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Q58.1776
Q58
How many genes does the drug Ropinirole target and what are they?
There are 3 gene targets for the drug Ropinirole: DRD2, DRD3, and DRD4.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ropinirole%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1462', 'drugName': 'Ropinirole', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'DRD2 (ENSG00000149295), DRD3 (ENSG00000151577), DRD4 (ENSG00000069696)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 1997, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': ...
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Genetic Target
Q58.351
Q58
How many genes does the drug Raloxifene target and what are they?
ESR2 is the only gene target of drug Raloxifene.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%raloxifene%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1839', 'drugName': 'Raloxifene Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ESR2 (ENSG00000140009)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1997, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_5777', 'drugNa...
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Genetic Target
Q58.392
Q58
How many genes does the drug Aselizumab target and what are they?
The drug Aselizumab is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene SELL.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%aselizumab%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1635', 'drugName': 'Aselizumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'SELL (ENSG00000188404)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1033
Q58
How many genes does the drug Betamethasone target and what are they?
NR3C1 is the only gene target of drug Betamethasone.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%betamethasone%" OR LOWER(tradeNames_string) LIKE...
[{'UUID': 'DrugGeneTargets_v2_6021', 'drugName': 'Betamethasone Dipropionate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'NR3C1 (ENSG00000113580)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1975, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_2412', 'dru...
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Genetic Target
Q58.901
Q58
How many genes does the drug Tetrazepam target and what are they?
There are 16 gene targets for the drug Tetrazepam: GABRA1, GABRB2, GABRG2, GABRB3, GABRA4, GABRG3, GABRQ, GABRA3, GABRP, GABRD, GABRG1, GABRB1, GABRE, GABRA2, GABRA5, and GABRA6.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tetrazepam%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_3278', 'drugName': 'Tetrazepam', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089), GABRA3 (E...
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Genetic Target
Q58.835
Q58
How many genes does the drug Arsenic Trioxide target and what are they?
TXNRD1 is the only gene target of drug Arsenic Trioxide.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%arsenic trioxide%" OR LOWER(tradeNames_string) L...
[{'UUID': 'DrugGeneTargets_v2_975', 'drugName': 'Arsenic Trioxide', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'TXNRD1 (ENSG00000198431)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2000, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1894
Q58
How many genes does the drug Bay-1217389 target and what are they?
The drug Bay-1217389 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene TTK.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%bay-1217389%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_1430', 'drugName': 'Bay-1217389', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'TTK (ENSG00000112742)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drugIsApproved': False}]
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Genetic Target
Q58.481
Q58
How many genes does the drug Pateclizumab target and what are they?
The drug Pateclizumab is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene LTA.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%pateclizumab%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_937', 'drugName': 'Pateclizumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'LTA (ENSG00000226979)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1472
Q58
How many genes does the drug Belnacasan target and what are they?
The drug Belnacasan is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene CASP1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%belnacasan%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5967', 'drugName': 'Belnacasan', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CASP1 (ENSG00000137752)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1887
Q58
How many genes does the drug Pramlintide Acetate target and what are they?
There are 4 gene targets for the drug Pramlintide Acetate: CALCR, RAMP1, RAMP2, and RAMP3.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%pramlintide acetate%" OR LOWER(tradeNames_string...
[{'UUID': 'DrugGeneTargets_v2_2394', 'drugName': 'Pramlintide Acetate', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'CALCR (ENSG00000004948), RAMP1 (ENSG00000132329), RAMP2 (ENSG00000131477), RAMP3 (ENSG00000122679)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 2005, 'maxClinicalTrialPhase': 4, 'dru...
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Q58.1398
Q58
How many genes does the drug Obinutuzumab target and what are they?
MS4A1 is the only gene target of drug Obinutuzumab.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%obinutuzumab%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_847', 'drugName': 'Obinutuzumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'MS4A1 (ENSG00000156738)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2013, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.659
Q58
How many genes does the drug Thiothixene target and what are they?
