Datasets:

uuid
stringlengths
4
8
template_uuid
stringclasses
40 values
question
stringlengths
13
193
answer
stringlengths
29
2.2k
benchmark_query
stringlengths
133
622
execution_results
stringlengths
2
1.14M
query_type
stringclasses
2 values
sql_category
stringclasses
26 values
bio_category
stringclasses
14 values
Q1.931
Q1
Is NCAM1 a druggable gene?
There are currently no approved drugs targeting NCAM1, but there are 3 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%NCAM1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_189', 'drugName': 'Oncolysin S', 'drugIsApproved': False, 'newLinkedTargets_string': 'NCAM1 (ENSG00000149294)', 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_3306', 'drugName': 'Bb-10901', 'drugIsApproved': False, 'newLinkedTargets_string': 'NCAM1 (ENSG00000149294)', 'maxClinic...
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Approval Status, Genetic Target
Q1.576
Q1
Is HCK a druggable gene?
There are currently 2 approved drugs which target HCK, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%HCK %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3959', 'drugName': 'Bosutinib', 'drugIsApproved': True, 'newLinkedTargets_string': 'ABL1 (ENSG00000097007), BCR (ENSG00000186716), HCK (ENSG00000101336), SRC (ENSG00000197122), LYN (ENSG00000254087)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4603', 'drugName': 'Dasatinib',...
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Approval Status, Genetic Target
Q1.506
Q1
Is GABRG3 a druggable gene?
There are currently 66 approved drugs which target GABRG3, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%GABRG3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1494', 'drugName': 'Thiopental', 'drugIsApproved': True, 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089), GABRA3 (ENSG00000011677)...
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Approval Status, Genetic Target
Q1.787
Q1
Is KEAP1 a druggable gene?
There are currently 3 approved drugs which target KEAP1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%KEAP1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3182', 'drugName': 'Dimethyl Fumarate', 'drugIsApproved': True, 'newLinkedTargets_string': 'KEAP1 (ENSG00000079999)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5578', 'drugName': 'Diroximel Fumarate', 'drugIsApproved': True, 'newLinkedTargets_string': 'KEAP1 (ENSG0000007999...
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Approval Status, Genetic Target
Q1.4
Q1
Is ABCB1 a druggable gene?
There are currently no approved drugs targeting ABCB1, but there are 5 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%ABCB1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3894', 'drugName': 'Tariquidar', 'drugIsApproved': False, 'newLinkedTargets_string': 'ABCB1 (ENSG00000085563)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_5486', 'drugName': 'Zosuquidar', 'drugIsApproved': False, 'newLinkedTargets_string': 'ABCB1 (ENSG00000085563)', 'maxClin...
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Approval Status, Genetic Target
Q1.1369
Q1
Is SLC34A2 a druggable gene?
There are currently no approved drugs targeting SLC34A2, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%SLC34A2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3443', 'drugName': 'Lifastuzumab Vedotin', 'drugIsApproved': False, 'newLinkedTargets_string': 'SLC34A2 (ENSG00000157765), TUBB4B (ENSG00000188229), TUBB1 (ENSG00000101162), TUBA3C (ENSG00000198033), TUBA4A (ENSG00000127824), TUBB3 (ENSG00000258947), TUBA1A (ENSG00000167552), TUBB4A (ENSG0...
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Approval Status, Genetic Target
Q1.469
Q1
Is FGR a druggable gene?
There is 1 drug, Dasatinib, that targets FGR, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%FGR %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4602', 'drugName': 'Dasatinib', 'drugIsApproved': True, 'newLinkedTargets_string': 'PDGFRB (ENSG00000113721), FYN (ENSG00000010810), SRC (ENSG00000197122), LCK (ENSG00000182866), YES1 (ENSG00000176105), BLK (ENSG00000136573), HCK (ENSG00000101336), LYN (ENSG00000254087), FRK (ENSG000001118...
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Approval Status, Genetic Target
Q1.323
Q1
Is CSF2RB a druggable gene?
There is 1 drug, Sargramostim, that targets CSF2RB, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CSF2RB %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5636', 'drugName': 'Sargramostim', 'drugIsApproved': True, 'newLinkedTargets_string': 'CSF2RA (ENSG00000198223), CSF2RB (ENSG00000100368)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4751', 'drugName': 'Mavrilimumab', 'drugIsApproved': False, 'newLinkedTargets_string': 'CSF2...
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Approval Status, Genetic Target
Q1.6
Q1
Is ABCC8 a druggable gene?
There are currently 11 approved drugs which target ABCC8, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%ABCC8 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_951', 'drugName': 'Chlorpropamide', 'drugIsApproved': True, 'newLinkedTargets_string': 'KCNJ11 (ENSG00000187486), ABCC8 (ENSG00000006071)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5473', 'drugName': 'Glimepiride', 'drugIsApproved': True, 'newLinkedTargets_string': 'KCNJ11...
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Approval Status, Genetic Target
Q1.1003
Q1
Is NPY5R a druggable gene?
There are currently no approved drugs targeting NPY5R, but there are 3 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%NPY5R %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_836', 'drugName': 'Mk-0557', 'drugIsApproved': False, 'newLinkedTargets_string': 'NPY5R (ENSG00000164129)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_848', 'drugName': 'Velneperit', 'drugIsApproved': False, 'newLinkedTargets_string': 'NPY5R (ENSG00000164129)', 'maxClinicalT...
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Approval Status, Genetic Target
Q1.550
Q1
Is GRIN2B a druggable gene?
There are currently 14 approved drugs which target GRIN2B, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%GRIN2B %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_70', 'drugName': 'Orphenadrine', 'drugIsApproved': True, 'newLinkedTargets_string': 'SCN1A (ENSG00000144285), SCN5A (ENSG00000183873), SCN4A (ENSG00000007314), SCN7A (ENSG00000136546), SCN2A (ENSG00000136531), SCN9A (ENSG00000169432), SCN3A (ENSG00000153253), SCN11A (ENSG00000168356), SCN8...
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Approval Status, Genetic Target
Q1.1095
Q1
Is PLK1 a druggable gene?
