochloride, and Zimeldine Hydrochloride.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%HTR3C %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2386', 'drugName': 'Clothiapine', 'newLinkedTargets_string': 'HTR2B (ENSG00000135914), HTR2A (ENSG00000102468), HTR2C (ENSG00000147246), DRD4 (ENSG00000069696), HTR3A (ENSG00000166736), HTR3E (ENSG00000186038), HTR3B (ENSG00000149305), HTR3D (ENSG00000186090), HTR3C (ENSG00000178084)', 'dr...
general
Select, Similarity Search, Order By
Genetic Target
Q4.594
Q4
What drugs target the gene HLA-DRB4?
There are no approved drugs targeting HLA-DRB4, but the drug Apolizumab, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%HLA-DRB4 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_363', 'drugName': 'Apolizumab', 'newLinkedTargets_string': 'HLA-DRB3 (ENSG00000231679), HLA-DRB5 (ENSG00000198502), HLA-DRB1 (ENSG00000196126), HLA-DRB4 (ENSG00000231021)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
general
Select, Similarity Search, Order By
Genetic Target
Q4.1510
Q4
What drugs target the gene TXK?
There are no approved drugs targeting TXK, but the drug Pf-06651600, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TXK %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4380', 'drugName': 'Pf-06651600', 'newLinkedTargets_string': 'ITK (ENSG00000113263), BMX (ENSG00000102010), TEC (ENSG00000135605), TXK (ENSG00000074966), BTK (ENSG00000010671), JAK3 (ENSG00000105639)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_4381'...
general
Select, Similarity Search, Order By
Genetic Target
Q4.893
Q4
What drugs target the gene MMP1?
The drugs that target MMP1 are Doxycycline Anhydrous, Doxycycline Hyclate, Doxycycline, and Doxycycline Calcium.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%MMP1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2398', 'drugName': 'Doxycycline Hyclate', 'newLinkedTargets_string': 'MMP13 (ENSG00000137745), MMP1 (ENSG00000196611), MMP7 (ENSG00000137673), MMP8 (ENSG00000118113)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3046', 'drugName': 'Doxycycline', 'newLi...
general
Select, Similarity Search, Order By
Genetic Target
Q4.814
Q4
What drugs target the gene LAP3?
There are no approved drugs targeting LAP3, but the drug Tosedostat, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%LAP3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_582', 'drugName': 'Tosedostat', 'newLinkedTargets_string': 'ANPEP (ENSG00000166825), NPEPPS (ENSG00000141279), RNPEP (ENSG00000176393), METAP1 (ENSG00000164024), LNPEP (ENSG00000113441), DNPEP (ENSG00000123992), ENPEP (ENSG00000138792), XPNPEP1 (ENSG00000108039), LAP3 (ENSG00000002549), ME...
general
Select, Similarity Search, Order By
Genetic Target
Q4.905
Q4
What drugs target the gene MSLN?
There are no FDA approved drugs targeting the gene MSLN. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Rg-7600, Lmb-100, Amatuximab, Anetumab Ravtansine, and Ss1(Dsfv)-Pe38.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%MSLN %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1866', 'drugName': 'Lmb-100', 'newLinkedTargets_string': 'MSLN (ENSG00000102854), EEF2 (ENSG00000167658)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_1867', 'drugName': 'Lmb-100', 'newLinkedTargets_string': 'MSLN (ENSG00000102854), EEF2 (ENSG00000167...
general
Select, Similarity Search, Order By
Genetic Target
Q4.1195
Q4
What drugs target the gene PTGFR?
The drugs that target PTGFR are Latanoprost, Bimatoprost, Dinoprost, Latanoprostene Bunod, Carboprost Tromethamine, Dinoprost Tromethamine, Travoprost, Tafluprost, and Carboprost.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PTGFR %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3870', 'drugName': 'Travoprost', 'newLinkedTargets_string': 'PTGFR (ENSG00000122420)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5593', 'drugName': 'Carboprost', 'newLinkedTargets_string': 'PTGFR (ENSG00000122420)', 'drugIsApproved': True, 'maxClinic...
general
Select, Similarity Search, Order By
Genetic Target
Q4.296
Q4
What drugs target the gene COL4A1?
The drugs that target COL4A1 are Collagenase Clostridium Histolyticum and Ocriplasmin.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%COL4A1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5818', 'drugName': 'Ocriplasmin', 'newLinkedTargets_string': 'FN1 (ENSG00000115414), COL1A2 (ENSG00000164692), COL1A1 (ENSG00000108821), COL2A1 (ENSG00000139219), COL3A1 (ENSG00000168542), COL4A1 (ENSG00000187498), COL5A1 (ENSG00000130635), COL6A1 (ENSG00000142156), COL11A1 (ENSG0000006071...
general
Select, Similarity Search, Order By
Genetic Target
Q4.1126
Q4
What drugs target the gene PRKAB1?
