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Q58.995
Q58
How many genes does the drug Adc3680 target and what are they?
The drug Adc3680 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene PTGDR2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%adc3680%" OR LOWER(tradeNames_string) LIKE "%adc...
[{'UUID': 'DrugGeneTargets_v2_5282', 'drugName': 'Adc3680', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PTGDR2 (ENSG00000183134)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Q58.1707
Q58
How many genes does the drug Succinylcholine Chloride target and what are they?
There are 5 gene targets for the drug Succinylcholine Chloride: CHRNA1, CHRNG, CHRNB1, CHRND, and CHRNE.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%succinylcholine chloride%" OR LOWER(tradeNames_s...
[{'UUID': 'DrugGeneTargets_v2_2723', 'drugName': 'Succinylcholine Chloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CHRNA1 (ENSG00000138435), CHRNG (ENSG00000196811), CHRNB1 (ENSG00000170175), CHRND (ENSG00000135902), CHRNE (ENSG00000108556)', 'numberLinkedTargets': 5, 'yearOfFirstApproval':...
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Genetic Target
Q58.1285
Q58
How many genes does the drug Acetaminophen target and what are they?
There are 4 gene targets for the drug Acetaminophen: PTGS2, PTGS1, TRPV1, and FAAH.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%acetaminophen%" OR LOWER(tradeNames_string) LIKE...
[{'UUID': 'DrugGeneTargets_v2_146', 'drugName': 'Acetaminophen', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PTGS2 (ENSG00000073756), PTGS1 (ENSG00000095303), TRPV1 (ENSG00000196689), FAAH (ENSG00000117480)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 1968, 'maxClinicalTrialPhase': 4, 'drug...
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Genetic Target
Q58.1645
Q58
How many genes does the drug Molindone Hydrochloride target and what are they?
There are 2 gene targets for the drug Molindone Hydrochloride: DRD2 and HTR2A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%molindone hydrochloride%" OR LOWER(tradeNames_st...
[{'UUID': 'DrugGeneTargets_v2_3041', 'drugName': 'Molindone Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'DRD2 (ENSG00000149295), HTR2A (ENSG00000102468)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1974, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneT...
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Genetic Target
Q58.886
Q58
How many genes does the drug L19Il2 target and what are they?
The drug L19Il2 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene FN1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%l19il2%" OR LOWER(tradeNames_string) LIKE "%l19i...
[{'UUID': 'DrugGeneTargets_v2_3654', 'drugName': 'L19Il2', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'FN1 (ENSG00000115414)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.827
Q58
How many genes does the drug Denufosol Tetrasodium target and what are they?
The drug Denufosol Tetrasodium is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene P2RY2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%denufosol tetrasodium%" OR LOWER(tradeNames_stri...
[{'UUID': 'DrugGeneTargets_v2_2459', 'drugName': 'Denufosol Tetrasodium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'P2RY2 (ENSG00000175591)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.1660
Q58
How many genes does the drug Bitolterol target and what are they?
ADRB2 is the only gene target of drug Bitolterol.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%bitolterol%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5529', 'drugName': 'Bitolterol', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRB2 (ENSG00000169252)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1984, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_3535', 'drugName': 'Bitolte...
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Genetic Target
Q58.972
Q58
How many genes does the drug Miridesap target and what are they?
The drug Miridesap is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene APCS.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%miridesap%" OR LOWER(tradeNames_string) LIKE "%m...
[{'UUID': 'DrugGeneTargets_v2_1308', 'drugName': 'Miridesap', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'APCS (ENSG00000132703)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1049
Q58
How many genes does the drug Pseudoephedrine target and what are they?
SLC6A2 is the only gene target of drug Pseudoephedrine.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%pseudoephedrine%" OR LOWER(tradeNames_string) LI...
[{'UUID': 'DrugGeneTargets_v2_1353', 'drugName': 'Pseudoephedrine Sulfate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SLC6A2 (ENSG00000103546)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1963, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_5086', 'drugN...
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Genetic Target
Q58.671
Q58
How many genes does the drug Mavacamten target and what are they?
There are 7 gene targets for the drug Mavacamten: MYH7, MYH6, MYH7B, MYL3, MYL2, MYL7, and MYL4.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%mavacamten%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1036', 'drugName': 'Mavacamten', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'MYH7 (ENSG00000092054), MYH6 (ENSG00000197616), MYH7B (ENSG00000078814), MYL3 (ENSG00000160808), MYL2 (ENSG00000111245), MYL7 (ENSG00000106631), MYL4 (ENSG00000198336)', 'numberLinkedTargets...
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Genetic Target
Q58.145
Q58
How many genes does the drug Asoprisnil target and what are they?
The drug Asoprisnil is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene PGR.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%asoprisnil%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_4647', 'drugName': 'Asoprisnil', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PGR (ENSG00000082175)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.1518
Q58
How many genes does the drug Alfacalcidol target and what are they?
VDR is the only gene target of drug Alfacalcidol.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%alfacalcidol%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_4543', 'drugName': 'Alfacalcidol', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'VDR (ENSG00000111424)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.1999
Q58
How many genes does the drug Tamoxifen Citrate target and what are they?
ESR1 is the only gene target of drug Tamoxifen Citrate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tamoxifen citrate%" OR LOWER(tradeNames_string) ...
[{'UUID': 'DrugGeneTargets_v2_5201', 'drugName': 'Tamoxifen Citrate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ESR1 (ENSG00000091831)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1977, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.871
Q58
How many genes does the drug Paramethasone Acetate target and what are they?
