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Q58.142
Q58
How many genes does the drug Dronedarone Hydrochloride target and what are they?
There are 16 gene targets for the drug Dronedarone Hydrochloride: CACNA1C, CACNA1S, CACNA1D, CACNA1F, HCN4, SCN1A, SCN5A, SCN4A, SCN7A, SCN2A, SCN9A, SCN3A, SCN11A, SCN8A, SCN10A, and KCNJ2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%dronedarone hydrochloride%" OR LOWER(tradeNames_...
[{'UUID': 'DrugGeneTargets_v2_3873', 'drugName': 'Dronedarone Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CACNA1C (ENSG00000151067), CACNA1S (ENSG00000081248), CACNA1D (ENSG00000157388), CACNA1F (ENSG00000102001), HCN4 (ENSG00000138622), SCN1A (ENSG00000144285), SCN5A (ENSG0000018...
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Genetic Target
Q58.1736
Q58
How many genes does the drug Penbutolol Sulfate target and what are they?
There are 2 gene targets for the drug Penbutolol Sulfate: ADRB2 and ADRB1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%penbutolol sulfate%" OR LOWER(tradeNames_string)...
[{'UUID': 'DrugGeneTargets_v2_1057', 'drugName': 'Penbutolol Sulfate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRB2 (ENSG00000169252), ADRB1 (ENSG00000043591)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1987, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTarge...
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Genetic Target
Q58.537
Q58
How many genes does the drug Taletrectinib target and what are they?
The drug Taletrectinib is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 4 genes: NTRK1, NTRK2, NTRK3, and ROS1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%taletrectinib%" OR LOWER(tradeNames_string) LIKE...
[{'UUID': 'DrugGeneTargets_v2_4934', 'drugName': 'Taletrectinib', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'NTRK1 (ENSG00000198400), NTRK2 (ENSG00000148053), NTRK3 (ENSG00000140538), ROS1 (ENSG00000047936)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIs...
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Genetic Target
Q58.227
Q58
How many genes does the drug Tolazamide target and what are they?
There are 2 gene targets for the drug Tolazamide: KCNJ11 and ABCC8.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tolazamide%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2335', 'drugName': 'Tolazamide', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'KCNJ11 (ENSG00000187486), ABCC8 (ENSG00000006071)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1966, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.730
Q58
How many genes does the drug Nilutamide target and what are they?
AR is the only gene target of drug Nilutamide.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%nilutamide%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5601', 'drugName': 'Nilutamide', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'AR (ENSG00000169083)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1996, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.793
Q58
How many genes does the drug Glucagon Hydrochloride target and what are they?
GCGR is the only gene target of drug Glucagon Hydrochloride.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%glucagon hydrochloride%" OR LOWER(tradeNames_str...
[{'UUID': 'DrugGeneTargets_v2_2238', 'drugName': 'Glucagon Hydrochloride', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'GCGR (ENSG00000215644)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1960, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_4736', 'drugName': 'Das...
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Genetic Target
Q58.1718
Q58
How many genes does the drug Cyclopentolate target and what are they?
CHRM3 is the only gene target of drug Cyclopentolate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%cyclopentolate%" OR LOWER(tradeNames_string) LIK...
[{'UUID': 'DrugGeneTargets_v2_5172', 'drugName': 'Cyclopentolate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CHRM3 (ENSG00000133019)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1974, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_6338', 'drugName': 'Cyc...
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Genetic Target
Q58.994
Q58
How many genes does the drug Enalaprilat target and what are they?
ACE is the only gene target of drug Enalaprilat.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%enalaprilat%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_2276', 'drugName': 'Enalaprilat', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ACE (ENSG00000159640)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_1101', 'drugName': 'Enalaprilat...
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Genetic Target
Q58.415
Q58
How many genes does the drug Loperamide target and what are they?
OPRM1 is the only gene target of drug Loperamide.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%loperamide%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_3319', 'drugName': 'Loperamide', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'OPRM1 (ENSG00000112038)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1976, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_6052', 'drugName': 'Loperam...
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Genetic Target
Q58.329
Q58
How many genes does the drug Yttrium Y 90 Epratuzumab Tetraxetan target and what are they?
The drug Yttrium Y 90 Epratuzumab Tetraxetan is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene CD22.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%yttrium y 90 epratuzumab tetraxetan%" OR LOWER(t...
[{'UUID': 'DrugGeneTargets_v2_1182', 'drugName': 'Yttrium Y 90 Epratuzumab Tetraxetan', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'CD22 (ENSG00000012124)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1098
Q58
How many genes does the drug Clevidipine target and what are they?
There are 4 gene targets for the drug Clevidipine: CACNA1C, CACNA1S, CACNA1D, and CACNA1F.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%clevidipine%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_250', 'drugName': 'Clevidipine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CACNA1C (ENSG00000151067), CACNA1S (ENSG00000081248), CACNA1D (ENSG00000157388), CACNA1F (ENSG00000102001)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 2008, 'maxClinicalTrialPhase': 4...
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Genetic Target
Q58.303
Q58
How many genes does the drug Tibulizumab target and what are they?
The drug Tibulizumab is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 2 genes: IL17A and TNFSF13B.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tibulizumab%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_3619', 'drugName': 'Tibulizumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'IL17A (ENSG00000112115), TNFSF13B (ENSG00000102524)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}, {'UUID': 'DrugGeneTargets_v2_3620',...
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Genetic Target
Q58.1259
Q58
How many genes does the drug Dexamethasone target and what are they?