There are currently no approved drugs targeting PLK1, but there are 8 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%PLK1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2040', 'drugName': 'Volasertib', 'drugIsApproved': False, 'newLinkedTargets_string': 'PLK1 (ENSG00000166851)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_5804', 'drugName': 'Bi-2536', 'drugIsApproved': False, 'newLinkedTargets_string': 'PLK1 (ENSG00000166851)', 'maxClinicalT...
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Approval Status, Genetic Target
Q1.40
Q1
Is ADRB3 a druggable gene?
There are currently 27 approved drugs which target ADRB3, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%ADRB3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3354', 'drugName': 'Carteolol', 'drugIsApproved': True, 'newLinkedTargets_string': 'ADRB1 (ENSG00000043591), ADRB2 (ENSG00000169252), ADRB3 (ENSG00000188778)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3364', 'drugName': 'Dilevalol Hydrochloride', 'drugIsApproved': True, 'n...
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Approval Status, Genetic Target
Q1.545
Q1
Is GRIK3 a druggable gene?
There is 1 drug, Topiramate, that targets GRIK3, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%GRIK3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1594', 'drugName': 'Topiramate', 'drugIsApproved': True, 'newLinkedTargets_string': 'GRIK1 (ENSG00000171189), GRIK5 (ENSG00000105737), GRIK4 (ENSG00000149403), GRIK2 (ENSG00000164418), GRIK3 (ENSG00000163873), CA4 (ENSG00000167434), SCN1A (ENSG00000144285), SCN5A (ENSG00000183873), SCN4A (...
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Approval Status, Genetic Target
Q1.244
Q1
Is CDK4 a druggable gene?
There are currently 6 approved drugs which target CDK4, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CDK4 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3487', 'drugName': 'Ribociclib', 'drugIsApproved': True, 'newLinkedTargets_string': 'CDK4 (ENSG00000135446), CDK6 (ENSG00000105810)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3860', 'drugName': 'Trilaciclib Dihydrochloride', 'drugIsApproved': True, 'newLinkedTargets_string...
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Approval Status, Genetic Target
Q1.138
Q1
Is CA5B a druggable gene?
There are currently 2 approved drugs which target CA5B, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CA5B %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6095', 'drugName': 'Sulthiame', 'drugIsApproved': True, 'newLinkedTargets_string': 'CA2 (ENSG00000104267), CA7 (ENSG00000168748), CA1 (ENSG00000133742), CA3 (ENSG00000164879), CA6 (ENSG00000131686), CA12 (ENSG00000074410), CA14 (ENSG00000118298), CA9 (ENSG00000107159), CA4 (ENSG00000167434...
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Approval Status, Genetic Target
Q1.1329
Q1
Is S1PR5 a druggable gene?
There are currently 3 approved drugs which target S1PR5, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%S1PR5 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5906', 'drugName': 'Fingolimod Lauryl Sulfate', 'drugIsApproved': True, 'newLinkedTargets_string': 'S1PR5 (ENSG00000180739), S1PR2 (ENSG00000267534), S1PR4 (ENSG00000125910), S1PR3 (ENSG00000213694), S1PR1 (ENSG00000170989)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4765',...
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Approval Status, Genetic Target
Q1.623
Q1
Is HTR3A a druggable gene?
There are currently 21 approved drugs which target HTR3A, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%HTR3A %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2172', 'drugName': 'Vortioxetine', 'drugIsApproved': True, 'newLinkedTargets_string': 'HTR1A (ENSG00000178394), SLC6A4 (ENSG00000108576), HTR3A (ENSG00000166736)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2170', 'drugName': 'Vortioxetine', 'drugIsApproved': True, 'newLinke...
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Approval Status, Genetic Target
Q1.829
Q1
Is LRP1 a druggable gene?
There are currently no approved drugs targeting LRP1, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%LRP1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_429', 'drugName': 'Ang1005', 'drugIsApproved': False, 'newLinkedTargets_string': 'LRP1 (ENSG00000123384), TUBB4B (ENSG00000188229), TUBB1 (ENSG00000101162), TUBA3C (ENSG00000198033), TUBA4A (ENSG00000127824), TUBB3 (ENSG00000258947), TUBA1A (ENSG00000167552), TUBB4A (ENSG00000104833), TUBB...
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Approval Status, Genetic Target
Q1.699
Q1
Is IL4 a druggable gene?
There are currently no approved drugs targeting IL4, but there are 2 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%IL4 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5968', 'drugName': 'Pascolizumab', 'drugIsApproved': False, 'newLinkedTargets_string': 'IL4 (ENSG00000113520)', 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_932', 'drugName': 'Romilkimab', 'drugIsApproved': False, 'newLinkedTargets_string': 'IL4 (ENSG00000113520), IL13 (ENSG00...
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Approval Status, Genetic Target
Q1.1093
Q1
Is PLAT a druggable gene?
There is 1 drug, Aminocaproic Acid, that targets PLAT, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%PLAT %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5590', 'drugName': 'Aminocaproic Acid', 'drugIsApproved': True, 'newLinkedTargets_string': 'PLAT (ENSG00000104368), PLG (ENSG00000122194)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5591', 'drugName': 'Aminocaproic Acid', 'drugIsApproved': True, 'newLinkedTargets_string': '...
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Approval Status, Genetic Target
Q1.1474
Q1
Is TPH2 a druggable gene?
There are currently 3 approved drugs which target TPH2, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%TPH2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3468', 'drugName': 'Telotristat', 'drugIsApproved': True, 'newLinkedTargets_string': 'TPH2 (ENSG00000139287), TPH1 (ENSG00000129167)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1302', 'drugName': 'Telotristat Ethyl', 'drugIsApproved': True, 'newLinkedTargets_string': 'TPH2 ...
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Approval Status, Genetic Target
Q1.585
Q1
Is HDAC4 a druggable gene?
There are currently 4 approved drugs which target HDAC4, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%HDAC4 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4906', 'drugName': 'Panobinostat', 'drugIsApproved': True, 'newLinkedTargets_string': 'HDAC1 (ENSG00000116478), HDAC3 (ENSG00000171720), HDAC6 (ENSG00000094631), HDAC2 (ENSG00000196591), HDAC5 (ENSG00000108840), HDAC7 (ENSG00000061273), HDAC8 (ENSG00000147099), HDAC11 (ENSG00000163517), HD...
