Datasets:

uuid
stringlengths
4
8
template_uuid
stringclasses
40 values
question
stringlengths
13
193
answer
stringlengths
29
2.2k
benchmark_query
stringlengths
133
622
execution_results
stringlengths
2
1.14M
query_type
stringclasses
2 values
sql_category
stringclasses
26 values
bio_category
stringclasses
14 values
Q1.834
Q1
Is LTB4R2 a druggable gene?
There are currently no approved drugs targeting LTB4R2, but there are 2 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%LTB4R2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1192', 'drugName': 'Nomacopan', 'drugIsApproved': False, 'newLinkedTargets_string': 'LTB4R2 (ENSG00000213906), LTB4R (ENSG00000213903), C5 (ENSG00000106804)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_1191', 'drugName': 'Nomacopan', 'drugIsApproved': False, 'newLinkedTarget...
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Approval Status, Genetic Target
Q1.1260
Q1
Is RPL37 a druggable gene?
There is 1 drug, Ataluren, that targets RPL37, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%RPL37 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'drugIsApproved': True, 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG...
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Approval Status, Genetic Target
Q1.1519
Q1
Is UGCG a druggable gene?
There are currently 3 approved drugs which target UGCG, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%UGCG %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4249', 'drugName': 'Eliglustat', 'drugIsApproved': True, 'newLinkedTargets_string': 'UGCG (ENSG00000148154)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5675', 'drugName': 'Miglustat', 'drugIsApproved': True, 'newLinkedTargets_string': 'UGCG (ENSG00000148154)', 'maxClinicalT...
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Approval Status, Genetic Target
Q1.716
Q1
Is ITGA2B a druggable gene?
There are currently 4 approved drugs which target ITGA2B, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%ITGA2B %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2661', 'drugName': 'Abciximab', 'drugIsApproved': True, 'newLinkedTargets_string': 'ITGB3 (ENSG00000259207), ITGA2B (ENSG00000005961), ITGAV (ENSG00000138448)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1804', 'drugName': 'Eptifibatide', 'drugIsApproved': True, 'newLinkedTa...
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Approval Status, Genetic Target
Q1.181
Q1
Is CASP6 a druggable gene?
There are currently no approved drugs targeting CASP6, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CASP6 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_45', 'drugName': 'Emricasan', 'drugIsApproved': False, 'newLinkedTargets_string': 'CASP4 (ENSG00000196954), CASP9 (ENSG00000132906), CASP3 (ENSG00000164305), CASP5 (ENSG00000137757), CASP6 (ENSG00000138794), CASP7 (ENSG00000165806), CASP8 (ENSG00000064012), CASP1 (ENSG00000137752), CASP2 (...
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Approval Status, Genetic Target
Q1.422
Q1
Is EPOR a druggable gene?
There are currently 8 approved drugs which target EPOR, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%EPOR %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4490', 'drugName': 'Darbepoetin Alfa', 'drugIsApproved': True, 'newLinkedTargets_string': 'EPOR (ENSG00000187266)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2704', 'drugName': 'Epoetin Delta', 'drugIsApproved': True, 'newLinkedTargets_string': 'EPOR (ENSG00000187266)', 'ma...
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Approval Status, Genetic Target
Q1.1278
Q1
Is RPS14 a druggable gene?
There is 1 drug, Ataluren, that targets RPS14, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%RPS14 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'drugIsApproved': True, 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG...
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Approval Status, Genetic Target
Q1.441
Q1
Is F3 a druggable gene?
There is 1 drug, Tisotumab Vedotin, that targets F3, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%F3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4157', 'drugName': 'Tisotumab Vedotin', 'drugIsApproved': True, 'newLinkedTargets_string': 'F3 (ENSG00000117525), TUBB4B (ENSG00000188229), TUBB1 (ENSG00000101162), TUBA3C (ENSG00000198033), TUBA4A (ENSG00000127824), TUBB3 (ENSG00000258947), TUBA1A (ENSG00000167552), TUBB4A (ENSG0000010483...
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Approval Status, Genetic Target
Q1.593
Q1
Is HLA-DRB3 a druggable gene?
There are currently no approved drugs targeting HLA-DRB3, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%HLA-DRB3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_363', 'drugName': 'Apolizumab', 'drugIsApproved': False, 'newLinkedTargets_string': 'HLA-DRB3 (ENSG00000231679), HLA-DRB5 (ENSG00000198502), HLA-DRB1 (ENSG00000196126), HLA-DRB4 (ENSG00000231021)', 'maxClinicalTrialPhase': 2}]
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Approval Status, Genetic Target
Q1.843
Q1
Is MAGEA3 a druggable gene?
There are currently no approved drugs targeting MAGEA3, but there are 2 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%MAGEA3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4022', 'drugName': 'Astuprotimut-R', 'drugIsApproved': False, 'newLinkedTargets_string': 'MAGEA3 (ENSG00000221867)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_4575', 'drugName': 'Biropepimut-S', 'drugIsApproved': False, 'newLinkedTargets_string': 'MAGEA3 (ENSG00000221867)',...
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Approval Status, Genetic Target
Q1.365
Q1
Is DLL4 a druggable gene?
There are currently no approved drugs targeting DLL4, but there are 2 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%DLL4 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3542', 'drugName': 'Demcizumab', 'drugIsApproved': False, 'newLinkedTargets_string': 'DLL4 (ENSG00000128917)', 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_5324', 'drugName': 'Enoticumab', 'drugIsApproved': False, 'newLinkedTargets_string': 'DLL4 (ENSG00000128917)', 'maxClinic...
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Approval Status, Genetic Target
Q1.1206
Q1
Is PTPRC a druggable gene?
There are currently no approved drugs targeting PTPRC, but there are 2 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%PTPRC %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2505', 'drugName': 'Bc8 131I', 'drugIsApproved': False, 'newLinkedTargets_string': 'PTPRC (ENSG00000081237)', 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_1374', 'drugName': 'Ahn-12', 'drugIsApproved': False, 'newLinkedTargets_string': 'PTPRC (ENSG00000081237)', 'maxClinicalTr...
