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Q58.70
Q58
How many genes does the drug Ergotamine Tartrate target and what are they?
There are 7 gene targets for the drug Ergotamine Tartrate: ADRA1A, ADRA2A, ADRA2C, ADRA1D, ADRA1B, ADRA2B, and HTR1D.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ergotamine tartrate%" OR LOWER(tradeNames_string...
[{'UUID': 'DrugGeneTargets_v2_3552', 'drugName': 'Ergotamine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HTR1D (ENSG00000179546), ADRA1A (ENSG00000120907), ADRA2A (ENSG00000150594), ADRA2C (ENSG00000184160), ADRA1D (ENSG00000171873), ADRA1B (ENSG00000170214), ADRA2B (ENSG00000274286)', 'numberL...
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Genetic Target
Q58.938
Q58
How many genes does the drug Insulin Zinc Susp Extended Beef target and what are they?
INSR is the only gene target of drug Insulin Zinc Susp Extended Beef.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%insulin zinc susp extended beef%" OR LOWER(trade...
[{'UUID': 'DrugGeneTargets_v2_1883', 'drugName': 'Insulin Zinc Susp Extended Beef', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'INSR (ENSG00000171105)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1982, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1447
Q58
How many genes does the drug Dydrogesterone target and what are they?
PGR is the only gene target of drug Dydrogesterone.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%dydrogesterone%" OR LOWER(tradeNames_string) LIK...
[{'UUID': 'DrugGeneTargets_v2_4940', 'drugName': 'Dydrogesterone', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PGR (ENSG00000082175)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1982, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1782
Q58
How many genes does the drug Andolast target and what are they?
The drug Andolast is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene KCNMA1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%andolast%" OR LOWER(tradeNames_string) LIKE "%an...
[{'UUID': 'DrugGeneTargets_v2_5782', 'drugName': 'Andolast', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'KCNMA1 (ENSG00000156113)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.468
Q58
How many genes does the drug Hydroxyurea target and what are they?
There are 3 gene targets for the drug Hydroxyurea: RRM1, RRM2B, and RRM2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%hydroxyurea%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_5698', 'drugName': 'Hydroxyurea', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'RRM1 (ENSG00000167325), RRM2B (ENSG00000048392), RRM2 (ENSG00000171848)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 1967, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1396
Q58
How many genes does the drug Troxacitabine target and what are they?
The drug Troxacitabine is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 11 genes: POLA1, POLD4, POLD3, POLD1, POLD2, POLE, POLA2, PRIM1, PRIM2, POLE2, and POLE3.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%troxacitabine%" OR LOWER(tradeNames_string) LIKE...
[{'UUID': 'DrugGeneTargets_v2_5766', 'drugName': 'Troxacitabine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'POLA1 (ENSG00000101868), POLD4 (ENSG00000175482), POLD3 (ENSG00000077514), POLD1 (ENSG00000062822), POLD2 (ENSG00000106628), POLE (ENSG00000177084), POLA2 (ENSG00000014138), PRIM1 (ENSG00...
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Genetic Target
Q58.1614
Q58
How many genes does the drug Polatuzumab Vedotin target and what are they?
There are 16 gene targets for the drug Polatuzumab Vedotin: CD79B, TUBB4B, TUBB1, TUBA3C, TUBA4A, TUBB3, TUBA1A, TUBB4A, TUBB8, TUBB, TUBA1B, TUBA1C, TUBA3E, TUBB2A, TUBB2B, and TUBB6.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%polatuzumab vedotin%" OR LOWER(tradeNames_string...
[{'UUID': 'DrugGeneTargets_v2_560', 'drugName': 'Polatuzumab Vedotin', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'CD79B (ENSG00000007312), TUBB4B (ENSG00000188229), TUBB1 (ENSG00000101162), TUBA3C (ENSG00000198033), TUBA4A (ENSG00000127824), TUBB3 (ENSG00000258947), TUBA1A (ENSG00000167552), TUBB4A (E...
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Genetic Target
Q58.549
Q58
How many genes does the drug Prs-211375 target and what are they?
The drug Prs-211375 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene CNR2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%prs-211375%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5005', 'drugName': 'Prs-211375', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CNR2 (ENSG00000188822)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.538
Q58
How many genes does the drug Procaine target and what are they?
There are 10 gene targets for the drug Procaine: SCN1A, SCN5A, SCN4A, SCN7A, SCN2A, SCN9A, SCN3A, SCN11A, SCN8A, and SCN10A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%procaine%" OR LOWER(tradeNames_string) LIKE "%pr...
[{'UUID': 'DrugGeneTargets_v2_1754', 'drugName': 'Benoxinate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SCN1A (ENSG00000144285), SCN5A (ENSG00000183873), SCN4A (ENSG00000007314), SCN7A (ENSG00000136546), SCN2A (ENSG00000136531), SCN9A (ENSG00000169432), SCN3A (ENSG00000153253), SCN11A (ENSG000...
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Genetic Target
Q58.1230
Q58
How many genes does the drug Darbepoetin Alfa target and what are they?
EPOR is the only gene target of drug Darbepoetin Alfa.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%darbepoetin alfa%" OR LOWER(tradeNames_string) L...
[{'UUID': 'DrugGeneTargets_v2_4490', 'drugName': 'Darbepoetin Alfa', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'EPOR (ENSG00000187266)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2001, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.957
Q58
How many genes does the drug Pavinetant target and what are they?
The drug Pavinetant is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene TACR3.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%pavinetant%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_3855', 'drugName': 'Pavinetant', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'TACR3 (ENSG00000169836)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1635
Q58
How many genes does the drug Etilevodopa target and what are they?