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Approval Status, Genetic Target
Q1.1513
Q1
Is TYK2 a druggable gene?
There are currently 4 approved drugs which target TYK2, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%TYK2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6269', 'drugName': 'Deucravacitinib', 'drugIsApproved': True, 'newLinkedTargets_string': 'TYK2 (ENSG00000105397)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1979', 'drugName': 'Deucravacitinib', 'drugIsApproved': True, 'newLinkedTargets_string': 'TYK2 (ENSG00000105397)', 'm...
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Approval Status, Genetic Target
Q1.815
Q1
Is LCK a druggable gene?
There are currently 3 approved drugs which target LCK, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%LCK %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4603', 'drugName': 'Dasatinib', 'drugIsApproved': True, 'newLinkedTargets_string': 'PDGFRB (ENSG00000113721), FYN (ENSG00000010810), SRC (ENSG00000197122), LCK (ENSG00000182866), YES1 (ENSG00000176105), BLK (ENSG00000136573), HCK (ENSG00000101336), LYN (ENSG00000254087), FRK (ENSG000001118...
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Approval Status, Genetic Target
Q1.1463
Q1
Is TNNI2 a druggable gene?
There are currently no approved drugs targeting TNNI2, but there are 2 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%TNNI2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_451', 'drugName': 'Reldesemtiv', 'drugIsApproved': False, 'newLinkedTargets_string': 'TNNI2 (ENSG00000130598), TNNT3 (ENSG00000130595), TNNC2 (ENSG00000101470)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_6283', 'drugName': 'Tirasemtiv', 'drugIsApproved': False, 'newLinkedTa...
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Approval Status, Genetic Target
Q1.378
Q1
Is E2F1 a druggable gene?
There are currently no approved drugs targeting E2F1, but there are 2 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%E2F1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4614', 'drugName': 'Edifoligide Sodium', 'drugIsApproved': False, 'newLinkedTargets_string': 'E2F1 (ENSG00000101412), E2F2 (ENSG00000007968), E2F3 (ENSG00000112242), E2F4 (ENSG00000205250), E2F5 (ENSG00000133740), E2F6 (ENSG00000169016), E2F7 (ENSG00000165891), E2F8 (ENSG00000129173)', 'ma...
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Approval Status, Genetic Target
Q1.316
Q1
Is CREBBP a druggable gene?
There are currently no approved drugs targeting CREBBP, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CREBBP %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3141', 'drugName': 'Pri-724', 'drugIsApproved': False, 'newLinkedTargets_string': 'CREBBP (ENSG00000005339), CTNNB1 (ENSG00000168036)', 'maxClinicalTrialPhase': 2}]
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Approval Status, Genetic Target
Q1.444
Q1
Is F8 a druggable gene?
There is 1 drug, Drotrecogin Alfa (Activated), that targets F8, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%F8 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1085', 'drugName': 'Brentuximab Vedotin', 'drugIsApproved': True, 'newLinkedTargets_string': 'TNFRSF8 (ENSG00000120949), TUBB4B (ENSG00000188229), TUBB1 (ENSG00000101162), TUBA3C (ENSG00000198033), TUBA4A (ENSG00000127824), TUBB3 (ENSG00000258947), TUBA1A (ENSG00000167552), TUBB4A (ENSG000...
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Approval Status, Genetic Target
Q1.321
Q1
Is CSF2 a druggable gene?
There are currently no approved drugs targeting CSF2, but there are 6 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CSF2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3438', 'drugName': 'Lenzilumab', 'drugIsApproved': False, 'newLinkedTargets_string': 'CSF2 (ENSG00000164400)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_4644', 'drugName': 'Otilimab', 'drugIsApproved': False, 'newLinkedTargets_string': 'CSF2 (ENSG00000164400)', 'maxClinical...
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Approval Status, Genetic Target
Q1.1186
Q1
Is PSMD8 a druggable gene?
There are currently 4 approved drugs which target PSMD8, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%PSMD8 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_559', 'drugName': 'Bortezomib', 'drugIsApproved': True, 'newLinkedTargets_string': 'PSMD1 (ENSG00000173692), PSMB2 (ENSG00000126067), PSMB1 (ENSG00000008018), PSMB5 (ENSG00000100804), PSMB8 (ENSG00000204264), PSMB9 (ENSG00000240065), PSMB6 (ENSG00000142507), PSMD14 (ENSG00000115233), PSMA1...
general
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Approval Status, Genetic Target
Q1.1317
Q1
Is RTN4 a druggable gene?
There are currently no approved drugs targeting RTN4, but there are 2 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%RTN4 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6319', 'drugName': 'Ozanezumab', 'drugIsApproved': False, 'newLinkedTargets_string': 'RTN4 (ENSG00000115310)', 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_5814', 'drugName': 'Atinumab', 'drugIsApproved': False, 'newLinkedTargets_string': 'RTN4 (ENSG00000115310)', 'maxClinical...
general
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Approval Status, Genetic Target
Q1.1158
Q1
Is PSMA8 a druggable gene?
There are currently 4 approved drugs which target PSMA8, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%PSMA8 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3334', 'drugName': 'Ixazomib', 'drugIsApproved': True, 'newLinkedTargets_string': 'PSMD1 (ENSG00000173692), PSMB2 (ENSG00000126067), PSMB1 (ENSG00000008018), PSMB5 (ENSG00000100804), PSMB8 (ENSG00000204264), PSMB9 (ENSG00000240065), PSMB6 (ENSG00000142507), PSMD14 (ENSG00000115233), PSMA1 ...
general
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Approval Status, Genetic Target
Q1.426
Q1
Is ERBB3 a druggable gene?
There is 1 drug, Vandetanib, that targets ERBB3, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%ERBB3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1933', 'drugName': 'Vandetanib', 'drugIsApproved': True, 'newLinkedTargets_string': 'TEK (ENSG00000120156), ERBB2 (ENSG00000141736), EGFR (ENSG00000146648), ERBB4 (ENSG00000178568), ERBB3 (ENSG00000065361), EPHA2 (ENSG00000142627), EPHB2 (ENSG00000133216), EPHA5 (ENSG00000145242), EPHA4 (E...
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Approval Status, Genetic Target
Q1.556
Q1
Is GRM3 a druggable gene?