There are no approved drugs targeting PRKAB1, but the drug Acadesine, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PRKAB1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5888', 'drugName': 'Acadesine', 'newLinkedTargets_string': 'PRKAA2 (ENSG00000162409), PRKAB2 (ENSG00000131791), PRKAG1 (ENSG00000181929), PRKAG2 (ENSG00000106617), PRKAB1 (ENSG00000111725), PRKAA1 (ENSG00000132356), PRKAG3 (ENSG00000115592)', 'drugIsApproved': False, 'maxClinicalTrialPhase...
general
Select, Similarity Search, Order By
Genetic Target
Q4.898
Q4
What drugs target the gene MMP3?
There are no FDA approved drugs targeting the gene MMP3. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Cts-1027 and Marimastat.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%MMP3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5863', 'drugName': 'Marimastat', 'newLinkedTargets_string': 'MMP9 (ENSG00000100985), MMP3 (ENSG00000149968), MMP7 (ENSG00000137673), MMP1 (ENSG00000196611), MMP2 (ENSG00000087245), MMP12 (ENSG00000262406)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_...
general
Select, Similarity Search, Order By
Genetic Target
Q4.90
Q4
What drugs target the gene ATP4A?
The drugs that target ATP4A are Dexlansoprazole, Pantoprazole Sodium, Esomeprazole, Esomeprazole Strontium, Lansoprazole, Omeprazole Magnesium, Rabeprazole, Esomeprazole Sodium, Esomeprazole Magnesium, Omeprazole, Pantoprazole, Rabeprazole Sodium, Vonoprazan, and Vonoprazan Fumarate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ATP4A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5144', 'drugName': 'Rabeprazole Sodium', 'newLinkedTargets_string': 'ATP4A (ENSG00000105675), ATP4B (ENSG00000186009)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4835', 'drugName': 'Pantoprazole', 'newLinkedTargets_string': 'ATP4A (ENSG00000105675), ...
general
Select, Similarity Search, Order By
Genetic Target
Q4.1007
Q4
What drugs target the gene NR1H4?
The drugs that target NR1H4 are Chenodiol, Obeticholic Acid, and Ursodiol.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NR1H4 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4210', 'drugName': 'Ursodiol', 'newLinkedTargets_string': 'NR1H4 (ENSG00000012504)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3863', 'drugName': 'Obeticholic Acid', 'newLinkedTargets_string': 'NR1H4 (ENSG00000012504)', 'drugIsApproved': True, 'maxCl...
general
Select, Similarity Search, Order By
Genetic Target
Q4.990
Q4
What drugs target the gene NOTCH2?
There are no approved drugs targeting NOTCH2, but the drug Tarextumab, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NOTCH2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4401', 'drugName': 'Tarextumab', 'newLinkedTargets_string': 'NOTCH2 (ENSG00000134250), NOTCH3 (ENSG00000074181)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 1}, {'UUID': 'DrugGeneTargets_v2_4402', 'drugName': 'Tarextumab', 'newLinkedTargets_string': 'NOTCH2 (ENSG00000134250), NOTCH3...
general
Select, Similarity Search, Order By
Genetic Target
Q4.1427
Q4
What drugs target the gene TGFBR1?
There are no FDA approved drugs targeting the gene TGFBR1. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Vactosertib and Galunisertib.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TGFBR1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_166', 'drugName': 'Vactosertib', 'newLinkedTargets_string': 'TGFBR1 (ENSG00000106799)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_818', 'drugName': 'Galunisertib', 'newLinkedTargets_string': 'TGFBR1 (ENSG00000106799)', 'drugIsApproved': False, 'maxC...
general
Select, Similarity Search, Order By
Genetic Target
Q4.683
Q4
What drugs target the gene IL1B?
The drugs that target IL1B are Rilonacept and Canakinumab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%IL1B %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5122', 'drugName': 'Canakinumab', 'newLinkedTargets_string': 'IL1B (ENSG00000125538)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3681', 'drugName': 'Rilonacept', 'newLinkedTargets_string': 'IL1B (ENSG00000125538)', 'drugIsApproved': True, 'maxClinica...
general
Select, Similarity Search, Order By
Genetic Target
Q4.1423
Q4
What drugs target the gene TGFA?