The drug Etilevodopa is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene DRD3.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%etilevodopa%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_3987', 'drugName': 'Etilevodopa', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'DRD3 (ENSG00000151577)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1418
Q58
How many genes does the drug Chenodiol target and what are they?
NR1H4 is the only gene target of drug Chenodiol.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%chenodiol%" OR LOWER(tradeNames_string) LIKE "%c...
[{'UUID': 'DrugGeneTargets_v2_976', 'drugName': 'Chenodiol', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'NR1H4 (ENSG00000012504)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1983, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.422
Q58
How many genes does the drug Esomeprazole Sodium target and what are they?
There are 2 gene targets for the drug Esomeprazole Sodium: ATP4A and ATP4B.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%esomeprazole sodium%" OR LOWER(tradeNames_string...
[{'UUID': 'DrugGeneTargets_v2_3760', 'drugName': 'Esomeprazole Sodium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ATP4A (ENSG00000105675), ATP4B (ENSG00000186009)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2005, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1935
Q58
How many genes does the drug Doxacurium Chloride target and what are they?
There are 5 gene targets for the drug Doxacurium Chloride: CHRNA1, CHRNG, CHRNB1, CHRND, and CHRNE.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%doxacurium chloride%" OR LOWER(tradeNames_string...
[{'UUID': 'DrugGeneTargets_v2_5531', 'drugName': 'Doxacurium Chloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CHRNA1 (ENSG00000138435), CHRNG (ENSG00000196811), CHRNB1 (ENSG00000170175), CHRND (ENSG00000135902), CHRNE (ENSG00000108556)', 'numberLinkedTargets': 5, 'yearOfFirstApproval': 1991...
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Genetic Target
Q58.1532
Q58
How many genes does the drug Orphenadrine Citrate target and what are they?
There are 19 gene targets for the drug Orphenadrine Citrate: GRIN1, GRIN2A, GRIN2B, GRIN2D, GRIN3B, GRIN2C, GRIN3A, HRH1, SLC6A2, SCN1A, SCN5A, SCN4A, SCN7A, SCN2A, SCN9A, SCN3A, SCN11A, SCN8A, and SCN10A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%orphenadrine citrate%" OR LOWER(tradeNames_strin...
[{'UUID': 'DrugGeneTargets_v2_6210', 'drugName': 'Orphenadrine Citrate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GRIN1 (ENSG00000176884), GRIN2A (ENSG00000183454), GRIN2B (ENSG00000273079), GRIN2D (ENSG00000105464), GRIN3B (ENSG00000116032), GRIN2C (ENSG00000161509), GRIN3A (ENSG00000198785),...
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Genetic Target
Q58.1580
Q58
How many genes does the drug S-222611 target and what are they?
The drug S-222611 is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 2 genes: ERBB2 and EGFR.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%s-222611%" OR LOWER(tradeNames_string) LIKE "%s-...
[{'UUID': 'DrugGeneTargets_v2_2712', 'drugName': 'S-222611', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ERBB2 (ENSG00000141736), EGFR (ENSG00000146648)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drugIsApproved': False}, {'UUID': 'DrugGeneTargets_v2_2713', ...
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Genetic Target
Q58.1659
Q58
How many genes does the drug Clonazepam target and what are they?
There are 16 gene targets for the drug Clonazepam: GABRA1, GABRB2, GABRG2, GABRB3, GABRA4, GABRG3, GABRQ, GABRA3, GABRP, GABRD, GABRG1, GABRB1, GABRE, GABRA2, GABRA5, and GABRA6.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%clonazepam%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1496', 'drugName': 'Clonazepam', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089), GABRA3 (E...
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Q58.1116
Q58
How many genes does the drug Tocainide Hydrochloride target and what are they?
There are 10 gene targets for the drug Tocainide Hydrochloride: SCN1A, SCN5A, SCN4A, SCN7A, SCN2A, SCN9A, SCN3A, SCN11A, SCN8A, and SCN10A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tocainide hydrochloride%" OR LOWER(tradeNames_st...
[{'UUID': 'DrugGeneTargets_v2_4128', 'drugName': 'Tocainide Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SCN1A (ENSG00000144285), SCN5A (ENSG00000183873), SCN4A (ENSG00000007314), SCN7A (ENSG00000136546), SCN2A (ENSG00000136531), SCN9A (ENSG00000169432), SCN3A (ENSG00000153253), SC...
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Q58.722
Q58
How many genes does the drug Idasanutlin target and what are they?
The drug Idasanutlin is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 2 genes: TP53 and MDM2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%idasanutlin%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_3191', 'drugName': 'Idasanutlin', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'TP53 (ENSG00000141510), MDM2 (ENSG00000135679)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Q58.1247
Q58
How many genes does the drug Phenytoin target and what are they?
There are 10 gene targets for the drug Phenytoin: SCN1A, SCN5A, SCN4A, SCN7A, SCN2A, SCN9A, SCN3A, SCN11A, SCN8A, and SCN10A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%phenytoin%" OR LOWER(tradeNames_string) LIKE "%p...
[{'UUID': 'DrugGeneTargets_v2_1082', 'drugName': 'Phenytoin Sodium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SCN1A (ENSG00000144285), SCN5A (ENSG00000183873), SCN4A (ENSG00000007314), SCN7A (ENSG00000136546), SCN2A (ENSG00000136531), SCN9A (ENSG00000169432), SCN3A (ENSG00000153253), SCN11A (E...
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Genetic Target
Q58.1236
Q58
How many genes does the drug Codeine Sulfate target and what are they?
There are 3 gene targets for the drug Codeine Sulfate: OPRK1, OPRD1, and OPRM1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%codeine sulfate%" OR LOWER(tradeNames_string) LI...