There are currently no approved drugs targeting GRM3, but there are 4 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%GRM3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6226', 'drugName': 'Pomaglumetad Methionil', 'drugIsApproved': False, 'newLinkedTargets_string': 'GRM2 (ENSG00000164082), GRM3 (ENSG00000198822)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_6227', 'drugName': 'Pomaglumetad Methionil', 'drugIsApproved': False, 'newLinkedTarge...
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Approval Status, Genetic Target
Q1.598
Q1
Is HNF4A a druggable gene?
There is 1 drug, Alverine, that targets HNF4A, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%HNF4A %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4846', 'drugName': 'Alverine', 'drugIsApproved': True, 'newLinkedTargets_string': 'HTR1A (ENSG00000178394), HNF4A (ENSG00000101076)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4847', 'drugName': 'Alverine', 'drugIsApproved': True, 'newLinkedTargets_string': 'HTR1A (ENSG0000...
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Approval Status, Genetic Target
Q1.922
Q1
Is MYH6 a druggable gene?
There is 1 drug, Mavacamten, that targets MYH6, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%MYH6 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1036', 'drugName': 'Mavacamten', 'drugIsApproved': True, 'newLinkedTargets_string': 'MYH7 (ENSG00000092054), MYH6 (ENSG00000197616), MYH7B (ENSG00000078814), MYL3 (ENSG00000160808), MYL2 (ENSG00000111245), MYL7 (ENSG00000106631), MYL4 (ENSG00000198336)', 'maxClinicalTrialPhase': 4}, {'UUID...
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Approval Status, Genetic Target
Q1.674
Q1
Is IL15 a druggable gene?
There are currently no approved drugs targeting IL15, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%IL15 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3251', 'drugName': 'Ordesekimab', 'drugIsApproved': False, 'newLinkedTargets_string': 'IL15 (ENSG00000164136)', 'maxClinicalTrialPhase': 2}]
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Approval Status, Genetic Target
Q1.1091
Q1
Is PLA2G5 a druggable gene?
There are currently no approved drugs targeting PLA2G5, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%PLA2G5 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6244', 'drugName': 'Varespladib Methyl', 'drugIsApproved': False, 'newLinkedTargets_string': 'PLA2G5 (ENSG00000127472), PLA2G10 (ENSG00000069764), PLA2G2A (ENSG00000188257)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_6245', 'drugName': 'Varespladib Methyl', 'drugIsApproved'...
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Approval Status, Genetic Target
Q1.1248
Q1
Is RPL27A a druggable gene?
There is 1 drug, Ataluren, that targets RPL27A, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%RPL27A %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'drugIsApproved': True, 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG...
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Approval Status, Genetic Target
Q1.1402
Q1
Is STAT3 a druggable gene?
There are currently no approved drugs targeting STAT3, but there are 2 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%STAT3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4959', 'drugName': 'Danvatirsen', 'drugIsApproved': False, 'newLinkedTargets_string': 'STAT3 (ENSG00000168610)', 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_199', 'drugName': 'Danvatirsen Sodium', 'drugIsApproved': False, 'newLinkedTargets_string': 'STAT3 (ENSG00000168610)', ...
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Approval Status, Genetic Target
Q1.229
Q1
Is CDH3 a druggable gene?
There are currently no approved drugs targeting CDH3, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CDH3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1343', 'drugName': 'Pf-03732010', 'drugIsApproved': False, 'newLinkedTargets_string': 'CDH3 (ENSG00000062038)', 'maxClinicalTrialPhase': 1}]
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Approval Status, Genetic Target
Q1.1207
Q1
Is RAF1 a druggable gene?
There are currently 3 approved drugs which target RAF1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%RAF1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_812', 'drugName': 'Regorafenib', 'drugIsApproved': True, 'newLinkedTargets_string': 'EPHA2 (ENSG00000142627), TEK (ENSG00000120156), MAPK11 (ENSG00000185386), RAF1 (ENSG00000132155), FRK (ENSG00000111816), PDGFRB (ENSG00000113721), PDGFRA (ENSG00000134853), KIT (ENSG00000157404), FGFR1 (EN...
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Approval Status, Genetic Target
Q1.1198
Q1
Is PTGS2 a druggable gene?
There are currently 71 approved drugs which target PTGS2, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%PTGS2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2672', 'drugName': 'Parecoxib Sodium', 'drugIsApproved': True, 'newLinkedTargets_string': 'PTGS2 (ENSG00000073756)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5955', 'drugName': 'Valdecoxib', 'drugIsApproved': True, 'newLinkedTargets_string': 'PTGS2 (ENSG00000073756)', 'max...
general
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Approval Status, Genetic Target
Q1.1154
Q1
Is PSMA4 a druggable gene?
There are currently 4 approved drugs which target PSMA4, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%PSMA4 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3334', 'drugName': 'Ixazomib', 'drugIsApproved': True, 'newLinkedTargets_string': 'PSMD1 (ENSG00000173692), PSMB2 (ENSG00000126067), PSMB1 (ENSG00000008018), PSMB5 (ENSG00000100804), PSMB8 (ENSG00000204264), PSMB9 (ENSG00000240065), PSMB6 (ENSG00000142507), PSMD14 (ENSG00000115233), PSMA1 ...
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Approval Status, Genetic Target
Q1.712
Q1
Is INSR a druggable gene?
There are currently 37 approved drugs which target INSR, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%INSR %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_495', 'drugName': 'Insulin Glargine', 'drugIsApproved': True, 'newLinkedTargets_string': 'INSR (ENSG00000171105)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5849', 'drugName': 'Insulin Susp Isophane Semisynthetic Purified Human', 'drugIsApproved': True, 'newLinkedTargets_st...
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Approval Status, Genetic Target
Q1.67
Q1
Is AOC3 a druggable gene?
There are currently no approved drugs targeting AOC3, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%AOC3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5390', 'drugName': 'Vepalimomab', 'drugIsApproved': False, 'newLinkedTargets_string': 'AOC3 (ENSG00000131471)', 'maxClinicalTrialPhase': 2}]
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Approval Status, Genetic Target
Q1.395
Q1
Is EGLN2 a druggable gene?