There are no approved drugs targeting TGFA, but the drug Fepixnebart, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TGFA %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_509', 'drugName': 'Fepixnebart', 'newLinkedTargets_string': 'TGFA (ENSG00000163235), EREG (ENSG00000124882)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_510', 'drugName': 'Fepixnebart', 'newLinkedTargets_string': 'TGFA (ENSG00000163235), EREG (ENSG00...
general
Select, Similarity Search, Order By
Genetic Target
Q4.720
Q4
What drugs target the gene ITGAM?
There are no approved drugs targeting ITGAM, but the drug Rovelizumab, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ITGAM %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_553', 'drugName': 'Rovelizumab', 'newLinkedTargets_string': 'ITGB2 (ENSG00000160255), ITGAM (ENSG00000169896), ITGAL (ENSG00000005844)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_554', 'drugName': 'Rovelizumab', 'newLinkedTargets_string': 'ITGB2 (EN...
general
Select, Similarity Search, Order By
Genetic Target
Q4.973
Q4
What drugs target the gene NDUFS7?
The drugs that target NDUFS7 are Metformin and Metformin Hydrochloride.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NDUFS7 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (ENSG00000165264), NDUFA4 (...
general
Select, Similarity Search, Order By
Genetic Target
Q4.292
Q4
What drugs target the gene COL27A1?
The drugs that target COL27A1 are Collagenase Clostridium Histolyticum and Ocriplasmin.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%COL27A1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5818', 'drugName': 'Ocriplasmin', 'newLinkedTargets_string': 'FN1 (ENSG00000115414), COL1A2 (ENSG00000164692), COL1A1 (ENSG00000108821), COL2A1 (ENSG00000139219), COL3A1 (ENSG00000168542), COL4A1 (ENSG00000187498), COL5A1 (ENSG00000130635), COL6A1 (ENSG00000142156), COL11A1 (ENSG0000006071...
general
Select, Similarity Search, Order By
Genetic Target
Q4.1454
Q4
What drugs target the gene TNFSF12?
There are no FDA approved drugs targeting the gene TNFSF12. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Biib-023 and Ro-5458640.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TNFSF12 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1562', 'drugName': 'Biib-023', 'newLinkedTargets_string': 'TNFSF12 (ENSG00000239697)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_5094', 'drugName': 'Ro-5458640', 'newLinkedTargets_string': 'TNFSF12 (ENSG00000239697)', 'drugIsApproved': False, 'maxCl...
general
Select, Similarity Search, Order By
Genetic Target
Q4.615
Q4
What drugs target the gene HTR1A?
The drugs that target HTR1A are Buspirone, Vortioxetine Hydrobromide, Zimeldine, Amisulpride, Vortioxetine, Aripiprazole, Methysergide Maleate, Dexfenfluramine, Ergoloid Mesylates, Methysergide, Dexfenfluramine Hydrochloride, Buspirone Hydrochloride, Aripiprazole Lauroxil, Alverine, Vilazodone, Ergoloid, Vilazodone Hyd...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%HTR1A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4681', 'drugName': 'Aripiprazole Lauroxil', 'newLinkedTargets_string': 'DRD2 (ENSG00000149295), HTR2A (ENSG00000102468), HTR1A (ENSG00000178394)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2808', 'drugName': 'Methysergide Maleate', 'newLinkedTargets_...
general
Select, Similarity Search, Order By
Genetic Target
Q4.350
Q4
What drugs target the gene CYP3A5?
The drugs that target CYP3A5 are Ritonavir and Cobicistat.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CYP3A5 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2751', 'drugName': 'Ritonavir', 'newLinkedTargets_string': 'CYP3A4 (ENSG00000160868), CYP3A5 (ENSG00000106258), CYP3A43 (ENSG00000021461), CYP3A7 (ENSG00000160870)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2752', 'drugName': 'Ritonavir', 'newLinked...
general
Select, Similarity Search, Order By
Genetic Target
Q4.587
Q4
What drugs target the gene HDAC6?
The drugs that target HDAC6 are Belinostat, Vorinostat, Panobinostat, Panobinostat Lactate, and Romidepsin.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%HDAC6 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1601', 'drugName': 'Belinostat', 'newLinkedTargets_string': 'HDAC1 (ENSG00000116478), HDAC3 (ENSG00000171720), HDAC6 (ENSG00000094631), HDAC2 (ENSG00000196591), HDAC5 (ENSG00000108840), HDAC7 (ENSG00000061273), HDAC8 (ENSG00000147099), HDAC11 (ENSG00000163517), HDAC4 (ENSG00000068024), HDA...
general
Select, Similarity Search, Order By
Genetic Target
Q4.1518
Q4
What drugs target the gene UBA3?