NR3C1 is the only gene target of drug Dexamethasone.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%dexamethasone%" OR LOWER(tradeNames_string) LIKE...
[{'UUID': 'DrugGeneTargets_v2_3466', 'drugName': 'Dexamethasone Sodium Phosphate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'NR3C1 (ENSG00000113580)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1959, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_535', '...
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Genetic Target
Q58.1996
Q58
How many genes does the drug Clidinium target and what are they?
There are 2 gene targets for the drug Clidinium: CHRM3 and CHRM1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%clidinium%" OR LOWER(tradeNames_string) LIKE "%c...
[{'UUID': 'DrugGeneTargets_v2_73', 'drugName': 'Clidinium Bromide', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CHRM3 (ENSG00000133019), CHRM1 (ENSG00000168539)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1982, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_...
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Genetic Target
Q58.26
Q58
How many genes does the drug Oxybutynin target and what are they?
There are 2 gene targets for the drug Oxybutynin: CHRM3 and CHRM2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%oxybutynin%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_3', 'drugName': 'Oxybutynin', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CHRM3 (ENSG00000133019), CHRM2 (ENSG00000181072)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1975, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_2', '...
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Genetic Target
Q58.1860
Q58
How many genes does the drug Degarelix target and what are they?
GNRHR is the only gene target of drug Degarelix.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%degarelix%" OR LOWER(tradeNames_string) LIKE "%d...
[{'UUID': 'DrugGeneTargets_v2_6054', 'drugName': 'Degarelix Acetate', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'GNRHR (ENSG00000109163)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2008, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_1491', 'drugName': 'Degarel...
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Genetic Target
Q58.721
Q58
How many genes does the drug Erenumab target and what are they?
CALCRL is the only gene target of drug Erenumab.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%erenumab%" OR LOWER(tradeNames_string) LIKE "%er...
[{'UUID': 'DrugGeneTargets_v2_5361', 'drugName': 'Erenumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'CALCRL (ENSG00000064989)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2018, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.996
Q58
How many genes does the drug Relatlimab target and what are they?
LAG3 is the only gene target of drug Relatlimab.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%relatlimab%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2446', 'drugName': 'Relatlimab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'LAG3 (ENSG00000089692)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2022, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.196
Q58
How many genes does the drug Diltiazem Malate target and what are they?
There are 4 gene targets for the drug Diltiazem Malate: CACNA1C, CACNA1S, CACNA1D, and CACNA1F.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%diltiazem malate%" OR LOWER(tradeNames_string) L...
[{'UUID': 'DrugGeneTargets_v2_3324', 'drugName': 'Diltiazem Malate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CACNA1C (ENSG00000151067), CACNA1S (ENSG00000081248), CACNA1D (ENSG00000157388), CACNA1F (ENSG00000102001)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 1996, 'maxClinicalTrialPha...
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Q58.446
Q58
How many genes does the drug Anileridine target and what are they?
There are 2 gene targets for the drug Anileridine: OPRM1 and OPRK1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%anileridine%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_4939', 'drugName': 'Anileridine Phosphate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'OPRM1 (ENSG00000112038), OPRK1 (ENSG00000082556)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1982, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTa...
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Genetic Target
Q58.579
Q58
How many genes does the drug St1535 target and what are they?
The drug St1535 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene ADORA2A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%st1535%" OR LOWER(tradeNames_string) LIKE "%st15...
[{'UUID': 'DrugGeneTargets_v2_3125', 'drugName': 'St1535', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADORA2A (ENSG00000128271)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drugIsApproved': False}]
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Genetic Target
Q58.955
Q58
How many genes does the drug Etavopivat target and what are they?
The drug Etavopivat is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene PKLR.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%etavopivat%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_660', 'drugName': 'Etavopivat', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PKLR (ENSG00000143627)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Q58.509
Q58
How many genes does the drug Sar-407899 target and what are they?
The drug Sar-407899 is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 2 genes: ROCK2 and ROCK1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%sar-407899%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_996', 'drugName': 'Sar-407899', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ROCK2 (ENSG00000134318), ROCK1 (ENSG00000067900)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}, {'UUID': 'DrugGeneTargets_v2_5513'...
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Q58.612
Q58
How many genes does the drug Lamotrigine target and what are they?
There are 10 gene targets for the drug Lamotrigine: SCN1A, SCN5A, SCN4A, SCN7A, SCN2A, SCN9A, SCN3A, SCN11A, SCN8A, and SCN10A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%lamotrigine%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_5462', 'drugName': 'Lamotrigine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SCN1A (ENSG00000144285), SCN5A (ENSG00000183873), SCN4A (ENSG00000007314), SCN7A (ENSG00000136546), SCN2A (ENSG00000136531), SCN9A (ENSG00000169432), SCN3A (ENSG00000153253), SCN11A (ENSG00...
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Genetic Target
Q58.1864
Q58
How many genes does the drug Dimethindene target and what are they?
HRH1 is the only gene target of drug Dimethindene.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%dimethindene%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_588', 'drugName': 'Dimethindene', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HRH1 (ENSG00000196639)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1725
Q58
How many genes does the drug Panobinostat Lactate target and what are they?
There are 11 gene targets for the drug Panobinostat Lactate: HDAC1, HDAC3, HDAC6, HDAC2, HDAC5, HDAC7, HDAC8, HDAC11, HDAC4, HDAC9, and HDAC10.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%panobinostat lactate%" OR LOWER(tradeNames_strin...