NR3C1 is the only gene target of drug Paramethasone Acetate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%paramethasone acetate%" OR LOWER(tradeNames_stri...
[{'UUID': 'DrugGeneTargets_v2_2298', 'drugName': 'Paramethasone Acetate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'NR3C1 (ENSG00000113580)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1982, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.427
Q58
How many genes does the drug Ertugliflozin target and what are they?
SLC5A2 is the only gene target of drug Ertugliflozin.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ertugliflozin%" OR LOWER(tradeNames_string) LIKE...
[{'UUID': 'DrugGeneTargets_v2_3216', 'drugName': 'Ertugliflozin', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SLC5A2 (ENSG00000140675)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2017, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.643
Q58
How many genes does the drug Daclizumab target and what are they?
There are 3 gene targets for the drug Daclizumab: IL2RA, IL2RG, and IL2RB.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%daclizumab%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5681', 'drugName': 'Daclizumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'IL2RA (ENSG00000134460), IL2RG (ENSG00000147168), IL2RB (ENSG00000100385)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 1997, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.1408
Q58
How many genes does the drug Pbf-509 target and what are they?
The drug Pbf-509 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene ADORA2A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%pbf-509%" OR LOWER(tradeNames_string) LIKE "%pbf...
[{'UUID': 'DrugGeneTargets_v2_5617', 'drugName': 'Pbf-509', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADORA2A (ENSG00000128271)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drugIsApproved': False}]
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Q58.806
Q58
How many genes does the drug Levetiracetam target and what are they?
There are 2 gene targets for the drug Levetiracetam: CACNA1B and SV2A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%levetiracetam%" OR LOWER(tradeNames_string) LIKE...
[{'UUID': 'DrugGeneTargets_v2_283', 'drugName': 'Levetiracetam', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CACNA1B (ENSG00000148408), SV2A (ENSG00000159164)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1999, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2...
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Q58.1067
Q58
How many genes does the drug Dovitinib target and what are they?
The drug Dovitinib is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 8 genes: PDGFRB, PDGFRA, KIT, FLT3, FGFR3, FLT1, FLT4, and KDR.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%dovitinib%" OR LOWER(tradeNames_string) LIKE "%d...
[{'UUID': 'DrugGeneTargets_v2_5744', 'drugName': 'Dovitinib', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PDGFRB (ENSG00000113721), PDGFRA (ENSG00000134853), KIT (ENSG00000157404), FLT3 (ENSG00000122025), FGFR3 (ENSG00000068078), FLT1 (ENSG00000102755), FLT4 (ENSG00000037280), KDR (ENSG0000012805...
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Q58.622
Q58
How many genes does the drug Candesartan Cilexetil target and what are they?
AGTR1 is the only gene target of drug Candesartan Cilexetil.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%candesartan cilexetil%" OR LOWER(tradeNames_stri...
[{'UUID': 'DrugGeneTargets_v2_2579', 'drugName': 'Candesartan Cilexetil', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'AGTR1 (ENSG00000144891)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1998, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_3868', 'drugName...
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Q58.298
Q58
How many genes does the drug Rg7185 target and what are they?
The drug Rg7185 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene PTGDR2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%rg7185%" OR LOWER(tradeNames_string) LIKE "%rg71...
[{'UUID': 'DrugGeneTargets_v2_2003', 'drugName': 'Rg7185', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PTGDR2 (ENSG00000183134)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drugIsApproved': False}]
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Q58.912
Q58
How many genes does the drug Bazlitoran target and what are they?
The drug Bazlitoran is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 3 genes: TLR8, TLR9, and TLR7.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%bazlitoran%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5581', 'drugName': 'Bazlitoran', 'drugMolecularType': 'Unknown', 'newLinkedTargets_string': 'TLR8 (ENSG00000101916), TLR9 (ENSG00000239732), TLR7 (ENSG00000196664)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}, {'UUID': 'DrugGene...
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Q58.917
Q58
How many genes does the drug Tirbanibulin target and what are they?
SRC is the only gene target of drug Tirbanibulin.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tirbanibulin%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_5805', 'drugName': 'Tirbanibulin', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SRC (ENSG00000197122)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2020, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.1903
Q58
How many genes does the drug Vandetanib target and what are they?
There are 25 gene targets for the drug Vandetanib: TEK, ERBB2, EGFR, ERBB4, ERBB3, EPHA2, EPHB2, EPHA5, EPHA4, EPHA8, EPHA6, EPHA7, EPHB3, EPHA3, EPHB1, EPHB4, EPHA1, EPHB6, EPHA10, SRC, RET, FLT1, FLT4, KDR, and PTK6.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%vandetanib%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1936', 'drugName': 'Vandetanib', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'TEK (ENSG00000120156), ERBB2 (ENSG00000141736), EGFR (ENSG00000146648), ERBB4 (ENSG00000178568), ERBB3 (ENSG00000065361), EPHA2 (ENSG00000142627), EPHB2 (ENSG00000133216), EPHA5 (ENSG0000014...
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Genetic Target
Q58.91
Q58
How many genes does the drug Seribantumab target and what are they?
The drug Seribantumab is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene ERBB3.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%seribantumab%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_4106', 'drugName': 'Seribantumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'ERBB3 (ENSG00000065361)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.42
Q58
How many genes does the drug Emactuzumab target and what are they?
