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Q58.625
Q58
How many genes does the drug Mbx-2982 target and what are they?
The drug Mbx-2982 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene GPR119.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%mbx-2982%" OR LOWER(tradeNames_string) LIKE "%mb...
[{'UUID': 'DrugGeneTargets_v2_4851', 'drugName': 'Mbx-2982', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GPR119 (ENSG00000147262)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Q58.487
Q58
How many genes does the drug Eltrombopag target and what are they?
MPL is the only gene target of drug Eltrombopag.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%eltrombopag%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_2769', 'drugName': 'Eltrombopag Olamine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'MPL (ENSG00000117400)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2008, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_1104', 'drugName': '...
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Genetic Target
Q58.1579
Q58
How many genes does the drug Bms-777607 target and what are they?
The drug Bms-777607 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene MET.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%bms-777607%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5979', 'drugName': 'Bms-777607', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'MET (ENSG00000105976)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.512
Q58
How many genes does the drug Clofibrate target and what are they?
PPARA is the only gene target of drug Clofibrate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%clofibrate%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2331', 'drugName': 'Clofibrate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PPARA (ENSG00000186951)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1967, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.740
Q58
How many genes does the drug Nadolol target and what are they?
There are 2 gene targets for the drug Nadolol: ADRB2 and ADRB1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%nadolol%" OR LOWER(tradeNames_string) LIKE "%nad...
[{'UUID': 'DrugGeneTargets_v2_424', 'drugName': 'Nadolol', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRB2 (ENSG00000169252), ADRB1 (ENSG00000043591)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1979, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_425', ...
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Q58.762
Q58
How many genes does the drug Naphazoline target and what are they?
There are 6 gene targets for the drug Naphazoline: ADRA1A, ADRA2A, ADRA2C, ADRA1D, ADRA1B, and ADRA2B.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%naphazoline%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_327', 'drugName': 'Naphazoline Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRA1A (ENSG00000120907), ADRA2A (ENSG00000150594), ADRA2C (ENSG00000184160), ADRA1D (ENSG00000171873), ADRA1B (ENSG00000170214), ADRA2B (ENSG00000274286)', 'numberLinkedTarget...
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Genetic Target
Q58.1990
Q58
How many genes does the drug Ursodiol target and what are they?
NR1H4 is the only gene target of drug Ursodiol.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ursodiol%" OR LOWER(tradeNames_string) LIKE "%ur...
[{'UUID': 'DrugGeneTargets_v2_4210', 'drugName': 'Ursodiol', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'NR1H4 (ENSG00000012504)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1987, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.784
Q58
How many genes does the drug Methylpromazine target and what are they?
HRH1 is the only gene target of drug Methylpromazine.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%methylpromazine%" OR LOWER(tradeNames_string) LI...
[{'UUID': 'DrugGeneTargets_v2_2846', 'drugName': 'Methylpromazine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HRH1 (ENSG00000196639)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1982, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_3705', 'drugName': 'Tri...
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Genetic Target
Q58.1763
Q58
How many genes does the drug Esomeprazole Strontium target and what are they?
There are 2 gene targets for the drug Esomeprazole Strontium: ATP4A and ATP4B.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%esomeprazole strontium%" OR LOWER(tradeNames_str...
[{'UUID': 'DrugGeneTargets_v2_2645', 'drugName': 'Esomeprazole Strontium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ATP4A (ENSG00000105675), ATP4B (ENSG00000186009)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2013, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.848
Q58
How many genes does the drug Tilarginine Acetate target and what are they?
The drug Tilarginine Acetate is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 3 genes: NOS1, NOS2, and NOS3.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tilarginine acetate%" OR LOWER(tradeNames_string...
[{'UUID': 'DrugGeneTargets_v2_1662', 'drugName': 'Tilarginine Acetate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'NOS1 (ENSG00000089250), NOS2 (ENSG00000007171), NOS3 (ENSG00000164867)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Q58.315
Q58
How many genes does the drug Rizatriptan target and what are they?
There are 2 gene targets for the drug Rizatriptan: HTR1D and HTR1B.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%rizatriptan%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_1141', 'drugName': 'Rizatriptan Benzoate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HTR1D (ENSG00000179546), HTR1B (ENSG00000135312)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1998, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTar...
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Q58.816
Q58
How many genes does the drug Cabozantinib S-Malate target and what are they?
There are 2 gene targets for the drug Cabozantinib S-Malate: MET and KDR.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%cabozantinib s-malate%" OR LOWER(tradeNames_stri...
[{'UUID': 'DrugGeneTargets_v2_3579', 'drugName': 'Cabozantinib S-Malate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'MET (ENSG00000105976), KDR (ENSG00000128052)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2012, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTarget...
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Q58.411
Q58
How many genes does the drug Oxycodone Hydrochloride target and what are they?
OPRM1 is the only gene target of drug Oxycodone Hydrochloride.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%oxycodone hydrochloride%" OR LOWER(tradeNames_st...
[{'UUID': 'DrugGeneTargets_v2_4049', 'drugName': 'Oxycodone Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'OPRM1 (ENSG00000112038)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1950, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_3599', 'drugNa...
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Genetic Target
Q58.826
Q58
How many genes does the drug Montelukast Sodium target and what are they?