[{'UUID': 'DrugGeneTargets_v2_5237', 'drugName': 'Panobinostat Lactate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HDAC1 (ENSG00000116478), HDAC3 (ENSG00000171720), HDAC6 (ENSG00000094631), HDAC2 (ENSG00000196591), HDAC5 (ENSG00000108840), HDAC7 (ENSG00000061273), HDAC8 (ENSG00000147099), HDAC1...
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Genetic Target
Q58.1885
Q58
How many genes does the drug Metyrosine target and what are they?
TH is the only gene target of drug Metyrosine.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%metyrosine%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2694', 'drugName': 'Metyrosine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'TH (ENSG00000180176)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1979, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.853
Q58
How many genes does the drug Tocilizumab target and what are they?
IL6R is the only gene target of drug Tocilizumab.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tocilizumab%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_2072', 'drugName': 'Tocilizumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'IL6R (ENSG00000160712)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2005, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.4
Q58
How many genes does the drug Diazoxide target and what are they?
There are 2 gene targets for the drug Diazoxide: KCNJ11 and KCNJ8.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%diazoxide%" OR LOWER(tradeNames_string) LIKE "%d...
[{'UUID': 'DrugGeneTargets_v2_1171', 'drugName': 'Diazoxide', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'KCNJ11 (ENSG00000187486), KCNJ8 (ENSG00000121361)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1973, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_11...
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Genetic Target
Q58.1569
Q58
How many genes does the drug Tranylcypromine target and what are they?
There are 2 gene targets for the drug Tranylcypromine: MAOA and MAOB.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tranylcypromine%" OR LOWER(tradeNames_string) LI...
[{'UUID': 'DrugGeneTargets_v2_3703', 'drugName': 'Tranylcypromine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'MAOA (ENSG00000189221), MAOB (ENSG00000069535)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1961, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2...
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Genetic Target
Q58.1461
Q58
How many genes does the drug Milnacipran Hydrochloride target and what are they?
There are 2 gene targets for the drug Milnacipran Hydrochloride: SLC6A2 and SLC6A4.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%milnacipran hydrochloride%" OR LOWER(tradeNames_...
[{'UUID': 'DrugGeneTargets_v2_4226', 'drugName': 'Milnacipran Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SLC6A2 (ENSG00000103546), SLC6A4 (ENSG00000108576)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2009, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'Drug...
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Genetic Target
Q58.473
Q58
How many genes does the drug Maprotiline Hydrochloride target and what are they?
SLC6A2 is the only gene target of drug Maprotiline Hydrochloride.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%maprotiline hydrochloride%" OR LOWER(tradeNames_...
[{'UUID': 'DrugGeneTargets_v2_4631', 'drugName': 'Maprotiline Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SLC6A2 (ENSG00000103546)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1980, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.325
Q58
How many genes does the drug Vosoritide target and what are they?
NPR2 is the only gene target of drug Vosoritide.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%vosoritide%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_6124', 'drugName': 'Vosoritide', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'NPR2 (ENSG00000159899)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2021, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.6
Q58
How many genes does the drug Benoxaprofen target and what are they?
ALOX12 is the only gene target of drug Benoxaprofen.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%benoxaprofen%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_5509', 'drugName': 'Benoxaprofen', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ALOX12 (ENSG00000108839)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1982, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.225
Q58
How many genes does the drug Azd-8330 target and what are they?
The drug Azd-8330 is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 2 genes: MAP2K1 and MAP2K2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%azd-8330%" OR LOWER(tradeNames_string) LIKE "%az...
[{'UUID': 'DrugGeneTargets_v2_4849', 'drugName': 'Azd-8330', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'MAP2K1 (ENSG00000169032), MAP2K2 (ENSG00000126934)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drugIsApproved': False}, {'UUID': 'DrugGeneTargets_v2_4850...
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Genetic Target
Q58.1376
Q58
How many genes does the drug Atogepant target and what are they?
CALCRL is the only gene target of drug Atogepant.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%atogepant%" OR LOWER(tradeNames_string) LIKE "%a...
[{'UUID': 'DrugGeneTargets_v2_2683', 'drugName': 'Atogepant', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CALCRL (ENSG00000064989)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2021, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.553
Q58
How many genes does the drug Flecainide target and what are they?
SCN5A is the only gene target of drug Flecainide.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%flecainide%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5669', 'drugName': 'Flecainide', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SCN5A (ENSG00000183873)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1985, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_605', 'drugName': 'Flecaini...
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Genetic Target
Q58.231
Q58
How many genes does the drug Pf-04991532 target and what are they?
The drug Pf-04991532 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene GCK.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%pf-04991532%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_4171', 'drugName': 'Pf-04991532', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GCK (ENSG00000106633)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.40
Q58
How many genes does the drug Mitapivat target and what are they?
PKLR is the only gene target of drug Mitapivat.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%mitapivat%" OR LOWER(tradeNames_string) LIKE "%m...
[{'UUID': 'DrugGeneTargets_v2_4932', 'drugName': 'Mitapivat', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PKLR (ENSG00000143627)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2022, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_2811', 'drugName': 'Mitapivat...
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Genetic Target
Q58.548
Q58
How many genes does the drug Amelparib Dihydrochloride Dihydrate target and what are they?
The drug Amelparib Dihydrochloride Dihydrate is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene PARP1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%amelparib dihydrochloride dihydrate%" OR LOWER(t...