[{'UUID': 'DrugGeneTargets_v2_3666', 'drugName': 'Codeine Sulfate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'OPRK1 (ENSG00000082556), OPRD1 (ENSG00000116329), OPRM1 (ENSG00000112038)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 2009, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1076
Q58
How many genes does the drug Belzutifan target and what are they?
EPAS1 is the only gene target of drug Belzutifan.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%belzutifan%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_342', 'drugName': 'Belzutifan', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'EPAS1 (ENSG00000116016)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2021, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1907
Q58
How many genes does the drug Patidegib target and what are they?
The drug Patidegib is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene SMO.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%patidegib%" OR LOWER(tradeNames_string) LIKE "%p...
[{'UUID': 'DrugGeneTargets_v2_6104', 'drugName': 'Patidegib', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SMO (ENSG00000128602)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.264
Q58
How many genes does the drug Vatelizumab target and what are they?
The drug Vatelizumab is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene ITGA2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%vatelizumab%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_4470', 'drugName': 'Vatelizumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'ITGA2 (ENSG00000164171)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1437
Q58
How many genes does the drug Collagenase Clostridium Histolyticum target and what are they?
There are 25 gene targets for the drug Collagenase Clostridium Histolyticum: COL1A2, COL1A1, COL2A1, COL3A1, COL4A1, COL5A1, COL6A1, COL11A1, COL15A1, COL18A1, COL24A1, COL27A1, COL28A1, COL4A2, COL5A2, COL6A2, COL11A2, COL4A3, COL5A3, COL6A3, COL4A4, COL4A5, COL6A5, COL4A6, and COL6A6.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%collagenase clostridium histolyticum%" OR LOWER(...
[{'UUID': 'DrugGeneTargets_v2_1275', 'drugName': 'Collagenase Clostridium Histolyticum', 'drugMolecularType': 'Enzyme', 'newLinkedTargets_string': 'COL1A2 (ENSG00000164692), COL1A1 (ENSG00000108821), COL2A1 (ENSG00000139219), COL3A1 (ENSG00000168542), COL4A1 (ENSG00000187498), COL5A1 (ENSG00000130635), COL6A1 (ENSG0000...
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Genetic Target
Q58.1339
Q58
How many genes does the drug Pitavastatin Sodium target and what are they?
HMGCR is the only gene target of drug Pitavastatin Sodium.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%pitavastatin sodium%" OR LOWER(tradeNames_string...
[{'UUID': 'DrugGeneTargets_v2_1489', 'drugName': 'Pitavastatin Sodium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HMGCR (ENSG00000113161)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2017, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.243
Q58
How many genes does the drug Rocuronium target and what are they?
There are 5 gene targets for the drug Rocuronium: CHRNA1, CHRNG, CHRNB1, CHRND, and CHRNE.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%rocuronium%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1958', 'drugName': 'Rocuronium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CHRNA1 (ENSG00000138435), CHRNG (ENSG00000196811), CHRNB1 (ENSG00000170175), CHRND (ENSG00000135902), CHRNE (ENSG00000108556)', 'numberLinkedTargets': 5, 'yearOfFirstApproval': 1994, 'maxCli...
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Genetic Target
Q58.1010
Q58
How many genes does the drug Lercanidipine Hydrochloride target and what are they?
There are 4 gene targets for the drug Lercanidipine Hydrochloride: CACNA1C, CACNA1S, CACNA1D, and CACNA1F.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%lercanidipine hydrochloride%" OR LOWER(tradeName...
[{'UUID': 'DrugGeneTargets_v2_4021', 'drugName': 'Lercanidipine Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CACNA1C (ENSG00000151067), CACNA1S (ENSG00000081248), CACNA1D (ENSG00000157388), CACNA1F (ENSG00000102001)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 0, 'maxClinical...
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Genetic Target
Q58.685
Q58
How many genes does the drug Medi-8968 target and what are they?
The drug Medi-8968 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene IL1R1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%medi-8968%" OR LOWER(tradeNames_string) LIKE "%m...
[{'UUID': 'DrugGeneTargets_v2_2001', 'drugName': 'Medi-8968', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'IL1R1 (ENSG00000115594)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1268
Q58
How many genes does the drug Olanzapine target and what are they?
There are 5 gene targets for the drug Olanzapine: DRD2, DRD3, DRD4, HTR2C, and HTR2A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%olanzapine%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1531', 'drugName': 'Olanzapine Pamoate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HTR2C (ENSG00000147246), HTR2A (ENSG00000102468), DRD2 (ENSG00000149295), DRD3 (ENSG00000151577), DRD4 (ENSG00000069696)', 'numberLinkedTargets': 5, 'yearOfFirstApproval': 2009, 'max...
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Genetic Target
Q58.1475
Q58
How many genes does the drug Cerivastatin Sodium target and what are they?
HMGCR is the only gene target of drug Cerivastatin Sodium.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%cerivastatin sodium%" OR LOWER(tradeNames_string...
[{'UUID': 'DrugGeneTargets_v2_3117', 'drugName': 'Cerivastatin Sodium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HMGCR (ENSG00000113161)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1997, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1502
Q58
How many genes does the drug Tinzaparin Sodium target and what are they?
SERPINC1 is the only gene target of drug Tinzaparin Sodium.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tinzaparin sodium%" OR LOWER(tradeNames_string) ...
[{'UUID': 'DrugGeneTargets_v2_3678', 'drugName': 'Tinzaparin Sodium', 'drugMolecularType': 'Oligosaccharide', 'newLinkedTargets_string': 'SERPINC1 (ENSG00000117601)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2000, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.370
Q58
How many genes does the drug Canrenoate target and what are they?