CYSLTR1 is the only gene target of drug Montelukast Sodium.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%montelukast sodium%" OR LOWER(tradeNames_string)...
[{'UUID': 'DrugGeneTargets_v2_2453', 'drugName': 'Montelukast Sodium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CYSLTR1 (ENSG00000173198)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1998, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.1143
Q58
How many genes does the drug Margetuximab target and what are they?
ERBB2 is the only gene target of drug Margetuximab.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%margetuximab%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_5571', 'drugName': 'Margetuximab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'ERBB2 (ENSG00000141736)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2020, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.313
Q58
How many genes does the drug Ibrutinib target and what are they?
BTK is the only gene target of drug Ibrutinib.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ibrutinib%" OR LOWER(tradeNames_string) LIKE "%i...
[{'UUID': 'DrugGeneTargets_v2_2044', 'drugName': 'Ibrutinib', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'BTK (ENSG00000010671)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2013, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.229
Q58
How many genes does the drug Lonaprisan target and what are they?
The drug Lonaprisan is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene PGR.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%lonaprisan%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2999', 'drugName': 'Lonaprisan', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PGR (ENSG00000082175)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Q58.1699
Q58
How many genes does the drug Macitentan target and what are they?
There are 2 gene targets for the drug Macitentan: EDNRB and EDNRA.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%macitentan%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5056', 'drugName': 'Macitentan', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'EDNRB (ENSG00000136160), EDNRA (ENSG00000151617)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2010, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_13...
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Genetic Target
Q58.1451
Q58
How many genes does the drug Omarigliptin target and what are they?
The drug Omarigliptin is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene DPP4.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%omarigliptin%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_3734', 'drugName': 'Omarigliptin', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'DPP4 (ENSG00000197635)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.1976
Q58
How many genes does the drug Avdoralimab target and what are they?
The drug Avdoralimab is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene C5AR1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%avdoralimab%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_4794', 'drugName': 'Avdoralimab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'C5AR1 (ENSG00000197405)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Q58.814
Q58
How many genes does the drug Casimersen target and what are they?
DMD is the only gene target of drug Casimersen.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%casimersen%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_4498', 'drugName': 'Casimersen', 'drugMolecularType': 'Oligonucleotide', 'newLinkedTargets_string': 'DMD (ENSG00000198947)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2021, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.1847
Q58
How many genes does the drug Cyclosporine target and what are they?
PPIA is the only gene target of drug Cyclosporine.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%cyclosporine%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_1993', 'drugName': 'Cyclosporine', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'PPIA (ENSG00000196262)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1983, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.151
Q58
How many genes does the drug Brexucabtagene Autoleucel target and what are they?
The drug Brexucabtagene Autoleucel is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene CD19.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%brexucabtagene autoleucel%" OR LOWER(tradeNames_...
[{'UUID': 'DrugGeneTargets_v2_5372', 'drugName': 'Brexucabtagene Autoleucel', 'drugMolecularType': 'Gene', 'newLinkedTargets_string': 'CD19 (ENSG00000177455)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Q58.781
Q58
How many genes does the drug Ibuprofen Sodium target and what are they?
There are 2 gene targets for the drug Ibuprofen Sodium: PTGS2 and PTGS1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ibuprofen sodium%" OR LOWER(tradeNames_string) L...
[{'UUID': 'DrugGeneTargets_v2_566', 'drugName': 'Ibuprofen Sodium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PTGS2 (ENSG00000073756), PTGS1 (ENSG00000095303)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2012, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.727
Q58
How many genes does the drug Cocaine target and what are they?
There are 10 gene targets for the drug Cocaine: SCN1A, SCN5A, SCN4A, SCN7A, SCN2A, SCN9A, SCN3A, SCN11A, SCN8A, and SCN10A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%cocaine%" OR LOWER(tradeNames_string) LIKE "%coc...
[{'UUID': 'DrugGeneTargets_v2_3300', 'drugName': 'Apomorphine Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'DRD2 (ENSG00000149295), DRD3 (ENSG00000151577), DRD4 (ENSG00000069696)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 2004, 'maxClinicalTrialPhase': 4, 'drugIsApproved': T...
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Q58.820
Q58
How many genes does the drug Benzquinamide Hydrochloride target and what are they?
DRD2 is the only gene target of drug Benzquinamide Hydrochloride.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%benzquinamide hydrochloride%" OR LOWER(tradeName...
[{'UUID': 'DrugGeneTargets_v2_1440', 'drugName': 'Benzquinamide Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'DRD2 (ENSG00000149295)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1974, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1636
Q58
How many genes does the drug Rivastigmine Tartrate target and what are they?
There are 2 gene targets for the drug Rivastigmine Tartrate: BCHE and ACHE.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%rivastigmine tartrate%" OR LOWER(tradeNames_stri...
[{'UUID': 'DrugGeneTargets_v2_1705', 'drugName': 'Rivastigmine Tartrate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'BCHE (ENSG00000114200), ACHE (ENSG00000087085)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2000, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.825
Q58
How many genes does the drug Lifitegrast target and what are they?