There are 2 gene targets for the drug Thiothixene: DRD2 and HTR2A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%thiothixene%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_2625', 'drugName': 'Thiothixene', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'DRD2 (ENSG00000149295), HTR2A (ENSG00000102468)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1967, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_26...
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Genetic Target
Q58.175
Q58
How many genes does the drug Laropiprant target and what are they?
PTGDR is the only gene target of drug Laropiprant.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%laropiprant%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_1831', 'drugName': 'Laropiprant', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PTGDR (ENSG00000168229)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1159
Q58
How many genes does the drug Tazarotene target and what are they?
There are 3 gene targets for the drug Tazarotene: RARG, RARB, and RARA.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tazarotene%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5124', 'drugName': 'Tazarotene', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'RARG (ENSG00000172819), RARB (ENSG00000077092), RARA (ENSG00000131759)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 1997, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.39
Q58
How many genes does the drug Inotuzumab target and what are they?
CD22 is the only gene target of drug Inotuzumab.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%inotuzumab%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_6318', 'drugName': 'Inotuzumab Ozogamicin', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'CD22 (ENSG00000012124)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2017, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_1534', 'drugName': 'Ino...
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Q58.720
Q58
How many genes does the drug Fluphenazine Enanthate target and what are they?
DRD2 is the only gene target of drug Fluphenazine Enanthate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%fluphenazine enanthate%" OR LOWER(tradeNames_str...
[{'UUID': 'DrugGeneTargets_v2_905', 'drugName': 'Fluphenazine Enanthate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'DRD2 (ENSG00000149295)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1967, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.93
Q58
How many genes does the drug Ziprasidone target and what are they?
There are 3 gene targets for the drug Ziprasidone: HTR2A, DRD2, and HTR2C.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ziprasidone%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_1685', 'drugName': 'Ziprasidone', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HTR2A (ENSG00000102468), DRD2 (ENSG00000149295), HTR2C (ENSG00000147246)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 2001, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID...
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Q58.1937
Q58
How many genes does the drug Naloxone Hydrochloride target and what are they?
There are 3 gene targets for the drug Naloxone Hydrochloride: OPRK1, OPRD1, and OPRM1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%naloxone hydrochloride%" OR LOWER(tradeNames_str...
[{'UUID': 'DrugGeneTargets_v2_3927', 'drugName': 'Naloxone Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'OPRK1 (ENSG00000082556), OPRD1 (ENSG00000116329), OPRM1 (ENSG00000112038)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 1971, 'maxClinicalTrialPhase': 4, 'drugIsApproved': T...
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Q58.1215
Q58
How many genes does the drug Isoetharine target and what are they?
ADRB2 is the only gene target of drug Isoetharine.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%isoetharine%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_3508', 'drugName': 'Isoetharine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRB2 (ENSG00000169252)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1979, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_2925', 'drugName': 'Isoeth...
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Q58.882
Q58
How many genes does the drug Quinidine Polygalacturonate target and what are they?
There are 10 gene targets for the drug Quinidine Polygalacturonate: SCN1A, SCN5A, SCN4A, SCN7A, SCN2A, SCN9A, SCN3A, SCN11A, SCN8A, and SCN10A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%quinidine polygalacturonate%" OR LOWER(tradeName...
[{'UUID': 'DrugGeneTargets_v2_154', 'drugName': 'Quinidine Polygalacturonate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SCN1A (ENSG00000144285), SCN5A (ENSG00000183873), SCN4A (ENSG00000007314), SCN7A (ENSG00000136546), SCN2A (ENSG00000136531), SCN9A (ENSG00000169432), SCN3A (ENSG00000153253),...
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Q58.1353
Q58
How many genes does the drug Cinnarizine target and what are they?
There are 5 gene targets for the drug Cinnarizine: HRH1, CACNA1C, CACNA1S, CACNA1D, and CACNA1F.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%cinnarizine%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_4535', 'drugName': 'Cinnarizine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HRH1 (ENSG00000196639), CACNA1C (ENSG00000151067), CACNA1S (ENSG00000081248), CACNA1D (ENSG00000157388), CACNA1F (ENSG00000102001)', 'numberLinkedTargets': 5, 'yearOfFirstApproval': 0, 'max...