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Approval Status, Genetic Target
Q1.1228
Q1
Is RPE65 a druggable gene?
There are currently no approved drugs targeting RPE65, but there are 3 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%RPE65 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3372', 'drugName': 'Emixustat', 'drugIsApproved': False, 'newLinkedTargets_string': 'RPE65 (ENSG00000116745)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_1065', 'drugName': 'Voretigene Neparvovec', 'drugIsApproved': False, 'newLinkedTargets_string': 'RPE65 (ENSG00000116745)'...
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Approval Status, Genetic Target
Q1.348
Q1
Is CYP3A4 a druggable gene?
There are currently 2 approved drugs which target CYP3A4, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CYP3A4 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2752', 'drugName': 'Ritonavir', 'drugIsApproved': True, 'newLinkedTargets_string': 'CYP3A4 (ENSG00000160868), CYP3A5 (ENSG00000106258), CYP3A43 (ENSG00000021461), CYP3A7 (ENSG00000160870)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2751', 'drugName': 'Ritonavir', 'drugIsApp...
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Approval Status, Genetic Target
Q1.473
Q1
Is FLT3 a druggable gene?
There are currently 13 approved drugs which target FLT3, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%FLT3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3450', 'drugName': 'Sunitinib', 'drugIsApproved': True, 'newLinkedTargets_string': 'RET (ENSG00000165731), FLT1 (ENSG00000102755), FLT4 (ENSG00000037280), KDR (ENSG00000128052), CSF1R (ENSG00000182578), FLT3 (ENSG00000122025), KIT (ENSG00000157404), PDGFRB (ENSG00000113721), PDGFRA (ENSG00...
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Approval Status, Genetic Target
Q1.535
Q1
Is GPR119 a druggable gene?
There are currently no approved drugs targeting GPR119, but there are 2 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%GPR119 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4851', 'drugName': 'Mbx-2982', 'drugIsApproved': False, 'newLinkedTargets_string': 'GPR119 (ENSG00000147262)', 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_5541', 'drugName': 'Gsk-1292263', 'drugIsApproved': False, 'newLinkedTargets_string': 'GPR119 (ENSG00000147262)', 'maxCli...
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Approval Status, Genetic Target
Q1.812
Q1
Is LAMC2 a druggable gene?
There is 1 drug, Ocriplasmin, that targets LAMC2, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%LAMC2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5818', 'drugName': 'Ocriplasmin', 'drugIsApproved': True, 'newLinkedTargets_string': 'FN1 (ENSG00000115414), COL1A2 (ENSG00000164692), COL1A1 (ENSG00000108821), COL2A1 (ENSG00000139219), COL3A1 (ENSG00000168542), COL4A1 (ENSG00000187498), COL5A1 (ENSG00000130635), COL6A1 (ENSG00000142156),...
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Approval Status, Genetic Target
Q1.1325
Q1
Is S1PR1 a druggable gene?
There are currently 8 approved drugs which target S1PR1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%S1PR1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4765', 'drugName': 'Fingolimod Hydrochloride', 'drugIsApproved': True, 'newLinkedTargets_string': 'S1PR5 (ENSG00000180739), S1PR2 (ENSG00000267534), S1PR4 (ENSG00000125910), S1PR3 (ENSG00000213694), S1PR1 (ENSG00000170989)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1976', ...
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Approval Status, Genetic Target
Q1.609
Q1
Is HSP90AA1 a druggable gene?
There are currently no approved drugs targeting HSP90AA1, but there are 10 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%HSP90AA1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1279', 'drugName': 'Retaspimycin Hydrochloride', 'drugIsApproved': False, 'newLinkedTargets_string': 'HSP90AA1 (ENSG00000080824), HSP90AB1 (ENSG00000096384)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_2657', 'drugName': 'Tanespimycin', 'drugIsApproved': False, 'newLinkedTar...
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Approval Status, Genetic Target
Q1.588
Q1
Is HDAC7 a druggable gene?
There are currently 4 approved drugs which target HDAC7, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%HDAC7 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4906', 'drugName': 'Panobinostat', 'drugIsApproved': True, 'newLinkedTargets_string': 'HDAC1 (ENSG00000116478), HDAC3 (ENSG00000171720), HDAC6 (ENSG00000094631), HDAC2 (ENSG00000196591), HDAC5 (ENSG00000108840), HDAC7 (ENSG00000061273), HDAC8 (ENSG00000147099), HDAC11 (ENSG00000163517), HD...
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Approval Status, Genetic Target
Q1.653
Q1
Is IFNAR1 a druggable gene?
There are currently 11 approved drugs which target IFNAR1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%IFNAR1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4596', 'drugName': 'Interferon Alfa-2B', 'drugIsApproved': True, 'newLinkedTargets_string': 'IFNAR1 (ENSG00000142166), IFNAR2 (ENSG00000159110)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2953', 'drugName': 'Peginterferon Alfa-2B', 'drugIsApproved': True, 'newLinkedTargets_...
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Approval Status, Genetic Target
Q1.245
Q1
Is CDK5 a druggable gene?
There are currently no approved drugs targeting CDK5, but there are 7 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CDK5 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_48', 'drugName': 'Dinaciclib', 'drugIsApproved': False, 'newLinkedTargets_string': 'CDK5 (ENSG00000164885), CDK1 (ENSG00000170312), CDK9 (ENSG00000136807), CDK2 (ENSG00000123374)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_46', 'drugName': 'Dinaciclib', 'drugIsApproved': Fa...
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Approval Status, Genetic Target
Q1.831
Q1
Is LTA4H a druggable gene?
There are currently no approved drugs targeting LTA4H, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%LTA4H %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5456', 'drugName': 'Acebilustat', 'drugIsApproved': False, 'newLinkedTargets_string': 'LTA4H (ENSG00000111144)', 'maxClinicalTrialPhase': 2}]
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Approval Status, Genetic Target
Q1.557
Q1
Is GRM4 a druggable gene?