There are 2 gene targets for the drug Lifitegrast: ITGAL and ITGB2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%lifitegrast%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_2931', 'drugName': 'Lifitegrast', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ITGAL (ENSG00000005844), ITGB2 (ENSG00000160255)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2016, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.581
Q58
How many genes does the drug Calcifediol target and what are they?
VDR is the only gene target of drug Calcifediol.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%calcifediol%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_2157', 'drugName': 'Calcifediol', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'VDR (ENSG00000111424)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1980, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_6195', 'drugName': 'Calcifed...
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Genetic Target
Q58.563
Q58
How many genes does the drug Aprepitant target and what are they?
TACR1 is the only gene target of drug Aprepitant.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%aprepitant%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1299', 'drugName': 'Aprepitant', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'TACR1 (ENSG00000115353)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2003, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_5495', 'drugName': 'Fosapre...
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Genetic Target
Q58.1758
Q58
How many genes does the drug Lumasiran target and what are they?
HAO1 is the only gene target of drug Lumasiran.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%lumasiran%" OR LOWER(tradeNames_string) LIKE "%l...
[{'UUID': 'DrugGeneTargets_v2_1382', 'drugName': 'Lumasiran', 'drugMolecularType': 'Oligonucleotide', 'newLinkedTargets_string': 'HAO1 (ENSG00000101323)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_1071', 'drugName': 'Lumasiran S...
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Genetic Target
Q58.1727
Q58
How many genes does the drug Prenylamine target and what are they?
There are 2 gene targets for the drug Prenylamine: SCN5A and CALM1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%prenylamine%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_5448', 'drugName': 'Prenylamine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SCN5A (ENSG00000183873), CALM1 (ENSG00000198668)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_5449...
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Genetic Target
Q58.1349
Q58
How many genes does the drug Lornoxicam target and what are they?
There are 2 gene targets for the drug Lornoxicam: PTGS2 and PTGS1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%lornoxicam%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5752', 'drugName': 'Lornoxicam', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PTGS2 (ENSG00000073756), PTGS1 (ENSG00000095303)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1161
Q58
How many genes does the drug Orvepitant target and what are they?
The drug Orvepitant is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene TACR1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%orvepitant%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2045', 'drugName': 'Orvepitant', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'TACR1 (ENSG00000115353)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.945
Q58
How many genes does the drug Insulin Zinc Susp Purified Beef/Pork target and what are they?
INSR is the only gene target of drug Insulin Zinc Susp Purified Beef/Pork.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%insulin zinc susp purified beef/pork%" OR LOWER(...
[{'UUID': 'DrugGeneTargets_v2_2821', 'drugName': 'Insulin Zinc Susp Purified Beef/Pork', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'INSR (ENSG00000171105)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1982, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.290
Q58
How many genes does the drug Isoproterenol Hydrochloride target and what are they?
There are 3 gene targets for the drug Isoproterenol Hydrochloride: ADRB1, ADRB2, and ADRB3.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%isoproterenol hydrochloride%" OR LOWER(tradeName...
[{'UUID': 'DrugGeneTargets_v2_1200', 'drugName': 'Isoproterenol Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRB1 (ENSG00000043591), ADRB2 (ENSG00000169252), ADRB3 (ENSG00000188778)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 1956, 'maxClinicalTrialPhase': 4, 'drugIsApprove...
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Genetic Target
Q58.1947
Q58
How many genes does the drug Futuximab target and what are they?
The drug Futuximab is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene EGFR.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%futuximab%" OR LOWER(tradeNames_string) LIKE "%f...
[{'UUID': 'DrugGeneTargets_v2_973', 'drugName': 'Futuximab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'EGFR (ENSG00000146648)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.973
Q58
How many genes does the drug Insulin Zinc Susp Purified Pork target and what are they?
INSR is the only gene target of drug Insulin Zinc Susp Purified Pork.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%insulin zinc susp purified pork%" OR LOWER(trade...
[{'UUID': 'DrugGeneTargets_v2_1233', 'drugName': 'Insulin Zinc Susp Purified Pork', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'INSR (ENSG00000171105)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1979, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.605
Q58
How many genes does the drug Burosumab target and what are they?
FGF23 is the only gene target of drug Burosumab.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%burosumab%" OR LOWER(tradeNames_string) LIKE "%b...
[{'UUID': 'DrugGeneTargets_v2_4495', 'drugName': 'Burosumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'FGF23 (ENSG00000118972)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2018, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1312
Q58
How many genes does the drug Darotropium target and what are they?
The drug Darotropium is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 5 genes: CHRM3, CHRM4, CHRM1, CHRM2, and CHRM5.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%darotropium%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_2791', 'drugName': 'Darotropium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CHRM3 (ENSG00000133019), CHRM4 (ENSG00000180720), CHRM1 (ENSG00000168539), CHRM2 (ENSG00000181072), CHRM5 (ENSG00000184984)', 'numberLinkedTargets': 5, 'yearOfFirstApproval': 0, 'maxClinica...
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Genetic Target
Q58.1244
Q58
How many genes does the drug Loxapine Succinate target and what are they?
There are 5 gene targets for the drug Loxapine Succinate: HTR2C, HTR2A, DRD2, DRD3, and DRD4.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%loxapine succinate%" OR LOWER(tradeNames_string)...
