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Q4.1316
Q4
What drugs target the gene RSPO3?
There are no approved drugs targeting RSPO3, but the drug Rosmantuzumab, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RSPO3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5619', 'drugName': 'Rosmantuzumab', 'newLinkedTargets_string': 'RSPO3 (ENSG00000146374), LGR4 (ENSG00000205213)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}]
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Q4.1426
Q4
What drugs target the gene TGFB3?
The drug that targets TGFB3 is Luspatercept.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TGFB3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6093', 'drugName': 'Luspatercept', 'newLinkedTargets_string': 'TGFB1 (ENSG00000105329), TGFB2 (ENSG00000092969), TGFB3 (ENSG00000119699)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3207', 'drugName': 'Bintrafusp Alfa', 'newLinkedTargets_string': 'TGF...
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Q4.976
Q4
What drugs target the gene NDUFV2?
The drugs that target NDUFV2 are Metformin and Metformin Hydrochloride.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NDUFV2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (ENSG00000165264), NDUFA4 (...
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Q4.931
Q4
What drugs target the gene NCAM1?
There are no FDA approved drugs targeting the gene NCAM1. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Oncolysin S, Bb-10901, and Lorvotuzumab Mertansine.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NCAM1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_189', 'drugName': 'Oncolysin S', 'newLinkedTargets_string': 'NCAM1 (ENSG00000149294)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_3306', 'drugName': 'Bb-10901', 'newLinkedTargets_string': 'NCAM1 (ENSG00000149294)', 'drugIsApproved': False, 'maxClinic...
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Q4.576
Q4
What drugs target the gene HCK?
The drugs that target HCK are Bosutinib and Dasatinib.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%HCK %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3959', 'drugName': 'Bosutinib', 'newLinkedTargets_string': 'ABL1 (ENSG00000097007), BCR (ENSG00000186716), HCK (ENSG00000101336), SRC (ENSG00000197122), LYN (ENSG00000254087)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4603', 'drugName': 'Dasatinib',...
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Q4.506
Q4
What drugs target the gene GABRG3?
The drugs that target GABRG3 are Meprobamate, Acamprosate Calcium, Enflurane, Methohexital, Metharbital, Butabarbital, Flurazepam Hydrochloride, Pentobarbital Sodium, Acamprosate, Primidone, Temazepam, Flunitrazepam, Ganaxolone, Diazepam, Methyprylon, Thiopental, Clonazepam, Topiramate, Remimazolam Besylate, Brexanolon...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%GABRG3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1494', 'drugName': 'Thiopental', 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089), GABRA3 (ENSG00000011677), GABRP (ENSG00000094755...
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Q4.787
Q4
What drugs target the gene KEAP1?
The drugs that target KEAP1 are Monomethyl Fumarate, Dimethyl Fumarate, and Diroximel Fumarate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%KEAP1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3182', 'drugName': 'Dimethyl Fumarate', 'newLinkedTargets_string': 'KEAP1 (ENSG00000079999)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5578', 'drugName': 'Diroximel Fumarate', 'newLinkedTargets_string': 'KEAP1 (ENSG00000079999)', 'drugIsApproved': T...
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Q4.4
Q4
What drugs target the gene ABCB1?
There are no FDA approved drugs targeting the gene ABCB1. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Valspodar, Tariquidar, Biricodar, Zosuquidar, and Encequidar.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ABCB1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3894', 'drugName': 'Tariquidar', 'newLinkedTargets_string': 'ABCB1 (ENSG00000085563)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_5486', 'drugName': 'Zosuquidar', 'newLinkedTargets_string': 'ABCB1 (ENSG00000085563)', 'drugIsApproved': False, 'maxClin...
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Q4.1369
Q4
What drugs target the gene SLC34A2?
There are no approved drugs targeting SLC34A2, but the drug Lifastuzumab Vedotin, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%SLC34A2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3443', 'drugName': 'Lifastuzumab Vedotin', 'newLinkedTargets_string': 'SLC34A2 (ENSG00000157765), TUBB4B (ENSG00000188229), TUBB1 (ENSG00000101162), TUBA3C (ENSG00000198033), TUBA4A (ENSG00000127824), TUBB3 (ENSG00000258947), TUBA1A (ENSG00000167552), TUBB4A (ENSG00000104833), TUBB8 (ENSG0...
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Q4.469
Q4
What drugs target the gene FGR?
The drug that targets FGR is Dasatinib.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%FGR %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4602', 'drugName': 'Dasatinib', 'newLinkedTargets_string': 'PDGFRB (ENSG00000113721), FYN (ENSG00000010810), SRC (ENSG00000197122), LCK (ENSG00000182866), YES1 (ENSG00000176105), BLK (ENSG00000136573), HCK (ENSG00000101336), LYN (ENSG00000254087), FRK (ENSG00000111816), FGR (ENSG0000000093...
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Q4.323
Q4
What drugs target the gene CSF2RB?
The drug that targets CSF2RB is Sargramostim.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CSF2RB %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5636', 'drugName': 'Sargramostim', 'newLinkedTargets_string': 'CSF2RA (ENSG00000198223), CSF2RB (ENSG00000100368)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4751', 'drugName': 'Mavrilimumab', 'newLinkedTargets_string': 'CSF2RA (ENSG00000198223), CSF...
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Q4.6
Q4
What drugs target the gene ABCC8?
The drugs that target ABCC8 are Tolbutamide, Glyburide, Chlorpropamide, Acetohexamide, Glipizide, Tolazamide, Repaglinide, Gliclazide, Tolbutamide Sodium, Sterile, Glimepiride, and Nateglinide.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ABCC8 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_951', 'drugName': 'Chlorpropamide', 'newLinkedTargets_string': 'KCNJ11 (ENSG00000187486), ABCC8 (ENSG00000006071)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5473', 'drugName': 'Glimepiride', 'newLinkedTargets_string': 'KCNJ11 (ENSG00000187486), ABCC...
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Q4.1003
Q4
What drugs target the gene NPY5R?
There are no FDA approved drugs targeting the gene NPY5R. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Mk-0557, Velneperit, and S-237648.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NPY5R %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_836', 'drugName': 'Mk-0557', 'newLinkedTargets_string': 'NPY5R (ENSG00000164129)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_848', 'drugName': 'Velneperit', 'newLinkedTargets_string': 'NPY5R (ENSG00000164129)', 'drugIsApproved': False, 'maxClinicalT...
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Q4.550
Q4
What drugs target the gene GRIN2B?