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Q58.1891
Q58
How many genes does the drug Omaveloxolone target and what are they?
The drug Omaveloxolone is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene NFE2L2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%omaveloxolone%" OR LOWER(tradeNames_string) LIKE...
[{'UUID': 'DrugGeneTargets_v2_6069', 'drugName': 'Omaveloxolone', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'NFE2L2 (ENSG00000116044)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Q58.1102
Q58
How many genes does the drug Evacetrapib target and what are they?
The drug Evacetrapib is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene CETP.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%evacetrapib%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_5790', 'drugName': 'Evacetrapib', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CETP (ENSG00000087237)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Q58.1165
Q58
How many genes does the drug Pimasertib target and what are they?
The drug Pimasertib is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 2 genes: MAP2K1 and MAP2K2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%pimasertib%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_3059', 'drugName': 'Pimasertib', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'MAP2K1 (ENSG00000169032), MAP2K2 (ENSG00000126934)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}, {'UUID': 'DrugGeneTargets_v2_30...
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Genetic Target
Q58.1365
Q58
How many genes does the drug Hexylcaine Hydrochloride target and what are they?
There are 10 gene targets for the drug Hexylcaine Hydrochloride: SCN1A, SCN5A, SCN4A, SCN7A, SCN2A, SCN9A, SCN3A, SCN11A, SCN8A, and SCN10A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%hexylcaine hydrochloride%" OR LOWER(tradeNames_s...
[{'UUID': 'DrugGeneTargets_v2_702', 'drugName': 'Hexylcaine Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SCN1A (ENSG00000144285), SCN5A (ENSG00000183873), SCN4A (ENSG00000007314), SCN7A (ENSG00000136546), SCN2A (ENSG00000136531), SCN9A (ENSG00000169432), SCN3A (ENSG00000153253), SC...
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Genetic Target
Q58.1959
Q58
How many genes does the drug Norepinephrine Bitartrate target and what are they?
There are 9 gene targets for the drug Norepinephrine Bitartrate: ADRA1A, ADRA2A, ADRB1, ADRB2, ADRA2C, ADRA1D, ADRA1B, ADRA2B, and ADRB3.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%norepinephrine bitartrate%" OR LOWER(tradeNames_...
[{'UUID': 'DrugGeneTargets_v2_1843', 'drugName': 'Norepinephrine Bitartrate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRA1A (ENSG00000120907), ADRA2A (ENSG00000150594), ADRB1 (ENSG00000043591), ADRB2 (ENSG00000169252), ADRA2C (ENSG00000184160), ADRA1D (ENSG00000171873), ADRA1B (ENSG000001702...
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Genetic Target
Q58.505
Q58
How many genes does the drug Gc1118 target and what are they?
The drug Gc1118 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene EGFR.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%gc1118%" OR LOWER(tradeNames_string) LIKE "%gc11...
[{'UUID': 'DrugGeneTargets_v2_6070', 'drugName': 'Gc1118', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'EGFR (ENSG00000146648)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.342
Q58
How many genes does the drug Tepotinib Hydrochloride target and what are they?
MET is the only gene target of drug Tepotinib Hydrochloride.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tepotinib hydrochloride%" OR LOWER(tradeNames_st...
[{'UUID': 'DrugGeneTargets_v2_1908', 'drugName': 'Tepotinib Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'MET (ENSG00000105976)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2021, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1198
Q58
How many genes does the drug Tretinoin target and what are they?
There are 3 gene targets for the drug Tretinoin: RARG, RARB, and RARA.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tretinoin%" OR LOWER(tradeNames_string) LIKE "%t...
[{'UUID': 'DrugGeneTargets_v2_5360', 'drugName': 'Tretinoin', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'RARG (ENSG00000172819), RARB (ENSG00000077092), RARA (ENSG00000131759)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 1971, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': '...
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Genetic Target
Q58.29
Q58
How many genes does the drug Testosterone Enanthate target and what are they?
AR is the only gene target of drug Testosterone Enanthate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%testosterone enanthate%" OR LOWER(tradeNames_str...