[{'UUID': 'DrugGeneTargets_v2_488', 'drugName': 'Loxapine Succinate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HTR2C (ENSG00000147246), HTR2A (ENSG00000102468), DRD2 (ENSG00000149295), DRD3 (ENSG00000151577), DRD4 (ENSG00000069696)', 'numberLinkedTargets': 5, 'yearOfFirstApproval': 1975, 'maxC...
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Genetic Target
Q58.1638
Q58
How many genes does the drug Metformin target and what are they?
There are 51 gene targets for the drug Metformin: GPD2, MT-ND6, NDUFA10, NDUFS8, MT-ND4L, NDUFA6, MT-ND1, NDUFB6, NDUFA4, NDUFA11, NDUFB7, MT-ND2, NDUFS2, MT-ND5, NDUFA8, NDUFB5, MT-ND4, MT-ND3, NDUFAB1, NDUFA1, NDUFS4, NDUFB3, NDUFC1, NDUFA2, NDUFS5, NDUFS7, NDUFS6, NDUFB1, NDUFS3, NDUFA3, NDUFB4, NDUFB8, NDUFB2, NDUF...
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%metformin%" OR LOWER(tradeNames_string) LIKE "%m...
[{'UUID': 'DrugGeneTargets_v2_1886', 'drugName': 'Metformin', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (E...
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Genetic Target
Q58.1588
Q58
How many genes does the drug Ketoprofen target and what are they?
There are 2 gene targets for the drug Ketoprofen: PTGS2 and PTGS1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ketoprofen%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5314', 'drugName': 'Dexketoprofen', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PTGS2 (ENSG00000073756), PTGS1 (ENSG00000095303)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_58...
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Genetic Target
Q58.1316
Q58
How many genes does the drug Reserpine target and what are they?
SLC18A2 is the only gene target of drug Reserpine.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%reserpine%" OR LOWER(tradeNames_string) LIKE "%r...
[{'UUID': 'DrugGeneTargets_v2_1911', 'drugName': 'Reserpine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SLC18A2 (ENSG00000165646)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1960, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1779
Q58
How many genes does the drug Zyh7 target and what are they?
The drug Zyh7 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene PPARA.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%zyh7%" OR LOWER(tradeNames_string) LIKE "%zyh7%"...
[{'UUID': 'DrugGeneTargets_v2_2834', 'drugName': 'Zyh7', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PPARA (ENSG00000186951)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1647
Q58
How many genes does the drug Tenecteplase target and what are they?
PLG is the only gene target of drug Tenecteplase.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tenecteplase%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_5412', 'drugName': 'Tenecteplase', 'drugMolecularType': 'Enzyme', 'newLinkedTargets_string': 'PLG (ENSG00000122194)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2000, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1255
Q58
How many genes does the drug Procainamide Hydrochloride target and what are they?
There are 10 gene targets for the drug Procainamide Hydrochloride: SCN1A, SCN5A, SCN4A, SCN7A, SCN2A, SCN9A, SCN3A, SCN11A, SCN8A, and SCN10A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%procainamide hydrochloride%" OR LOWER(tradeNames...
[{'UUID': 'DrugGeneTargets_v2_4967', 'drugName': 'Procainamide Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SCN1A (ENSG00000144285), SCN5A (ENSG00000183873), SCN4A (ENSG00000007314), SCN7A (ENSG00000136546), SCN2A (ENSG00000136531), SCN9A (ENSG00000169432), SCN3A (ENSG00000153253),...
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Genetic Target
Q58.1675
Q58
How many genes does the drug Conatumumab target and what are they?
The drug Conatumumab is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene TNFRSF10B.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%conatumumab%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_2732', 'drugName': 'Conatumumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'TNFRSF10B (ENSG00000120889)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1801
Q58
How many genes does the drug Conteltinib target and what are they?
The drug Conteltinib is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 4 genes: ALK, PTK2, IGF1R, and PTK2B.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%conteltinib %" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_3030', 'drugName': 'Conteltinib ', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ALK (ENSG00000171094), PTK2 (ENSG00000169398), IGF1R (ENSG00000140443), PTK2B (ENSG00000120899)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drugIsApp...
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Genetic Target
Q58.759
Q58
How many genes does the drug Mecamylamine Hydrochloride target and what are they?
There are 2 gene targets for the drug Mecamylamine Hydrochloride: CHRNB4 and CHRNA3.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%mecamylamine hydrochloride%" OR LOWER(tradeNames...
[{'UUID': 'DrugGeneTargets_v2_1272', 'drugName': 'Mecamylamine Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CHRNB4 (ENSG00000117971), CHRNA3 (ENSG00000080644)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1956, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.616
Q58
How many genes does the drug Tilarginine target and what are they?
The drug Tilarginine is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 3 genes: NOS1, NOS2, and NOS3.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tilarginine%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_890', 'drugName': 'Tilarginine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'NOS1 (ENSG00000089250), NOS2 (ENSG00000007171), NOS3 (ENSG00000164867)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}, {'UUID': 'D...
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Genetic Target
Q58.1045
Q58
How many genes does the drug Nortriptyline Hydrochloride target and what are they?
There are 2 gene targets for the drug Nortriptyline Hydrochloride: SLC6A2 and SLC6A4.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%nortriptyline hydrochloride%" OR LOWER(tradeName...