There is 1 drug, Roxadustat, that targets EGLN2, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%EGLN2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5393', 'drugName': 'Roxadustat', 'drugIsApproved': True, 'newLinkedTargets_string': 'EGLN2 (ENSG00000269858), P4HTM (ENSG00000178467), EGLN1 (ENSG00000135766), EGLN3 (ENSG00000129521)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2677', 'drugName': 'Daprodustat', 'drugIsAppro...
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Approval Status, Genetic Target
Q1.583
Q1
Is HDAC2 a druggable gene?
There are currently 5 approved drugs which target HDAC2, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%HDAC2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2373', 'drugName': 'Vorinostat', 'drugIsApproved': True, 'newLinkedTargets_string': 'HDAC1 (ENSG00000116478), HDAC2 (ENSG00000196591), HDAC3 (ENSG00000171720), HDAC6 (ENSG00000094631)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2372', 'drugName': 'Vorinostat', 'drugIsApprov...
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Approval Status, Genetic Target
Q1.1019
Q1
Is OPRK1 a druggable gene?
There are currently 33 approved drugs which target OPRK1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%OPRK1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2630', 'drugName': 'Levallorphan', 'drugIsApproved': True, 'newLinkedTargets_string': 'OPRK1 (ENSG00000082556), OPRM1 (ENSG00000112038)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_749', 'drugName': 'Butorphanol', 'drugIsApproved': True, 'newLinkedTargets_string': 'OPRM1 (EN...
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Approval Status, Genetic Target
Q1.213
Q1
Is CD3G a druggable gene?
There are currently 4 approved drugs which target CD3G, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CD3G %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3214', 'drugName': 'Muromonab-Cd3', 'drugIsApproved': True, 'newLinkedTargets_string': 'CD3E (ENSG00000198851), CD3G (ENSG00000160654), CD3D (ENSG00000167286)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_6103', 'drugName': 'Teclistamab', 'drugIsApproved': True, 'newLinkedTar...
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Approval Status, Genetic Target
Q1.1187
Q1
Is PTAFR a druggable gene?
There are currently no approved drugs targeting PTAFR, but there are 2 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%PTAFR %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2192', 'drugName': 'Rupatadine', 'drugIsApproved': False, 'newLinkedTargets_string': 'HRH1 (ENSG00000196639), PTAFR (ENSG00000169403)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_2191', 'drugName': 'Rupatadine', 'drugIsApproved': False, 'newLinkedTargets_string': 'HRH1 (ENSG...
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Approval Status, Genetic Target
Q1.957
Q1
Is NDUFB2 a druggable gene?
There are currently 2 approved drugs which target NDUFB2, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%NDUFB2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'drugIsApproved': True, 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (EN...
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Approval Status, Genetic Target
Q1.539
Q1
Is GRIA1 a druggable gene?
There are currently 2 approved drugs which target GRIA1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%GRIA1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1597', 'drugName': 'Topiramate', 'drugIsApproved': True, 'newLinkedTargets_string': 'GRIK1 (ENSG00000171189), GRIK5 (ENSG00000105737), GRIK4 (ENSG00000149403), GRIK2 (ENSG00000164418), GRIK3 (ENSG00000163873), CA4 (ENSG00000167434), SCN1A (ENSG00000144285), SCN5A (ENSG00000183873), SCN4A (...
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Approval Status, Genetic Target
Q1.1237
Q1
Is RPL17 a druggable gene?
There is 1 drug, Ataluren, that targets RPL17, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%RPL17 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'drugIsApproved': True, 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG...
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Approval Status, Genetic Target
Q1.685
Q1
Is IL1RAP a druggable gene?
There is 1 drug, Spesolimab, that targets IL1RAP, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%IL1RAP %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2421', 'drugName': 'Spesolimab', 'drugIsApproved': True, 'newLinkedTargets_string': 'IL1RL2 (ENSG00000115598), IL1RAP (ENSG00000196083)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_102', 'drugName': 'Imsidolimab', 'drugIsApproved': False, 'newLinkedTargets_string': 'IL1RL2 (...
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Approval Status, Genetic Target
Q1.87
Q1
Is ATP2A1 a druggable gene?
There are currently no approved drugs targeting ATP2A1, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%ATP2A1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3997', 'drugName': 'Mipsagargin', 'drugIsApproved': False, 'newLinkedTargets_string': 'ATP2A3 (ENSG00000074370), ATP2A1 (ENSG00000196296), ATP2A2 (ENSG00000174437)', 'maxClinicalTrialPhase': 2}]
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Approval Status, Genetic Target
Q1.1383
Q1
Is SMO a druggable gene?
There are currently 5 approved drugs which target SMO, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%SMO %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2876', 'drugName': 'Glasdegib Maleate', 'drugIsApproved': True, 'newLinkedTargets_string': 'SMO (ENSG00000128602)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3933', 'drugName': 'Sonidegib Phosphate', 'drugIsApproved': True, 'newLinkedTargets_string': 'SMO (ENSG00000128602)'...
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Approval Status, Genetic Target
Q1.274
Q1
Is CHRNB4 a druggable gene?
There are currently 6 approved drugs which target CHRNB4, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CHRNB4 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5467', 'drugName': 'Trimethaphan Camsylate', 'drugIsApproved': True, 'newLinkedTargets_string': 'CHRNB4 (ENSG00000117971), CHRNA3 (ENSG00000080644)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4467', 'drugName': 'Trimethaphan', 'drugIsApproved': True, 'newLinkedTargets_strin...
general
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Approval Status, Genetic Target
Q1.944
Q1
Is NDUFA5 a druggable gene?
There are currently 2 approved drugs which target NDUFA5, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%NDUFA5 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'drugIsApproved': True, 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (EN...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.684
Q1
Is IL1R1 a druggable gene?
There is 1 drug, Anakinra, that targets IL1R1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%IL1R1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2379', 'drugName': 'Anakinra', 'drugIsApproved': True, 'newLinkedTargets_string': 'IL1R1 (ENSG00000115594)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2001', 'drugName': 'Medi-8968', 'drugIsApproved': False, 'newLinkedTargets_string': 'IL1R1 (ENSG00000115594)', 'maxClinical...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1384
Q1
Is SNAP25 a druggable gene?