NR3C2 is the only gene target of drug Canrenoate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%canrenoate%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_82', 'drugName': 'Canrenoate Potassium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'NR3C2 (ENSG00000151623)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_4944', 'drugName': 'Ca...
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Genetic Target
Q58.1009
Q58
How many genes does the drug Magrolimab target and what are they?
The drug Magrolimab is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene CD47.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%magrolimab%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_4258', 'drugName': 'Magrolimab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'CD47 (ENSG00000196776)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.1239
Q58
How many genes does the drug Ethchlorvynol target and what are they?
There are 16 gene targets for the drug Ethchlorvynol: GABRA1, GABRB2, GABRG2, GABRB3, GABRA4, GABRG3, GABRQ, GABRA3, GABRP, GABRD, GABRG1, GABRB1, GABRE, GABRA2, GABRA5, and GABRA6.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ethchlorvynol%" OR LOWER(tradeNames_string) LIKE...
[{'UUID': 'DrugGeneTargets_v2_3295', 'drugName': 'Ethchlorvynol', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089), GABRA3...
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Genetic Target
Q58.595
Q58
How many genes does the drug Dazodalibep target and what are they?
The drug Dazodalibep is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene CD40LG.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%dazodalibep%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_4887', 'drugName': 'Dazodalibep', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'CD40LG (ENSG00000102245)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.728
Q58
How many genes does the drug Estazolam target and what are they?
There are 16 gene targets for the drug Estazolam: GABRA1, GABRB2, GABRG2, GABRB3, GABRA4, GABRG3, GABRQ, GABRA3, GABRP, GABRD, GABRG1, GABRB1, GABRE, GABRA2, GABRA5, and GABRA6.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%estazolam%" OR LOWER(tradeNames_string) LIKE "%e...
[{'UUID': 'DrugGeneTargets_v2_6282', 'drugName': 'Estazolam', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089), GABRA3 (EN...
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Genetic Target
Q58.486
Q58
How many genes does the drug Trilostane target and what are they?
HSD3B2 is the only gene target of drug Trilostane.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%trilostane%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2278', 'drugName': 'Trilostane', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HSD3B2 (ENSG00000203859)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1984, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.573
Q58
How many genes does the drug Mecasermin Rinfabate target and what are they?
IGF1R is the only gene target of drug Mecasermin Rinfabate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%mecasermin rinfabate%" OR LOWER(tradeNames_strin...
[{'UUID': 'DrugGeneTargets_v2_672', 'drugName': 'Mecasermin Rinfabate', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'IGF1R (ENSG00000140443)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2005, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.74
Q58
How many genes does the drug Estramustine Phosphate target and what are they?
ESR2 is the only gene target of drug Estramustine Phosphate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%estramustine phosphate%" OR LOWER(tradeNames_str...
[{'UUID': 'DrugGeneTargets_v2_5377', 'drugName': 'Estramustine Phosphate Sodium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ESR2 (ENSG00000140009)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1981, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_5789', 'd...
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Genetic Target
Q58.635
Q58
How many genes does the drug Gemtuzumab Ozogamicin target and what are they?
CD33 is the only gene target of drug Gemtuzumab Ozogamicin.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%gemtuzumab ozogamicin%" OR LOWER(tradeNames_stri...
[{'UUID': 'DrugGeneTargets_v2_6112', 'drugName': 'Gemtuzumab Ozogamicin', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'CD33 (ENSG00000105383)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2000, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.262
Q58
How many genes does the drug Budigalimab target and what are they?
The drug Budigalimab is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene PDCD1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%budigalimab%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_6333', 'drugName': 'Budigalimab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'PDCD1 (ENSG00000188389)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.52
Q58
How many genes does the drug Methapyrilene Hydrochloride target and what are they?
HRH1 is the only gene target of drug Methapyrilene Hydrochloride.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%methapyrilene hydrochloride%" OR LOWER(tradeName...
[{'UUID': 'DrugGeneTargets_v2_2856', 'drugName': 'Methapyrilene Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HRH1 (ENSG00000196639)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.201
Q58
How many genes does the drug Cdx-3379 target and what are they?
The drug Cdx-3379 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene ERBB3.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%cdx-3379%" OR LOWER(tradeNames_string) LIKE "%cd...
[{'UUID': 'DrugGeneTargets_v2_1385', 'drugName': 'Cdx-3379', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'ERBB3 (ENSG00000065361)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.432
Q58
How many genes does the drug Lecozotan target and what are they?
The drug Lecozotan is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene HTR1A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%lecozotan%" OR LOWER(tradeNames_string) LIKE "%l...
[{'UUID': 'DrugGeneTargets_v2_1643', 'drugName': 'Lecozotan', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HTR1A (ENSG00000178394)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}, {'UUID': 'DrugGeneTargets_v2_6152', 'drugName': 'Lecozotan ...
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Genetic Target
Q58.1563
Q58
How many genes does the drug Fenclofenac target and what are they?
There are 2 gene targets for the drug Fenclofenac: PTGS2 and PTGS1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%fenclofenac%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_1508', 'drugName': 'Fenclofenac', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PTGS2 (ENSG00000073756), PTGS1 (ENSG00000095303)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1978, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.336
Q58
How many genes does the drug Mbx-2044 target and what are they?
The drug Mbx-2044 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene PPARG.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%mbx-2044%" OR LOWER(tradeNames_string) LIKE "%mb...
[{'UUID': 'DrugGeneTargets_v2_5830', 'drugName': 'Mbx-2044', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PPARG (ENSG00000132170)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1557
Q58
How many genes does the drug Bms-582949 target and what are they?