There are currently no approved drugs targeting GRM4, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%GRM4 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3750', 'drugName': 'Foliglurax', 'drugIsApproved': False, 'newLinkedTargets_string': 'GRM4 (ENSG00000124493)', 'maxClinicalTrialPhase': 2}]
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Approval Status, Genetic Target
Q1.953
Q1
Is NDUFAF4 a druggable gene?
There are currently 2 approved drugs which target NDUFAF4, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%NDUFAF4 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'drugIsApproved': True, 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (EN...
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Approval Status, Genetic Target
Q1.919
Q1
Is MUC1 a druggable gene?
There are currently no approved drugs targeting MUC1, but there are 14 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%MUC1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1399', 'drugName': 'Pemtumomab', 'drugIsApproved': False, 'newLinkedTargets_string': 'MUC1 (ENSG00000185499)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_1059', 'drugName': 'Tecemotide', 'drugIsApproved': False, 'newLinkedTargets_string': 'MUC1 (ENSG00000185499)', 'maxClinic...
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Approval Status, Genetic Target
Q1.440
Q1
Is F2RL3 a druggable gene?
There are currently no approved drugs targeting F2RL3, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%F2RL3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1642', 'drugName': 'Bms-986141', 'drugIsApproved': False, 'newLinkedTargets_string': 'F2RL3 (ENSG00000127533)', 'maxClinicalTrialPhase': 2}]
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Approval Status, Genetic Target
Q1.1456
Q1
Is TNFSF13B a druggable gene?
There is 1 drug, Belimumab, that targets TNFSF13B, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%TNFSF13B %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6001', 'drugName': 'Belimumab', 'drugIsApproved': True, 'newLinkedTargets_string': 'TNFSF13B (ENSG00000102524)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_550', 'drugName': 'Blisibimod', 'drugIsApproved': False, 'newLinkedTargets_string': 'TNFSF13B (ENSG00000102524)', 'maxC...
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Approval Status, Genetic Target
Q1.1382
Q1
Is SMN2 a druggable gene?
There are currently 4 approved drugs which target SMN2, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%SMN2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6328', 'drugName': 'Nusinersen Sodium', 'drugIsApproved': True, 'newLinkedTargets_string': 'SMN2 (ENSG00000205571)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2674', 'drugName': 'Nusinersen', 'drugIsApproved': True, 'newLinkedTargets_string': 'SMN2 (ENSG00000205571)', 'maxC...
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Approval Status, Genetic Target
Q1.310
Q1
Is COMT a druggable gene?
There are currently 3 approved drugs which target COMT, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%COMT %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4197', 'drugName': 'Tolcapone', 'drugIsApproved': True, 'newLinkedTargets_string': 'COMT (ENSG00000093010)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2548', 'drugName': 'Opicapone', 'drugIsApproved': True, 'newLinkedTargets_string': 'COMT (ENSG00000093010)', 'maxClinicalTr...
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Approval Status, Genetic Target
Q1.432
Q1
Is ESRRG a druggable gene?
There are currently no approved drugs targeting ESRRG, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%ESRRG %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5111', 'drugName': 'Afimoxifene', 'drugIsApproved': False, 'newLinkedTargets_string': 'ESRRG (ENSG00000196482), ESR2 (ENSG00000140009), ESR1 (ENSG00000091831)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_5112', 'drugName': 'Afimoxifene', 'drugIsApproved': False, 'newLinkedTa...
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Approval Status, Genetic Target
Q1.910
Q1
Is MT-ND3 a druggable gene?
There are currently 2 approved drugs which target MT-ND3, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%MT-ND3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'drugIsApproved': True, 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (EN...
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Approval Status, Genetic Target
Q1.400
Q1
Is EML4 a druggable gene?
There are currently 5 approved drugs which target EML4, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%EML4 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2435', 'drugName': 'Ceritinib', 'drugIsApproved': True, 'newLinkedTargets_string': 'ALK (ENSG00000171094), EML4 (ENSG00000143924), NPM1 (ENSG00000181163)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4672', 'drugName': 'Alectinib', 'drugIsApproved': True, 'newLinkedTargets_st...
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Approval Status, Genetic Target
Q1.425
Q1
Is ERBB2 a druggable gene?
There are currently 14 approved drugs which target ERBB2, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%ERBB2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5756', 'drugName': 'Trastuzumab Emtansine', 'drugIsApproved': True, 'newLinkedTargets_string': 'ERBB2 (ENSG00000141736), TUBB4B (ENSG00000188229), TUBB1 (ENSG00000101162), TUBA3C (ENSG00000198033), TUBA4A (ENSG00000127824), TUBB3 (ENSG00000258947), TUBA1A (ENSG00000167552), TUBB4A (ENSG000...
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Approval Status, Genetic Target
Q1.372
Q1
Is DPYD a druggable gene?
There are currently no approved drugs targeting DPYD, but there are 2 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%DPYD %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4866', 'drugName': 'Gimeracil', 'drugIsApproved': False, 'newLinkedTargets_string': 'DPYD (ENSG00000188641)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_1418', 'drugName': 'Eniluracil', 'drugIsApproved': False, 'newLinkedTargets_string': 'DPYD (ENSG00000188641)', 'maxClinica...
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Approval Status, Genetic Target
Q1.55
Q1
Is ALDH5A1 a druggable gene?
There are currently 3 approved drugs which target ALDH5A1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%ALDH5A1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6237', 'drugName': 'Valproic Acid', 'drugIsApproved': True, 'newLinkedTargets_string': 'ALDH5A1 (ENSG00000112294)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5683', 'drugName': 'Divalproex Sodium', 'drugIsApproved': True, 'newLinkedTargets_string': 'ALDH5A1 (ENSG00000112294...
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Approval Status, Genetic Target
Q1.696
Q1
Is IL31RA a druggable gene?
There are currently no approved drugs targeting IL31RA, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%IL31RA %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_830', 'drugName': 'Nemolizumab', 'drugIsApproved': False, 'newLinkedTargets_string': 'IL31RA (ENSG00000164509)', 'maxClinicalTrialPhase': 3}]
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Approval Status, Genetic Target
Q1.589
Q1
Is HDAC8 a druggable gene?