[{'UUID': 'DrugGeneTargets_v2_5959', 'drugName': 'Testosterone Enanthate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'AR (ENSG00000169083)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1953, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1227
Q58
How many genes does the drug Lapatinib target and what are they?
There are 2 gene targets for the drug Lapatinib: EGFR and ERBB2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%lapatinib%" OR LOWER(tradeNames_string) LIKE "%l...
[{'UUID': 'DrugGeneTargets_v2_2161', 'drugName': 'Lapatinib Ditosylate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'EGFR (ENSG00000146648), ERBB2 (ENSG00000141736)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2007, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTarg...
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Genetic Target
Q58.1434
Q58
How many genes does the drug Glpg-1205 target and what are they?
The drug Glpg-1205 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene GPR84.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%glpg-1205%" OR LOWER(tradeNames_string) LIKE "%g...
[{'UUID': 'DrugGeneTargets_v2_1454', 'drugName': 'Glpg-1205', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GPR84 (ENSG00000139572)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1954
Q58
How many genes does the drug Apolizumab target and what are they?
The drug Apolizumab is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 4 genes: HLA-DRB3, HLA-DRB5, HLA-DRB1, and HLA-DRB4.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%apolizumab%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_363', 'drugName': 'Apolizumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'HLA-DRB3 (ENSG00000231679), HLA-DRB5 (ENSG00000198502), HLA-DRB1 (ENSG00000196126), HLA-DRB4 (ENSG00000231021)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'dru...
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Genetic Target
Q58.954
Q58
How many genes does the drug Protriptyline Hydrochloride target and what are they?
There are 2 gene targets for the drug Protriptyline Hydrochloride: SLC6A2 and SLC6A4.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%protriptyline hydrochloride%" OR LOWER(tradeName...
[{'UUID': 'DrugGeneTargets_v2_5492', 'drugName': 'Protriptyline Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SLC6A2 (ENSG00000103546), SLC6A4 (ENSG00000108576)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1967, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'Dr...
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Genetic Target
Q58.172
Q58
How many genes does the drug Terodiline target and what are they?
There are 31 gene targets for the drug Terodiline: CHRM3, CHRM4, CHRM1, CHRM2, CHRM5, CACNA1H, CACNA2D1, CACNA1C, CACNA2D3, CACNA1S, CACNA2D2, CACNA1D, CACNA1A, CACNA1B, CACNA1G, CACNA2D4, CACNA1I, CACNA1F, CACNA1E, CACNB4, CACNB2, CACNB1, CACNB3, CACNG7, CACNG5, CACNG2, CACNG4, CACNG8, CACNG3, CACNG6, and CACNG1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%terodiline%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_6292', 'drugName': 'Terodiline', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CHRM3 (ENSG00000133019), CHRM4 (ENSG00000180720), CHRM1 (ENSG00000168539), CHRM2 (ENSG00000181072), CHRM5 (ENSG00000184984), CACNA1H (ENSG00000196557), CACNA2D1 (ENSG00000153956), CACNA1C (E...
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Genetic Target
Q58.1406
Q58
How many genes does the drug Ascrinvacumab target and what are they?
The drug Ascrinvacumab is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene ACVRL1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ascrinvacumab%" OR LOWER(tradeNames_string) LIKE...
[{'UUID': 'DrugGeneTargets_v2_526', 'drugName': 'Ascrinvacumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'ACVRL1 (ENSG00000139567)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1207
Q58
How many genes does the drug Benzydamine Hydrochloride target and what are they?
There are 2 gene targets for the drug Benzydamine Hydrochloride: PTGS2 and PTGS1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%benzydamine hydrochloride%" OR LOWER(tradeNames_...
[{'UUID': 'DrugGeneTargets_v2_3576', 'drugName': 'Benzydamine Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PTGS2 (ENSG00000073756), PTGS1 (ENSG00000095303)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1263
Q58
How many genes does the drug Galantamine target and what are they?