The drugs that target GRIN2B are Orphenadrine, Acamprosate Calcium, Felbamate, Amantadine Hydrochloride, Esketamine Hydrochloride, Acamprosate, Ketamine Hydrochloride, Memantine, Ketamine, Amantadine, Orphenadrine Hydrochloride, Esketamine, Memantine Hydrochloride, and Orphenadrine Citrate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%GRIN2B %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_70', 'drugName': 'Orphenadrine', 'newLinkedTargets_string': 'SCN1A (ENSG00000144285), SCN5A (ENSG00000183873), SCN4A (ENSG00000007314), SCN7A (ENSG00000136546), SCN2A (ENSG00000136531), SCN9A (ENSG00000169432), SCN3A (ENSG00000153253), SCN11A (ENSG00000168356), SCN8A (ENSG00000196876), SCN...
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Q4.1095
Q4
What drugs target the gene PLK1?
There are no FDA approved drugs targeting the gene PLK1. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Tak-960, Mk-1496, Volasertib, Cafusertib, Gsk-461364, Hmn-214, Bi-2536, and Onvansertib.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PLK1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2040', 'drugName': 'Volasertib', 'newLinkedTargets_string': 'PLK1 (ENSG00000166851)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_5804', 'drugName': 'Bi-2536', 'newLinkedTargets_string': 'PLK1 (ENSG00000166851)', 'drugIsApproved': False, 'maxClinicalT...
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Q4.40
Q4
What drugs target the gene ADRB3?
The drugs that target ADRB3 are Vibegron, Dipivefrin, Epinephrine, Carvedilol Phosphate, Mirabegron, Isoproterenol Hydrochloride, Dipivefrin Hydrochloride, Labetalol, Carteolol Hydrochloride, Norepinephrine Bitartrate, Epinephrine Bitartrate, Hydroxyamphetamine, Norepinephrine, Isoproterenol, Hydroxyamphetamine Hydrobr...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ADRB3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3354', 'drugName': 'Carteolol', 'newLinkedTargets_string': 'ADRB1 (ENSG00000043591), ADRB2 (ENSG00000169252), ADRB3 (ENSG00000188778)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3364', 'drugName': 'Dilevalol Hydrochloride', 'newLinkedTargets_string':...
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Q4.545
Q4
What drugs target the gene GRIK3?
The drug that targets GRIK3 is Topiramate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%GRIK3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1594', 'drugName': 'Topiramate', 'newLinkedTargets_string': 'GRIK1 (ENSG00000171189), GRIK5 (ENSG00000105737), GRIK4 (ENSG00000149403), GRIK2 (ENSG00000164418), GRIK3 (ENSG00000163873), CA4 (ENSG00000167434), SCN1A (ENSG00000144285), SCN5A (ENSG00000183873), SCN4A (ENSG00000007314), SCN7A ...
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Q4.244
Q4
What drugs target the gene CDK4?
The drugs that target CDK4 are Trilaciclib, Ribociclib Succinate, Palbociclib, Ribociclib, Trilaciclib Dihydrochloride, and Abemaciclib.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CDK4 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3487', 'drugName': 'Ribociclib', 'newLinkedTargets_string': 'CDK4 (ENSG00000135446), CDK6 (ENSG00000105810)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3860', 'drugName': 'Trilaciclib Dihydrochloride', 'newLinkedTargets_string': 'CDK6 (ENSG0000010581...
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Q4.138
Q4
What drugs target the gene CA5B?
The drugs that target CA5B are Ethoxzolamide and Sulthiame.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CA5B %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6095', 'drugName': 'Sulthiame', 'newLinkedTargets_string': 'CA2 (ENSG00000104267), CA7 (ENSG00000168748), CA1 (ENSG00000133742), CA3 (ENSG00000164879), CA6 (ENSG00000131686), CA12 (ENSG00000074410), CA14 (ENSG00000118298), CA9 (ENSG00000107159), CA4 (ENSG00000167434), CA13 (ENSG00000185015...
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Q4.1329
Q4
What drugs target the gene S1PR5?
The drugs that target S1PR5 are Fingolimod Hydrochloride, Fingolimod, and Fingolimod Lauryl Sulfate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%S1PR5 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5906', 'drugName': 'Fingolimod Lauryl Sulfate', 'newLinkedTargets_string': 'S1PR5 (ENSG00000180739), S1PR2 (ENSG00000267534), S1PR4 (ENSG00000125910), S1PR3 (ENSG00000213694), S1PR1 (ENSG00000170989)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4765',...
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Q4.623
Q4
What drugs target the gene HTR3A?
The drugs that target HTR3A are Granisetron Hydrochloride, Vortioxetine Hydrobromide, Zimeldine, Amisulpride, Granisetron, Vortioxetine, Clothiapine, Dexfenfluramine, Dolasetron Mesylate, Tropisetron, Metoclopramide, Palonosetron Hydrochloride, Dexfenfluramine Hydrochloride, Palonosetron, Ondansetron, Alosetron, Ondans...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%HTR3A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2172', 'drugName': 'Vortioxetine', 'newLinkedTargets_string': 'HTR1A (ENSG00000178394), SLC6A4 (ENSG00000108576), HTR3A (ENSG00000166736)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2170', 'drugName': 'Vortioxetine', 'newLinkedTargets_string': 'HTR1A...
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Q4.829
Q4
What drugs target the gene LRP1?
There are no approved drugs targeting LRP1, but the drug Ang1005, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%LRP1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_429', 'drugName': 'Ang1005', 'newLinkedTargets_string': 'LRP1 (ENSG00000123384), TUBB4B (ENSG00000188229), TUBB1 (ENSG00000101162), TUBA3C (ENSG00000198033), TUBA4A (ENSG00000127824), TUBB3 (ENSG00000258947), TUBA1A (ENSG00000167552), TUBB4A (ENSG00000104833), TUBB8 (ENSG00000261456), TUBB...
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Q4.699
Q4
What drugs target the gene IL4?
There are no FDA approved drugs targeting the gene IL4. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Romilkimab and Pascolizumab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%IL4 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5968', 'drugName': 'Pascolizumab', 'newLinkedTargets_string': 'IL4 (ENSG00000113520)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_932', 'drugName': 'Romilkimab', 'newLinkedTargets_string': 'IL4 (ENSG00000113520), IL13 (ENSG00000169194)', 'drugIsAppro...
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Q4.1093
Q4
What drugs target the gene PLAT?
The drug that targets PLAT is Aminocaproic Acid.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PLAT %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5590', 'drugName': 'Aminocaproic Acid', 'newLinkedTargets_string': 'PLAT (ENSG00000104368), PLG (ENSG00000122194)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5591', 'drugName': 'Aminocaproic Acid', 'newLinkedTargets_string': 'PLAT (ENSG00000104368), ...