[{'UUID': 'DrugGeneTargets_v2_2907', 'drugName': 'Amelparib Dihydrochloride Dihydrate', 'drugMolecularType': 'Unknown', 'newLinkedTargets_string': 'PARP1 (ENSG00000143799)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.245
Q58
How many genes does the drug Idelalisib target and what are they?
PIK3CD is the only gene target of drug Idelalisib.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%idelalisib%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_3742', 'drugName': 'Idelalisib', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PIK3CD (ENSG00000171608)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2014, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.905
Q58
How many genes does the drug Methantheline target and what are they?
HRH2 is the only gene target of drug Methantheline.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%methantheline%" OR LOWER(tradeNames_string) LIKE...
[{'UUID': 'DrugGeneTargets_v2_3052', 'drugName': 'Methantheline', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HRH2 (ENSG00000113749)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1951, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_3603', 'drugName': 'Metha...
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Genetic Target
Q58.1429
Q58
How many genes does the drug Disulfiram target and what are they?
ALDH2 is the only gene target of drug Disulfiram.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%disulfiram%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5934', 'drugName': 'Disulfiram', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ALDH2 (ENSG00000111275)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1951, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.139
Q58
How many genes does the drug Regramostim target and what are they?
The drug Regramostim is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene CSF3R.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%regramostim%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_3609', 'drugName': 'Regramostim', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'CSF3R (ENSG00000119535)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.1191
Q58
How many genes does the drug Pf-4191834 target and what are they?
The drug Pf-4191834 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene ALOX5.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%pf-4191834%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_697', 'drugName': 'Pf-4191834', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ALOX5 (ENSG00000012779)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1757
Q58
How many genes does the drug Cep-1347 target and what are they?
The drug Cep-1347 is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 5 genes: MAP3K13, MAP3K12, MAP3K10, MAP3K9, and MAP3K11.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%cep-1347%" OR LOWER(tradeNames_string) LIKE "%ce...
[{'UUID': 'DrugGeneTargets_v2_6091', 'drugName': 'Cep-1347', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'MAP3K13 (ENSG00000073803), MAP3K12 (ENSG00000139625), MAP3K10 (ENSG00000130758), MAP3K9 (ENSG00000006432), MAP3K11 (ENSG00000173327)', 'numberLinkedTargets': 5, 'yearOfFirstApproval': 0, 'maxC...
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Genetic Target
Q58.1573
Q58
How many genes does the drug Fluoxymesterone target and what are they?
AR is the only gene target of drug Fluoxymesterone.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%fluoxymesterone%" OR LOWER(tradeNames_string) LI...
[{'UUID': 'DrugGeneTargets_v2_3575', 'drugName': 'Fluoxymesterone', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'AR (ENSG00000169083)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1956, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1443
Q58
How many genes does the drug Evenamide target and what are they?
The drug Evenamide is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 10 genes: SCN1A, SCN5A, SCN4A, SCN7A, SCN2A, SCN9A, SCN3A, SCN11A, SCN8A, and SCN10A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%evenamide%" OR LOWER(tradeNames_string) LIKE "%e...
[{'UUID': 'DrugGeneTargets_v2_1248', 'drugName': 'Evenamide', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SCN1A (ENSG00000144285), SCN5A (ENSG00000183873), SCN4A (ENSG00000007314), SCN7A (ENSG00000136546), SCN2A (ENSG00000136531), SCN9A (ENSG00000169432), SCN3A (ENSG00000153253), SCN11A (ENSG0000...
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Genetic Target
Q58.836
Q58
How many genes does the drug Trimethaphan Camsylate target and what are they?
There are 2 gene targets for the drug Trimethaphan Camsylate: CHRNB4 and CHRNA3.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%trimethaphan camsylate%" OR LOWER(tradeNames_str...
[{'UUID': 'DrugGeneTargets_v2_5467', 'drugName': 'Trimethaphan Camsylate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CHRNB4 (ENSG00000117971), CHRNA3 (ENSG00000080644)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1982, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.451
Q58
How many genes does the drug Methaqualone Hydrochloride target and what are they?
There are 16 gene targets for the drug Methaqualone Hydrochloride: GABRA1, GABRB2, GABRG2, GABRB3, GABRA4, GABRG3, GABRQ, GABRA3, GABRP, GABRD, GABRG1, GABRB1, GABRE, GABRA2, GABRA5, and GABRA6.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%methaqualone hydrochloride%" OR LOWER(tradeNames...
[{'UUID': 'DrugGeneTargets_v2_2025', 'drugName': 'Methaqualone Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG0000026...
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Genetic Target
Q58.849
Q58
How many genes does the drug Mycophenolate Sodium target and what are they?
There are 2 gene targets for the drug Mycophenolate Sodium: IMPDH1 and IMPDH2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%mycophenolate sodium%" OR LOWER(tradeNames_strin...
[{'UUID': 'DrugGeneTargets_v2_2561', 'drugName': 'Mycophenolate Sodium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'IMPDH1 (ENSG00000106348), IMPDH2 (ENSG00000178035)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2004, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1087
Q58
How many genes does the drug Goserelin Acetate target and what are they?
GNRHR is the only gene target of drug Goserelin Acetate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%goserelin acetate%" OR LOWER(tradeNames_string) ...
[{'UUID': 'DrugGeneTargets_v2_246', 'drugName': 'Goserelin Acetate', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'GNRHR (ENSG00000109163)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1989, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_2259', 'drugName': 'Gosereli...
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Genetic Target
Q58.1420
Q58
How many genes does the drug Buserelin target and what are they?