There are currently 4 approved drugs which target HDAC8, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%HDAC8 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6063', 'drugName': 'Romidepsin', 'drugIsApproved': True, 'newLinkedTargets_string': 'HDAC1 (ENSG00000116478), HDAC3 (ENSG00000171720), HDAC6 (ENSG00000094631), HDAC2 (ENSG00000196591), HDAC5 (ENSG00000108840), HDAC7 (ENSG00000061273), HDAC8 (ENSG00000147099), HDAC11 (ENSG00000163517), HDAC...
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Approval Status, Genetic Target
Q1.314
Q1
Is CR1 a druggable gene?
There are currently no approved drugs targeting CR1, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CR1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_542', 'drugName': 'Fosaprepitant', 'drugIsApproved': True, 'newLinkedTargets_string': 'TACR1 (ENSG00000115353)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1941', 'drugName': 'Fosnetupitant', 'drugIsApproved': True, 'newLinkedTargets_string': 'TACR1 (ENSG00000115353)', 'maxC...
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Approval Status, Genetic Target
Q1.979
Q1
Is NFE2L2 a druggable gene?
There are currently no approved drugs targeting NFE2L2, but there are 2 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%NFE2L2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4920', 'drugName': 'Bardoxolone Methyl', 'drugIsApproved': False, 'newLinkedTargets_string': 'NFE2L2 (ENSG00000116044), KEAP1 (ENSG00000079999), PPARG (ENSG00000132170), IKBKB (ENSG00000104365)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_4922', 'drugName': 'Bardoxolone Meth...
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Approval Status, Genetic Target
Q1.968
Q1
Is NDUFS2 a druggable gene?
There are currently 2 approved drugs which target NDUFS2, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%NDUFS2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'drugIsApproved': True, 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (EN...
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Approval Status, Genetic Target
Q1.111
Q1
Is BHMT a druggable gene?
There are currently 2 approved drugs which target BHMT, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%BHMT %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3565', 'drugName': 'Betaine', 'drugIsApproved': True, 'newLinkedTargets_string': 'BHMT (ENSG00000145692), BHMT2 (ENSG00000132840)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1270', 'drugName': 'Betaine Hydrochloride', 'drugIsApproved': True, 'newLinkedTargets_string': 'BHMT...
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Approval Status, Genetic Target
Q1.481
Q1
Is FSHR a druggable gene?
There are currently 4 approved drugs which target FSHR, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%FSHR %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1764', 'drugName': 'Menotropins', 'drugIsApproved': True, 'newLinkedTargets_string': 'LHCGR (ENSG00000138039), FSHR (ENSG00000170820)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2306', 'drugName': 'Corifollitropin Alfa', 'drugIsApproved': True, 'newLinkedTargets_string': 'F...
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Approval Status, Genetic Target
Q1.715
Q1
Is ITGA2 a druggable gene?
There are currently no approved drugs targeting ITGA2, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%ITGA2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4470', 'drugName': 'Vatelizumab', 'drugIsApproved': False, 'newLinkedTargets_string': 'ITGA2 (ENSG00000164171)', 'maxClinicalTrialPhase': 2}]
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Approval Status, Genetic Target
Q1.102
Q1
Is BCL2 a druggable gene?
There is 1 drug, Venetoclax, that targets BCL2, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%BCL2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5609', 'drugName': 'Venetoclax', 'drugIsApproved': True, 'newLinkedTargets_string': 'BCL2 (ENSG00000171791)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2964', 'drugName': 'Obatoclax Mesylate', 'drugIsApproved': False, 'newLinkedTargets_string': 'BCL2 (ENSG00000171791), BCL2...
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Approval Status, Genetic Target
Q1.480
Q1
Is FRK a druggable gene?
There are currently 2 approved drugs which target FRK, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%FRK %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_803', 'drugName': 'Regorafenib', 'drugIsApproved': True, 'newLinkedTargets_string': 'EPHA2 (ENSG00000142627), TEK (ENSG00000120156), MAPK11 (ENSG00000185386), RAF1 (ENSG00000132155), FRK (ENSG00000111816), PDGFRB (ENSG00000113721), PDGFRA (ENSG00000134853), KIT (ENSG00000157404), FGFR1 (EN...
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Approval Status, Genetic Target
Q1.846
Q1
Is MAOB a druggable gene?
There are currently 17 approved drugs which target MAOB, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%MAOB %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1874', 'drugName': 'Safinamide Mesylate', 'drugIsApproved': True, 'newLinkedTargets_string': 'MAOB (ENSG00000069535)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5670', 'drugName': 'Pargyline', 'drugIsApproved': True, 'newLinkedTargets_string': 'MAOA (ENSG00000189221), MAOB ...
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Approval Status, Genetic Target
Q1.1409
Q1
Is SYK a druggable gene?
There are currently 2 approved drugs which target SYK, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%SYK %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4030', 'drugName': 'Fostamatinib Disodium', 'drugIsApproved': True, 'newLinkedTargets_string': 'SYK (ENSG00000165025)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1146', 'drugName': 'Fostamatinib', 'drugIsApproved': True, 'newLinkedTargets_string': 'SYK (ENSG00000165025)', '...
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Approval Status, Genetic Target
Q1.268
Q1
Is CHRNA5 a druggable gene?
There are currently no approved drugs targeting CHRNA5, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CHRNA5 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3835', 'drugName': 'Pozanicline', 'drugIsApproved': False, 'newLinkedTargets_string': 'CHRNB2 (ENSG00000160716), CHRNA6 (ENSG00000147434), CHRNA4 (ENSG00000101204), CHRNA5 (ENSG00000169684)', 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_3836', 'drugName': 'Pozanicline', 'drugI...
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Approval Status, Genetic Target
Q1.1392
Q1
Is SRC a druggable gene?