[{'UUID': 'DrugGeneTargets_v2_5991', 'drugName': 'Nortriptyline Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SLC6A2 (ENSG00000103546), SLC6A4 (ENSG00000108576)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1964, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'Dr...
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Genetic Target
Q58.788
Q58
How many genes does the drug Ezogabine target and what are they?
There are 5 gene targets for the drug Ezogabine: KCNQ1, KCNQ2, KCNQ3, KCNQ5, and KCNQ4.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ezogabine%" OR LOWER(tradeNames_string) LIKE "%e...
[{'UUID': 'DrugGeneTargets_v2_3665', 'drugName': 'Ezogabine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'KCNQ1 (ENSG00000053918), KCNQ2 (ENSG00000075043), KCNQ3 (ENSG00000184156), KCNQ5 (ENSG00000185760), KCNQ4 (ENSG00000117013)', 'numberLinkedTargets': 5, 'yearOfFirstApproval': 2011, 'maxClinic...
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Genetic Target
Q58.1690
Q58
How many genes does the drug Somatostatin target and what are they?
The drug Somatostatin is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 5 genes: SSTR5, SSTR2, SSTR4, SSTR1, and SSTR3.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%somatostatin%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_1300', 'drugName': 'Somatostatin', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'SSTR5 (ENSG00000162009), SSTR2 (ENSG00000180616), SSTR4 (ENSG00000132671), SSTR1 (ENSG00000139874), SSTR3 (ENSG00000278195)', 'numberLinkedTargets': 5, 'yearOfFirstApproval': 0, 'maxClinicalTrial...
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Genetic Target
Q58.997
Q58
How many genes does the drug Biricodar target and what are they?
The drug Biricodar is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 2 genes: ABCC1 and ABCB1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%biricodar%" OR LOWER(tradeNames_string) LIKE "%b...
[{'UUID': 'DrugGeneTargets_v2_5418', 'drugName': 'Biricodar', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ABCC1 (ENSG00000103222), ABCB1 (ENSG00000085563)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}, {'UUID': 'DrugGeneTargets_v2_5419'...
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Genetic Target
Q58.499
Q58
How many genes does the drug Alisporivir target and what are they?
The drug Alisporivir is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene PPIA.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%alisporivir%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_5603', 'drugName': 'Alisporivir', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'PPIA (ENSG00000196262)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.1320
Q58
How many genes does the drug Mirabegron target and what are they?
ADRB3 is the only gene target of drug Mirabegron.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%mirabegron%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1178', 'drugName': 'Mirabegron', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRB3 (ENSG00000188778)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2012, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.281
Q58
How many genes does the drug Camoteskimab target and what are they?
The drug Camoteskimab is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene IL18.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%camoteskimab%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_6087', 'drugName': 'Camoteskimab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'IL18 (ENSG00000150782)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drugIsApproved': False}]
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Genetic Target
Q58.1848
Q58
How many genes does the drug Dexbrompheniramine Maleate target and what are they?
HRH1 is the only gene target of drug Dexbrompheniramine Maleate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%dexbrompheniramine maleate%" OR LOWER(tradeNames...
[{'UUID': 'DrugGeneTargets_v2_431', 'drugName': 'Dexbrompheniramine Maleate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HRH1 (ENSG00000196639)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1963, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.363
Q58
How many genes does the drug Anileridine Phosphate target and what are they?
There are 2 gene targets for the drug Anileridine Phosphate: OPRM1 and OPRK1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%anileridine phosphate%" OR LOWER(tradeNames_stri...
[{'UUID': 'DrugGeneTargets_v2_4938', 'drugName': 'Anileridine Phosphate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'OPRM1 (ENSG00000112038), OPRK1 (ENSG00000082556)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1982, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTa...
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Genetic Target
Q58.1179
Q58
How many genes does the drug Montelukast target and what are they?
CYSLTR1 is the only gene target of drug Montelukast.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%montelukast%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_2453', 'drugName': 'Montelukast Sodium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CYSLTR1 (ENSG00000173198)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1998, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_2189', 'drugName'...
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Genetic Target
Q58.239
Q58
How many genes does the drug Acamprosate target and what are they?
There are 23 gene targets for the drug Acamprosate: GRIN1, GRIN2A, GRIN2B, GRIN2D, GRIN3B, GRIN2C, GRIN3A, GABRA1, GABRB2, GABRG2, GABRB3, GABRA4, GABRG3, GABRQ, GABRA3, GABRP, GABRD, GABRG1, GABRB1, GABRE, GABRA2, GABRA5, and GABRA6.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%acamprosate%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_163', 'drugName': 'Acamprosate Calcium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089), G...
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Genetic Target
Q58.557
Q58
How many genes does the drug Mk-6913 target and what are they?
The drug Mk-6913 is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 2 genes: ESR2 and ESR1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%mk-6913%" OR LOWER(tradeNames_string) LIKE "%mk-...
[{'UUID': 'DrugGeneTargets_v2_3696', 'drugName': 'Mk-6913', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ESR2 (ENSG00000140009), ESR1 (ENSG00000091831)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1870
Q58
How many genes does the drug Ibutilide Fumarate target and what are they?