The drug Emactuzumab is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene CSF1R.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%emactuzumab%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_5215', 'drugName': 'Emactuzumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'CSF1R (ENSG00000182578)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.1803
Q58
How many genes does the drug Pf-03715455 target and what are they?
The drug Pf-03715455 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene MAPK14.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%pf-03715455%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_5605', 'drugName': 'Pf-03715455', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'MAPK14 (ENSG00000112062)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1934
Q58
How many genes does the drug Daunorubicin Citrate target and what are they?
TOP2A is the only gene target of drug Daunorubicin Citrate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%daunorubicin citrate%" OR LOWER(tradeNames_strin...
[{'UUID': 'DrugGeneTargets_v2_1471', 'drugName': 'Daunorubicin Citrate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'TOP2A (ENSG00000131747)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1996, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.134
Q58
How many genes does the drug Pinacidil target and what are they?
There are 2 gene targets for the drug Pinacidil: KCNJ11 and ABCC9.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%pinacidil%" OR LOWER(tradeNames_string) LIKE "%p...
[{'UUID': 'DrugGeneTargets_v2_1076', 'drugName': 'Pinacidil', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'KCNJ11 (ENSG00000187486), ABCC9 (ENSG00000069431)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1989, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_59...
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Genetic Target
Q58.1566
Q58
How many genes does the drug Zoledronic Acid target and what are they?
FDPS is the only gene target of drug Zoledronic Acid.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%zoledronic acid%" OR LOWER(tradeNames_string) LI...
[{'UUID': 'DrugGeneTargets_v2_4706', 'drugName': 'Zoledronic Acid', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'FDPS (ENSG00000160752)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2001, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.977
Q58
How many genes does the drug Pantoprazole Sodium target and what are they?
There are 2 gene targets for the drug Pantoprazole Sodium: ATP4A and ATP4B.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%pantoprazole sodium%" OR LOWER(tradeNames_string...
[{'UUID': 'DrugGeneTargets_v2_1903', 'drugName': 'Pantoprazole Sodium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ATP4A (ENSG00000105675), ATP4B (ENSG00000186009)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2000, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1070
Q58
How many genes does the drug Ruxolitinib Phosphate target and what are they?
There are 2 gene targets for the drug Ruxolitinib Phosphate: JAK1 and JAK2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ruxolitinib phosphate%" OR LOWER(tradeNames_stri...
[{'UUID': 'DrugGeneTargets_v2_1727', 'drugName': 'Ruxolitinib Phosphate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'JAK1 (ENSG00000162434), JAK2 (ENSG00000096968)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2011, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTarg...
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Genetic Target
Q58.1856
Q58
How many genes does the drug Parecoxib Sodium target and what are they?
PTGS2 is the only gene target of drug Parecoxib Sodium.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%parecoxib sodium%" OR LOWER(tradeNames_string) L...
[{'UUID': 'DrugGeneTargets_v2_2672', 'drugName': 'Parecoxib Sodium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PTGS2 (ENSG00000073756)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1346
Q58
How many genes does the drug Cinacalcet target and what are they?
CASR is the only gene target of drug Cinacalcet.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%cinacalcet%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_841', 'drugName': 'Cinacalcet Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CASR (ENSG00000036828)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2004, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_247', 'drugName...
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Genetic Target
Q58.1831
Q58
How many genes does the drug Lenvatinib target and what are they?
There are 3 gene targets for the drug Lenvatinib: FLT1, FLT4, and KDR.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%lenvatinib%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_3026', 'drugName': 'Lenvatinib Mesylate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'FLT1 (ENSG00000102755), FLT4 (ENSG00000037280), KDR (ENSG00000128052)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 2015, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {...
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Genetic Target
Q58.167
Q58
How many genes does the drug Nesvacumab target and what are they?
The drug Nesvacumab is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene ANGPT2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%nesvacumab%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1274', 'drugName': 'Nesvacumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'ANGPT2 (ENSG00000091879)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.731
Q58
How many genes does the drug Sitaxentan Sodium target and what are they?
There are 2 gene targets for the drug Sitaxentan Sodium: EDNRB and EDNRA.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%sitaxentan sodium%" OR LOWER(tradeNames_string) ...
[{'UUID': 'DrugGeneTargets_v2_5500', 'drugName': 'Sitaxentan Sodium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'EDNRB (ENSG00000136160), EDNRA (ENSG00000151617)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2006, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.294
Q58
How many genes does the drug Wnt-974 target and what are they?
The drug Wnt-974 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene PORCN.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%wnt-974%" OR LOWER(tradeNames_string) LIKE "%wnt...
[{'UUID': 'DrugGeneTargets_v2_447', 'drugName': 'Wnt-974', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PORCN (ENSG00000102312)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1142
Q58
How many genes does the drug Fenoldopam target and what are they?
DRD1 is the only gene target of drug Fenoldopam.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%fenoldopam%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_4966', 'drugName': 'Fenoldopam', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'DRD1 (ENSG00000184845)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1997, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_4006', 'drugName': 'Fenoldop...
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Genetic Target
Q58.1536
Q58
How many genes does the drug Procyclidine Hydrochloride target and what are they?
CHRM1 is the only gene target of drug Procyclidine Hydrochloride.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%procyclidine hydrochloride%" OR LOWER(tradeNames...
[{'UUID': 'DrugGeneTargets_v2_4919', 'drugName': 'Procyclidine Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CHRM1 (ENSG00000168539)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1955, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1897
Q58
How many genes does the drug Asenapine Maleate target and what are they?