ACHE is the only gene target of drug Galantamine.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%galantamine%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_1632', 'drugName': 'Galantamine Hydrobromide', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ACHE (ENSG00000087085)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2001, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_3143', 'drugNa...
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Genetic Target
Q58.1400
Q58
How many genes does the drug Sotalol Hydrochloride target and what are they?
There are 3 gene targets for the drug Sotalol Hydrochloride: ADRB1, KCNH2, and ADRB2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%sotalol hydrochloride%" OR LOWER(tradeNames_stri...
[{'UUID': 'DrugGeneTargets_v2_4569', 'drugName': 'Sotalol Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRB1 (ENSG00000043591), KCNH2 (ENSG00000055118), ADRB2 (ENSG00000169252)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 1992, 'maxClinicalTrialPhase': 4, 'drugIsApproved': Tr...
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Genetic Target
Q58.920
Q58
How many genes does the drug Tirasemtiv target and what are they?
The drug Tirasemtiv is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 3 genes: TNNI2, TNNT3, and TNNC2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tirasemtiv%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_6283', 'drugName': 'Tirasemtiv', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'TNNI2 (ENSG00000130598), TNNT3 (ENSG00000130595), TNNC2 (ENSG00000101470)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.497
Q58
How many genes does the drug Fluocinonide target and what are they?
NR3C1 is the only gene target of drug Fluocinonide.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%fluocinonide%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_4918', 'drugName': 'Fluocinonide', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'NR3C1 (ENSG00000113580)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1971, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.962
Q58
How many genes does the drug Ruxolitinib target and what are they?
There are 2 gene targets for the drug Ruxolitinib: JAK1 and JAK2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ruxolitinib%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_1728', 'drugName': 'Ruxolitinib Phosphate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'JAK1 (ENSG00000162434), JAK2 (ENSG00000096968)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2011, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTarg...
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Genetic Target
Q58.1106
Q58
How many genes does the drug Trospium target and what are they?
There are 2 gene targets for the drug Trospium: CHRM3 and CHRM2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%trospium%" OR LOWER(tradeNames_string) LIKE "%tr...
[{'UUID': 'DrugGeneTargets_v2_6081', 'drugName': 'Trospium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CHRM3 (ENSG00000133019), CHRM2 (ENSG00000181072)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2004, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_6080...
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Genetic Target
Q58.1041
Q58
How many genes does the drug Aclidinium Bromide target and what are they?
CHRM3 is the only gene target of drug Aclidinium Bromide.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%aclidinium bromide%" OR LOWER(tradeNames_string)...
[{'UUID': 'DrugGeneTargets_v2_6136', 'drugName': 'Aclidinium Bromide', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CHRM3 (ENSG00000133019)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2012, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.594
Q58
How many genes does the drug Oliceridine target and what are they?
OPRM1 is the only gene target of drug Oliceridine.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%oliceridine%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_4900', 'drugName': 'Oliceridine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'OPRM1 (ENSG00000112038)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2020, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.757
Q58
How many genes does the drug Tofacitinib target and what are they?
There are 4 gene targets for the drug Tofacitinib: JAK3, JAK1, JAK2, and TYK2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tofacitinib%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_4953', 'drugName': 'Tofacitinib', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'JAK3 (ENSG00000105639), JAK1 (ENSG00000162434), JAK2 (ENSG00000096968), TYK2 (ENSG00000105397)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 2012, 'maxClinicalTrialPhase': 4, 'drugIsAp...
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Genetic Target
Q58.664
Q58
How many genes does the drug Tolbutamide target and what are they?
There are 2 gene targets for the drug Tolbutamide: KCNJ11 and ABCC8.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tolbutamide%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_427', 'drugName': 'Tolbutamide', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'KCNJ11 (ENSG00000187486), ABCC8 (ENSG00000006071)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1961, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_3...
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Genetic Target
Q58.237
Q58
How many genes does the drug Minaprine target and what are they?
There are 8 gene targets for the drug Minaprine: MAOA, DRD2, DRD1, HTR2B, HTR2A, HTR2C, CHRM1, and ACHE.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%minaprine%" OR LOWER(tradeNames_string) LIKE "%m...