The drug Bms-582949 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene MAPK14.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%bms-582949%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_673', 'drugName': 'Bms-582949', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'MAPK14 (ENSG00000112062)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1539
Q58
How many genes does the drug Chlorzoxazone target and what are they?
KCNN4 is the only gene target of drug Chlorzoxazone.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%chlorzoxazone%" OR LOWER(tradeNames_string) LIKE...
[{'UUID': 'DrugGeneTargets_v2_326', 'drugName': 'Chlorzoxazone', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'KCNN4 (ENSG00000104783)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1958, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.426
Q58
How many genes does the drug Alvespimycin target and what are they?
The drug Alvespimycin is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 2 genes: HSP90AA1 and HSP90AB1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%alvespimycin%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_5099', 'drugName': 'Alvespimycin', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HSP90AA1 (ENSG00000080824), HSP90AB1 (ENSG00000096384)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.637
Q58
How many genes does the drug Vatiquinone target and what are they?
The drug Vatiquinone is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene NQO1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%vatiquinone%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_2788', 'drugName': 'Vatiquinone', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'NQO1 (ENSG00000181019)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.941
Q58
How many genes does the drug Plovamer Acetate target and what are they?
The drug Plovamer Acetate is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene HLA-DRB1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%plovamer acetate%" OR LOWER(tradeNames_string) L...
[{'UUID': 'DrugGeneTargets_v2_5057', 'drugName': 'Plovamer Acetate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HLA-DRB1 (ENSG00000196126)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.993
Q58
How many genes does the drug Amantadine Hydrochloride target and what are they?
There are 7 gene targets for the drug Amantadine Hydrochloride: GRIN1, GRIN2A, GRIN2B, GRIN2D, GRIN3B, GRIN2C, and GRIN3A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%amantadine hydrochloride%" OR LOWER(tradeNames_s...
[{'UUID': 'DrugGeneTargets_v2_768', 'drugName': 'Amantadine Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GRIN1 (ENSG00000176884), GRIN2A (ENSG00000183454), GRIN2B (ENSG00000273079), GRIN2D (ENSG00000105464), GRIN3B (ENSG00000116032), GRIN2C (ENSG00000161509), GRIN3A (ENSG0000019878...
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Genetic Target
Q58.868
Q58
How many genes does the drug Avoralstat target and what are they?
The drug Avoralstat is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene KLKB1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%avoralstat%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1318', 'drugName': 'Avoralstat', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'KLKB1 (ENSG00000164344)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.1951
Q58
How many genes does the drug Brompheniramine target and what are they?
HRH1 is the only gene target of drug Brompheniramine.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%brompheniramine%" OR LOWER(tradeNames_string) LI...
[{'UUID': 'DrugGeneTargets_v2_6367', 'drugName': 'Brompheniramine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HRH1 (ENSG00000196639)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1957, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_1014', 'drugName': 'Bro...
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Genetic Target
Q58.558
Q58
How many genes does the drug Mapatumumab target and what are they?
The drug Mapatumumab is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene TNFRSF10A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%mapatumumab%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_5538', 'drugName': 'Mapatumumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'TNFRSF10A (ENSG00000104689)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.433
Q58
How many genes does the drug Mifamurtide target and what are they?
NOD2 is the only gene target of drug Mifamurtide.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%mifamurtide%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_1449', 'drugName': 'Mifamurtide', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'NOD2 (ENSG00000167207)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_4474', 'drugName': 'Mifamurtid...
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Genetic Target
Q58.1777
Q58
How many genes does the drug Sulfasalazine target and what are they?
There are 3 gene targets for the drug Sulfasalazine: ALOX5, PTGS2, and PTGS1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%sulfasalazine%" OR LOWER(tradeNames_string) LIKE...
[{'UUID': 'DrugGeneTargets_v2_3015', 'drugName': 'Sulfasalazine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ALOX5 (ENSG00000012779), PTGS2 (ENSG00000073756), PTGS1 (ENSG00000095303)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 1950, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'U...
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Genetic Target
Q58.1834
Q58
How many genes does the drug Tas-115 target and what are they?
The drug Tas-115 is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 2 genes: MET and KDR.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tas-115%" OR LOWER(tradeNames_string) LIKE "%tas...
[{'UUID': 'DrugGeneTargets_v2_532', 'drugName': 'Tas-115', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'MET (ENSG00000105976), KDR (ENSG00000128052)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drugIsApproved': False}, {'UUID': 'DrugGeneTargets_v2_533', 'drugN...
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Genetic Target
Q58.1977
Q58
How many genes does the drug Fibrinolysin, Human target and what are they?
There are 3 gene targets for the drug Fibrinolysin, Human: FGA, FGB, and FGG.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%fibrinolysin, human%" OR LOWER(tradeNames_string...
[{'UUID': 'DrugGeneTargets_v2_1199', 'drugName': 'Fibrinolysin, Human', 'drugMolecularType': 'Unknown', 'newLinkedTargets_string': 'FGA (ENSG00000171560), FGB (ENSG00000171564), FGG (ENSG00000171557)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 1964, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1506
Q58
How many genes does the drug Remimazolam target and what are they?
There are 16 gene targets for the drug Remimazolam: GABRA1, GABRB2, GABRG2, GABRB3, GABRA4, GABRG3, GABRQ, GABRA3, GABRP, GABRD, GABRG1, GABRB1, GABRE, GABRA2, GABRA5, and GABRA6.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%remimazolam%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_3380', 'drugName': 'Remimazolam', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089), GABRA3 (...
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Genetic Target
Q58.1622
Q58
How many genes does the drug Dipivefrin target and what are they?