There are 2 gene targets for the drug Asenapine Maleate: HTR2A and DRD2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%asenapine maleate%" OR LOWER(tradeNames_string) ...
[{'UUID': 'DrugGeneTargets_v2_4103', 'drugName': 'Asenapine Maleate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HTR2A (ENSG00000102468), DRD2 (ENSG00000149295)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2009, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets...
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Genetic Target
Q58.1006
Q58
How many genes does the drug Metaraminol Bitartrate target and what are they?
There are 3 gene targets for the drug Metaraminol Bitartrate: ADRA1A, ADRA1D, and ADRA1B.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%metaraminol bitartrate%" OR LOWER(tradeNames_str...
[{'UUID': 'DrugGeneTargets_v2_1846', 'drugName': 'Metaraminol Bitartrate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRA1A (ENSG00000120907), ADRA1D (ENSG00000171873), ADRA1B (ENSG00000170214)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 1954, 'maxClinicalTrialPhase': 4, 'drugIsApproved'...
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Genetic Target
Q58.1421
Q58
How many genes does the drug Nafarelin Acetate target and what are they?
GNRHR is the only gene target of drug Nafarelin Acetate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%nafarelin acetate%" OR LOWER(tradeNames_string) ...
[{'UUID': 'DrugGeneTargets_v2_669', 'drugName': 'Nafarelin Acetate', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'GNRHR (ENSG00000109163)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1990, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.785
Q58
How many genes does the drug Benazepril target and what are they?
ACE is the only gene target of drug Benazepril.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%benazepril%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5353', 'drugName': 'Benazepril Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ACE (ENSG00000159640)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1991, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_5259', 'drugNam...
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Genetic Target
Q58.846
Q58
How many genes does the drug Vemurafenib target and what are they?
BRAF is the only gene target of drug Vemurafenib.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%vemurafenib%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_3298', 'drugName': 'Vemurafenib', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'BRAF (ENSG00000157764)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2011, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.352
Q58
How many genes does the drug Cariprazine Hydrochloride target and what are they?
There are 2 gene targets for the drug Cariprazine Hydrochloride: DRD2 and DRD3.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%cariprazine hydrochloride%" OR LOWER(tradeNames_...
[{'UUID': 'DrugGeneTargets_v2_4947', 'drugName': 'Cariprazine Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'DRD2 (ENSG00000149295), DRD3 (ENSG00000151577)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2015, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGene...
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Genetic Target
Q58.1945
Q58
How many genes does the drug Epinephrine target and what are they?
There are 9 gene targets for the drug Epinephrine: ADRA1A, ADRA2A, ADRB1, ADRB2, ADRA2C, ADRA1D, ADRA1B, ADRA2B, and ADRB3.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%epinephrine%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_1884', 'drugName': 'Epinephrine Bitartrate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRA1A (ENSG00000120907), ADRA2A (ENSG00000150594), ADRB1 (ENSG00000043591), ADRB2 (ENSG00000169252), ADRA2C (ENSG00000184160), ADRA1D (ENSG00000171873), ADRA1B (ENSG00000170214)...
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Genetic Target
Q58.577
Q58
How many genes does the drug Levallorphan Tartrate target and what are they?
There are 2 gene targets for the drug Levallorphan Tartrate: OPRM1 and OPRK1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%levallorphan tartrate%" OR LOWER(tradeNames_stri...
[{'UUID': 'DrugGeneTargets_v2_5565', 'drugName': 'Levallorphan Tartrate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'OPRM1 (ENSG00000112038), OPRK1 (ENSG00000082556)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1982, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTa...
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Genetic Target
Q58.1923
Q58
How many genes does the drug Vintafolide target and what are they?
The drug Vintafolide is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene FOLR1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%vintafolide%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_53', 'drugName': 'Vintafolide', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'FOLR1 (ENSG00000110195)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.1888
Q58
How many genes does the drug Me-344 target and what are they?
The drug Me-344 is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 50 genes: MT-ND6, NDUFA10, NDUFS8, MT-ND4L, NDUFA6, MT-ND1, NDUFB6, NDUFA4, NDUFA11, NDUFB7, MT-ND2, NDUFS2, MT-ND5, NDUFA8, NDUFB5, MT-ND4, MT-ND3, NDUFAB1, NDUFA1, NDUFS4, NDUFB3, NDUFC1, NDUFA2, ND...
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%me-344%" OR LOWER(tradeNames_string) LIKE "%me-3...
[{'UUID': 'DrugGeneTargets_v2_3900', 'drugName': 'Me-344', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (ENSG00000165264), NDUFA4 (EN...
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Genetic Target
Q58.1470
Q58
How many genes does the drug Rasagiline target and what are they?
MAOB is the only gene target of drug Rasagiline.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%rasagiline%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_4089', 'drugName': 'Rasagiline Mesylate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'MAOB (ENSG00000069535)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2006, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_1464', 'drugName': ...
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Genetic Target
Q58.1818
Q58
How many genes does the drug Selegiline target and what are they?
MAOB is the only gene target of drug Selegiline.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%selegiline%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_991', 'drugName': 'Selegiline Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'MAOB (ENSG00000069535)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1989, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_4707', 'drugNam...
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Genetic Target
Q58.1317
Q58
How many genes does the drug Olopatadine target and what are they?
HRH1 is the only gene target of drug Olopatadine.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%olopatadine%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_6184', 'drugName': 'Olopatadine Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HRH1 (ENSG00000196639)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1996, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_4800', 'drugN...