KCNH2 is the only gene target of drug Ibutilide Fumarate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ibutilide fumarate%" OR LOWER(tradeNames_string)...
[{'UUID': 'DrugGeneTargets_v2_5277', 'drugName': 'Ibutilide Fumarate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'KCNH2 (ENSG00000055118)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1995, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1915
Q58
How many genes does the drug Hokt3 target and what are they?
The drug Hokt3 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene CD3E.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%hokt3%" OR LOWER(tradeNames_string) LIKE "%hokt3...
[{'UUID': 'DrugGeneTargets_v2_4396', 'drugName': 'Hokt3', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'CD3E (ENSG00000198851)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}, {'UUID': 'DrugGeneTargets_v2_3514', 'drugName': 'Teplizumab', 'drugMol...
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Genetic Target
Q58.211
Q58
How many genes does the drug Erfonrilimab target and what are they?
The drug Erfonrilimab is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 2 genes: CD274 and CTLA4.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%erfonrilimab%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_2574', 'drugName': 'Erfonrilimab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'CD274 (ENSG00000120217), CTLA4 (ENSG00000163599)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}, {'UUID': 'DrugGeneTargets_v2_2575', '...
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Genetic Target
Q58.1922
Q58
How many genes does the drug Siponimod Fumarate target and what are they?
S1PR1 is the only gene target of drug Siponimod Fumarate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%siponimod fumarate%" OR LOWER(tradeNames_string)...
[{'UUID': 'DrugGeneTargets_v2_4451', 'drugName': 'Siponimod Fumarate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'S1PR1 (ENSG00000170989)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2019, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1561
Q58
How many genes does the drug Benzthiazide target and what are they?
SLC12A3 is the only gene target of drug Benzthiazide.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%benzthiazide%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_2994', 'drugName': 'Benzthiazide', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SLC12A3 (ENSG00000070915)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1960, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.60
Q58
How many genes does the drug Baclofen target and what are they?
There are 2 gene targets for the drug Baclofen: GABBR1 and GABBR2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%baclofen%" OR LOWER(tradeNames_string) LIKE "%ba...
[{'UUID': 'DrugGeneTargets_v2_3627', 'drugName': 'Baclofen', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GABBR1 (ENSG00000204681), GABBR2 (ENSG00000136928)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1977, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_33...
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Genetic Target
Q58.1835
Q58
How many genes does the drug Brivaracetam target and what are they?
SV2A is the only gene target of drug Brivaracetam.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%brivaracetam%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_4908', 'drugName': 'Brivaracetam', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SV2A (ENSG00000159164)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2016, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1906
Q58
How many genes does the drug Cjm-112 target and what are they?
The drug Cjm-112 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene IL17A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%cjm-112%" OR LOWER(tradeNames_string) LIKE "%cjm...
[{'UUID': 'DrugGeneTargets_v2_1574', 'drugName': 'Cjm-112', 'drugMolecularType': 'Unknown', 'newLinkedTargets_string': 'IL17A (ENSG00000112115)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1578
Q58
How many genes does the drug Briakinumab target and what are they?
The drug Briakinumab is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 3 genes: IL12B, IL23A, and IL12A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%briakinumab%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_1844', 'drugName': 'Briakinumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'IL12B (ENSG00000113302), IL23A (ENSG00000110944), IL12A (ENSG00000168811)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}, {'UUID': 'Dru...
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Genetic Target
Q58.368
Q58
How many genes does the drug Meclizine Hydrochloride target and what are they?
HRH1 is the only gene target of drug Meclizine Hydrochloride.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%meclizine hydrochloride%" OR LOWER(tradeNames_st...
[{'UUID': 'DrugGeneTargets_v2_5400', 'drugName': 'Meclizine Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HRH1 (ENSG00000196639)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1957, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.511
Q58
How many genes does the drug Methixene target and what are they?
There are 2 gene targets for the drug Methixene: CHRM1 and HTR2C.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%methixene%" OR LOWER(tradeNames_string) LIKE "%m...
[{'UUID': 'DrugGeneTargets_v2_1167', 'drugName': 'Methixene', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CHRM1 (ENSG00000168539), HTR2C (ENSG00000147246)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1982, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_116...
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Genetic Target
Q58.815
Q58
How many genes does the drug Marizomib target and what are they?
The drug Marizomib is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 19 genes: PSMB2, PSMB1, PSMB5, PSMB8, PSMB9, PSMB6, PSMA1, PSMA2, PSMA3, PSMA4, PSMA5, PSMA6, PSMA7, PSMA8, PSMB10, PSMB11, PSMB3, PSMB4, and PSMB7.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%marizomib%" OR LOWER(tradeNames_string) LIKE "%m...
[{'UUID': 'DrugGeneTargets_v2_4687', 'drugName': 'Marizomib', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PSMB2 (ENSG00000126067), PSMB1 (ENSG00000008018), PSMB5 (ENSG00000100804), PSMB8 (ENSG00000204264), PSMB9 (ENSG00000240065), PSMB6 (ENSG00000142507), PSMA1 (ENSG00000129084), PSMA2 (ENSG00000...
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Genetic Target
Q58.1122
Q58
How many genes does the drug Isoxsuprine target and what are they?