There are currently 4 approved drugs which target SRC, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%SRC %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3956', 'drugName': 'Bosutinib', 'drugIsApproved': True, 'newLinkedTargets_string': 'ABL1 (ENSG00000097007), BCR (ENSG00000186716), HCK (ENSG00000101336), SRC (ENSG00000197122), LYN (ENSG00000254087)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3958', 'drugName': 'Bosutinib',...
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Approval Status, Genetic Target
Q1.298
Q1
Is COL4A3 a druggable gene?
There are currently 2 approved drugs which target COL4A3, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%COL4A3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5818', 'drugName': 'Ocriplasmin', 'drugIsApproved': True, 'newLinkedTargets_string': 'FN1 (ENSG00000115414), COL1A2 (ENSG00000164692), COL1A1 (ENSG00000108821), COL2A1 (ENSG00000139219), COL3A1 (ENSG00000168542), COL4A1 (ENSG00000187498), COL5A1 (ENSG00000130635), COL6A1 (ENSG00000142156),...
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Approval Status, Genetic Target
Q1.547
Q1
Is GRIK5 a druggable gene?
There is 1 drug, Topiramate, that targets GRIK5, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%GRIK5 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1594', 'drugName': 'Topiramate', 'drugIsApproved': True, 'newLinkedTargets_string': 'GRIK1 (ENSG00000171189), GRIK5 (ENSG00000105737), GRIK4 (ENSG00000149403), GRIK2 (ENSG00000164418), GRIK3 (ENSG00000163873), CA4 (ENSG00000167434), SCN1A (ENSG00000144285), SCN5A (ENSG00000183873), SCN4A (...
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Approval Status, Genetic Target
Q1.974
Q1
Is NDUFS8 a druggable gene?
There are currently 2 approved drugs which target NDUFS8, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%NDUFS8 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'drugIsApproved': True, 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (EN...
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Approval Status, Genetic Target
Q1.1465
Q1
Is TNNT2 a druggable gene?
There are currently no approved drugs targeting TNNT2, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%TNNT2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2198', 'drugName': 'Levosimendan', 'drugIsApproved': False, 'newLinkedTargets_string': 'PDE3A (ENSG00000172572), PDE3B (ENSG00000152270), TNNC1 (ENSG00000114854), TNNI3 (ENSG00000129991), TNNT2 (ENSG00000118194)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_2199', 'drugName':...
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Approval Status, Genetic Target
Q1.980
Q1
Is NFKB1 a druggable gene?
There are currently no approved drugs targeting NFKB1, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%NFKB1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1568', 'drugName': 'Edasalonexent', 'drugIsApproved': False, 'newLinkedTargets_string': 'NFKB2 (ENSG00000077150), NFKB1 (ENSG00000109320), RELA (ENSG00000173039)', 'maxClinicalTrialPhase': 3}]
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Approval Status, Genetic Target
Q1.379
Q1
Is E2F2 a druggable gene?
There are currently no approved drugs targeting E2F2, but there are 2 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%E2F2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4614', 'drugName': 'Edifoligide Sodium', 'drugIsApproved': False, 'newLinkedTargets_string': 'E2F1 (ENSG00000101412), E2F2 (ENSG00000007968), E2F3 (ENSG00000112242), E2F4 (ENSG00000205250), E2F5 (ENSG00000133740), E2F6 (ENSG00000169016), E2F7 (ENSG00000165891), E2F8 (ENSG00000129173)', 'ma...
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Approval Status, Genetic Target
Q1.288
Q1
Is COL18A1 a druggable gene?
There are currently 2 approved drugs which target COL18A1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%COL18A1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5818', 'drugName': 'Ocriplasmin', 'drugIsApproved': True, 'newLinkedTargets_string': 'FN1 (ENSG00000115414), COL1A2 (ENSG00000164692), COL1A1 (ENSG00000108821), COL2A1 (ENSG00000139219), COL3A1 (ENSG00000168542), COL4A1 (ENSG00000187498), COL5A1 (ENSG00000130635), COL6A1 (ENSG00000142156),...
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Approval Status, Genetic Target
Q1.1475
Q1
Is TPO a druggable gene?
There are currently 3 approved drugs which target TPO, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%TPO %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3174', 'drugName': 'Methimazole', 'drugIsApproved': True, 'newLinkedTargets_string': 'TPO (ENSG00000115705)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2546', 'drugName': 'Carbimazole', 'drugIsApproved': True, 'newLinkedTargets_string': 'TPO (ENSG00000115705)', 'maxClinical...
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Approval Status, Genetic Target
Q1.1246
Q1
Is RPL26 a druggable gene?
There is 1 drug, Ataluren, that targets RPL26, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%RPL26 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'drugIsApproved': True, 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG...
general
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Approval Status, Genetic Target
Q1.128
Q1
Is C5 a druggable gene?
There are currently 2 approved drugs which target C5, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%C5 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2422', 'drugName': 'Carfilzomib', 'drugIsApproved': True, 'newLinkedTargets_string': 'PSMD1 (ENSG00000173692), PSMB2 (ENSG00000126067), PSMB1 (ENSG00000008018), PSMB5 (ENSG00000100804), PSMB8 (ENSG00000204264), PSMB9 (ENSG00000240065), PSMB6 (ENSG00000142507), PSMD14 (ENSG00000115233), PSM...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.329
Q1
Is CTLA4 a druggable gene?
There are currently 2 approved drugs which target CTLA4, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CTLA4 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6378', 'drugName': 'Ipilimumab', 'drugIsApproved': True, 'newLinkedTargets_string': 'CTLA4 (ENSG00000163599)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_680', 'drugName': 'Tremelimumab', 'drugIsApproved': True, 'newLinkedTargets_string': 'CTLA4 (ENSG00000163599)', 'maxClini...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.294
Q1
Is COL2A1 a druggable gene?
There are currently 2 approved drugs which target COL2A1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%COL2A1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5818', 'drugName': 'Ocriplasmin', 'drugIsApproved': True, 'newLinkedTargets_string': 'FN1 (ENSG00000115414), COL1A2 (ENSG00000164692), COL1A1 (ENSG00000108821), COL2A1 (ENSG00000139219), COL3A1 (ENSG00000168542), COL4A1 (ENSG00000187498), COL5A1 (ENSG00000130635), COL6A1 (ENSG00000142156),...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.813
Q1
Is LAMC3 a druggable gene?