[{'UUID': 'DrugGeneTargets_v2_4771', 'drugName': 'Minaprine Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'DRD2 (ENSG00000149295), DRD1 (ENSG00000184845), CHRM1 (ENSG00000168539), ACHE (ENSG00000087085), MAOA (ENSG00000189221), HTR2B (ENSG00000135914), HTR2A (ENSG00000102468), HTR2C ...
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Genetic Target
Q58.739
Q58
How many genes does the drug Bromodiphenhydramine Hydrochloride target and what are they?
HRH1 is the only gene target of drug Bromodiphenhydramine Hydrochloride.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%bromodiphenhydramine hydrochloride%" OR LOWER(tr...
[{'UUID': 'DrugGeneTargets_v2_1015', 'drugName': 'Bromodiphenhydramine Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HRH1 (ENSG00000196639)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1954, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1989
Q58
How many genes does the drug Heparin Calcium target and what are they?
SERPINC1 is the only gene target of drug Heparin Calcium.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%heparin calcium%" OR LOWER(tradeNames_string) LI...
[{'UUID': 'DrugGeneTargets_v2_843', 'drugName': 'Heparin Calcium', 'drugMolecularType': 'Oligosaccharide', 'newLinkedTargets_string': 'SERPINC1 (ENSG00000117601)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1982, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1633
Q58
How many genes does the drug Givosiran Sodium target and what are they?
ALAS1 is the only gene target of drug Givosiran Sodium.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%givosiran sodium%" OR LOWER(tradeNames_string) L...
[{'UUID': 'DrugGeneTargets_v2_5803', 'drugName': 'Givosiran Sodium', 'drugMolecularType': 'Oligonucleotide', 'newLinkedTargets_string': 'ALAS1 (ENSG00000023330)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2019, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1166
Q58
How many genes does the drug Tasimelteon target and what are they?
There are 2 gene targets for the drug Tasimelteon: MTNR1A and MTNR1B.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tasimelteon%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_6185', 'drugName': 'Tasimelteon', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'MTNR1A (ENSG00000168412), MTNR1B (ENSG00000134640)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2014, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1471
Q58
How many genes does the drug Gz-389988 target and what are they?
The drug Gz-389988 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene NTRK1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%gz-389988%" OR LOWER(tradeNames_string) LIKE "%g...
[{'UUID': 'DrugGeneTargets_v2_4929', 'drugName': 'Gz-389988', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'NTRK1 (ENSG00000198400)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1913
Q58
How many genes does the drug Buprenorphine target and what are they?
There are 2 gene targets for the drug Buprenorphine: OPRM1 and OPRK1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%buprenorphine%" OR LOWER(tradeNames_string) LIKE...
[{'UUID': 'DrugGeneTargets_v2_3501', 'drugName': 'Buprenorphine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'OPRM1 (ENSG00000112038), OPRK1 (ENSG00000082556)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1981, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2...
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Genetic Target
Q58.1628
Q58
How many genes does the drug Epacadostat target and what are they?
The drug Epacadostat is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene IDO1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%epacadostat%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_856', 'drugName': 'Epacadostat', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'IDO1 (ENSG00000131203)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.943
Q58
How many genes does the drug Guselkumab target and what are they?
There are 2 gene targets for the drug Guselkumab: IL12B and IL23A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%guselkumab%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2147', 'drugName': 'Guselkumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'IL12B (ENSG00000113302), IL23A (ENSG00000110944)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2017, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1219
Q58
How many genes does the drug Midodrine Hydrochloride target and what are they?
There are 3 gene targets for the drug Midodrine Hydrochloride: ADRA1A, ADRA1D, and ADRA1B.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%midodrine hydrochloride%" OR LOWER(tradeNames_st...
[{'UUID': 'DrugGeneTargets_v2_5117', 'drugName': 'Midodrine Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRA1A (ENSG00000120907), ADRA1D (ENSG00000171873), ADRA1B (ENSG00000170214)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 1996, 'maxClinicalTrialPhase': 4, 'drugIsApproved...