There are currently 6 approved drugs which target SNAP25, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%SNAP25 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2163', 'drugName': 'Onabotulinumtoxina', 'drugIsApproved': True, 'newLinkedTargets_string': 'SNAP25 (ENSG00000132639)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5684', 'drugName': 'Abobotulinumtoxina', 'drugIsApproved': True, 'newLinkedTargets_string': 'SNAP25 (ENSG0000013...
general
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Approval Status, Genetic Target
Q1.634
Q1
Is ICAM3 a druggable gene?
There are currently no approved drugs targeting ICAM3, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%ICAM3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1930', 'drugName': 'Icm3', 'drugIsApproved': False, 'newLinkedTargets_string': 'ICAM3 (ENSG00000076662)', 'maxClinicalTrialPhase': 2}]
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1053
Q1
Is PDE6A a druggable gene?
There are currently 2 approved drugs which target PDE6A, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%PDE6A %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6107', 'drugName': 'Dipyridamole', 'drugIsApproved': True, 'newLinkedTargets_string': 'PDE5A (ENSG00000138735), PDE4A (ENSG00000065989), PDE3A (ENSG00000172572), PDE6H (ENSG00000139053), PDE6G (ENSG00000185527), PDE2A (ENSG00000186642), PDE7A (ENSG00000205268), PDE1A (ENSG00000115252), PDE...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1435
Q1
Is TLR4 a druggable gene?
There are currently no approved drugs targeting TLR4, but there are 3 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%TLR4 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5358', 'drugName': 'Resatorvid', 'drugIsApproved': False, 'newLinkedTargets_string': 'TLR4 (ENSG00000136869)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_1063', 'drugName': 'Eritoran Tetrasodium', 'drugIsApproved': False, 'newLinkedTargets_string': 'TLR4 (ENSG00000136869), L...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1058
Q1
Is PDE6H a druggable gene?
There are currently 2 approved drugs which target PDE6H, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%PDE6H %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6107', 'drugName': 'Dipyridamole', 'drugIsApproved': True, 'newLinkedTargets_string': 'PDE5A (ENSG00000138735), PDE4A (ENSG00000065989), PDE3A (ENSG00000172572), PDE6H (ENSG00000139053), PDE6G (ENSG00000185527), PDE2A (ENSG00000186642), PDE7A (ENSG00000205268), PDE1A (ENSG00000115252), PDE...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.275
Q1
Is CHRND a druggable gene?
There are currently 28 approved drugs which target CHRND, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CHRND %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2723', 'drugName': 'Succinylcholine Chloride', 'drugIsApproved': True, 'newLinkedTargets_string': 'CHRNA1 (ENSG00000138435), CHRNG (ENSG00000196811), CHRNB1 (ENSG00000170175), CHRND (ENSG00000135902), CHRNE (ENSG00000108556)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_922',...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.746
Q1
Is KCNC4 a druggable gene?
There are currently 5 approved drugs which target KCNC4, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%KCNC4 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5118', 'drugName': 'Guanidine Hydrochloride', 'drugIsApproved': True, 'newLinkedTargets_string': 'KCNQ1 (ENSG00000053918), KCND3 (ENSG00000171385), KCNH2 (ENSG00000055118), KCNA2 (ENSG00000177301), KCNA1 (ENSG00000111262), KCNQ2 (ENSG00000075043), KCNQ3 (ENSG00000184156), KCNA7 (ENSG000001...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.364
Q1
Is DLL3 a druggable gene?
There are currently no approved drugs targeting DLL3, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%DLL3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4409', 'drugName': 'Rovalpituzumab Tesirine', 'drugIsApproved': False, 'newLinkedTargets_string': 'DLL3 (ENSG00000090932)', 'maxClinicalTrialPhase': 3}]
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.626
Q1
Is HTR3D a druggable gene?
There are currently 7 approved drugs which target HTR3D, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%HTR3D %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2386', 'drugName': 'Clothiapine', 'drugIsApproved': True, 'newLinkedTargets_string': 'HTR2B (ENSG00000135914), HTR2A (ENSG00000102468), HTR2C (ENSG00000147246), DRD4 (ENSG00000069696), HTR3A (ENSG00000166736), HTR3E (ENSG00000186038), HTR3B (ENSG00000149305), HTR3D (ENSG00000186090), HTR3C...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.3
Q1
Is ABCA1 a druggable gene?
There is 1 drug, Probucol, that targets ABCA1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%ABCA1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_632', 'drugName': 'Probucol', 'drugIsApproved': True, 'newLinkedTargets_string': 'ABCA1 (ENSG00000165029)', 'maxClinicalTrialPhase': 4}]
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.7
Q1
Is ABCC9 a druggable gene?
There are currently 2 approved drugs which target ABCC9, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%ABCC9 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1076', 'drugName': 'Pinacidil', 'drugIsApproved': True, 'newLinkedTargets_string': 'KCNJ11 (ENSG00000187486), ABCC9 (ENSG00000069431)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5958', 'drugName': 'Pinacidil', 'drugIsApproved': True, 'newLinkedTargets_string': 'KCNJ11 (ENSG...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.313
Q1
Is CPT2 a druggable gene?
There are currently 2 approved drugs which target CPT2, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CPT2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1726', 'drugName': 'Perhexiline Maleate', 'drugIsApproved': True, 'newLinkedTargets_string': 'MTOR (ENSG00000198793), CPT2 (ENSG00000157184), CPT1B (ENSG00000205560)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_919', 'drugName': 'Perhexiline', 'drugIsApproved': True, 'newLin...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.717
Q1
Is ITGA4 a druggable gene?
There are currently 2 approved drugs which target ITGA4, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%ITGA4 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5016', 'drugName': 'Natalizumab', 'drugIsApproved': True, 'newLinkedTargets_string': 'ITGA4 (ENSG00000115232), ITGB7 (ENSG00000139626), ITGB1 (ENSG00000150093)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5015', 'drugName': 'Natalizumab', 'drugIsApproved': True, 'newLinkedTa...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.669
Q1
Is IL12A a druggable gene?