GNRHR is the only gene target of drug Buserelin.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%buserelin%" OR LOWER(tradeNames_string) LIKE "%b...
[{'UUID': 'DrugGeneTargets_v2_5687', 'drugName': 'Buserelin', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'GNRHR (ENSG00000109163)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1154
Q58
How many genes does the drug Fosbretabulin target and what are they?
The drug Fosbretabulin is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 15 genes: TUBB4B, TUBB1, TUBA3C, TUBA4A, TUBB3, TUBA1A, TUBB4A, TUBB8, TUBB, TUBA1B, TUBA1C, TUBA3E, TUBB2A, TUBB2B, and TUBB6.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%fosbretabulin%" OR LOWER(tradeNames_string) LIKE...
[{'UUID': 'DrugGeneTargets_v2_3390', 'drugName': 'Fosbretabulin', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'TUBB4B (ENSG00000188229), TUBB1 (ENSG00000101162), TUBA3C (ENSG00000198033), TUBA4A (ENSG00000127824), TUBB3 (ENSG00000258947), TUBA1A (ENSG00000167552), TUBB4A (ENSG00000104833), TUBB8 (...
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Genetic Target
Q58.1826
Q58
How many genes does the drug Dorzolamide Hydrochloride target and what are they?
CA2 is the only gene target of drug Dorzolamide Hydrochloride.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%dorzolamide hydrochloride%" OR LOWER(tradeNames_...
[{'UUID': 'DrugGeneTargets_v2_1719', 'drugName': 'Dorzolamide Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CA2 (ENSG00000104267)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1994, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.588
Q58
How many genes does the drug Ralpancizumab target and what are they?
The drug Ralpancizumab is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene PCSK9.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ralpancizumab%" OR LOWER(tradeNames_string) LIKE...
[{'UUID': 'DrugGeneTargets_v2_4790', 'drugName': 'Ralpancizumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'PCSK9 (ENSG00000169174)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drugIsApproved': False}]
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Genetic Target
Q58.1892
Q58
How many genes does the drug Pentostatin target and what are they?
ADA is the only gene target of drug Pentostatin.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%pentostatin%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_251', 'drugName': 'Pentostatin', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADA (ENSG00000196839)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1991, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1970
Q58
How many genes does the drug Diflunisal target and what are they?
There are 2 gene targets for the drug Diflunisal: PTGS2 and PTGS1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%diflunisal%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_602', 'drugName': 'Diflunisal', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PTGS2 (ENSG00000073756), PTGS1 (ENSG00000095303)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1982, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.668
Q58
How many genes does the drug Cobolimab target and what are they?
The drug Cobolimab is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene HAVCR2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%cobolimab%" OR LOWER(tradeNames_string) LIKE "%c...
[{'UUID': 'DrugGeneTargets_v2_5425', 'drugName': 'Cobolimab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'HAVCR2 (ENSG00000135077)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.442
Q58
How many genes does the drug Dextromethorphan Hydrobromide target and what are they?
There are 2 gene targets for the drug Dextromethorphan Hydrobromide: GRIN2A and SIGMAR1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%dextromethorphan hydrobromide%" OR LOWER(tradeNa...
[{'UUID': 'DrugGeneTargets_v2_5995', 'drugName': 'Dextromethorphan Hydrobromide', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GRIN2A (ENSG00000183454), SIGMAR1 (ENSG00000147955)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1984, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': ...
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Genetic Target
Q58.1857
Q58
How many genes does the drug Dantrolene Sodium target and what are they?
There are 2 gene targets for the drug Dantrolene Sodium: RYR3 and RYR1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%dantrolene sodium%" OR LOWER(tradeNames_string) ...
[{'UUID': 'DrugGeneTargets_v2_4504', 'drugName': 'Dantrolene Sodium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'RYR3 (ENSG00000198838), RYR1 (ENSG00000196218)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1974, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_...
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Genetic Target
Q58.382
Q58
How many genes does the drug Calcitonin Human target and what are they?
CALCR is the only gene target of drug Calcitonin Human.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%calcitonin human%" OR LOWER(tradeNames_string) L...
[{'UUID': 'DrugGeneTargets_v2_1951', 'drugName': 'Calcitonin Human', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'CALCR (ENSG00000004948)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1986, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1478
Q58
How many genes does the drug Bms-813160 target and what are they?
The drug Bms-813160 is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 2 genes: CCR2 and CCR5.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%bms-813160%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1069', 'drugName': 'Bms-813160', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CCR2 (ENSG00000121807), CCR5 (ENSG00000160791)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}, {'UUID': 'DrugGeneTargets_v2_1070',...
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Genetic Target
Q58.974
Q58
How many genes does the drug Ciprofibrate target and what are they?
PPARA is the only gene target of drug Ciprofibrate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ciprofibrate%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_4561', 'drugName': 'Ciprofibrate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PPARA (ENSG00000186951)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1210
Q58
How many genes does the drug Aus-131 target and what are they?
The drug Aus-131 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene ESR2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%aus-131%" OR LOWER(tradeNames_string) LIKE "%aus...
[{'UUID': 'DrugGeneTargets_v2_6316', 'drugName': 'Aus-131', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ESR2 (ENSG00000140009)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.318
Q58
How many genes does the drug Acotiamide target and what are they?
The drug Acotiamide is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene ACHE.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%acotiamide%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_3004', 'drugName': 'Acotiamide Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ACHE (ENSG00000087085)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}, {'UUID': 'DrugGeneTargets_v2_5855', 'drugName...