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Genetic Target
Q58.1074
Q58
How many genes does the drug Elimusertib target and what are they?
The drug Elimusertib is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene ATR.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%elimusertib%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_4961', 'drugName': 'Elimusertib', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ATR (ENSG00000175054)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drugIsApproved': False}]
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Genetic Target
Q58.111
Q58
How many genes does the drug Theophylline Glycinate target and what are they?
There are 10 gene targets for the drug Theophylline Glycinate: ADORA1, ADORA2B, ADORA3, ADORA2A, PDE4A, PDE4D, PDE4B, PDE4C, PDE3A, and PDE3B.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%theophylline glycinate%" OR LOWER(tradeNames_str...
[{'UUID': 'DrugGeneTargets_v2_2662', 'drugName': 'Theophylline Glycinate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADORA1 (ENSG00000163485), ADORA2B (ENSG00000170425), ADORA3 (ENSG00000282608), ADORA2A (ENSG00000128271), PDE4A (ENSG00000065989), PDE4D (ENSG00000113448), PDE4B (ENSG00000184588...
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Genetic Target
Q58.1944
Q58
How many genes does the drug Levosimendan target and what are they?
The drug Levosimendan is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 5 genes: PDE3A, PDE3B, TNNC1, TNNI3, and TNNT2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%levosimendan%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_2198', 'drugName': 'Levosimendan', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PDE3A (ENSG00000172572), PDE3B (ENSG00000152270), TNNC1 (ENSG00000114854), TNNI3 (ENSG00000129991), TNNT2 (ENSG00000118194)', 'numberLinkedTargets': 5, 'yearOfFirstApproval': 0, 'maxClinic...
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Genetic Target
Q58.574
Q58
How many genes does the drug Carbetocin target and what are they?
OXTR is the only gene target of drug Carbetocin.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%carbetocin%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_6062', 'drugName': 'Carbetocin', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'OXTR (ENSG00000180914)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1177
Q58
How many genes does the drug Ispinesib target and what are they?
The drug Ispinesib is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene KIF11.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ispinesib%" OR LOWER(tradeNames_string) LIKE "%i...
[{'UUID': 'DrugGeneTargets_v2_3893', 'drugName': 'Ispinesib', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'KIF11 (ENSG00000138160)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1184
Q58
How many genes does the drug Insulin Zinc Susp Extended Recombinant Human target and what are they?
INSR is the only gene target of drug Insulin Zinc Susp Extended Recombinant Human.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%insulin zinc susp extended recombinant human%" O...
[{'UUID': 'DrugGeneTargets_v2_4713', 'drugName': 'Insulin Zinc Susp Extended Recombinant Human', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'INSR (ENSG00000171105)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1987, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.897
Q58
How many genes does the drug Balsalazide Disodium target and what are they?
There are 4 gene targets for the drug Balsalazide Disodium: PPARG, PTGS2, PTGS1, and ALOX5.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%balsalazide disodium%" OR LOWER(tradeNames_strin...
[{'UUID': 'DrugGeneTargets_v2_1296', 'drugName': 'Balsalazide Disodium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PPARG (ENSG00000132170), PTGS2 (ENSG00000073756), PTGS1 (ENSG00000095303), ALOX5 (ENSG00000012779)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 2000, 'maxClinicalTrialPhase':...
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Genetic Target
Q58.956
Q58
How many genes does the drug Etomidate target and what are they?
There are 16 gene targets for the drug Etomidate: GABRA1, GABRB2, GABRG2, GABRB3, GABRA4, GABRG3, GABRQ, GABRA3, GABRP, GABRD, GABRG1, GABRB1, GABRE, GABRA2, GABRA5, and GABRA6.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%etomidate%" OR LOWER(tradeNames_string) LIKE "%e...
[{'UUID': 'DrugGeneTargets_v2_5114', 'drugName': 'Etomidate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089), GABRA3 (EN...
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Genetic Target
Q58.1057
Q58
How many genes does the drug Naluzotan target and what are they?
The drug Naluzotan is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene HTR1A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%naluzotan%" OR LOWER(tradeNames_string) LIKE "%n...