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Genetic Target
Q58.1501
Q58
How many genes does the drug Fgi-101-1A6 target and what are they?
The drug Fgi-101-1A6 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene TSG101.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%fgi-101-1a6%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_1451', 'drugName': 'Fgi-101-1A6', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'TSG101 (ENSG00000074319)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drugIsApproved': False}]
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Genetic Target
Q58.464
Q58
How many genes does the drug Testosterone Propionate target and what are they?
AR is the only gene target of drug Testosterone Propionate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%testosterone propionate%" OR LOWER(tradeNames_st...
[{'UUID': 'DrugGeneTargets_v2_2128', 'drugName': 'Testosterone Propionate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'AR (ENSG00000169083)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1974, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.381
Q58
How many genes does the drug Levomilnacipran target and what are they?
There are 2 gene targets for the drug Levomilnacipran: SLC6A2 and SLC6A4.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%levomilnacipran%" OR LOWER(tradeNames_string) LI...
[{'UUID': 'DrugGeneTargets_v2_5568', 'drugName': 'Levomilnacipran Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SLC6A4 (ENSG00000108576), SLC6A2 (ENSG00000103546)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2013, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': '...
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Genetic Target
Q58.1344
Q58
How many genes does the drug Tol-101 target and what are they?
The drug Tol-101 is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 4 genes: TRAV29DV5, TRAC, TRBV7-9, and TRGV3.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tol-101%" OR LOWER(tradeNames_string) LIKE "%tol...
[{'UUID': 'DrugGeneTargets_v2_5971', 'drugName': 'Tol-101', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'TRAV29DV5 (ENSG00000211810), TRAC (ENSG00000277734), TRBV7-9 (ENSG00000278030), TRGV3 (ENSG00000211699)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApprov...
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Genetic Target
Q58.337
Q58
How many genes does the drug Riociguat target and what are they?
There are 4 gene targets for the drug Riociguat: GUCY1B1, GUCY1B2, GUCY1A2, and GUCY1A1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%riociguat%" OR LOWER(tradeNames_string) LIKE "%r...
[{'UUID': 'DrugGeneTargets_v2_3991', 'drugName': 'Riociguat', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GUCY1B1 (ENSG00000061918), GUCY1B2 (ENSG00000123201), GUCY1A2 (ENSG00000152402), GUCY1A1 (ENSG00000164116)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 2013, 'maxClinicalTrialPhase': 4,...
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Genetic Target
Q58.1284
Q58
How many genes does the drug Tcd-717 target and what are they?
The drug Tcd-717 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene CHKA.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tcd-717%" OR LOWER(tradeNames_string) LIKE "%tcd...
[{'UUID': 'DrugGeneTargets_v2_6258', 'drugName': 'Tcd-717', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CHKA (ENSG00000110721)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drugIsApproved': False}]
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Genetic Target
Q58.1762
Q58
How many genes does the drug Phentermine target and what are they?
SLC6A2 is the only gene target of drug Phentermine.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%phentermine%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_4285', 'drugName': 'Mephentermine Sulfate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRA1A (ENSG00000120907), ADRA2A (ENSG00000150594), ADRB1 (ENSG00000043591), ADRB2 (ENSG00000169252), ADRA2C (ENSG00000184160), ADRA1D (ENSG00000171873), ADRA1B (ENSG00000170214),...
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Genetic Target
Q58.1459
Q58
How many genes does the drug Desoxycorticosterone Pivalate target and what are they?
NR3C2 is the only gene target of drug Desoxycorticosterone Pivalate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%desoxycorticosterone pivalate%" OR LOWER(tradeNa...
[{'UUID': 'DrugGeneTargets_v2_3356', 'drugName': 'Desoxycorticosterone Pivalate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'NR3C2 (ENSG00000151623)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1982, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.823
Q58
How many genes does the drug Glembatumumab Vedotin target and what are they?
The drug Glembatumumab Vedotin is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 16 genes: GPNMB, TUBB4B, TUBB1, TUBA3C, TUBA4A, TUBB3, TUBA1A, TUBB4A, TUBB8, TUBB, TUBA1B, TUBA1C, TUBA3E, TUBB2A, TUBB2B, and TUBB6.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%glembatumumab vedotin%" OR LOWER(tradeNames_stri...
[{'UUID': 'DrugGeneTargets_v2_6314', 'drugName': 'Glembatumumab Vedotin', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'GPNMB (ENSG00000136235), TUBB4B (ENSG00000188229), TUBB1 (ENSG00000101162), TUBA3C (ENSG00000198033), TUBA4A (ENSG00000127824), TUBB3 (ENSG00000258947), TUBA1A (ENSG00000167552), TUBB4A...
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Genetic Target
Q58.1114
Q58
How many genes does the drug Axitinib target and what are they?
There are 3 gene targets for the drug Axitinib: FLT1, FLT4, and KDR.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%axitinib%" OR LOWER(tradeNames_string) LIKE "%ax...
[{'UUID': 'DrugGeneTargets_v2_4943', 'drugName': 'Axitinib', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'FLT1 (ENSG00000102755), FLT4 (ENSG00000037280), KDR (ENSG00000128052)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 2012, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1524
Q58
How many genes does the drug Brentuximab Vedotin target and what are they?
There are 16 gene targets for the drug Brentuximab Vedotin: TNFRSF8, TUBB4B, TUBB1, TUBA3C, TUBA4A, TUBB3, TUBA1A, TUBB4A, TUBB8, TUBB, TUBA1B, TUBA1C, TUBA3E, TUBB2A, TUBB2B, and TUBB6.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%brentuximab vedotin%" OR LOWER(tradeNames_string...