There are 4 gene targets for the drug Isoxsuprine: ADRB2, ADRA1A, ADRA1D, and ADRA1B.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%isoxsuprine%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_5346', 'drugName': 'Isoxsuprine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRB2 (ENSG00000169252), ADRA1A (ENSG00000120907), ADRA1D (ENSG00000171873), ADRA1B (ENSG00000170214)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drug...
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Genetic Target
Q58.1731
Q58
How many genes does the drug Humax-Il8 target and what are they?
The drug Humax-Il8 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene CXCL8.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%humax-il8%" OR LOWER(tradeNames_string) LIKE "%h...
[{'UUID': 'DrugGeneTargets_v2_4247', 'drugName': 'Humax-Il8', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'CXCL8 (ENSG00000169429)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1216
Q58
How many genes does the drug Lypressin target and what are they?
There are 3 gene targets for the drug Lypressin: AVPR2, AVPR1A, and AVPR1B.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%lypressin%" OR LOWER(tradeNames_string) LIKE "%l...
[{'UUID': 'DrugGeneTargets_v2_5948', 'drugName': 'Terlipressin', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'AVPR1A (ENSG00000166148), AVPR1B (ENSG00000198049), AVPR2 (ENSG00000126895)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 2022, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': ...
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Genetic Target
Q58.1212
Q58
How many genes does the drug Liatermin target and what are they?
The drug Liatermin is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene GFRA1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%liatermin%" OR LOWER(tradeNames_string) LIKE "%l...
[{'UUID': 'DrugGeneTargets_v2_4217', 'drugName': 'Liatermin', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'GFRA1 (ENSG00000151892)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drugIsApproved': False}]
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Genetic Target
Q58.971
Q58
How many genes does the drug Hydroxyzine Pamoate target and what are they?
HRH1 is the only gene target of drug Hydroxyzine Pamoate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%hydroxyzine pamoate%" OR LOWER(tradeNames_string...
[{'UUID': 'DrugGeneTargets_v2_1501', 'drugName': 'Hydroxyzine Pamoate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HRH1 (ENSG00000196639)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1959, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.805
Q58
How many genes does the drug Itolizumab target and what are they?
The drug Itolizumab is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene CD6.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%itolizumab%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_4017', 'drugName': 'Itolizumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'CD6 (ENSG00000013725)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.121
Q58
How many genes does the drug Obexelimab target and what are they?
The drug Obexelimab is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 2 genes: CD19 and FCGR2B.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%obexelimab%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2610', 'drugName': 'Obexelimab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'CD19 (ENSG00000177455), FCGR2B (ENSG00000072694)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}, {'UUID': 'DrugGeneTargets_v2_2611', 'dr...
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Genetic Target
Q58.1322
Q58
How many genes does the drug Rosuvastatin target and what are they?
HMGCR is the only gene target of drug Rosuvastatin.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%rosuvastatin%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_5208', 'drugName': 'Rosuvastatin Calcium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HMGCR (ENSG00000113161)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2003, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_6280', 'drugName'...
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Genetic Target
Q58.1221
Q58
How many genes does the drug Dyphylline target and what are they?
There are 5 gene targets for the drug Dyphylline: PDE4A, PDE4D, PDE4B, PDE4C, and PDE3A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%dyphylline%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2641', 'drugName': 'Dyphylline', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PDE4A (ENSG00000065989), PDE4D (ENSG00000113448), PDE4B (ENSG00000184588), PDE4C (ENSG00000105650), PDE3A (ENSG00000172572)', 'numberLinkedTargets': 5, 'yearOfFirstApproval': 1951, 'maxClini...
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Genetic Target
Q58.528
Q58
How many genes does the drug Vardenafil Hydrochloride target and what are they?
PDE5A is the only gene target of drug Vardenafil Hydrochloride.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%vardenafil hydrochloride%" OR LOWER(tradeNames_s...
[{'UUID': 'DrugGeneTargets_v2_4542', 'drugName': 'Vardenafil Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PDE5A (ENSG00000138735)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2003, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.519
Q58
How many genes does the drug Sar-260301 target and what are they?
The drug Sar-260301 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene PIK3CB.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%sar-260301%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_911', 'drugName': 'Sar-260301', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PIK3CB (ENSG00000051382)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drugIsApproved': False}]
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Genetic Target
Q58.84
Q58
How many genes does the drug Grapiprant target and what are they?
The drug Grapiprant is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene PTGER4.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%grapiprant%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_3097', 'drugName': 'Grapiprant', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PTGER4 (ENSG00000171522)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.717
Q58
How many genes does the drug Gw501516 target and what are they?
The drug Gw501516 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene PPARD.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%gw501516%" OR LOWER(tradeNames_string) LIKE "%gw...
[{'UUID': 'DrugGeneTargets_v2_3549', 'drugName': 'Gw501516', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PPARD (ENSG00000112033)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1185
Q58
How many genes does the drug Imatinib Mesylate target and what are they?
There are 4 gene targets for the drug Imatinib Mesylate: ABL1, PDGFRB, KIT, and BCR.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%imatinib mesylate%" OR LOWER(tradeNames_string) ...