There are no approved drugs targeting UBA3, but the drug Pevonedistat, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%UBA3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3764', 'drugName': 'Pevonedistat', 'newLinkedTargets_string': 'UBA3 (ENSG00000144744), NAE1 (ENSG00000159593)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}]
general
Select, Similarity Search, Order By
Genetic Target
Q4.1358
Q4
What drugs target the gene SLAMF7?
The drug that targets SLAMF7 is Elotuzumab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%SLAMF7 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5815', 'drugName': 'Elotuzumab', 'newLinkedTargets_string': 'SLAMF7 (ENSG00000026751)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1646', 'drugName': 'Azintuxizumab Vedotin', 'newLinkedTargets_string': 'TUBB4B (ENSG00000188229), TUBB1 (ENSG00000101162...
general
Select, Similarity Search, Order By
Genetic Target
Q4.1379
Q4
What drugs target the gene SLC9A3?
The drugs that target SLC9A3 are Tenapanor Hydrochloride and Tenapanor.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%SLC9A3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4791', 'drugName': 'Tenapanor', 'newLinkedTargets_string': 'SLC9A3 (ENSG00000066230)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3816', 'drugName': 'Tenapanor Hydrochloride', 'newLinkedTargets_string': 'SLC9A3 (ENSG00000066230)', 'drugIsApproved': Tr...
general
Select, Similarity Search, Order By
Genetic Target
Q4.619
Q4
What drugs target the gene HTR1F?
The drugs that target HTR1F are Zimeldine, Amisulpride, Lasmiditan Succinate, Eletriptan, Almotriptan, Dexfenfluramine, Almotriptan Malate, Dexfenfluramine Hydrochloride, Eletriptan Hydrobromide, Lasmiditan, and Zimeldine Hydrochloride.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%HTR1F %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2456', 'drugName': 'Eletriptan', 'newLinkedTargets_string': 'HTR1F (ENSG00000179097), HTR1D (ENSG00000179546), HTR1B (ENSG00000135312)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3458', 'drugName': 'Almotriptan Malate', 'newLinkedTargets_string': 'HT...
general
Select, Similarity Search, Order By
Genetic Target
Q4.460
Q4
What drugs target the gene FGB?
The drug that targets FGB is Fibrinolysin and Human.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%FGB %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1199', 'drugName': 'Fibrinolysin, Human', 'newLinkedTargets_string': 'FGA (ENSG00000171560), FGB (ENSG00000171564), FGG (ENSG00000171557)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5760', 'drugName': 'Fibrinogen, Human', 'newLinkedTargets_string': '...
general
Select, Similarity Search, Order By
Genetic Target
Q4.377
Q4
What drugs target the gene DRD5?
The drugs that target DRD5 are Amoxapine, Pimozide, Ergoloid Mesylates, Pergolide, Ergoloid, and Pergolide Mesylate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%DRD5 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3173', 'drugName': 'Pimozide', 'newLinkedTargets_string': 'DRD2 (ENSG00000149295), DRD3 (ENSG00000151577), DRD5 (ENSG00000169676), DRD4 (ENSG00000069696), DRD1 (ENSG00000184845), HTR2A (ENSG00000102468)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_237...
general
Select, Similarity Search, Order By
Genetic Target
Q4.335
Q4
What drugs target the gene CX3CL1?
There are no approved drugs targeting CX3CL1, but the drug Quetmolimab, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CX3CL1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_537', 'drugName': 'Quetmolimab', 'newLinkedTargets_string': 'CX3CL1 (ENSG00000006210)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
general
Select, Similarity Search, Order By
Genetic Target
Q4.782
Q4
What drugs target the gene KCNS3?
The drugs that target KCNS3 are Dalfampridine, Guanidine, Amifampridine Phosphate, Guanidine Hydrochloride, and Amifampridine.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%KCNS3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5118', 'drugName': 'Guanidine Hydrochloride', 'newLinkedTargets_string': 'KCNQ1 (ENSG00000053918), KCND3 (ENSG00000171385), KCNH2 (ENSG00000055118), KCNA2 (ENSG00000177301), KCNA1 (ENSG00000111262), KCNQ2 (ENSG00000075043), KCNQ3 (ENSG00000184156), KCNA7 (ENSG00000104848), KCNQ5 (ENSG00000...
general
Select, Similarity Search, Order By
Genetic Target
Q4.1356
Q4
What drugs target the gene SIGMAR1?