There are 9 gene targets for the drug Dipivefrin: ADRA1A, ADRA2A, ADRB1, ADRB2, ADRA2C, ADRA1D, ADRA1B, ADRA2B, and ADRB3.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%dipivefrin%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_842', 'drugName': 'Dipivefrin', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRA1A (ENSG00000120907), ADRA2A (ENSG00000150594), ADRB1 (ENSG00000043591), ADRB2 (ENSG00000169252), ADRA2C (ENSG00000184160), ADRA1D (ENSG00000171873), ADRA1B (ENSG00000170214), ADRA2B (ENS...
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Genetic Target
Q58.404
Q58
How many genes does the drug Tolterodine Tartrate target and what are they?
There are 2 gene targets for the drug Tolterodine Tartrate: CHRM3 and CHRM2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tolterodine tartrate%" OR LOWER(tradeNames_strin...
[{'UUID': 'DrugGeneTargets_v2_3301', 'drugName': 'Tolterodine Tartrate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CHRM3 (ENSG00000133019), CHRM2 (ENSG00000181072)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1998, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTar...
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Genetic Target
Q58.1791
Q58
How many genes does the drug Carteolol Hydrochloride target and what are they?
There are 3 gene targets for the drug Carteolol Hydrochloride: ADRB1, ADRB2, and ADRB3.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%carteolol hydrochloride%" OR LOWER(tradeNames_st...
[{'UUID': 'DrugGeneTargets_v2_1755', 'drugName': 'Carteolol Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRB1 (ENSG00000043591), ADRB2 (ENSG00000169252), ADRB3 (ENSG00000188778)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 1988, 'maxClinicalTrialPhase': 4, 'drugIsApproved': ...
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Genetic Target
Q58.195
Q58
How many genes does the drug Pravastatin Sodium target and what are they?
HMGCR is the only gene target of drug Pravastatin Sodium.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%pravastatin sodium%" OR LOWER(tradeNames_string)...
[{'UUID': 'DrugGeneTargets_v2_1605', 'drugName': 'Pravastatin Sodium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HMGCR (ENSG00000113161)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1991, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1281
Q58
How many genes does the drug Nalmefene Hydrochloride target and what are they?
There are 3 gene targets for the drug Nalmefene Hydrochloride: OPRK1, OPRD1, and OPRM1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%nalmefene hydrochloride%" OR LOWER(tradeNames_st...
[{'UUID': 'DrugGeneTargets_v2_4044', 'drugName': 'Nalmefene', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'OPRK1 (ENSG00000082556), OPRD1 (ENSG00000116329), OPRM1 (ENSG00000112038)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 1995, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID'...
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Genetic Target
Q58.1381
Q58
How many genes does the drug Propafenone target and what are they?
There are 12 gene targets for the drug Propafenone: ADRB2, SCN1A, SCN5A, SCN4A, SCN7A, SCN2A, SCN9A, SCN3A, SCN11A, SCN8A, SCN10A, and ADRB1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%propafenone%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_2589', 'drugName': 'Propafenone Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRB1 (ENSG00000043591), ADRB2 (ENSG00000169252), SCN1A (ENSG00000144285), SCN5A (ENSG00000183873), SCN4A (ENSG00000007314), SCN7A (ENSG00000136546), SCN2A (ENSG00000136531), ...
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Genetic Target
Q58.677
Q58
How many genes does the drug Cannabidiol target and what are they?
CNR1 is the only gene target of drug Cannabidiol.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%cannabidiol%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_4055', 'drugName': 'Cannabidiol', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CNR1 (ENSG00000118432)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2018, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.795
Q58
How many genes does the drug Benserazide target and what are they?
DDC is the only gene target of drug Benserazide.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%benserazide%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_2020', 'drugName': 'Benserazide', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'DDC (ENSG00000132437)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1463
Q58
How many genes does the drug Vonoprazan Fumarate target and what are they?
There are 2 gene targets for the drug Vonoprazan Fumarate: ATP4A and ATP4B.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%vonoprazan fumarate%" OR LOWER(tradeNames_string...
[{'UUID': 'DrugGeneTargets_v2_5640', 'drugName': 'Vonoprazan Fumarate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ATP4A (ENSG00000105675), ATP4B (ENSG00000186009)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2022, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1457
Q58
How many genes does the drug Terazosin Hydrochloride target and what are they?
There are 3 gene targets for the drug Terazosin Hydrochloride: ADRA1A, ADRA1D, and ADRA1B.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%terazosin hydrochloride%" OR LOWER(tradeNames_st...
[{'UUID': 'DrugGeneTargets_v2_1256', 'drugName': 'Terazosin Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRA1A (ENSG00000120907), ADRA1D (ENSG00000171873), ADRA1B (ENSG00000170214)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 1987, 'maxClinicalTrialPhase': 4, 'drugIsApproved...
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Genetic Target
Q58.144
Q58
How many genes does the drug Triclofos target and what are they?
There are 16 gene targets for the drug Triclofos: GABRA1, GABRB2, GABRG2, GABRB3, GABRA4, GABRG3, GABRQ, GABRA3, GABRP, GABRD, GABRG1, GABRB1, GABRE, GABRA2, GABRA5, and GABRA6.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%triclofos%" OR LOWER(tradeNames_string) LIKE "%t...
[{'UUID': 'DrugGeneTargets_v2_2585', 'drugName': 'Triclofos Sodium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089), GAB...
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Genetic Target
Q58.1188
Q58
How many genes does the drug Pasireotide Pamoate target and what are they?
There are 4 gene targets for the drug Pasireotide Pamoate: SSTR3, SSTR5, SSTR2, and SSTR1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%pasireotide pamoate%" OR LOWER(tradeNames_string...