[{'UUID': 'DrugGeneTargets_v2_3270', 'drugName': 'Imatinib Mesylate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ABL1 (ENSG00000097007), PDGFRB (ENSG00000113721), KIT (ENSG00000157404), BCR (ENSG00000186716)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 2001, 'maxClinicalTrialPhase': 4, 'dr...
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Genetic Target
Q58.386
Q58
How many genes does the drug Loxapine target and what are they?
There are 5 gene targets for the drug Loxapine: HTR2A, HTR2C, DRD2, DRD3, and DRD4.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%loxapine%" OR LOWER(tradeNames_string) LIKE "%lo...
[{'UUID': 'DrugGeneTargets_v2_490', 'drugName': 'Loxapine Succinate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HTR2C (ENSG00000147246), HTR2A (ENSG00000102468), DRD2 (ENSG00000149295), DRD3 (ENSG00000151577), DRD4 (ENSG00000069696)', 'numberLinkedTargets': 5, 'yearOfFirstApproval': 1975, 'maxC...
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Genetic Target
Q58.1022
Q58
How many genes does the drug Ergotamine target and what are they?
There are 7 gene targets for the drug Ergotamine: HTR1D, ADRA1A, ADRA2A, ADRA2C, ADRA1D, ADRA1B, and ADRA2B.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ergotamine%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_3132', 'drugName': 'Ergotamine Tartrate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRA1A (ENSG00000120907), ADRA2A (ENSG00000150594), ADRA2C (ENSG00000184160), ADRA1D (ENSG00000171873), ADRA1B (ENSG00000170214), ADRA2B (ENSG00000274286), HTR1D (ENSG00000179546)',...
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Genetic Target
Q58.1689
Q58
How many genes does the drug Chlorpropamide target and what are they?
There are 2 gene targets for the drug Chlorpropamide: KCNJ11 and ABCC8.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%chlorpropamide%" OR LOWER(tradeNames_string) LIK...
[{'UUID': 'DrugGeneTargets_v2_951', 'drugName': 'Chlorpropamide', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'KCNJ11 (ENSG00000187486), ABCC8 (ENSG00000006071)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1958, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.87
Q58
How many genes does the drug Irdabisant target and what are they?
The drug Irdabisant is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene HRH3.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%irdabisant%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1518', 'drugName': 'Irdabisant', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HRH3 (ENSG00000101180)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drugIsApproved': False}]
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Genetic Target
Q58.1684
Q58
How many genes does the drug Crenezumab target and what are they?
The drug Crenezumab is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene APP.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%crenezumab%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_158', 'drugName': 'Crenezumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'APP (ENSG00000142192)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.333
Q58
How many genes does the drug Flindokalner target and what are they?
The drug Flindokalner is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 5 genes: KCNMA1, KCNQ2, KCNQ3, KCNQ4, and KCNQ5.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%flindokalner%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_2869', 'drugName': 'Flindokalner', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'KCNMA1 (ENSG00000156113), KCNQ2 (ENSG00000075043), KCNQ3 (ENSG00000184156), KCNQ4 (ENSG00000117013), KCNQ5 (ENSG00000185760)', 'numberLinkedTargets': 5, 'yearOfFirstApproval': 0, 'maxClini...
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Genetic Target
Q58.7
Q58
How many genes does the drug Levamlodipine Maleate target and what are they?
There are 4 gene targets for the drug Levamlodipine Maleate: CACNA1C, CACNA1S, CACNA1D, and CACNA1F.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%levamlodipine maleate%" OR LOWER(tradeNames_stri...
[{'UUID': 'DrugGeneTargets_v2_6132', 'drugName': 'Levamlodipine Maleate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CACNA1C (ENSG00000151067), CACNA1S (ENSG00000081248), CACNA1D (ENSG00000157388), CACNA1F (ENSG00000102001)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 2019, 'maxClinicalTri...
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Genetic Target
Q58.737
Q58
How many genes does the drug Edicotinib target and what are they?
The drug Edicotinib is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene CSF1R.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%edicotinib%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_477', 'drugName': 'Edicotinib', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CSF1R (ENSG00000182578)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.750
Q58
How many genes does the drug Ulipristal Acetate target and what are they?
PGR is the only gene target of drug Ulipristal Acetate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ulipristal acetate%" OR LOWER(tradeNames_string)...
[{'UUID': 'DrugGeneTargets_v2_470', 'drugName': 'Ulipristal', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PGR (ENSG00000082175)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_4281', 'drugName': 'Ulipristal Ac...
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Genetic Target
Q58.1414
Q58
How many genes does the drug Patritumab target and what are they?
The drug Patritumab is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene ERBB3.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%patritumab%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2705', 'drugName': 'Patritumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'ERBB3 (ENSG00000065361)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}, {'UUID': 'DrugGeneTargets_v2_1952', 'drugName': 'Patritumab Deru...
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Genetic Target
Q58.1751
Q58
How many genes does the drug Isopropamide Iodide target and what are they?
There are 2 gene targets for the drug Isopropamide Iodide: CHRM1 and CHRM3.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%isopropamide iodide%" OR LOWER(tradeNames_string...
[{'UUID': 'DrugGeneTargets_v2_4390', 'drugName': 'Isopropamide Iodide', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CHRM1 (ENSG00000168539), CHRM3 (ENSG00000133019)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1957, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTarg...
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