The drugs that target SIGMAR1 are Fenfluramine, Pentazocine Lactate, Pentazocine, Carbetapentane, Pentazocine Hydrochloride, Dextromethorphan Polistirex, Fenfluramine Hydrochloride, Dextromethorphan, Carbetapentane Citrate, and Dextromethorphan Hydrobromide.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%SIGMAR1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5072', 'drugName': 'Dextromethorphan', 'newLinkedTargets_string': 'GRIN2A (ENSG00000183454), SIGMAR1 (ENSG00000147955)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5996', 'drugName': 'Dextromethorphan Hydrobromide', 'newLinkedTargets_string': 'GRIN2A ...
general
Select, Similarity Search, Order By
Genetic Target
Q4.735
Q4
What drugs target the gene KCNA2?
The drugs that target KCNA2 are Dalfampridine, Guanidine, Amifampridine Phosphate, Guanidine Hydrochloride, and Amifampridine.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%KCNA2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5118', 'drugName': 'Guanidine Hydrochloride', 'newLinkedTargets_string': 'KCNQ1 (ENSG00000053918), KCND3 (ENSG00000171385), KCNH2 (ENSG00000055118), KCNA2 (ENSG00000177301), KCNA1 (ENSG00000111262), KCNQ2 (ENSG00000075043), KCNQ3 (ENSG00000184156), KCNA7 (ENSG00000104848), KCNQ5 (ENSG00000...
general
Select, Similarity Search, Order By
Genetic Target
Q4.1425
Q4
What drugs target the gene TGFB2?
The drug that targets TGFB2 is Luspatercept.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TGFB2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6093', 'drugName': 'Luspatercept', 'newLinkedTargets_string': 'TGFB1 (ENSG00000105329), TGFB2 (ENSG00000092969), TGFB3 (ENSG00000119699)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3208', 'drugName': 'Bintrafusp Alfa', 'newLinkedTargets_string': 'TGF...
general
Select, Similarity Search, Order By
Genetic Target
Q4.586
Q4
What drugs target the gene HDAC5?
The drugs that target HDAC5 are Belinostat, Panobinostat, Panobinostat Lactate, and Romidepsin.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%HDAC5 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4906', 'drugName': 'Panobinostat', 'newLinkedTargets_string': 'HDAC1 (ENSG00000116478), HDAC3 (ENSG00000171720), HDAC6 (ENSG00000094631), HDAC2 (ENSG00000196591), HDAC5 (ENSG00000108840), HDAC7 (ENSG00000061273), HDAC8 (ENSG00000147099), HDAC11 (ENSG00000163517), HDAC4 (ENSG00000068024), H...
general
Select, Similarity Search, Order By
Genetic Target
Q4.330
Q4
What drugs target the gene CTNNB1?
There are no approved drugs targeting CTNNB1, but the drug Pri-724, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CTNNB1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3141', 'drugName': 'Pri-724', 'newLinkedTargets_string': 'CREBBP (ENSG00000005339), CTNNB1 (ENSG00000168036)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
general
Select, Similarity Search, Order By
Genetic Target
Q4.320
Q4
What drugs target the gene CSF1R?
The drugs that target CSF1R are Pazopanib Hydrochloride, Pexidartinib, Sunitinib, Sunitinib Malate, Pexidartinib Hydrochloride, and Pazopanib.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CSF1R %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3920', 'drugName': 'Sunitinib Malate', 'newLinkedTargets_string': 'PDGFRB (ENSG00000113721), PDGFRA (ENSG00000134853), RET (ENSG00000165731), FLT1 (ENSG00000102755), FLT4 (ENSG00000037280), KDR (ENSG00000128052), CSF1R (ENSG00000182578), FLT3 (ENSG00000122025), KIT (ENSG00000157404)', 'dru...
general
Select, Similarity Search, Order By
Genetic Target
Q4.1181
Q4
What drugs target the gene PSMD2?
The drugs that target PSMD2 are Bortezomib, Carfilzomib, Ixazomib, and Ixazomib Citrate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PSMD2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_559', 'drugName': 'Bortezomib', 'newLinkedTargets_string': 'PSMD1 (ENSG00000173692), PSMB2 (ENSG00000126067), PSMB1 (ENSG00000008018), PSMB5 (ENSG00000100804), PSMB8 (ENSG00000204264), PSMB9 (ENSG00000240065), PSMB6 (ENSG00000142507), PSMD14 (ENSG00000115233), PSMA1 (ENSG00000129084), PSMA...
general
Select, Similarity Search, Order By
Genetic Target
Q4.982
Q4
What drugs target the gene NGF?