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Genetic Target
Q58.698
Q58
How many genes does the drug Methdilazine target and what are they?
HRH1 is the only gene target of drug Methdilazine.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%methdilazine%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_2195', 'drugName': 'Methdilazine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HRH1 (ENSG00000196639)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1982, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_6240', 'drugName': 'Methdi...
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Genetic Target
Q58.1505
Q58
How many genes does the drug Ponatinib target and what are they?
There are 2 gene targets for the drug Ponatinib: ABL1 and BCR.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ponatinib%" OR LOWER(tradeNames_string) LIKE "%p...
[{'UUID': 'DrugGeneTargets_v2_2277', 'drugName': 'Ponatinib', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ABL1 (ENSG00000097007), BCR (ENSG00000186716)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2012, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_6150',...
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Genetic Target
Q58.430
Q58
How many genes does the drug Plecanatide target and what are they?
GUCY2C is the only gene target of drug Plecanatide.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%plecanatide%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_5758', 'drugName': 'Plecanatide', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'GUCY2C (ENSG00000070019)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2017, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.601
Q58
How many genes does the drug Enalapril target and what are they?
ACE is the only gene target of drug Enalapril.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%enalapril%" OR LOWER(tradeNames_string) LIKE "%e...
[{'UUID': 'DrugGeneTargets_v2_6274', 'drugName': 'Enalapril Maleate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ACE (ENSG00000159640)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1985, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_2276', 'drugName': 'En...
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Genetic Target
Q58.1964
Q58
How many genes does the drug Teduglutide target and what are they?
GLP2R is the only gene target of drug Teduglutide.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%teduglutide%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_1614', 'drugName': 'Teduglutide', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'GLP2R (ENSG00000065325)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2012, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.629
Q58
How many genes does the drug Botulinum Toxin Type A target and what are they?
SNAP25 is the only gene target of drug Botulinum Toxin Type A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%botulinum toxin type a%" OR LOWER(tradeNames_str...
[{'UUID': 'DrugGeneTargets_v2_3257', 'drugName': 'Botulinum Toxin Type A', 'drugMolecularType': 'Unknown', 'newLinkedTargets_string': 'SNAP25 (ENSG00000132639)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_2163', 'drugName': 'Onab...
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Genetic Target
Q58.1170
Q58
How many genes does the drug Chlorpheniramine target and what are they?
HRH1 is the only gene target of drug Chlorpheniramine.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%chlorpheniramine%" OR LOWER(tradeNames_string) L...
[{'UUID': 'DrugGeneTargets_v2_6213', 'drugName': 'Dexchlorpheniramine Maleate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HRH1 (ENSG00000196639)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1981, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_4827', 'dru...
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Genetic Target
Q58.1254
Q58
How many genes does the drug Ebastine target and what are they?
The drug Ebastine is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene HRH1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ebastine%" OR LOWER(tradeNames_string) LIKE "%eb...
[{'UUID': 'DrugGeneTargets_v2_6094', 'drugName': 'Ebastine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HRH1 (ENSG00000196639)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.230
Q58
How many genes does the drug Telotristat target and what are they?
There are 2 gene targets for the drug Telotristat: TPH2 and TPH1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%telotristat%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_3468', 'drugName': 'Telotristat', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'TPH2 (ENSG00000139287), TPH1 (ENSG00000129167)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_1302',...
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Genetic Target
Q58.1180
Q58
How many genes does the drug Spirapril Hydrochloride target and what are they?
ACE is the only gene target of drug Spirapril Hydrochloride.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%spirapril hydrochloride%" OR LOWER(tradeNames_st...
[{'UUID': 'DrugGeneTargets_v2_4466', 'drugName': 'Spirapril Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ACE (ENSG00000159640)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1994, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1332
Q58
How many genes does the drug Lurasidone target and what are they?
There are 2 gene targets for the drug Lurasidone: DRD2 and HTR2A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%lurasidone%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_3925', 'drugName': 'Lurasidone Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'DRD2 (ENSG00000149295), HTR2A (ENSG00000102468)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2010, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGene...
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Genetic Target
Q58.1587
Q58
How many genes does the drug Technetium Succimer target and what are they?
A2M is the only gene target of drug Technetium Succimer.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%technetium succimer%" OR LOWER(tradeNames_string...
[{'UUID': 'DrugGeneTargets_v2_4248', 'drugName': 'Technetium Succimer', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'A2M (ENSG00000175899)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1982, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.69
Q58
How many genes does the drug Gabapentin Enacarbil target and what are they?
There are 26 gene targets for the drug Gabapentin Enacarbil: CACNA1H, CACNA2D1, CACNA1C, CACNA2D3, CACNA1S, CACNA2D2, CACNA1D, CACNA1A, CACNA1B, CACNA1G, CACNA2D4, CACNA1I, CACNA1F, CACNA1E, CACNB4, CACNB2, CACNB1, CACNB3, CACNG7, CACNG5, CACNG2, CACNG4, CACNG8, CACNG3, CACNG6, and CACNG1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%gabapentin enacarbil%" OR LOWER(tradeNames_strin...
[{'UUID': 'DrugGeneTargets_v2_4133', 'drugName': 'Gabapentin Enacarbil', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CACNA1H (ENSG00000196557), CACNA2D1 (ENSG00000153956), CACNA1C (ENSG00000151067), CACNA2D3 (ENSG00000157445), CACNA1S (ENSG00000081248), CACNA2D2 (ENSG00000007402), CACNA1D (ENSG00...