[{'UUID': 'DrugGeneTargets_v2_1084', 'drugName': 'Brentuximab Vedotin', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'TNFRSF8 (ENSG00000120949), TUBB4B (ENSG00000188229), TUBB1 (ENSG00000101162), TUBA3C (ENSG00000198033), TUBA4A (ENSG00000127824), TUBB3 (ENSG00000258947), TUBA1A (ENSG00000167552), TUBB4A...
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Genetic Target
Q58.1941
Q58
How many genes does the drug Carmegliptin target and what are they?
The drug Carmegliptin is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene DPP4.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%carmegliptin%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_3419', 'drugName': 'Carmegliptin', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'DPP4 (ENSG00000197635)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1616
Q58
How many genes does the drug Sagopilone target and what are they?
The drug Sagopilone is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 15 genes: TUBB4B, TUBB1, TUBA3C, TUBA4A, TUBB3, TUBA1A, TUBB4A, TUBB8, TUBB, TUBA1B, TUBA1C, TUBA3E, TUBB2A, TUBB2B, and TUBB6.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%sagopilone%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_3189', 'drugName': 'Sagopilone', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'TUBB4B (ENSG00000188229), TUBB1 (ENSG00000101162), TUBA3C (ENSG00000198033), TUBA4A (ENSG00000127824), TUBB3 (ENSG00000258947), TUBA1A (ENSG00000167552), TUBB4A (ENSG00000104833), TUBB8 (ENS...
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Genetic Target
Q58.1898
Q58
How many genes does the drug Naproxen target and what are they?
There are 2 gene targets for the drug Naproxen: PTGS2 and PTGS1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%naproxen%" OR LOWER(tradeNames_string) LIKE "%na...
[{'UUID': 'DrugGeneTargets_v2_4517', 'drugName': 'Naproxen', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PTGS2 (ENSG00000073756), PTGS1 (ENSG00000095303)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1976, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_5291...
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Genetic Target
Q58.918
Q58
How many genes does the drug Methohexital Sodium target and what are they?
There are 16 gene targets for the drug Methohexital Sodium: GABRA1, GABRB2, GABRG2, GABRB3, GABRA4, GABRG3, GABRQ, GABRA3, GABRP, GABRD, GABRG1, GABRB1, GABRE, GABRA2, GABRA5, and GABRA6.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%methohexital sodium%" OR LOWER(tradeNames_string...
[{'UUID': 'DrugGeneTargets_v2_4143', 'drugName': 'Methohexital Sodium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089), ...
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Genetic Target
Q58.1930
Q58
How many genes does the drug Ziconotide Acetate target and what are they?
CACNA1B is the only gene target of drug Ziconotide Acetate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ziconotide acetate%" OR LOWER(tradeNames_string)...
[{'UUID': 'DrugGeneTargets_v2_4779', 'drugName': 'Ziconotide Acetate', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'CACNA1B (ENSG00000148408)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2004, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1126
Q58
How many genes does the drug Branebrutinib target and what are they?
The drug Branebrutinib is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene BTK.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%branebrutinib%" OR LOWER(tradeNames_string) LIKE...
[{'UUID': 'DrugGeneTargets_v2_2770', 'drugName': 'Branebrutinib', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'BTK (ENSG00000010671)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.332
Q58
How many genes does the drug Methamphetamine Hydrochloride target and what are they?
There are 3 gene targets for the drug Methamphetamine Hydrochloride: SLC6A4, SLC6A3, and SLC6A2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%methamphetamine hydrochloride%" OR LOWER(tradeNa...
[{'UUID': 'DrugGeneTargets_v2_5557', 'drugName': 'Methamphetamine Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SLC6A4 (ENSG00000108576), SLC6A3 (ENSG00000142319), SLC6A2 (ENSG00000103546)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 1943, 'maxClinicalTrialPhase': 4, 'drugIsAp...
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Genetic Target
Q58.1036
Q58
How many genes does the drug Rabusertib target and what are they?
The drug Rabusertib is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene CHEK1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%rabusertib%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1309', 'drugName': 'Rabusertib', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CHEK1 (ENSG00000149554)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.322
Q58
How many genes does the drug Aqw051 target and what are they?
The drug Aqw051 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene CHRNA7.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%aqw051%" OR LOWER(tradeNames_string) LIKE "%aqw0...
[{'UUID': 'DrugGeneTargets_v2_5615', 'drugName': 'Aqw051', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CHRNA7 (ENSG00000175344)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1531
Q58
How many genes does the drug Benazepril Hydrochloride target and what are they?
ACE is the only gene target of drug Benazepril Hydrochloride.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%benazepril hydrochloride%" OR LOWER(tradeNames_s...
[{'UUID': 'DrugGeneTargets_v2_5353', 'drugName': 'Benazepril Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ACE (ENSG00000159640)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1991, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1360
Q58
How many genes does the drug Diethylpropion target and what are they?
There are 2 gene targets for the drug Diethylpropion: SLC6A2 and SLC6A3.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%diethylpropion%" OR LOWER(tradeNames_string) LIK...
[{'UUID': 'DrugGeneTargets_v2_1630', 'drugName': 'Diethylpropion', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SLC6A2 (ENSG00000103546), SLC6A3 (ENSG00000142319)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1959, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets...