There are no FDA approved drugs targeting the gene NGF. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Fasinumab, Tanezumab, Medi-578, Fulranumab, and Pg-110.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NGF %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5018', 'drugName': 'Fulranumab', 'newLinkedTargets_string': 'NGF (ENSG00000134259)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_3772', 'drugName': 'Tanezumab', 'newLinkedTargets_string': 'NGF (ENSG00000134259)', 'drugIsApproved': False, 'maxClinicalT...
general
Select, Similarity Search, Order By
Genetic Target
Q4.13
Q4
What drugs target the gene ACLY?
The drug that targets ACLY is Bempedoic Acid.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ACLY %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5953', 'drugName': 'Bempedoic Acid', 'newLinkedTargets_string': 'ACLY (ENSG00000131473)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}]
general
Select, Similarity Search, Order By
Genetic Target
Q4.173
Q4
What drugs target the gene CASP1?
There are no FDA approved drugs targeting the gene CASP1. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Emricasan, Nivocasan, and Belnacasan.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CASP1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1849', 'drugName': 'Nivocasan', 'newLinkedTargets_string': 'CASP8 (ENSG00000064012), CASP1 (ENSG00000137752), CASP9 (ENSG00000132906)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_5967', 'drugName': 'Belnacasan', 'newLinkedTargets_string': 'CASP1 (ENS...
general
Select, Similarity Search, Order By
Genetic Target
Q4.262
Q4
What drugs target the gene CHRM4?
The drugs that target CHRM4 are Terodiline Hydrochloride and Terodiline.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CHRM4 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_311', 'drugName': 'Terodiline Hydrochloride', 'newLinkedTargets_string': 'CHRM3 (ENSG00000133019), CHRM4 (ENSG00000180720), CHRM1 (ENSG00000168539), CHRM2 (ENSG00000181072), CHRM5 (ENSG00000184984), CACNA1H (ENSG00000196557), CACNA2D1 (ENSG00000153956), CACNA1C (ENSG00000151067), CACNA2D3 ...
general
Select, Similarity Search, Order By
Genetic Target
Q4.996
Q4
What drugs target the gene NPEPPS?
There are no approved drugs targeting NPEPPS, but the drug Tosedostat, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NPEPPS %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_582', 'drugName': 'Tosedostat', 'newLinkedTargets_string': 'ANPEP (ENSG00000166825), NPEPPS (ENSG00000141279), RNPEP (ENSG00000176393), METAP1 (ENSG00000164024), LNPEP (ENSG00000113441), DNPEP (ENSG00000123992), ENPEP (ENSG00000138792), XPNPEP1 (ENSG00000108039), LAP3 (ENSG00000002549), ME...
general
Select, Similarity Search, Order By
Genetic Target
Q4.1148
Q4
What drugs target the gene PSEN1?
There are no FDA approved drugs targeting the gene PSEN1. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Tarenflurbil, Rg-4733, Nirogacestat, Avagacestat, Begacestat, and Semagacestat.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PSEN1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5562', 'drugName': 'Nirogacestat', 'newLinkedTargets_string': 'APH1A (ENSG00000117362), PSENEN (ENSG00000205155), APH1B (ENSG00000138613), PSEN1 (ENSG00000080815), NCSTN (ENSG00000162736), PSEN2 (ENSG00000143801)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTar...
general
Select, Similarity Search, Order By
Genetic Target
Q4.823
Q4
What drugs target the gene LINGO1?
There are no approved drugs targeting LINGO1, but the drug Opicinumab, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%LINGO1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2176', 'drugName': 'Opicinumab', 'newLinkedTargets_string': 'LINGO1 (ENSG00000169783)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
general
Select, Similarity Search, Order By
Genetic Target
Q4.140
Q4
What drugs target the gene CA7?
The drugs that target CA7 are Ethoxzolamide, Methazolamide, and Sulthiame.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CA7 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3089', 'drugName': 'Ethoxzolamide', 'newLinkedTargets_string': 'CA2 (ENSG00000104267), CA7 (ENSG00000168748), CA1 (ENSG00000133742), CA3 (ENSG00000164879), CA6 (ENSG00000131686), CA12 (ENSG00000074410), CA14 (ENSG00000118298), CA9 (ENSG00000107159), CA4 (ENSG00000167434), CA13 (ENSG0000018...
general
Select, Similarity Search, Order By
Genetic Target
Q4.552
Q4
What drugs target the gene GRIN2D?