There is 1 drug, Ocriplasmin, that targets LAMC3, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%LAMC3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5818', 'drugName': 'Ocriplasmin', 'drugIsApproved': True, 'newLinkedTargets_string': 'FN1 (ENSG00000115414), COL1A2 (ENSG00000164692), COL1A1 (ENSG00000108821), COL2A1 (ENSG00000139219), COL3A1 (ENSG00000168542), COL4A1 (ENSG00000187498), COL5A1 (ENSG00000130635), COL6A1 (ENSG00000142156),...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.751
Q1
Is KCNG1 a druggable gene?
There are currently 5 approved drugs which target KCNG1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%KCNG1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5118', 'drugName': 'Guanidine Hydrochloride', 'drugIsApproved': True, 'newLinkedTargets_string': 'KCNQ1 (ENSG00000053918), KCND3 (ENSG00000171385), KCNH2 (ENSG00000055118), KCNA2 (ENSG00000177301), KCNA1 (ENSG00000111262), KCNQ2 (ENSG00000075043), KCNQ3 (ENSG00000184156), KCNA7 (ENSG000001...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.606
Q1
Is HSD11B1 a druggable gene?
There is 1 drug, Carbenoxolone, that targets HSD11B1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%HSD11B1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5312', 'drugName': 'Carbenoxolone', 'drugIsApproved': True, 'newLinkedTargets_string': 'HSD11B2 (ENSG00000176387), HSD11B1 (ENSG00000117594)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5241', 'drugName': 'Bi-187004', 'drugIsApproved': False, 'newLinkedTargets_string': 'HSD1...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.357
Q1
Is DDR2 a druggable gene?
There is 1 drug, Regorafenib, that targets DDR2, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%DDR2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_805', 'drugName': 'Regorafenib', 'drugIsApproved': True, 'newLinkedTargets_string': 'EPHA2 (ENSG00000142627), TEK (ENSG00000120156), MAPK11 (ENSG00000185386), RAF1 (ENSG00000132155), FRK (ENSG00000111816), PDGFRB (ENSG00000113721), PDGFRA (ENSG00000134853), KIT (ENSG00000157404), FGFR1 (EN...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1400
Q1
Is SSTR4 a druggable gene?
There are currently 4 approved drugs which target SSTR4, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%SSTR4 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_693', 'drugName': 'Lutetium Dotatate', 'drugIsApproved': True, 'newLinkedTargets_string': 'SSTR5 (ENSG00000162009), SSTR2 (ENSG00000180616), SSTR4 (ENSG00000132671), SSTR1 (ENSG00000139874), SSTR3 (ENSG00000278195)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_759', 'drugName...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.172
Q1
Is CALM1 a druggable gene?
There are currently 2 approved drugs which target CALM1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CALM1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1971', 'drugName': 'Benziodarone', 'drugIsApproved': True, 'newLinkedTargets_string': 'CALM1 (ENSG00000198668)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5448', 'drugName': 'Prenylamine', 'drugIsApproved': True, 'newLinkedTargets_string': 'SCN5A (ENSG00000183873), CALM1 (E...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.870
Q1
Is MC1R a druggable gene?
There is 1 drug, Afamelanotide, that targets MC1R, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%MC1R %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6266', 'drugName': 'Afamelanotide', 'drugIsApproved': True, 'newLinkedTargets_string': 'MC1R (ENSG00000258839)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_935', 'drugName': 'Dersimelagon', 'drugIsApproved': False, 'newLinkedTargets_string': 'MC1R (ENSG00000258839)', 'maxCli...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.887
Q1
Is MIF a druggable gene?
There are currently no approved drugs targeting MIF, but there are 2 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%MIF %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5945', 'drugName': 'Iguratimod', 'drugIsApproved': False, 'newLinkedTargets_string': 'MIF (ENSG00000240972), TRAF3IP2 (ENSG00000056972), PTGS2 (ENSG00000073756)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_5947', 'drugName': 'Iguratimod', 'drugIsApproved': False, 'newLinkedT...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1301
Q1
Is RPS6 a druggable gene?
There is 1 drug, Ataluren, that targets RPS6, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%RPS6 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'drugIsApproved': True, 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.211
Q1
Is CD3D a druggable gene?
There are currently 4 approved drugs which target CD3D, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CD3D %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3214', 'drugName': 'Muromonab-Cd3', 'drugIsApproved': True, 'newLinkedTargets_string': 'CD3E (ENSG00000198851), CD3G (ENSG00000160654), CD3D (ENSG00000167286)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_6103', 'drugName': 'Teclistamab', 'drugIsApproved': True, 'newLinkedTar...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.622
Q1
Is HTR2C a druggable gene?
There are currently 45 approved drugs which target HTR2C, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%HTR2C %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3865', 'drugName': 'Risperidone', 'drugIsApproved': True, 'newLinkedTargets_string': 'HTR2A (ENSG00000102468), HTR2C (ENSG00000147246), DRD2 (ENSG00000149295)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_348', 'drugName': 'Methixene Hydrochloride', 'drugIsApproved': True, 'n...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.538
Q1
Is GRB2 a druggable gene?
There are currently no approved drugs targeting GRB2, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%GRB2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6066', 'drugName': 'Prexigebersen', 'drugIsApproved': False, 'newLinkedTargets_string': 'GRB2 (ENSG00000177885)', 'maxClinicalTrialPhase': 2}]
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.142
Q1
Is CACNA1A a druggable gene?
There are currently 9 approved drugs which target CACNA1A, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CACNA1A %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1799', 'drugName': 'Suloctidil', 'drugIsApproved': True, 'newLinkedTargets_string': 'CACNA1H (ENSG00000196557), CACNA2D1 (ENSG00000153956), CACNA1C (ENSG00000151067), CACNA2D3 (ENSG00000157445), CACNA1S (ENSG00000081248), CACNA2D2 (ENSG00000007402), CACNA1D (ENSG00000157388), CACNA1A (ENSG...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1106
Q1
Is POLE a druggable gene?