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Genetic Target
Q58.1734
Q58
How many genes does the drug Interferon Beta-1A target and what are they?
There are 2 gene targets for the drug Interferon Beta-1A: IFNAR1 and IFNAR2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%interferon beta-1a%" OR LOWER(tradeNames_string)...
[{'UUID': 'DrugGeneTargets_v2_635', 'drugName': 'Interferon Beta-1A', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'IFNAR1 (ENSG00000142166), IFNAR2 (ENSG00000159110)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1996, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_...
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Genetic Target
Q58.170
Q58
How many genes does the drug Morolimumab target and what are they?
The drug Morolimumab is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene RHD.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%morolimumab%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_4899', 'drugName': 'Morolimumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'RHD (ENSG00000187010)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drugIsApproved': False}]
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Genetic Target
Q58.13
Q58
How many genes does the drug Tizanidine target and what are they?
There are 3 gene targets for the drug Tizanidine: ADRA2A, ADRA2C, and ADRA2B.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tizanidine%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5012', 'drugName': 'Tizanidine Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRA2A (ENSG00000150594), ADRA2C (ENSG00000184160), ADRA2B (ENSG00000274286)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 1996, 'maxClinicalTrialPhase': 4, 'drugIsApprove...
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Genetic Target
Q58.1927
Q58
How many genes does the drug Betamethasone Acetate target and what are they?
NR3C1 is the only gene target of drug Betamethasone Acetate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%betamethasone acetate%" OR LOWER(tradeNames_stri...
[{'UUID': 'DrugGeneTargets_v2_4913', 'drugName': 'Betamethasone Acetate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'NR3C1 (ENSG00000113580)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1965, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.174
Q58
How many genes does the drug Clazakizumab target and what are they?
The drug Clazakizumab is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene IL6.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%clazakizumab%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_3651', 'drugName': 'Clazakizumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'IL6 (ENSG00000136244)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.656
Q58
How many genes does the drug Lonafarnib target and what are they?
There are 2 gene targets for the drug Lonafarnib: FNTA and FNTB.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%lonafarnib%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5762', 'drugName': 'Lonafarnib', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'FNTA (ENSG00000168522), FNTB (ENSG00000257365)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2020, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1062
Q58
How many genes does the drug Uk432097 target and what are they?
The drug Uk432097 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene ADORA2A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%uk432097%" OR LOWER(tradeNames_string) LIKE "%uk...
[{'UUID': 'DrugGeneTargets_v2_5630', 'drugName': 'Uk432097', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADORA2A (ENSG00000128271)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.263
Q58
How many genes does the drug Lercanidipine target and what are they?
There are 4 gene targets for the drug Lercanidipine: CACNA1C, CACNA1S, CACNA1D, and CACNA1F.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%lercanidipine%" OR LOWER(tradeNames_string) LIKE...
[{'UUID': 'DrugGeneTargets_v2_909', 'drugName': 'Lercanidipine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CACNA1C (ENSG00000151067), CACNA1S (ENSG00000081248), CACNA1D (ENSG00000157388), CACNA1F (ENSG00000102001)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4,...
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Genetic Target
Q58.1427
Q58
How many genes does the drug Dilevalol target and what are they?
There are 3 gene targets for the drug Dilevalol: ADRB2, ADRB1, and ADRB3.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%dilevalol%" OR LOWER(tradeNames_string) LIKE "%d...
[{'UUID': 'DrugGeneTargets_v2_6355', 'drugName': 'Dilevalol', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRB2 (ENSG00000169252), ADRB1 (ENSG00000043591), ADRB3 (ENSG00000188778)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 1990, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID'...
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Genetic Target
Q58.1582
Q58
How many genes does the drug Simlukafusp Alfa target and what are they?
The drug Simlukafusp Alfa is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 3 genes: FAP, IL2RG, and IL2RB.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%simlukafusp alfa%" OR LOWER(tradeNames_string) L...
[{'UUID': 'DrugGeneTargets_v2_4414', 'drugName': 'Simlukafusp Alfa', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'FAP (ENSG00000078098), IL2RG (ENSG00000147168), IL2RB (ENSG00000100385)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}, {'UUID': 'D...
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Genetic Target
Q58.909
Q58
How many genes does the drug Mephentermine Sulfate target and what are they?
There are 9 gene targets for the drug Mephentermine Sulfate: ADRA1A, ADRA2A, ADRB1, ADRB2, ADRA2C, ADRA1D, ADRA1B, ADRA2B, and ADRB3.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%mephentermine sulfate%" OR LOWER(tradeNames_stri...
[{'UUID': 'DrugGeneTargets_v2_4285', 'drugName': 'Mephentermine Sulfate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRA1A (ENSG00000120907), ADRA2A (ENSG00000150594), ADRB1 (ENSG00000043591), ADRB2 (ENSG00000169252), ADRA2C (ENSG00000184160), ADRA1D (ENSG00000171873), ADRA1B (ENSG00000170214),...
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Genetic Target
Q58.679
Q58
How many genes does the drug Copanlisib Hydrochloride target and what are they?
There are 2 gene targets for the drug Copanlisib Hydrochloride: PIK3CA and PIK3CD.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%copanlisib hydrochloride%" OR LOWER(tradeNames_s...
[{'UUID': 'DrugGeneTargets_v2_1213', 'drugName': 'Copanlisib Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PIK3CA (ENSG00000121879), PIK3CD (ENSG00000171608)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2017, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugG...