There is 1 drug, Ustekinumab, that targets IL12A, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%IL12A %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3327', 'drugName': 'Ustekinumab', 'drugIsApproved': True, 'newLinkedTargets_string': 'IL12B (ENSG00000113302), IL23A (ENSG00000110944), IL12A (ENSG00000168811)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3328', 'drugName': 'Ustekinumab', 'drugIsApproved': True, 'newLinkedTa...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.967
Q1
Is NDUFS1 a druggable gene?
There are currently 2 approved drugs which target NDUFS1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%NDUFS1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'drugIsApproved': True, 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (EN...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1516
Q1
Is TYR a druggable gene?
There are currently 2 approved drugs which target TYR, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%TYR %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5010', 'drugName': 'Mequinol', 'drugIsApproved': True, 'newLinkedTargets_string': 'TYR (ENSG00000077498)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3683', 'drugName': 'Monobenzone', 'drugIsApproved': True, 'newLinkedTargets_string': 'TYR (ENSG00000077498)', 'maxClinicalTri...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.217
Q1
Is CD44 a druggable gene?
There are currently no approved drugs targeting CD44, but there are 3 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CD44 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2202', 'drugName': 'Bivatuzumab', 'drugIsApproved': False, 'newLinkedTargets_string': 'CD44 (ENSG00000026508)', 'maxClinicalTrialPhase': 1}, {'UUID': 'DrugGeneTargets_v2_6223', 'drugName': 'Bivatuzumab Mertansine', 'drugIsApproved': False, 'newLinkedTargets_string': 'CD44 (ENSG00000026508)...
general
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Approval Status, Genetic Target
Q1.1460
Q1
Is TNKS2 a druggable gene?
There are currently no approved drugs targeting TNKS2, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%TNKS2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1419', 'drugName': '2X-121', 'drugIsApproved': False, 'newLinkedTargets_string': 'TNKS2 (ENSG00000107854), TNKS (ENSG00000173273), PARP1 (ENSG00000143799), PARP2 (ENSG00000129484)', 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_1420', 'drugName': '2X-121', 'drugIsApproved': Fal...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.28
Q1
Is ADORA1 a druggable gene?
There are currently 8 approved drugs which target ADORA1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%ADORA1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4548', 'drugName': 'Theophylline', 'drugIsApproved': True, 'newLinkedTargets_string': 'ADORA1 (ENSG00000163485), ADORA2B (ENSG00000170425), ADORA3 (ENSG00000282608), ADORA2A (ENSG00000128271), PDE3A (ENSG00000172572), PDE3B (ENSG00000152270), PDE4A (ENSG00000065989), PDE4D (ENSG00000113448...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1105
Q1
Is POLD4 a druggable gene?
There are currently 5 approved drugs which target POLD4, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%POLD4 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4', 'drugName': 'Gemcitabine Hydrochloride', 'drugIsApproved': True, 'newLinkedTargets_string': 'POLA1 (ENSG00000101868), POLD4 (ENSG00000175482), POLD3 (ENSG00000077514), POLD1 (ENSG00000062822), POLD2 (ENSG00000106628), POLE (ENSG00000177084), POLA2 (ENSG00000014138), PRIM1 (ENSG00000198...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.894
Q1
Is MMP12 a druggable gene?
There are currently no approved drugs targeting MMP12, but there are 3 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%MMP12 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5864', 'drugName': 'Marimastat', 'drugIsApproved': False, 'newLinkedTargets_string': 'MMP9 (ENSG00000100985), MMP3 (ENSG00000149968), MMP7 (ENSG00000137673), MMP1 (ENSG00000196611), MMP2 (ENSG00000087245), MMP12 (ENSG00000262406)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1071
Q1
Is PDPK1 a druggable gene?
There are currently no approved drugs targeting PDPK1, but there are 2 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%PDPK1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4659', 'drugName': 'Ucn-01', 'drugIsApproved': False, 'newLinkedTargets_string': 'PDPK1 (ENSG00000140992), CDK2 (ENSG00000123374), CDK4 (ENSG00000135446), PRKD3 (ENSG00000115825), PRKCI (ENSG00000163558), PRKCA (ENSG00000154229), PRKCG (ENSG00000126583), PRKCD (ENSG00000163932), PRKCB (ENS...
general
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Approval Status, Genetic Target
Q1.642
Q1
Is IFNA13 a druggable gene?
There are currently no approved drugs targeting IFNA13, but there are 3 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%IFNA13 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4431', 'drugName': 'Rontalizumab', 'drugIsApproved': False, 'newLinkedTargets_string': 'IFNA6 (ENSG00000120235), IFNA8 (ENSG00000120242), IFNA5 (ENSG00000147873), IFNA10 (ENSG00000186803), IFNA2 (ENSG00000188379), IFNA1 (ENSG00000197919), IFNA13 (ENSG00000233816), IFNA7 (ENSG00000214042), ...
general
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Approval Status, Genetic Target
Q1.786
Q1
Is KDR a druggable gene?
There are currently 19 approved drugs which target KDR, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%KDR %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_392', 'drugName': 'Pazopanib Hydrochloride', 'drugIsApproved': True, 'newLinkedTargets_string': 'FGFR1 (ENSG00000077782), FGFR3 (ENSG00000068078), KIT (ENSG00000157404), CSF1R (ENSG00000182578), FLT1 (ENSG00000102755), FLT4 (ENSG00000037280), KDR (ENSG00000128052), ITK (ENSG00000113263), P...
general
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Approval Status, Genetic Target
Q1.854
Q1
Is MAP3K5 a druggable gene?
There are currently no approved drugs targeting MAP3K5, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%MAP3K5 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5336', 'drugName': 'Selonsertib', 'drugIsApproved': False, 'newLinkedTargets_string': 'MAP3K5 (ENSG00000197442)', 'maxClinicalTrialPhase': 3}]
general
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Approval Status, Genetic Target
Q1.628
Q1
Is HTR4 a druggable gene?
There are currently 13 approved drugs which target HTR4, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%HTR4 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3506', 'drugName': 'Metoclopramide', 'drugIsApproved': True, 'newLinkedTargets_string': 'HTR4 (ENSG00000164270), HTR3A (ENSG00000166736), DRD2 (ENSG00000149295)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2042', 'drugName': 'Tegaserod Maleate', 'drugIsApproved': True, 'newL...
general
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Approval Status, Genetic Target
Q1.1043
Q1
Is PDE1B a druggable gene?