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Genetic Target
Q58.25
Q58
How many genes does the drug Ly-2606368 target and what are they?
The drug Ly-2606368 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene CHEK1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ly-2606368%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2443', 'drugName': 'Ly-2606368', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CHEK1 (ENSG00000149554)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.147
Q58
How many genes does the drug Fedratinib Hydrochloride target and what are they?
There are 2 gene targets for the drug Fedratinib Hydrochloride: JAK2 and FLT3.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%fedratinib hydrochloride%" OR LOWER(tradeNames_s...
[{'UUID': 'DrugGeneTargets_v2_4654', 'drugName': 'Fedratinib Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'JAK2 (ENSG00000096968), FLT3 (ENSG00000122025)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2019, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneT...
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Genetic Target
Q58.542
Q58
How many genes does the drug Warfarin target and what are they?
VKORC1 is the only gene target of drug Warfarin.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%warfarin%" OR LOWER(tradeNames_string) LIKE "%wa...
[{'UUID': 'DrugGeneTargets_v2_38', 'drugName': 'Warfarin Sodium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'VKORC1 (ENSG00000167397)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1954, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_3808', 'drugName': 'War...
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Genetic Target
Q58.818
Q58
How many genes does the drug Asg-5Me target and what are they?
The drug Asg-5Me is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 16 genes: SLC44A4, TUBB4B, TUBB1, TUBA3C, TUBA4A, TUBB3, TUBA1A, TUBB4A, TUBB8, TUBB, TUBA1B, TUBA1C, TUBA3E, TUBB2A, TUBB2B, and TUBB6.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%asg-5me%" OR LOWER(tradeNames_string) LIKE "%asg...
[{'UUID': 'DrugGeneTargets_v2_405', 'drugName': 'Asg-5Me', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'SLC44A4 (ENSG00000204385), TUBB4B (ENSG00000188229), TUBB1 (ENSG00000101162), TUBA3C (ENSG00000198033), TUBA4A (ENSG00000127824), TUBB3 (ENSG00000258947), TUBA1A (ENSG00000167552), TUBB4A (ENSG0000010...
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Genetic Target
Q58.1120
Q58
How many genes does the drug Pentobarbital Sodium target and what are they?
There are 16 gene targets for the drug Pentobarbital Sodium: GABRA1, GABRB2, GABRG2, GABRB3, GABRA4, GABRG3, GABRQ, GABRA3, GABRP, GABRD, GABRG1, GABRB1, GABRE, GABRA2, GABRA5, and GABRA6.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%pentobarbital sodium%" OR LOWER(tradeNames_strin...
[{'UUID': 'DrugGeneTargets_v2_757', 'drugName': 'Pentobarbital Sodium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089), ...
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Genetic Target
Q58.88
Q58
How many genes does the drug Interferon Alfa-2A target and what are they?
There are 2 gene targets for the drug Interferon Alfa-2A: IFNAR1 and IFNAR2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%interferon alfa-2a%" OR LOWER(tradeNames_string)...
[{'UUID': 'DrugGeneTargets_v2_4676', 'drugName': 'Interferon Alfa-2A', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'IFNAR1 (ENSG00000142166), IFNAR2 (ENSG00000159110)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1986, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2...
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Genetic Target
Q58.1183
Q58
How many genes does the drug Secobarbital target and what are they?
There are 16 gene targets for the drug Secobarbital: GABRA1, GABRB2, GABRG2, GABRB3, GABRA4, GABRG3, GABRQ, GABRA3, GABRP, GABRD, GABRG1, GABRB1, GABRE, GABRA2, GABRA5, and GABRA6.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%secobarbital%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_5547', 'drugName': 'Secobarbital', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089), GABRA3 ...
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Q58.1333
Q58
How many genes does the drug Modimelanotide target and what are they?
The drug Modimelanotide is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 2 genes: MC3R and MC1R.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%modimelanotide%" OR LOWER(tradeNames_string) LIK...
[{'UUID': 'DrugGeneTargets_v2_2087', 'drugName': 'Modimelanotide', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'MC3R (ENSG00000124089), MC1R (ENSG00000258839)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}, {'UUID': 'DrugGeneTargets_v2_2088', 'd...
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Q58.1806
Q58
How many genes does the drug X-82 target and what are they?
The drug X-82 is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 5 genes: FLT1, FLT4, KDR, PDGFRB, and PDGFRA.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%x-82%" OR LOWER(tradeNames_string) LIKE "%x-82%"...
[{'UUID': 'DrugGeneTargets_v2_5333', 'drugName': 'X-82', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'FLT1 (ENSG00000102755), FLT4 (ENSG00000037280), KDR (ENSG00000128052), PDGFRB (ENSG00000113721), PDGFRA (ENSG00000134853)', 'numberLinkedTargets': 5, 'yearOfFirstApproval': 0, 'maxClinicalTrialPha...
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Q58.1819
Q58
How many genes does the drug Pexidartinib Hydrochloride target and what are they?
There are 3 gene targets for the drug Pexidartinib Hydrochloride: KIT, FLT3, and CSF1R.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%pexidartinib hydrochloride%" OR LOWER(tradeNames...
[{'UUID': 'DrugGeneTargets_v2_4377', 'drugName': 'Pexidartinib Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'KIT (ENSG00000157404), FLT3 (ENSG00000122025), CSF1R (ENSG00000182578)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 2019, 'maxClinicalTrialPhase': 4, 'drugIsApproved': ...