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Genetic Target
Q58.261
Q58
How many genes does the drug Sitagliptin Phosphate target and what are they?
DPP4 is the only gene target of drug Sitagliptin Phosphate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%sitagliptin phosphate%" OR LOWER(tradeNames_stri...
[{'UUID': 'DrugGeneTargets_v2_2411', 'drugName': 'Sitagliptin Phosphate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'DPP4 (ENSG00000197635)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2006, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.851
Q58
How many genes does the drug Doxylamine Succinate target and what are they?
HRH1 is the only gene target of drug Doxylamine Succinate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%doxylamine succinate%" OR LOWER(tradeNames_strin...
[{'UUID': 'DrugGeneTargets_v2_3456', 'drugName': 'Doxylamine Succinate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HRH1 (ENSG00000196639)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1948, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.874
Q58
How many genes does the drug Dexamethasone Phosphoric Acid target and what are they?
NR3C1 is the only gene target of drug Dexamethasone Phosphoric Acid.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%dexamethasone phosphoric acid%" OR LOWER(tradeNa...
[{'UUID': 'DrugGeneTargets_v2_4269', 'drugName': 'Dexamethasone Phosphoric Acid', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'NR3C1 (ENSG00000113580)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1959, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1564
Q58
How many genes does the drug Sad448 target and what are they?
The drug Sad448 is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 2 genes: CNR1 and CNR2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%sad448%" OR LOWER(tradeNames_string) LIKE "%sad4...
[{'UUID': 'DrugGeneTargets_v2_234', 'drugName': 'Sad448', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CNR1 (ENSG00000118432), CNR2 (ENSG00000188822)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drugIsApproved': False}, {'UUID': 'DrugGeneTargets_v2_235', 'drug...
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Genetic Target
Q58.141
Q58
How many genes does the drug Chlorpromazine Hydrochloride target and what are they?
There are 4 gene targets for the drug Chlorpromazine Hydrochloride: DRD2, DRD3, DRD4, and HTR2A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%chlorpromazine hydrochloride%" OR LOWER(tradeNam...
[{'UUID': 'DrugGeneTargets_v2_2783', 'drugName': 'Chlorpromazine Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'DRD2 (ENSG00000149295), DRD3 (ENSG00000151577), DRD4 (ENSG00000069696), HTR2A (ENSG00000102468)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 1957, 'maxClinicalTrialPh...
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Genetic Target
Q58.900
Q58
How many genes does the drug Dienestrol target and what are they?
ESR1 is the only gene target of drug Dienestrol.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%dienestrol%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5260', 'drugName': 'Dienestrol', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ESR1 (ENSG00000091831)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1947, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1839
Q58
How many genes does the drug Nadroparin Calcium target and what are they?
The drug Nadroparin Calcium is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene SERPINC1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%nadroparin calcium%" OR LOWER(tradeNames_string)...
[{'UUID': 'DrugGeneTargets_v2_5178', 'drugName': 'Nadroparin Calcium', 'drugMolecularType': 'Oligosaccharide', 'newLinkedTargets_string': 'SERPINC1 (ENSG00000117601)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.555
Q58
How many genes does the drug Pitavastatin Magnesium target and what are they?
HMGCR is the only gene target of drug Pitavastatin Magnesium.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%pitavastatin magnesium%" OR LOWER(tradeNames_str...
[{'UUID': 'DrugGeneTargets_v2_1773', 'drugName': 'Pitavastatin Magnesium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HMGCR (ENSG00000113161)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2017, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.323
Q58
How many genes does the drug Ivabradine Hydrochloride target and what are they?
HCN4 is the only gene target of drug Ivabradine Hydrochloride.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ivabradine hydrochloride%" OR LOWER(tradeNames_s...
[{'UUID': 'DrugGeneTargets_v2_1183', 'drugName': 'Ivabradine Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HCN4 (ENSG00000138622)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2015, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1854
Q58
How many genes does the drug Zimlovisertib target and what are they?
The drug Zimlovisertib is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene IRAK4.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%zimlovisertib%" OR LOWER(tradeNames_string) LIKE...
[{'UUID': 'DrugGeneTargets_v2_4254', 'drugName': 'Zimlovisertib', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'IRAK4 (ENSG00000198001)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1235
Q58
How many genes does the drug Tesamorelin target and what are they?
GHRHR is the only gene target of drug Tesamorelin.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tesamorelin%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_2825', 'drugName': 'Tesamorelin', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'GHRHR (ENSG00000106128)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2010, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_4100', 'drugName': 'Tesamorelin A...
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Genetic Target
Q58.1726
Q58
How many genes does the drug Olezarsen target and what are they?
The drug Olezarsen is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene APOC3.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%olezarsen%" OR LOWER(tradeNames_string) LIKE "%o...
[{'UUID': 'DrugGeneTargets_v2_2017', 'drugName': 'Olezarsen', 'drugMolecularType': 'Oligonucleotide', 'newLinkedTargets_string': 'APOC3 (ENSG00000110245)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.564
Q58
How many genes does the drug Etretinate target and what are they?
There are 6 gene targets for the drug Etretinate: RXRB, RARG, RXRG, RARB, RARA, and RXRA.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%etretinate%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_343', 'drugName': 'Etretinate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'RXRB (ENSG00000204231), RARG (ENSG00000172819), RXRG (ENSG00000143171), RARB (ENSG00000077092), RARA (ENSG00000131759), RXRA (ENSG00000186350)', 'numberLinkedTargets': 6, 'yearOfFirstApproval...
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