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Q4.1474
Q4
What drugs target the gene TPH2?
The drugs that target TPH2 are Telotristat Etiprate, Telotristat Ethyl, and Telotristat.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TPH2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3468', 'drugName': 'Telotristat', 'newLinkedTargets_string': 'TPH2 (ENSG00000139287), TPH1 (ENSG00000129167)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1302', 'drugName': 'Telotristat Ethyl', 'newLinkedTargets_string': 'TPH2 (ENSG00000139287), TPH1 ...
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Q4.585
Q4
What drugs target the gene HDAC4?
The drugs that target HDAC4 are Belinostat, Panobinostat, Panobinostat Lactate, and Romidepsin.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%HDAC4 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4906', 'drugName': 'Panobinostat', 'newLinkedTargets_string': 'HDAC1 (ENSG00000116478), HDAC3 (ENSG00000171720), HDAC6 (ENSG00000094631), HDAC2 (ENSG00000196591), HDAC5 (ENSG00000108840), HDAC7 (ENSG00000061273), HDAC8 (ENSG00000147099), HDAC11 (ENSG00000163517), HDAC4 (ENSG00000068024), H...
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Q4.1513
Q4
What drugs target the gene TYK2?
The drugs that target TYK2 are Deucravacitinib, Tofacitinib Citrate, Upadacitinib, and Tofacitinib.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TYK2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6269', 'drugName': 'Deucravacitinib', 'newLinkedTargets_string': 'TYK2 (ENSG00000105397)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1979', 'drugName': 'Deucravacitinib', 'newLinkedTargets_string': 'TYK2 (ENSG00000105397)', 'drugIsApproved': True, 'm...
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Q4.815
Q4
What drugs target the gene LCK?
The drugs that target LCK are Pazopanib Hydrochloride, Dasatinib, and Pazopanib.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%LCK %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4603', 'drugName': 'Dasatinib', 'newLinkedTargets_string': 'PDGFRB (ENSG00000113721), FYN (ENSG00000010810), SRC (ENSG00000197122), LCK (ENSG00000182866), YES1 (ENSG00000176105), BLK (ENSG00000136573), HCK (ENSG00000101336), LYN (ENSG00000254087), FRK (ENSG00000111816), FGR (ENSG0000000093...
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Genetic Target
Q4.1463
Q4
What drugs target the gene TNNI2?
There are no FDA approved drugs targeting the gene TNNI2. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Reldesemtiv and Tirasemtiv.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TNNI2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_451', 'drugName': 'Reldesemtiv', 'newLinkedTargets_string': 'TNNI2 (ENSG00000130598), TNNT3 (ENSG00000130595), TNNC2 (ENSG00000101470)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_6283', 'drugName': 'Tirasemtiv', 'newLinkedTargets_string': 'TNNI2 (EN...
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Genetic Target
Q4.378
Q4
What drugs target the gene E2F1?
There are no FDA approved drugs targeting the gene E2F1. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Edifoligide and Edifoligide Sodium.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%E2F1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4614', 'drugName': 'Edifoligide Sodium', 'newLinkedTargets_string': 'E2F1 (ENSG00000101412), E2F2 (ENSG00000007968), E2F3 (ENSG00000112242), E2F4 (ENSG00000205250), E2F5 (ENSG00000133740), E2F6 (ENSG00000169016), E2F7 (ENSG00000165891), E2F8 (ENSG00000129173)', 'drugIsApproved': False, 'ma...
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Genetic Target
Q4.316
Q4
What drugs target the gene CREBBP?
There are no approved drugs targeting CREBBP, but the drug Pri-724, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CREBBP %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3141', 'drugName': 'Pri-724', 'newLinkedTargets_string': 'CREBBP (ENSG00000005339), CTNNB1 (ENSG00000168036)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
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Genetic Target
Q4.444
Q4
What drugs target the gene F8?
The drug that targets F8 is Drotrecogin Alfa (Activated).
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%F8 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1085', 'drugName': 'Brentuximab Vedotin', 'newLinkedTargets_string': 'TNFRSF8 (ENSG00000120949), TUBB4B (ENSG00000188229), TUBB1 (ENSG00000101162), TUBA3C (ENSG00000198033), TUBA4A (ENSG00000127824), TUBB3 (ENSG00000258947), TUBA1A (ENSG00000167552), TUBB4A (ENSG00000104833), TUBB8 (ENSG00...
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Genetic Target
Q4.321
Q4
What drugs target the gene CSF2?
There are no FDA approved drugs targeting the gene CSF2. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Plonmarlimab, Namilumab, Lenzilumab, Pexastimogene Devacirepvec, Otilimab, and Gimsilumab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CSF2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3438', 'drugName': 'Lenzilumab', 'newLinkedTargets_string': 'CSF2 (ENSG00000164400)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_4644', 'drugName': 'Otilimab', 'newLinkedTargets_string': 'CSF2 (ENSG00000164400)', 'drugIsApproved': False, 'maxClinical...
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Genetic Target
Q4.1186
Q4
What drugs target the gene PSMD8?
The drugs that target PSMD8 are Bortezomib, Carfilzomib, Ixazomib, and Ixazomib Citrate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PSMD8 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_559', 'drugName': 'Bortezomib', 'newLinkedTargets_string': 'PSMD1 (ENSG00000173692), PSMB2 (ENSG00000126067), PSMB1 (ENSG00000008018), PSMB5 (ENSG00000100804), PSMB8 (ENSG00000204264), PSMB9 (ENSG00000240065), PSMB6 (ENSG00000142507), PSMD14 (ENSG00000115233), PSMA1 (ENSG00000129084), PSMA...
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Genetic Target
Q4.1317
Q4
What drugs target the gene RTN4?
There are no FDA approved drugs targeting the gene RTN4. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Atinumab and Ozanezumab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RTN4 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6319', 'drugName': 'Ozanezumab', 'newLinkedTargets_string': 'RTN4 (ENSG00000115310)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_5814', 'drugName': 'Atinumab', 'newLinkedTargets_string': 'RTN4 (ENSG00000115310)', 'drugIsApproved': False, 'maxClinical...
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Genetic Target
Q4.1158
Q4
What drugs target the gene PSMA8?
The drugs that target PSMA8 are Bortezomib, Carfilzomib, Ixazomib, and Ixazomib Citrate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PSMA8 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3334', 'drugName': 'Ixazomib', 'newLinkedTargets_string': 'PSMD1 (ENSG00000173692), PSMB2 (ENSG00000126067), PSMB1 (ENSG00000008018), PSMB5 (ENSG00000100804), PSMB8 (ENSG00000204264), PSMB9 (ENSG00000240065), PSMB6 (ENSG00000142507), PSMD14 (ENSG00000115233), PSMA1 (ENSG00000129084), PSMA2...