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Genetic Target
Q58.1374
Q58
How many genes does the drug Tivozanib Hydrochloride target and what are they?
There are 5 gene targets for the drug Tivozanib Hydrochloride: FLT1, FLT4, KDR, KIT, and PDGFRB.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tivozanib hydrochloride%" OR LOWER(tradeNames_st...
[{'UUID': 'DrugGeneTargets_v2_2104', 'drugName': 'Tivozanib Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'FLT1 (ENSG00000102755), FLT4 (ENSG00000037280), KDR (ENSG00000128052), KIT (ENSG00000157404), PDGFRB (ENSG00000113721)', 'numberLinkedTargets': 5, 'yearOfFirstApproval': 2021, '...
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Genetic Target
Q58.1144
Q58
How many genes does the drug Prazepam target and what are they?
There are 16 gene targets for the drug Prazepam: GABRA1, GABRB2, GABRG2, GABRB3, GABRA4, GABRG3, GABRQ, GABRA3, GABRP, GABRD, GABRG1, GABRB1, GABRE, GABRA2, GABRA5, and GABRA6.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%prazepam%" OR LOWER(tradeNames_string) LIKE "%pr...
[{'UUID': 'DrugGeneTargets_v2_4830', 'drugName': 'Prazepam', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089), GABRA3 (ENS...
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Genetic Target
Q58.367
Q58
How many genes does the drug Nimacimab target and what are they?
The drug Nimacimab is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene CNR1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%nimacimab%" OR LOWER(tradeNames_string) LIKE "%n...
[{'UUID': 'DrugGeneTargets_v2_895', 'drugName': 'Nimacimab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'CNR1 (ENSG00000118432)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1790
Q58
How many genes does the drug Dopamine target and what are they?
ADRB1 is the only gene target of drug Dopamine.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%dopamine%" OR LOWER(tradeNames_string) LIKE "%do...
[{'UUID': 'DrugGeneTargets_v2_3237', 'drugName': 'Dopamine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRB1 (ENSG00000043591)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_4778', 'drugName': 'Dopamine Hyd...
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Genetic Target
Q58.1208
Q58
How many genes does the drug Diethylpropion Hydrochloride target and what are they?
There are 2 gene targets for the drug Diethylpropion Hydrochloride: SLC6A2 and SLC6A3.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%diethylpropion hydrochloride%" OR LOWER(tradeNam...
[{'UUID': 'DrugGeneTargets_v2_2343', 'drugName': 'Diethylpropion Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SLC6A2 (ENSG00000103546), SLC6A3 (ENSG00000142319)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1959, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'D...
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Genetic Target
Q58.1035
Q58
How many genes does the drug Triamterene target and what are they?
There are 3 gene targets for the drug Triamterene: SCNN1A, SCNN1B, and SCNN1G.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%triamterene%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_4230', 'drugName': 'Triamterene', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SCNN1A (ENSG00000111319), SCNN1B (ENSG00000168447), SCNN1G (ENSG00000166828)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 1964, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1039
Q58
How many genes does the drug Cinaciguat target and what are they?
The drug Cinaciguat is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 4 genes: GUCY1B1, GUCY1B2, GUCY1A2, and GUCY1A1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%cinaciguat%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_6276', 'drugName': 'Cinaciguat', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GUCY1B1 (ENSG00000061918), GUCY1B2 (ENSG00000123201), GUCY1A2 (ENSG00000152402), GUCY1A1 (ENSG00000164116)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, '...
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Q58.1761
Q58
How many genes does the drug Dinoprost Tromethamine target and what are they?
PTGFR is the only gene target of drug Dinoprost Tromethamine.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%dinoprost tromethamine%" OR LOWER(tradeNames_str...
[{'UUID': 'DrugGeneTargets_v2_3570', 'drugName': 'Dinoprost Tromethamine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PTGFR (ENSG00000122420)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1982, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.1357
Q58
How many genes does the drug Morphine Sulfate target and what are they?
OPRM1 is the only gene target of drug Morphine Sulfate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%morphine sulfate%" OR LOWER(tradeNames_string) L...
[{'UUID': 'DrugGeneTargets_v2_3650', 'drugName': 'Morphine Sulfate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'OPRM1 (ENSG00000112038)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1984, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.1875
Q58
How many genes does the drug Mometasone Furoate target and what are they?
NR3C1 is the only gene target of drug Mometasone Furoate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%mometasone furoate%" OR LOWER(tradeNames_string)...
[{'UUID': 'DrugGeneTargets_v2_2490', 'drugName': 'Mometasone Furoate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'NR3C1 (ENSG00000113580)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1987, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.672
Q58
How many genes does the drug Tosedostat target and what are they?
The drug Tosedostat is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 19 genes: ANPEP, NPEPPS, RNPEP, METAP1, LNPEP, DNPEP, ENPEP, XPNPEP1, LAP3, METAP2, XPNPEP2, ERAP2, ERAP1, LVRN, AOPEP, METAP1D, NPEPL1, RNPEPL1, and XPNPEP3.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tosedostat%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_582', 'drugName': 'Tosedostat', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ANPEP (ENSG00000166825), NPEPPS (ENSG00000141279), RNPEP (ENSG00000176393), METAP1 (ENSG00000164024), LNPEP (ENSG00000113441), DNPEP (ENSG00000123992), ENPEP (ENSG00000138792), XPNPEP1 (ENSG0...
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