There are currently 5 approved drugs which target POLE, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%POLE %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4', 'drugName': 'Gemcitabine Hydrochloride', 'drugIsApproved': True, 'newLinkedTargets_string': 'POLA1 (ENSG00000101868), POLD4 (ENSG00000175482), POLD3 (ENSG00000077514), POLD1 (ENSG00000062822), POLD2 (ENSG00000106628), POLE (ENSG00000177084), POLA2 (ENSG00000014138), PRIM1 (ENSG00000198...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1286
Q1
Is RPS20 a druggable gene?
There is 1 drug, Ataluren, that targets RPS20, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%RPS20 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'drugIsApproved': True, 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.673
Q1
Is IL13RA2 a druggable gene?
There are currently no approved drugs targeting IL13RA2, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%IL13RA2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2466', 'drugName': 'Cintredekin Besudotox', 'drugIsApproved': False, 'newLinkedTargets_string': 'IL4R (ENSG00000077238), IL13RA1 (ENSG00000131724), IL13RA2 (ENSG00000123496)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_2467', 'drugName': 'Cintredekin Besudotox', 'drugIsAppro...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1218
Q1
Is RGMA a druggable gene?
There are currently no approved drugs targeting RGMA, but there are 2 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%RGMA %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4257', 'drugName': 'Elezanumab', 'drugIsApproved': False, 'newLinkedTargets_string': 'RGMA (ENSG00000182175)', 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_4076', 'drugName': 'Unasnemab', 'drugIsApproved': False, 'newLinkedTargets_string': 'RGMA (ENSG00000182175)', 'maxClinica...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.710
Q1
Is INHBA a druggable gene?
There are currently no approved drugs targeting INHBA, but there are 2 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%INHBA %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1648', 'drugName': 'Garetosmab', 'drugIsApproved': False, 'newLinkedTargets_string': 'INHBA (ENSG00000122641)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_1051', 'drugName': 'Sotatercept', 'drugIsApproved': False, 'newLinkedTargets_string': 'INHBA (ENSG00000122641)', 'maxCli...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1488
Q1
Is TSG101 a druggable gene?
There are currently no approved drugs targeting TSG101, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%TSG101 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1451', 'drugName': 'Fgi-101-1A6', 'drugIsApproved': False, 'newLinkedTargets_string': 'TSG101 (ENSG00000074319)', 'maxClinicalTrialPhase': 1}]
general
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Approval Status, Genetic Target
Q1.1380
Q1
Is SMAD7 a druggable gene?
There are currently no approved drugs targeting SMAD7, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%SMAD7 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2010', 'drugName': 'Mongersen Sodium', 'drugIsApproved': False, 'newLinkedTargets_string': 'SMAD7 (ENSG00000101665)', 'maxClinicalTrialPhase': 3}]
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.201
Q1
Is CD200 a druggable gene?
There are currently no approved drugs targeting CD200, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CD200 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_546', 'drugName': 'Samalizumab', 'drugIsApproved': False, 'newLinkedTargets_string': 'CD200 (ENSG00000091972)', 'maxClinicalTrialPhase': 2}]
general
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Approval Status, Genetic Target
Q1.1354
Q1
Is SIGLEC10 a druggable gene?
There are currently no approved drugs targeting SIGLEC10, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%SIGLEC10 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5250', 'drugName': 'Cd24Fc', 'drugIsApproved': False, 'newLinkedTargets_string': 'HSP90AA1 (ENSG00000080824), HSP90AB1 (ENSG00000096384), SIGLEC10 (ENSG00000142512), HMGB1 (ENSG00000189403), HSPA1A (ENSG00000204389), HSPA1B (ENSG00000204388)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGen...
general
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Approval Status, Genetic Target
Q1.1245
Q1
Is RPL24 a druggable gene?
There is 1 drug, Ataluren, that targets RPL24, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%RPL24 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'drugIsApproved': True, 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.732
Q1
Is JAK3 a druggable gene?
There are currently 3 approved drugs which target JAK3, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%JAK3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3515', 'drugName': 'Tofacitinib Citrate', 'drugIsApproved': True, 'newLinkedTargets_string': 'JAK3 (ENSG00000105639), JAK1 (ENSG00000162434), JAK2 (ENSG00000096968), TYK2 (ENSG00000105397)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4653', 'drugName': 'Upadacitinib', 'drugI...
general
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Approval Status, Genetic Target
Q1.1389
Q1
Is SOST a druggable gene?
There is 1 drug, Romosozumab, that targets SOST, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%SOST %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6190', 'drugName': 'Romosozumab', 'drugIsApproved': True, 'newLinkedTargets_string': 'SOST (ENSG00000167941)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3825', 'drugName': 'Setrusumab', 'drugIsApproved': False, 'newLinkedTargets_string': 'SOST (ENSG00000167941)', 'maxClinic...
general
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Approval Status, Genetic Target
Q1.985
Q1
Is NOD2 a druggable gene?
There is 1 drug, Mifamurtide, that targets NOD2, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%NOD2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1449', 'drugName': 'Mifamurtide', 'drugIsApproved': True, 'newLinkedTargets_string': 'NOD2 (ENSG00000167207)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4474', 'drugName': 'Mifamurtide', 'drugIsApproved': True, 'newLinkedTargets_string': 'NOD2 (ENSG00000167207)', 'maxClinic...
general
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Approval Status, Genetic Target
Q1.11
Q1
Is ACE a druggable gene?
There are currently 22 approved drugs which target ACE, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%ACE %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2110', 'drugName': 'Fosinopril', 'drugIsApproved': True, 'newLinkedTargets_string': 'ACE (ENSG00000159640)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1101', 'drugName': 'Enalaprilat', 'drugIsApproved': True, 'newLinkedTargets_string': 'ACE (ENSG00000159640)', 'maxClinicalT...