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Genetic Target
Q4.426
Q4
What drugs target the gene ERBB3?
The drug that targets ERBB3 is Vandetanib.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ERBB3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1933', 'drugName': 'Vandetanib', 'newLinkedTargets_string': 'TEK (ENSG00000120156), ERBB2 (ENSG00000141736), EGFR (ENSG00000146648), ERBB4 (ENSG00000178568), ERBB3 (ENSG00000065361), EPHA2 (ENSG00000142627), EPHB2 (ENSG00000133216), EPHA5 (ENSG00000145242), EPHA4 (ENSG00000116106), EPHA8 (...
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Genetic Target
Q4.556
Q4
What drugs target the gene GRM3?
There are no FDA approved drugs targeting the gene GRM3. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Ly404039, Ly2969822, Pomaglumetad Methionil, and Decoglurant.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%GRM3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6226', 'drugName': 'Pomaglumetad Methionil', 'newLinkedTargets_string': 'GRM2 (ENSG00000164082), GRM3 (ENSG00000198822)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_6227', 'drugName': 'Pomaglumetad Methionil', 'newLinkedTargets_string': 'GRM2 (ENSG00...
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Genetic Target
Q4.598
Q4
What drugs target the gene HNF4A?
The drug that targets HNF4A is Alverine.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%HNF4A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4846', 'drugName': 'Alverine', 'newLinkedTargets_string': 'HTR1A (ENSG00000178394), HNF4A (ENSG00000101076)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4847', 'drugName': 'Alverine', 'newLinkedTargets_string': 'HTR1A (ENSG00000178394), HNF4A (ENSG000...
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Genetic Target
Q4.922
Q4
What drugs target the gene MYH6?
The drug that targets MYH6 is Mavacamten.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%MYH6 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1036', 'drugName': 'Mavacamten', 'newLinkedTargets_string': 'MYH7 (ENSG00000092054), MYH6 (ENSG00000197616), MYH7B (ENSG00000078814), MYL3 (ENSG00000160808), MYL2 (ENSG00000111245), MYL7 (ENSG00000106631), MYL4 (ENSG00000198336)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID...
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Genetic Target
Q4.674
Q4
What drugs target the gene IL15?
There are no approved drugs targeting IL15, but the drug Ordesekimab, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%IL15 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3251', 'drugName': 'Ordesekimab', 'newLinkedTargets_string': 'IL15 (ENSG00000164136)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
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Genetic Target
Q4.1091
Q4
What drugs target the gene PLA2G5?
There are no approved drugs targeting PLA2G5, but the drug Varespladib Methyl, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PLA2G5 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6244', 'drugName': 'Varespladib Methyl', 'newLinkedTargets_string': 'PLA2G5 (ENSG00000127472), PLA2G10 (ENSG00000069764), PLA2G2A (ENSG00000188257)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_6245', 'drugName': 'Varespladib Methyl', 'newLinkedTarget...
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Genetic Target
Q4.1248
Q4
What drugs target the gene RPL27A?
The drug that targets RPL27A is Ataluren.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RPL27A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG00000083845), RPS7 (ENSG...
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Genetic Target
Q4.1402
Q4
What drugs target the gene STAT3?
There are no FDA approved drugs targeting the gene STAT3. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Danvatirsen Sodium and Danvatirsen.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%STAT3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4959', 'drugName': 'Danvatirsen', 'newLinkedTargets_string': 'STAT3 (ENSG00000168610)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_199', 'drugName': 'Danvatirsen Sodium', 'newLinkedTargets_string': 'STAT3 (ENSG00000168610)', 'drugIsApproved': False, ...
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Genetic Target
Q4.229
Q4
What drugs target the gene CDH3?
There are no approved drugs targeting CDH3, but the drug Pf-03732010, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CDH3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1343', 'drugName': 'Pf-03732010', 'newLinkedTargets_string': 'CDH3 (ENSG00000062038)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 1}]
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Genetic Target
Q4.1207
Q4
What drugs target the gene RAF1?
The drugs that target RAF1 are Sorafenib, Regorafenib, and Sorafenib Tosylate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RAF1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_812', 'drugName': 'Regorafenib', 'newLinkedTargets_string': 'EPHA2 (ENSG00000142627), TEK (ENSG00000120156), MAPK11 (ENSG00000185386), RAF1 (ENSG00000132155), FRK (ENSG00000111816), PDGFRB (ENSG00000113721), PDGFRA (ENSG00000134853), KIT (ENSG00000157404), FGFR1 (ENSG00000077782), DDR2 (EN...
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Genetic Target
Q4.1198
Q4
What drugs target the gene PTGS2?
The drugs that target PTGS2 are Acetaminophen, Oxyphenbutazone, Aloxiprin, Lumiracoxib, Carprofen, Ibuprofen Sodium, Glafenine, Diflunisal, Sulindac, Suprofen, Etodolac, Meloxicam, Bromfenac Sodium, Balsalazide, Balsalazide Disodium, Bismuth Subsalicylate, Tolmetin Sodium, Dexibuprofen, Benzydamine, Fenclofenac, Aspiri...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PTGS2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2672', 'drugName': 'Parecoxib Sodium', 'newLinkedTargets_string': 'PTGS2 (ENSG00000073756)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5955', 'drugName': 'Valdecoxib', 'newLinkedTargets_string': 'PTGS2 (ENSG00000073756)', 'drugIsApproved': True, 'max...
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Genetic Target
Q4.1154
Q4
What drugs target the gene PSMA4?
The drugs that target PSMA4 are Bortezomib, Carfilzomib, Ixazomib, and Ixazomib Citrate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PSMA4 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3334', 'drugName': 'Ixazomib', 'newLinkedTargets_string': 'PSMD1 (ENSG00000173692), PSMB2 (ENSG00000126067), PSMB1 (ENSG00000008018), PSMB5 (ENSG00000100804), PSMB8 (ENSG00000204264), PSMB9 (ENSG00000240065), PSMB6 (ENSG00000142507), PSMD14 (ENSG00000115233), PSMA1 (ENSG00000129084), PSMA2...
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Genetic Target
Q4.712
Q4
What drugs target the gene INSR?