There are currently 2 approved drugs which target PDE1B, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%PDE1B %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6107', 'drugName': 'Dipyridamole', 'drugIsApproved': True, 'newLinkedTargets_string': 'PDE5A (ENSG00000138735), PDE4A (ENSG00000065989), PDE3A (ENSG00000172572), PDE6H (ENSG00000139053), PDE6G (ENSG00000185527), PDE2A (ENSG00000186642), PDE7A (ENSG00000205268), PDE1A (ENSG00000115252), PDE...
general
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Approval Status, Genetic Target
Q1.258
Q1
Is CHKA a druggable gene?
There are currently no approved drugs targeting CHKA, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CHKA %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6258', 'drugName': 'Tcd-717', 'drugIsApproved': False, 'newLinkedTargets_string': 'CHKA (ENSG00000110721)', 'maxClinicalTrialPhase': 1}]
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Q1.26
Q1
Is ADH7 a druggable gene?
There is 1 drug, Nitrefazole, that targets ADH7, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%ADH7 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6344', 'drugName': 'Nitrefazole', 'drugIsApproved': True, 'newLinkedTargets_string': 'ADH1A (ENSG00000187758), ADH4 (ENSG00000198099), ADH1B (ENSG00000196616), ADH1C (ENSG00000248144), ADH7 (ENSG00000196344), ADH5 (ENSG00000197894), ADH6 (ENSG00000172955)', 'maxClinicalTrialPhase': 4}]
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Q1.338
Q1
Is CXCL8 a druggable gene?
There are currently no approved drugs targeting CXCL8, but there are 2 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CXCL8 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4247', 'drugName': 'Humax-Il8', 'drugIsApproved': False, 'newLinkedTargets_string': 'CXCL8 (ENSG00000169429)', 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_4996', 'drugName': 'Abx-Il8', 'drugIsApproved': False, 'newLinkedTargets_string': 'CXCL8 (ENSG00000169429)', 'maxClinical...
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Q1.575
Q1
Is HCAR2 a druggable gene?
There are currently no approved drugs targeting HCAR2, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%HCAR2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5716', 'drugName': 'Sch-900271', 'drugIsApproved': False, 'newLinkedTargets_string': 'HCAR2 (ENSG00000182782)', 'maxClinicalTrialPhase': 2}]
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Q1.48
Q1
Is AKR1B1 a druggable gene?
There is 1 drug, Tolrestat, that targets AKR1B1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%AKR1B1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6334', 'drugName': 'Tolrestat', 'drugIsApproved': True, 'newLinkedTargets_string': 'AKR1B1 (ENSG00000085662)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2353', 'drugName': 'Sorbinil', 'drugIsApproved': False, 'newLinkedTargets_string': 'AKR1B1 (ENSG00000085662)', 'maxClinic...
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Q1.108
Q1
Is BCR a druggable gene?
There are currently 10 approved drugs which target BCR, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%BCR %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6150', 'drugName': 'Ponatinib Hydrochloride', 'drugIsApproved': True, 'newLinkedTargets_string': 'ABL1 (ENSG00000097007), BCR (ENSG00000186716)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2277', 'drugName': 'Ponatinib', 'drugIsApproved': True, 'newLinkedTargets_string': 'AB...
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Q1.351
Q1
Is CYP3A7 a druggable gene?
There are currently 2 approved drugs which target CYP3A7, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CYP3A7 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2751', 'drugName': 'Ritonavir', 'drugIsApproved': True, 'newLinkedTargets_string': 'CYP3A4 (ENSG00000160868), CYP3A5 (ENSG00000106258), CYP3A43 (ENSG00000021461), CYP3A7 (ENSG00000160870)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2752', 'drugName': 'Ritonavir', 'drugIsApp...
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Q1.56
Q1
Is ALK a druggable gene?
There are currently 7 approved drugs which target ALK, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%ALK %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2435', 'drugName': 'Ceritinib', 'drugIsApproved': True, 'newLinkedTargets_string': 'ALK (ENSG00000171094), EML4 (ENSG00000143924), NPM1 (ENSG00000181163)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1250', 'drugName': 'Alectinib Hydrochloride', 'drugIsApproved': True, 'newLi...
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Q1.1136
Q1
Is PRKCD a druggable gene?
There is 1 drug, Midostaurin, that targets PRKCD, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%PRKCD %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5668', 'drugName': 'Midostaurin', 'drugIsApproved': True, 'newLinkedTargets_string': 'KIT (ENSG00000157404), KDR (ENSG00000128052), PDGFRB (ENSG00000113721), PDGFRA (ENSG00000134853), FLT3 (ENSG00000122025), PRKD3 (ENSG00000115825), PRKCI (ENSG00000163558), PRKCA (ENSG00000154229), PRKCG (...
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Q1.215
Q1
Is CD40 a druggable gene?
There are currently no approved drugs targeting CD40, but there are 11 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CD40 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_507', 'drugName': 'Sotigalimab', 'drugIsApproved': False, 'newLinkedTargets_string': 'CD40 (ENSG00000101017)', 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_2640', 'drugName': 'Lucatumumab', 'drugIsApproved': False, 'newLinkedTargets_string': 'CD40 (ENSG00000101017)', 'maxClini...
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Q1.122
Q1
Is BRD4 a druggable gene?
There are currently no approved drugs targeting BRD4, but there are 6 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%BRD4 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_866', 'drugName': 'Pelabresib', 'drugIsApproved': False, 'newLinkedTargets_string': 'BRD2 (ENSG00000204256), BRD4 (ENSG00000141867), BRDT (ENSG00000137948), BRD3 (ENSG00000169925)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_746', 'drugName': 'Apabetalone', 'drugIsApproved':...
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Q1.897
Q1
Is MMP2 a druggable gene?
There are currently no approved drugs targeting MMP2, but there are 3 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%MMP2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5860', 'drugName': 'Marimastat', 'drugIsApproved': False, 'newLinkedTargets_string': 'MMP9 (ENSG00000100985), MMP3 (ENSG00000149968), MMP7 (ENSG00000137673), MMP1 (ENSG00000196611), MMP2 (ENSG00000087245), MMP12 (ENSG00000262406)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_...
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