The drugs that target GRIN2D are Orphenadrine, Acamprosate Calcium, Felbamate, Amantadine Hydrochloride, Esketamine Hydrochloride, Acamprosate, Ketamine Hydrochloride, Memantine, Ketamine, Amantadine, Orphenadrine Hydrochloride, Esketamine, Memantine Hydrochloride, and Orphenadrine Citrate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%GRIN2D %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6209', 'drugName': 'Orphenadrine Citrate', 'newLinkedTargets_string': 'GRIN1 (ENSG00000176884), GRIN2A (ENSG00000183454), GRIN2B (ENSG00000273079), GRIN2D (ENSG00000105464), GRIN3B (ENSG00000116032), GRIN2C (ENSG00000161509), GRIN3A (ENSG00000198785), HRH1 (ENSG00000196639), SLC6A2 (ENSG00...
general
Select, Similarity Search, Order By
Genetic Target
Q4.633
Q4
What drugs target the gene ICAM1?
There are no FDA approved drugs targeting the gene ICAM1. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Alicaforsen Sodium, Bi-505, Alicaforsen, Enlimomab, and Enlimomab Pegol.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ICAM1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2026', 'drugName': 'Alicaforsen', 'newLinkedTargets_string': 'ICAM1 (ENSG00000090339)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_5504', 'drugName': 'Enlimomab Pegol', 'newLinkedTargets_string': 'ICAM1 (ENSG00000090339)', 'drugIsApproved': False, 'm...
general
Select, Similarity Search, Order By
Genetic Target
Q4.873
Q4
What drugs target the gene MC4R?
The drugs that target MC4R are Bremelanotide Acetate, Setmelanotide, Setmelanotide Acetate, and Bremelanotide.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%MC4R %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2878', 'drugName': 'Setmelanotide Acetate', 'newLinkedTargets_string': 'MC4R (ENSG00000166603)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4990', 'drugName': 'Bremelanotide', 'newLinkedTargets_string': 'MC4R (ENSG00000166603)', 'drugIsApproved': True...
general
Select, Similarity Search, Order By
Genetic Target
Q4.804
Q4
What drugs target the gene LAMA3?
The drug that targets LAMA3 is Ocriplasmin.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%LAMA3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5818', 'drugName': 'Ocriplasmin', 'newLinkedTargets_string': 'FN1 (ENSG00000115414), COL1A2 (ENSG00000164692), COL1A1 (ENSG00000108821), COL2A1 (ENSG00000139219), COL3A1 (ENSG00000168542), COL4A1 (ENSG00000187498), COL5A1 (ENSG00000130635), COL6A1 (ENSG00000142156), COL11A1 (ENSG0000006071...
general
Select, Similarity Search, Order By
Genetic Target
Q4.561
Q4
What drugs target the gene GSR?
The drugs that target GSR are Carmustine and Oxiglutatione.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%GSR %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4261', 'drugName': 'Carmustine', 'newLinkedTargets_string': 'GSR (ENSG00000104687)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4895', 'drugName': 'Oxiglutatione', 'newLinkedTargets_string': 'GSR (ENSG00000104687)', 'drugIsApproved': True, 'maxClinica...
general
Select, Similarity Search, Order By
Genetic Target
Q4.141
Q4
What drugs target the gene CA9?
The drugs that target CA9 are Ethoxzolamide and Sulthiame.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CA9 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6095', 'drugName': 'Sulthiame', 'newLinkedTargets_string': 'CA2 (ENSG00000104267), CA7 (ENSG00000168748), CA1 (ENSG00000133742), CA3 (ENSG00000164879), CA6 (ENSG00000131686), CA12 (ENSG00000074410), CA14 (ENSG00000118298), CA9 (ENSG00000107159), CA4 (ENSG00000167434), CA13 (ENSG00000185015...
general
Select, Similarity Search, Order By
Genetic Target
Q4.1342
Q4
What drugs target the gene SCNN1G?
The drugs that target SCNN1G are Amiloride Hydrochloride, Amiloride, and Triamterene.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%SCNN1G %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2590', 'drugName': 'Amiloride Hydrochloride', 'newLinkedTargets_string': 'SCNN1A (ENSG00000111319), SCNN1B (ENSG00000168447), SCNN1G (ENSG00000166828)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4230', 'drugName': 'Triamterene', 'newLinkedTargets_str...
general
Select, Similarity Search, Order By
Genetic Target
Q4.1085
Q4
What drugs target the gene PIM2?