The drugs that target INSR are Insulin Glargine, Insulin Zinc Susp Beef, Insulin Lispro, Insulin Zinc Susp Extended Purified Beef, Insulin Aspart Protamine Recombinant, Insulin Zinc Susp Purified Pork, Insulin Zinc Susp Prompt Purified Pork, Insulin Susp Isophane Beef/Pork, Insulin Purified Pork, Insulin Zinc Susp Exte...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%INSR %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_495', 'drugName': 'Insulin Glargine', 'newLinkedTargets_string': 'INSR (ENSG00000171105)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5849', 'drugName': 'Insulin Susp Isophane Semisynthetic Purified Human', 'newLinkedTargets_string': 'INSR (ENSG000001...
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Genetic Target
Q4.67
Q4
What drugs target the gene AOC3?
There are no approved drugs targeting AOC3, but the drug Vepalimomab, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%AOC3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5390', 'drugName': 'Vepalimomab', 'newLinkedTargets_string': 'AOC3 (ENSG00000131471)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
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Genetic Target
Q4.395
Q4
What drugs target the gene EGLN2?
The drug that targets EGLN2 is Roxadustat.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%EGLN2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5393', 'drugName': 'Roxadustat', 'newLinkedTargets_string': 'EGLN2 (ENSG00000269858), P4HTM (ENSG00000178467), EGLN1 (ENSG00000135766), EGLN3 (ENSG00000129521)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2677', 'drugName': 'Daprodustat', 'newLinkedTa...
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Genetic Target
Q4.583
Q4
What drugs target the gene HDAC2?
The drugs that target HDAC2 are Belinostat, Vorinostat, Panobinostat, Panobinostat Lactate, and Romidepsin.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%HDAC2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2373', 'drugName': 'Vorinostat', 'newLinkedTargets_string': 'HDAC1 (ENSG00000116478), HDAC2 (ENSG00000196591), HDAC3 (ENSG00000171720), HDAC6 (ENSG00000094631)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2372', 'drugName': 'Vorinostat', 'newLinkedTar...
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Genetic Target
Q4.1019
Q4
What drugs target the gene OPRK1?
The drugs that target OPRK1 are Codeine Polistirex, Benzhydrocodone, Nalmefene Hydrochloride, Butorphanol, Nalbuphine, Dezocine, Anileridine, Butorphanol Tartrate, Codeine Phosphate, Nalbuphine Hydrochloride, Buprenorphine Hydrochloride, Hydrocodone Bitartrate, Hydrocodone Polistirex, Levallorphan, Samidorphan L-Malate...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%OPRK1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2630', 'drugName': 'Levallorphan', 'newLinkedTargets_string': 'OPRK1 (ENSG00000082556), OPRM1 (ENSG00000112038)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_749', 'drugName': 'Butorphanol', 'newLinkedTargets_string': 'OPRM1 (ENSG00000112038), OPRK1 (E...
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Genetic Target
Q4.213
Q4
What drugs target the gene CD3G?
The drugs that target CD3G are Catumaxomab, Muromonab-Cd3, Blinatumomab, and Teclistamab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CD3G %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3214', 'drugName': 'Muromonab-Cd3', 'newLinkedTargets_string': 'CD3E (ENSG00000198851), CD3G (ENSG00000160654), CD3D (ENSG00000167286)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_6103', 'drugName': 'Teclistamab', 'newLinkedTargets_string': 'CD3E (ENS...
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Genetic Target
Q4.1187
Q4
What drugs target the gene PTAFR?
There are no FDA approved drugs targeting the gene PTAFR. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Rupatadine and Minopafant.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PTAFR %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2192', 'drugName': 'Rupatadine', 'newLinkedTargets_string': 'HRH1 (ENSG00000196639), PTAFR (ENSG00000169403)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_2191', 'drugName': 'Rupatadine', 'newLinkedTargets_string': 'HRH1 (ENSG00000196639), PTAFR (ENSG...
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Genetic Target
Q4.957
Q4
What drugs target the gene NDUFB2?
The drugs that target NDUFB2 are Metformin and Metformin Hydrochloride.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NDUFB2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (ENSG00000165264), NDUFA4 (...
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Genetic Target
Q4.539
Q4
What drugs target the gene GRIA1?
The drugs that target GRIA1 are Topiramate and Perampanel.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%GRIA1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1597', 'drugName': 'Topiramate', 'newLinkedTargets_string': 'GRIK1 (ENSG00000171189), GRIK5 (ENSG00000105737), GRIK4 (ENSG00000149403), GRIK2 (ENSG00000164418), GRIK3 (ENSG00000163873), CA4 (ENSG00000167434), SCN1A (ENSG00000144285), SCN5A (ENSG00000183873), SCN4A (ENSG00000007314), SCN7A ...
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Genetic Target
Q4.1237
Q4
What drugs target the gene RPL17?
The drug that targets RPL17 is Ataluren.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RPL17 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG00000083845), RPS7 (ENSG...
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Genetic Target
Q4.685
Q4
What drugs target the gene IL1RAP?
The drug that targets IL1RAP is Spesolimab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%IL1RAP %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2421', 'drugName': 'Spesolimab', 'newLinkedTargets_string': 'IL1RL2 (ENSG00000115598), IL1RAP (ENSG00000196083)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_102', 'drugName': 'Imsidolimab', 'newLinkedTargets_string': 'IL1RL2 (ENSG00000115598), IL1RAP ...
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Genetic Target
Q4.87
Q4
What drugs target the gene ATP2A1?
There are no approved drugs targeting ATP2A1, but the drug Mipsagargin, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ATP2A1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3997', 'drugName': 'Mipsagargin', 'newLinkedTargets_string': 'ATP2A3 (ENSG00000074370), ATP2A1 (ENSG00000196296), ATP2A2 (ENSG00000174437)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
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Genetic Target
Q4.1383
Q4
What drugs target the gene SMO?
The drugs that target SMO are Glasdegib, Glasdegib Maleate, Sonidegib, Sonidegib Phosphate, and Vismodegib.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%SMO %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2876', 'drugName': 'Glasdegib Maleate', 'newLinkedTargets_string': 'SMO (ENSG00000128602)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3933', 'drugName': 'Sonidegib Phosphate', 'newLinkedTargets_string': 'SMO (ENSG00000128602)', 'drugIsApproved': True...
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Genetic Target
Q4.274
Q4
What drugs target the gene CHRNB4?
The drugs that target CHRNB4 are Mecamylamine, Mecamylamine Hydrochloride, Trimethaphan, Pentolinium Tartrate, Pentolinium, and Trimethaphan Camsylate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CHRNB4 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5467', 'drugName': 'Trimethaphan Camsylate', 'newLinkedTargets_string': 'CHRNB4 (ENSG00000117971), CHRNA3 (ENSG00000080644)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4467', 'drugName': 'Trimethaphan', 'newLinkedTargets_string': 'CHRNB4 (ENSG0000011...