[{'UUID': 'DrugGeneTargets_v2_6121', 'drugName': 'Pasireotide Pamoate', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'SSTR3 (ENSG00000278195), SSTR5 (ENSG00000162009), SSTR2 (ENSG00000180616), SSTR1 (ENSG00000139874)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 2014, 'maxClinicalTrialPhase': 4, 'dru...
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Genetic Target
Q58.3
Q58
How many genes does the drug Flurbiprofen Sodium target and what are they?
There are 2 gene targets for the drug Flurbiprofen Sodium: PTGS2 and PTGS1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%flurbiprofen sodium%" OR LOWER(tradeNames_string...
[{'UUID': 'DrugGeneTargets_v2_2737', 'drugName': 'Flurbiprofen Sodium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PTGS2 (ENSG00000073756), PTGS1 (ENSG00000095303)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1986, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.743
Q58
How many genes does the drug Flurbiprofen target and what are they?
There are 2 gene targets for the drug Flurbiprofen: PTGS2 and PTGS1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%flurbiprofen%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_2737', 'drugName': 'Flurbiprofen Sodium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PTGS2 (ENSG00000073756), PTGS1 (ENSG00000095303)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1986, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTarg...
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Genetic Target
Q58.1871
Q58
How many genes does the drug Iguratimod target and what are they?
The drug Iguratimod is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 3 genes: MIF, TRAF3IP2, and PTGS2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%iguratimod%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5945', 'drugName': 'Iguratimod', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'MIF (ENSG00000240972), TRAF3IP2 (ENSG00000056972), PTGS2 (ENSG00000073756)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}, {'UUID'...
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Genetic Target
Q58.1516
Q58
How many genes does the drug Urofollitropin target and what are they?
FSHR is the only gene target of drug Urofollitropin.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%urofollitropin%" OR LOWER(tradeNames_string) LIK...
[{'UUID': 'DrugGeneTargets_v2_5221', 'drugName': 'Urofollitropin', 'drugMolecularType': 'Unknown', 'newLinkedTargets_string': 'FSHR (ENSG00000170820)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1986, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.343
Q58
How many genes does the drug Pwt-33579 target and what are they?
The drug Pwt-33579 is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 2 genes: MTOR and PIK3CA.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%pwt-33579%" OR LOWER(tradeNames_string) LIKE "%p...
[{'UUID': 'DrugGeneTargets_v2_5396', 'drugName': 'Pwt-33579', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'MTOR (ENSG00000198793), PIK3CA (ENSG00000121879)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drugIsApproved': False}, {'UUID': 'DrugGeneTargets_v2_5397'...
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Genetic Target
Q58.626
Q58
How many genes does the drug Rilmenidine target and what are they?
The drug Rilmenidine is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene NISCH.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%rilmenidine%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_3253', 'drugName': 'Rilmenidine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'NISCH (ENSG00000010322)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.484
Q58
How many genes does the drug Desloratadine target and what are they?
HRH1 is the only gene target of drug Desloratadine.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%desloratadine%" OR LOWER(tradeNames_string) LIKE...
[{'UUID': 'DrugGeneTargets_v2_3239', 'drugName': 'Desloratadine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HRH1 (ENSG00000196639)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2001, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.532
Q58
How many genes does the drug Ulimorelin Hydrochloride target and what are they?
The drug Ulimorelin Hydrochloride is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene GHSR.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ulimorelin hydrochloride%" OR LOWER(tradeNames_s...
[{'UUID': 'DrugGeneTargets_v2_2076', 'drugName': 'Ulimorelin Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GHSR (ENSG00000121853)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.268
Q58
How many genes does the drug Bemiparin Sodium target and what are they?
SERPINC1 is the only gene target of drug Bemiparin Sodium.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%bemiparin sodium%" OR LOWER(tradeNames_string) L...
[{'UUID': 'DrugGeneTargets_v2_2284', 'drugName': 'Bemiparin Sodium', 'drugMolecularType': 'Oligosaccharide', 'newLinkedTargets_string': 'SERPINC1 (ENSG00000117601)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1390
Q58
How many genes does the drug Midostaurin target and what are they?
There are 16 gene targets for the drug Midostaurin: KIT, KDR, PDGFRB, PDGFRA, FLT3, PRKD3, PRKCI, PRKCA, PRKCG, PRKCD, PRKCB, PRKCZ, PRKCE, PRKCH, PRKD1, and PRKCQ.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%midostaurin%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_5667', 'drugName': 'Midostaurin', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'KIT (ENSG00000157404), KDR (ENSG00000128052), PDGFRB (ENSG00000113721), PDGFRA (ENSG00000134853), FLT3 (ENSG00000122025), PRKD3 (ENSG00000115825), PRKCI (ENSG00000163558), PRKCA (ENSG000001...
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Genetic Target
Q58.681
Q58
How many genes does the drug Benziodarone target and what are they?
CALM1 is the only gene target of drug Benziodarone.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%benziodarone%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_1971', 'drugName': 'Benziodarone', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CALM1 (ENSG00000198668)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.492
Q58
How many genes does the drug Levodopa target and what are they?
DRD3 is the only gene target of drug Levodopa.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%levodopa%" OR LOWER(tradeNames_string) LIKE "%le...
[{'UUID': 'DrugGeneTargets_v2_4351', 'drugName': 'Levodopa', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'DRD3 (ENSG00000151577)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1970, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_3987', 'drugName': 'Etilevodop...
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Q58.445
Q58
How many genes does the drug Danaparoid Sodium target and what are they?
SERPINC1 is the only gene target of drug Danaparoid Sodium.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%danaparoid sodium%" OR LOWER(tradeNames_string) ...