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Approval Status, Genetic Target
Q1.149
Q1
Is CACNA1H a druggable gene?
There are currently 16 approved drugs which target CACNA1H, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CACNA1H %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6292', 'drugName': 'Terodiline', 'drugIsApproved': True, 'newLinkedTargets_string': 'CHRM3 (ENSG00000133019), CHRM4 (ENSG00000180720), CHRM1 (ENSG00000168539), CHRM2 (ENSG00000181072), CHRM5 (ENSG00000184984), CACNA1H (ENSG00000196557), CACNA2D1 (ENSG00000153956), CACNA1C (ENSG00000151067)...
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Approval Status, Genetic Target
Q1.1152
Q1
Is PSMA2 a druggable gene?
There are currently 4 approved drugs which target PSMA2, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%PSMA2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3334', 'drugName': 'Ixazomib', 'drugIsApproved': True, 'newLinkedTargets_string': 'PSMD1 (ENSG00000173692), PSMB2 (ENSG00000126067), PSMB1 (ENSG00000008018), PSMB5 (ENSG00000100804), PSMB8 (ENSG00000204264), PSMB9 (ENSG00000240065), PSMB6 (ENSG00000142507), PSMD14 (ENSG00000115233), PSMA1 ...
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Approval Status, Genetic Target
Q1.284
Q1
Is CNR2 a druggable gene?
There are currently no approved drugs targeting CNR2, but there are 8 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CNR2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2533', 'drugName': 'Nonabine', 'drugIsApproved': False, 'newLinkedTargets_string': 'CNR2 (ENSG00000188822), CNR1 (ENSG00000118432)', 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_2534', 'drugName': 'Nonabine', 'drugIsApproved': False, 'newLinkedTargets_string': 'CNR2 (ENSG00000...
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Approval Status, Genetic Target
Q1.300
Q1
Is COL4A5 a druggable gene?
There are currently 2 approved drugs which target COL4A5, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%COL4A5 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5818', 'drugName': 'Ocriplasmin', 'drugIsApproved': True, 'newLinkedTargets_string': 'FN1 (ENSG00000115414), COL1A2 (ENSG00000164692), COL1A1 (ENSG00000108821), COL2A1 (ENSG00000139219), COL3A1 (ENSG00000168542), COL4A1 (ENSG00000187498), COL5A1 (ENSG00000130635), COL6A1 (ENSG00000142156),...
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Approval Status, Genetic Target
Q1.1157
Q1
Is PSMA7 a druggable gene?
There are currently 4 approved drugs which target PSMA7, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%PSMA7 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3334', 'drugName': 'Ixazomib', 'drugIsApproved': True, 'newLinkedTargets_string': 'PSMD1 (ENSG00000173692), PSMB2 (ENSG00000126067), PSMB1 (ENSG00000008018), PSMB5 (ENSG00000100804), PSMB8 (ENSG00000204264), PSMB9 (ENSG00000240065), PSMB6 (ENSG00000142507), PSMD14 (ENSG00000115233), PSMA1 ...
general
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Approval Status, Genetic Target
Q1.293
Q1
Is COL28A1 a druggable gene?
There are currently 2 approved drugs which target COL28A1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%COL28A1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5818', 'drugName': 'Ocriplasmin', 'drugIsApproved': True, 'newLinkedTargets_string': 'FN1 (ENSG00000115414), COL1A2 (ENSG00000164692), COL1A1 (ENSG00000108821), COL2A1 (ENSG00000139219), COL3A1 (ENSG00000168542), COL4A1 (ENSG00000187498), COL5A1 (ENSG00000130635), COL6A1 (ENSG00000142156),...
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Approval Status, Genetic Target
Q1.655
Q1
Is IFNB1 a druggable gene?
There are currently no approved drugs targeting IFNB1, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%IFNB1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4033', 'drugName': 'Pf-06823859', 'drugIsApproved': False, 'newLinkedTargets_string': 'IFNB1 (ENSG00000171855)', 'maxClinicalTrialPhase': 2}]
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Approval Status, Genetic Target
Q1.618
Q1
Is HTR1E a druggable gene?
There are currently 5 approved drugs which target HTR1E, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%HTR1E %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1378', 'drugName': 'Amisulpride', 'drugIsApproved': True, 'newLinkedTargets_string': 'HTR1F (ENSG00000179097), HTR2B (ENSG00000135914), HTR4 (ENSG00000164270), HTR1B (ENSG00000135312), HTR3A (ENSG00000166736), HTR1A (ENSG00000178394), HTR1D (ENSG00000179546), HTR2A (ENSG00000102468), HTR2C...
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Approval Status, Genetic Target
Q1.1063
Q1
Is PDE9A a druggable gene?
There are currently 2 approved drugs which target PDE9A, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%PDE9A %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4263', 'drugName': 'Pentoxifylline', 'drugIsApproved': True, 'newLinkedTargets_string': 'ADORA2B (ENSG00000170425), ADORA2A (ENSG00000128271), PDE5A (ENSG00000138735), PDE4A (ENSG00000065989), PDE3A (ENSG00000172572), PDE6H (ENSG00000139053), PDE6G (ENSG00000185527), PDE2A (ENSG00000186642...
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Approval Status, Genetic Target
Q1.1011
Q1
Is NRP1 a druggable gene?
There are currently no approved drugs targeting NRP1, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%NRP1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1821', 'drugName': 'Vesencumab', 'drugIsApproved': False, 'newLinkedTargets_string': 'NRP1 (ENSG00000099250)', 'maxClinicalTrialPhase': 1}]
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Approval Status, Genetic Target
Q1.1433
Q1
Is TLR2 a druggable gene?
There are currently no approved drugs targeting TLR2, but there are 2 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%TLR2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5402', 'drugName': 'Tomaralimab', 'drugIsApproved': False, 'newLinkedTargets_string': 'TLR2 (ENSG00000137462)', 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_5798', 'drugName': 'Vb-201', 'drugIsApproved': False, 'newLinkedTargets_string': 'TLR2 (ENSG00000137462), CD14 (ENSG0000...
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