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Genetic Target
Q4.944
Q4
What drugs target the gene NDUFA5?
The drugs that target NDUFA5 are Metformin and Metformin Hydrochloride.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NDUFA5 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (ENSG00000165264), NDUFA4 (...
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Genetic Target
Q4.684
Q4
What drugs target the gene IL1R1?
The drug that targets IL1R1 is Anakinra.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%IL1R1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2379', 'drugName': 'Anakinra', 'newLinkedTargets_string': 'IL1R1 (ENSG00000115594)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2001', 'drugName': 'Medi-8968', 'newLinkedTargets_string': 'IL1R1 (ENSG00000115594)', 'drugIsApproved': False, 'maxClinical...
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Genetic Target
Q4.1384
Q4
What drugs target the gene SNAP25?
The drugs that target SNAP25 are Onabotulinumtoxina, Prabotulinumtoxin A, Botulinum Toxin Type A, Daxibotulinumtoxina, Abobotulinumtoxina, and Incobotulinumtoxina.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%SNAP25 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2163', 'drugName': 'Onabotulinumtoxina', 'newLinkedTargets_string': 'SNAP25 (ENSG00000132639)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5684', 'drugName': 'Abobotulinumtoxina', 'newLinkedTargets_string': 'SNAP25 (ENSG00000132639)', 'drugIsApproved'...
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Genetic Target
Q4.634
Q4
What drugs target the gene ICAM3?
There are no approved drugs targeting ICAM3, but the drug Icm3, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ICAM3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1930', 'drugName': 'Icm3', 'newLinkedTargets_string': 'ICAM3 (ENSG00000076662)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
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Genetic Target
Q4.1053
Q4
What drugs target the gene PDE6A?
The drugs that target PDE6A are Pentoxifylline and Dipyridamole.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PDE6A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6107', 'drugName': 'Dipyridamole', 'newLinkedTargets_string': 'PDE5A (ENSG00000138735), PDE4A (ENSG00000065989), PDE3A (ENSG00000172572), PDE6H (ENSG00000139053), PDE6G (ENSG00000185527), PDE2A (ENSG00000186642), PDE7A (ENSG00000205268), PDE1A (ENSG00000115252), PDE9A (ENSG00000160191), PD...
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Genetic Target
Q4.1435
Q4
What drugs target the gene TLR4?
There are no FDA approved drugs targeting the gene TLR4. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Eritoran, Eritoran Tetrasodium, and Resatorvid.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TLR4 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5358', 'drugName': 'Resatorvid', 'newLinkedTargets_string': 'TLR4 (ENSG00000136869)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_1063', 'drugName': 'Eritoran Tetrasodium', 'newLinkedTargets_string': 'TLR4 (ENSG00000136869), LY96 (ENSG00000154589)', '...
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Genetic Target
Q4.1058
Q4
What drugs target the gene PDE6H?
The drugs that target PDE6H are Pentoxifylline and Dipyridamole.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PDE6H %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6107', 'drugName': 'Dipyridamole', 'newLinkedTargets_string': 'PDE5A (ENSG00000138735), PDE4A (ENSG00000065989), PDE3A (ENSG00000172572), PDE6H (ENSG00000139053), PDE6G (ENSG00000185527), PDE2A (ENSG00000186642), PDE7A (ENSG00000205268), PDE1A (ENSG00000115252), PDE9A (ENSG00000160191), PD...
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Genetic Target
Q4.275
Q4
What drugs target the gene CHRND?
The drugs that target CHRND are Pipecuronium, Decamethonium, Vecuronium, Rocuronium, Metocurine Iodide, Succinylcholine Chloride, Tubocurarine, Rocuronium Bromide, Cisatracurium, Cisatracurium Besylate, Mivacurium Chloride, Pancuronium, Gallamine, Vecuronium Bromide, Gallamine Triethiodide, Metocurine, Atracurium Besyl...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CHRND %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2723', 'drugName': 'Succinylcholine Chloride', 'newLinkedTargets_string': 'CHRNA1 (ENSG00000138435), CHRNG (ENSG00000196811), CHRNB1 (ENSG00000170175), CHRND (ENSG00000135902), CHRNE (ENSG00000108556)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_922',...
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Genetic Target
Q4.746
Q4
What drugs target the gene KCNC4?
The drugs that target KCNC4 are Dalfampridine, Guanidine, Amifampridine Phosphate, Guanidine Hydrochloride, and Amifampridine.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%KCNC4 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5118', 'drugName': 'Guanidine Hydrochloride', 'newLinkedTargets_string': 'KCNQ1 (ENSG00000053918), KCND3 (ENSG00000171385), KCNH2 (ENSG00000055118), KCNA2 (ENSG00000177301), KCNA1 (ENSG00000111262), KCNQ2 (ENSG00000075043), KCNQ3 (ENSG00000184156), KCNA7 (ENSG00000104848), KCNQ5 (ENSG00000...
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Q4.364
Q4
What drugs target the gene DLL3?
There are no approved drugs targeting DLL3, but the drug Rovalpituzumab Tesirine, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%DLL3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4409', 'drugName': 'Rovalpituzumab Tesirine', 'newLinkedTargets_string': 'DLL3 (ENSG00000090932)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}]
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Q4.626
Q4
What drugs target the gene HTR3D?
The drugs that target HTR3D are Zimeldine, Amisulpride, Clothiapine, Dexfenfluramine, Tropisetron, Dexfenfluramine Hydrochloride, and Zimeldine Hydrochloride.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%HTR3D %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2386', 'drugName': 'Clothiapine', 'newLinkedTargets_string': 'HTR2B (ENSG00000135914), HTR2A (ENSG00000102468), HTR2C (ENSG00000147246), DRD4 (ENSG00000069696), HTR3A (ENSG00000166736), HTR3E (ENSG00000186038), HTR3B (ENSG00000149305), HTR3D (ENSG00000186090), HTR3C (ENSG00000178084)', 'dr...
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Genetic Target
Q4.3
Q4
What drugs target the gene ABCA1?
The drug that targets ABCA1 is Probucol.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ABCA1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_632', 'drugName': 'Probucol', 'newLinkedTargets_string': 'ABCA1 (ENSG00000165029)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}]
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Genetic Target
Q4.7
Q4
What drugs target the gene ABCC9?
The drugs that target ABCC9 are Pinacidil and Minoxidil.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ABCC9 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1076', 'drugName': 'Pinacidil', 'newLinkedTargets_string': 'KCNJ11 (ENSG00000187486), ABCC9 (ENSG00000069431)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5958', 'drugName': 'Pinacidil', 'newLinkedTargets_string': 'KCNJ11 (ENSG00000187486), ABCC9 (ENS...