[{'UUID': 'DrugGeneTargets_v2_3361', 'drugName': 'Danaparoid Sodium', 'drugMolecularType': 'Unknown', 'newLinkedTargets_string': 'SERPINC1 (ENSG00000117601)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1996, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.274
Q58
How many genes does the drug Msc-2363318A target and what are they?
The drug Msc-2363318A is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 4 genes: AKT1, RPS6KB2, RPS6KB1, and AKT3.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%msc-2363318a%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_2448', 'drugName': 'Msc-2363318A', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'AKT1 (ENSG00000142208), RPS6KB2 (ENSG00000175634), RPS6KB1 (ENSG00000108443), AKT3 (ENSG00000117020)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drug...
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Genetic Target
Q58.187
Q58
How many genes does the drug Ag-24322 target and what are they?
The drug Ag-24322 is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 3 genes: CDK4, CDK2, and CDK1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ag-24322%" OR LOWER(tradeNames_string) LIKE "%ag...
[{'UUID': 'DrugGeneTargets_v2_1526', 'drugName': 'Ag-24322', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CDK4 (ENSG00000135446), CDK2 (ENSG00000123374), CDK1 (ENSG00000170312)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drugIsApproved': False}, {'UUID': 'Dru...
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Genetic Target
Q58.950
Q58
How many genes does the drug Huj591 177Lu target and what are they?
The drug Huj591 177Lu is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene FOLH1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%huj591 177lu%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_6225', 'drugName': 'Huj591 177Lu', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'FOLH1 (ENSG00000086205)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.247
Q58
How many genes does the drug Romidepsin target and what are they?
There are 11 gene targets for the drug Romidepsin: HDAC1, HDAC3, HDAC6, HDAC2, HDAC5, HDAC7, HDAC8, HDAC11, HDAC4, HDAC9, and HDAC10.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%romidepsin%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_6063', 'drugName': 'Romidepsin', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'HDAC1 (ENSG00000116478), HDAC3 (ENSG00000171720), HDAC6 (ENSG00000094631), HDAC2 (ENSG00000196591), HDAC5 (ENSG00000108840), HDAC7 (ENSG00000061273), HDAC8 (ENSG00000147099), HDAC11 (ENSG0000016351...
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Genetic Target
Q58.1100
Q58
How many genes does the drug Ulodesine target and what are they?
The drug Ulodesine is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene PNP.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ulodesine%" OR LOWER(tradeNames_string) LIKE "%u...
[{'UUID': 'DrugGeneTargets_v2_5299', 'drugName': 'Ulodesine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PNP (ENSG00000198805)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1018
Q58
How many genes does the drug Umeclidinium target and what are they?
CHRM3 is the only gene target of drug Umeclidinium.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%umeclidinium%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_5459', 'drugName': 'Umeclidinium Bromide', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CHRM3 (ENSG00000133019)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2013, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_2583', 'drugName'...
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Q58.590
Q58
How many genes does the drug Idarubicin target and what are they?
TOP2A is the only gene target of drug Idarubicin.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%idarubicin%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5440', 'drugName': 'Idarubicin Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'TOP2A (ENSG00000131747)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1990, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_459', 'drugNa...
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Genetic Target
Q58.1629
Q58
How many genes does the drug Treprostinil Diolamine target and what are they?
PTGIR is the only gene target of drug Treprostinil Diolamine.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%treprostinil diolamine%" OR LOWER(tradeNames_str...
[{'UUID': 'DrugGeneTargets_v2_2433', 'drugName': 'Treprostinil Diolamine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PTGIR (ENSG00000160013)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2013, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.535
Q58
How many genes does the drug Vasopressin Tannate target and what are they?
There are 3 gene targets for the drug Vasopressin Tannate: AVPR2, AVPR1B, and AVPR1A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%vasopressin tannate%" OR LOWER(tradeNames_string...
[{'UUID': 'DrugGeneTargets_v2_5785', 'drugName': 'Vasopressin Tannate', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'AVPR2 (ENSG00000126895), AVPR1B (ENSG00000198049), AVPR1A (ENSG00000166148)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 1982, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'...
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Genetic Target
Q58.899
Q58
How many genes does the drug Trihexyphenidyl Hydrochloride target and what are they?
CHRM1 is the only gene target of drug Trihexyphenidyl Hydrochloride.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%trihexyphenidyl hydrochloride%" OR LOWER(tradeNa...
[{'UUID': 'DrugGeneTargets_v2_6050', 'drugName': 'Trihexyphenidyl Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CHRM1 (ENSG00000168539)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1949, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1483
Q58
How many genes does the drug Izencitinib target and what are they?
The drug Izencitinib is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 4 genes: JAK3, JAK1, JAK2, and TYK2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%izencitinib%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_6205', 'drugName': 'Izencitinib', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'JAK3 (ENSG00000105639), JAK1 (ENSG00000162434), JAK2 (ENSG00000096968), TYK2 (ENSG00000105397)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsAppro...
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Genetic Target
Q58.1109
Q58
How many genes does the drug Amphetamine Aspartate target and what are they?
There are 2 gene targets for the drug Amphetamine Aspartate: SLC6A3 and SLC6A2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%amphetamine aspartate%" OR LOWER(tradeNames_stri...
[{'UUID': 'DrugGeneTargets_v2_1231', 'drugName': 'Amphetamine Aspartate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SLC6A3 (ENSG00000142319), SLC6A2 (ENSG00000103546)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1996, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGene...
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Genetic Target
Q58.421
Q58
How many genes does the drug Necitumumab target and what are they?
EGFR is the only gene target of drug Necitumumab.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%necitumumab%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_2498', 'drugName': 'Necitumumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'EGFR (ENSG00000146648)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2015, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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