There are no FDA approved drugs targeting the gene PIM2. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Sgi-1776, Azd-1208, and Lgh-447.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PIM2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_295', 'drugName': 'Sgi-1776', 'newLinkedTargets_string': 'PIM1 (ENSG00000137193), PIM2 (ENSG00000102096), PIM3 (ENSG00000198355)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 1}, {'UUID': 'DrugGeneTargets_v2_3068', 'drugName': 'Azd-1208', 'newLinkedTargets_string': 'PIM1 (ENSG0000013...
general
Select, Similarity Search, Order By
Genetic Target
Q4.226
Q4
What drugs target the gene CD86?
The drugs that target CD86 are Abatacept and Belatacept.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CD86 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3639', 'drugName': 'Abatacept', 'newLinkedTargets_string': 'CD80 (ENSG00000121594), CD86 (ENSG00000114013)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3638', 'drugName': 'Abatacept', 'newLinkedTargets_string': 'CD80 (ENSG00000121594), CD86 (ENSG00000...
general
Select, Similarity Search, Order By
Genetic Target
Q4.811
Q4
What drugs target the gene LAMC1?
The drug that targets LAMC1 is Ocriplasmin.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%LAMC1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5818', 'drugName': 'Ocriplasmin', 'newLinkedTargets_string': 'FN1 (ENSG00000115414), COL1A2 (ENSG00000164692), COL1A1 (ENSG00000108821), COL2A1 (ENSG00000139219), COL3A1 (ENSG00000168542), COL4A1 (ENSG00000187498), COL5A1 (ENSG00000130635), COL6A1 (ENSG00000142156), COL11A1 (ENSG0000006071...
general
Select, Similarity Search, Order By
Genetic Target
Q4.411
Q4
What drugs target the gene EPHA4?
The drug that targets EPHA4 is Vandetanib.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%EPHA4 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1936', 'drugName': 'Vandetanib', 'newLinkedTargets_string': 'TEK (ENSG00000120156), ERBB2 (ENSG00000141736), EGFR (ENSG00000146648), ERBB4 (ENSG00000178568), ERBB3 (ENSG00000065361), EPHA2 (ENSG00000142627), EPHB2 (ENSG00000133216), EPHA5 (ENSG00000145242), EPHA4 (ENSG00000116106), EPHA8 (...
general
Select, Similarity Search, Order By
Genetic Target
Q4.327
Q4
What drugs target the gene CTAG1A?
There are no approved drugs targeting CTAG1A, but the drug Rasdegafusp Alfa, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CTAG1A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5339', 'drugName': 'Rasdegafusp Alfa', 'newLinkedTargets_string': 'LY75 (ENSG00000054219), CTAG1B (ENSG00000184033), CTAG1A (ENSG00000268651)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_5340', 'drugName': 'Rasdegafusp Alfa', 'newLinkedTargets_string...
general
Select, Similarity Search, Order By
Genetic Target
Q4.301
Q4
What drugs target the gene COL4A6?
The drugs that target COL4A6 are Collagenase Clostridium Histolyticum and Ocriplasmin.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%COL4A6 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5818', 'drugName': 'Ocriplasmin', 'newLinkedTargets_string': 'FN1 (ENSG00000115414), COL1A2 (ENSG00000164692), COL1A1 (ENSG00000108821), COL2A1 (ENSG00000139219), COL3A1 (ENSG00000168542), COL4A1 (ENSG00000187498), COL5A1 (ENSG00000130635), COL6A1 (ENSG00000142156), COL11A1 (ENSG0000006071...
general
Select, Similarity Search, Order By
Genetic Target
Q4.913
Q4
What drugs target the gene MT-ND5?
The drugs that target MT-ND5 are Metformin and Metformin Hydrochloride.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%MT-ND5 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (ENSG00000165264), NDUFA4 (...
general
Select, Similarity Search, Order By
Genetic Target
Q4.762
Q4
What drugs target the gene KCNH8?
The drugs that target KCNH8 are Dalfampridine, Guanidine, Amifampridine Phosphate, Guanidine Hydrochloride, and Amifampridine.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%KCNH8 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5118', 'drugName': 'Guanidine Hydrochloride', 'newLinkedTargets_string': 'KCNQ1 (ENSG00000053918), KCND3 (ENSG00000171385), KCNH2 (ENSG00000055118), KCNA2 (ENSG00000177301), KCNA1 (ENSG00000111262), KCNQ2 (ENSG00000075043), KCNQ3 (ENSG00000184156), KCNA7 (ENSG00000104848), KCNQ5 (ENSG00000...
general
Select, Similarity Search, Order By
Genetic Target