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Genetic Target
Q4.313
Q4
What drugs target the gene CPT2?
The drugs that target CPT2 are Perhexiline and Perhexiline Maleate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CPT2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1726', 'drugName': 'Perhexiline Maleate', 'newLinkedTargets_string': 'MTOR (ENSG00000198793), CPT2 (ENSG00000157184), CPT1B (ENSG00000205560)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_919', 'drugName': 'Perhexiline', 'newLinkedTargets_string': 'MTO...
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Genetic Target
Q4.717
Q4
What drugs target the gene ITGA4?
The drugs that target ITGA4 are Natalizumab and Vedolizumab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ITGA4 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5016', 'drugName': 'Natalizumab', 'newLinkedTargets_string': 'ITGA4 (ENSG00000115232), ITGB7 (ENSG00000139626), ITGB1 (ENSG00000150093)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5015', 'drugName': 'Natalizumab', 'newLinkedTargets_string': 'ITGA4 (E...
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Genetic Target
Q4.669
Q4
What drugs target the gene IL12A?
The drug that targets IL12A is Ustekinumab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%IL12A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3327', 'drugName': 'Ustekinumab', 'newLinkedTargets_string': 'IL12B (ENSG00000113302), IL23A (ENSG00000110944), IL12A (ENSG00000168811)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3328', 'drugName': 'Ustekinumab', 'newLinkedTargets_string': 'IL12B (E...
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Genetic Target
Q4.967
Q4
What drugs target the gene NDUFS1?
The drugs that target NDUFS1 are Metformin and Metformin Hydrochloride.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NDUFS1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (ENSG00000165264), NDUFA4 (...
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Genetic Target
Q4.1516
Q4
What drugs target the gene TYR?
The drugs that target TYR are Monobenzone and Mequinol.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TYR %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5010', 'drugName': 'Mequinol', 'newLinkedTargets_string': 'TYR (ENSG00000077498)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3683', 'drugName': 'Monobenzone', 'newLinkedTargets_string': 'TYR (ENSG00000077498)', 'drugIsApproved': True, 'maxClinicalTri...
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Genetic Target
Q4.217
Q4
What drugs target the gene CD44?
There are no FDA approved drugs targeting the gene CD44. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Bivatuzumab, Pf-03475952, and Bivatuzumab Mertansine.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CD44 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2202', 'drugName': 'Bivatuzumab', 'newLinkedTargets_string': 'CD44 (ENSG00000026508)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 1}, {'UUID': 'DrugGeneTargets_v2_6223', 'drugName': 'Bivatuzumab Mertansine', 'newLinkedTargets_string': 'CD44 (ENSG00000026508), TUBB4B (ENSG00000188229...
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Genetic Target
Q4.1460
Q4
What drugs target the gene TNKS2?
There are no approved drugs targeting TNKS2, but the drug 2X-121, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TNKS2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1419', 'drugName': '2X-121', 'newLinkedTargets_string': 'TNKS2 (ENSG00000107854), TNKS (ENSG00000173273), PARP1 (ENSG00000143799), PARP2 (ENSG00000129484)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_1420', 'drugName': '2X-121', 'newLinkedTargets_str...
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Genetic Target
Q4.28
Q4
What drugs target the gene ADORA1?
The drugs that target ADORA1 are Theophylline Sodium Glycinate, Adenosine, Theophylline Glycinate, Oxtriphylline, Theophylline, Caffeine, Aminophylline, Caffeine, and Citrated.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ADORA1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4548', 'drugName': 'Theophylline', 'newLinkedTargets_string': 'ADORA1 (ENSG00000163485), ADORA2B (ENSG00000170425), ADORA3 (ENSG00000282608), ADORA2A (ENSG00000128271), PDE3A (ENSG00000172572), PDE3B (ENSG00000152270), PDE4A (ENSG00000065989), PDE4D (ENSG00000113448), PDE4B (ENSG0000018458...
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Genetic Target
Q4.1105
Q4
What drugs target the gene POLD4?
The drugs that target POLD4 are Gemcitabine Hydrochloride, Gemcitabine, Clofarabine, Fludarabine Phosphate, and Cytarabine.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%POLD4 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4', 'drugName': 'Gemcitabine Hydrochloride', 'newLinkedTargets_string': 'POLA1 (ENSG00000101868), POLD4 (ENSG00000175482), POLD3 (ENSG00000077514), POLD1 (ENSG00000062822), POLD2 (ENSG00000106628), POLE (ENSG00000177084), POLA2 (ENSG00000014138), PRIM1 (ENSG00000198056), PRIM2 (ENSG0000014...
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Genetic Target
Q4.894
Q4
What drugs target the gene MMP12?
There are no FDA approved drugs targeting the gene MMP12. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Azd-1236, Cts-1027, and Marimastat.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%MMP12 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5864', 'drugName': 'Marimastat', 'newLinkedTargets_string': 'MMP9 (ENSG00000100985), MMP3 (ENSG00000149968), MMP7 (ENSG00000137673), MMP1 (ENSG00000196611), MMP2 (ENSG00000087245), MMP12 (ENSG00000262406)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_...
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Q4.1071
Q4
What drugs target the gene PDPK1?
There are no FDA approved drugs targeting the gene PDPK1. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Ar-12 and Ucn-01.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PDPK1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4659', 'drugName': 'Ucn-01', 'newLinkedTargets_string': 'PDPK1 (ENSG00000140992), CDK2 (ENSG00000123374), CDK4 (ENSG00000135446), PRKD3 (ENSG00000115825), PRKCI (ENSG00000163558), PRKCA (ENSG00000154229), PRKCG (ENSG00000126583), PRKCD (ENSG00000163932), PRKCB (ENSG00000166501), PRKCZ (ENS...
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Q4.642
Q4
What drugs target the gene IFNA13?
There are no FDA approved drugs targeting the gene IFNA13. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Faralimomab, Rontalizumab, and Sifalimumab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%IFNA13 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4431', 'drugName': 'Rontalizumab', 'newLinkedTargets_string': 'IFNA6 (ENSG00000120235), IFNA8 (ENSG00000120242), IFNA5 (ENSG00000147873), IFNA10 (ENSG00000186803), IFNA2 (ENSG00000188379), IFNA1 (ENSG00000197919), IFNA13 (ENSG00000233816), IFNA7 (ENSG00000214042), IFNA21 (ENSG00000137080),...
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Q4.786
Q4
What drugs target the gene KDR?
The drugs that target KDR are Sorafenib, Pazopanib Hydrochloride, Regorafenib, Tivozanib, Ramucirumab, Sorafenib Tosylate, Vandetanib, Tivozanib Hydrochloride, Lenvatinib Mesylate, Sunitinib, Cabozantinib S-Malate, Sunitinib Malate, Nintedanib Esylate, Cabozantinib, Axitinib, Pazopanib, Midostaurin, Nintedanib, and Len...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%KDR %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_392', 'drugName': 'Pazopanib Hydrochloride', 'newLinkedTargets_string': 'FGFR1 (ENSG00000077782), FGFR3 (ENSG00000068078), KIT (ENSG00000157404), CSF1R (ENSG00000182578), FLT1 (ENSG00000102755), FLT4 (ENSG00000037280), KDR (ENSG00000128052), ITK (ENSG00000113263), PDGFRB (ENSG00000113721),...
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Q4.854
Q4
What drugs target the gene MAP3K5?
There are no approved drugs targeting MAP3K5, but the drug Selonsertib, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%MAP3K5 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5336', 'drugName': 'Selonsertib', 'newLinkedTargets_string': 'MAP3K5 (ENSG00000197442)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}]
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Q4.628
Q4
What drugs target the gene HTR4?
The drugs that target HTR4 are Prucalopride, Zimeldine, Amisulpride, Tegaserod Maleate, Prucalopride Succinate, Dexfenfluramine, Cisapride, Metoclopramide, Dexfenfluramine Hydrochloride, Tegaserod, Metoclopramide Hydrochloride, Clebopride, and Zimeldine Hydrochloride.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%HTR4 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3506', 'drugName': 'Metoclopramide', 'newLinkedTargets_string': 'HTR4 (ENSG00000164270), HTR3A (ENSG00000166736), DRD2 (ENSG00000149295)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2042', 'drugName': 'Tegaserod Maleate', 'newLinkedTargets_string': 'H...
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Q4.1043
Q4
What drugs target the gene PDE1B?
The drugs that target PDE1B are Pentoxifylline and Dipyridamole.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PDE1B %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6107', 'drugName': 'Dipyridamole', 'newLinkedTargets_string': 'PDE5A (ENSG00000138735), PDE4A (ENSG00000065989), PDE3A (ENSG00000172572), PDE6H (ENSG00000139053), PDE6G (ENSG00000185527), PDE2A (ENSG00000186642), PDE7A (ENSG00000205268), PDE1A (ENSG00000115252), PDE9A (ENSG00000160191), PD...
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Q4.258
Q4
What drugs target the gene CHKA?
There are no approved drugs targeting CHKA, but the drug Tcd-717, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CHKA %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6258', 'drugName': 'Tcd-717', 'newLinkedTargets_string': 'CHKA (ENSG00000110721)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 1}]
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Q4.26
Q4
What drugs target the gene ADH7?
The drug that targets ADH7 is Nitrefazole.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ADH7 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6344', 'drugName': 'Nitrefazole', 'newLinkedTargets_string': 'ADH1A (ENSG00000187758), ADH4 (ENSG00000198099), ADH1B (ENSG00000196616), ADH1C (ENSG00000248144), ADH7 (ENSG00000196344), ADH5 (ENSG00000197894), ADH6 (ENSG00000172955)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}]
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Q4.338
Q4
What drugs target the gene CXCL8?
There are no FDA approved drugs targeting the gene CXCL8. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Humax-Il8 and Abx-Il8.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CXCL8 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4247', 'drugName': 'Humax-Il8', 'newLinkedTargets_string': 'CXCL8 (ENSG00000169429)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_4996', 'drugName': 'Abx-Il8', 'newLinkedTargets_string': 'CXCL8 (ENSG00000169429)', 'drugIsApproved': False, 'maxClinical...
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Q4.575
Q4
What drugs target the gene HCAR2?
There are no approved drugs targeting HCAR2, but the drug Sch-900271, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%HCAR2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5716', 'drugName': 'Sch-900271', 'newLinkedTargets_string': 'HCAR2 (ENSG00000182782)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
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Q4.48
Q4
What drugs target the gene AKR1B1?
The drug that targets AKR1B1 is Tolrestat.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%AKR1B1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6334', 'drugName': 'Tolrestat', 'newLinkedTargets_string': 'AKR1B1 (ENSG00000085662)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2353', 'drugName': 'Sorbinil', 'newLinkedTargets_string': 'AKR1B1 (ENSG00000085662)', 'drugIsApproved': False, 'maxClinic...
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Q4.108
Q4
What drugs target the gene BCR?
The drugs that target BCR are Nilotinib Hydrochloride Monohydrate, Ponatinib, Imatinib, Imatinib Mesylate, Asciminib, Bosutinib, Asciminib Hydrochloride, Dasatinib, Nilotinib, and Ponatinib Hydrochloride.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%BCR %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6150', 'drugName': 'Ponatinib Hydrochloride', 'newLinkedTargets_string': 'ABL1 (ENSG00000097007), BCR (ENSG00000186716)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2277', 'drugName': 'Ponatinib', 'newLinkedTargets_string': 'ABL1 (ENSG00000097007), BC...
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Q4.351
Q4
What drugs target the gene CYP3A7?
The drugs that target CYP3A7 are Ritonavir and Cobicistat.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CYP3A7 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2751', 'drugName': 'Ritonavir', 'newLinkedTargets_string': 'CYP3A4 (ENSG00000160868), CYP3A5 (ENSG00000106258), CYP3A43 (ENSG00000021461), CYP3A7 (ENSG00000160870)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2752', 'drugName': 'Ritonavir', 'newLinked...
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Q4.56
Q4
What drugs target the gene ALK?
The drugs that target ALK are Lorlatinib, Entrectinib, Alectinib Hydrochloride, Brigatinib, Ceritinib, Alectinib, and Crizotinib.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ALK %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2435', 'drugName': 'Ceritinib', 'newLinkedTargets_string': 'ALK (ENSG00000171094), EML4 (ENSG00000143924), NPM1 (ENSG00000181163)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1250', 'drugName': 'Alectinib Hydrochloride', 'newLinkedTargets_string': 'AL...
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Q4.1136
Q4
What drugs target the gene PRKCD?
The drug that targets PRKCD is Midostaurin.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PRKCD %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5668', 'drugName': 'Midostaurin', 'newLinkedTargets_string': 'KIT (ENSG00000157404), KDR (ENSG00000128052), PDGFRB (ENSG00000113721), PDGFRA (ENSG00000134853), FLT3 (ENSG00000122025), PRKD3 (ENSG00000115825), PRKCI (ENSG00000163558), PRKCA (ENSG00000154229), PRKCG (ENSG00000126583), PRKCD ...
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