[{'UUID': 'DrugGeneTargets_v2_5444', 'drugName': 'Naluzotan', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HTR1A (ENSG00000178394)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.1354
Q58
How many genes does the drug Saxagliptin Hydrochloride target and what are they?
DPP4 is the only gene target of drug Saxagliptin Hydrochloride.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%saxagliptin hydrochloride%" OR LOWER(tradeNames_...
[{'UUID': 'DrugGeneTargets_v2_2239', 'drugName': 'Saxagliptin Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'DPP4 (ENSG00000197635)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2009, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1373
Q58
How many genes does the drug Follitropin Alfa target and what are they?
FSHR is the only gene target of drug Follitropin Alfa.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%follitropin alfa%" OR LOWER(tradeNames_string) L...
[{'UUID': 'DrugGeneTargets_v2_2306', 'drugName': 'Corifollitropin Alfa', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'FSHR (ENSG00000170820)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_206', 'drugName': 'Follitrop...
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Genetic Target
Q58.1448
Q58
How many genes does the drug M195 target and what are they?
The drug M195 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene CD33.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%m195%" OR LOWER(tradeNames_string) LIKE "%m195%"...
[{'UUID': 'DrugGeneTargets_v2_1520', 'drugName': 'Lintuzumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'CD33 (ENSG00000105383)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}, {'UUID': 'DrugGeneTargets_v2_6193', 'drugName': 'M195', 'drugMole...
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Genetic Target
Q58.891
Q58
How many genes does the drug Giloralimab target and what are they?
The drug Giloralimab is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene CD40.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%giloralimab%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_2944', 'drugName': 'Giloralimab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'CD40 (ENSG00000101017)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1673
Q58
How many genes does the drug Ataciguat target and what are they?
The drug Ataciguat is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 4 genes: GUCY1B1, GUCY1B2, GUCY1A2, and GUCY1A1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ataciguat%" OR LOWER(tradeNames_string) LIKE "%a...
[{'UUID': 'DrugGeneTargets_v2_3371', 'drugName': 'Ataciguat', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GUCY1B1 (ENSG00000061918), GUCY1B2 (ENSG00000123201), GUCY1A2 (ENSG00000152402), GUCY1A1 (ENSG00000164116)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'd...
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Genetic Target
Q58.857
Q58
How many genes does the drug Trx-1 target and what are they?
The drug Trx-1 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene CD4.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%trx-1%" OR LOWER(tradeNames_string) LIKE "%trx-1...
[{'UUID': 'DrugGeneTargets_v2_4140', 'drugName': 'Trx-1', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'CD4 (ENSG00000010610)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.741
Q58
How many genes does the drug Zolpidem Tartrate target and what are they?
There are 3 gene targets for the drug Zolpidem Tartrate: GABRA1, GABRG2, and GABRB1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%zolpidem tartrate%" OR LOWER(tradeNames_string) ...
[{'UUID': 'DrugGeneTargets_v2_5904', 'drugName': 'Zolpidem Tartrate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRG2 (ENSG00000113327), GABRB1 (ENSG00000163288)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 1992, 'maxClinicalTrialPhase': 4, 'drugIsApproved': Tru...
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Genetic Target
Q58.724
Q58
How many genes does the drug Imarikiren target and what are they?
The drug Imarikiren is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene REN.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%imarikiren%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_3903', 'drugName': 'Imarikiren Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'REN (ENSG00000143839)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}, {'UUID': 'DrugGeneTargets_v2_5101', 'drugName'...
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Genetic Target
Q58.460
Q58
How many genes does the drug Dibucaine Hydrochloride target and what are they?
There are 2 gene targets for the drug Dibucaine Hydrochloride: SCN5A and SCN10A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%dibucaine hydrochloride%" OR LOWER(tradeNames_st...
[{'UUID': 'DrugGeneTargets_v2_6109', 'drugName': 'Dibucaine Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SCN5A (ENSG00000183873), SCN10A (ENSG00000185313)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1982, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGen...
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Genetic Target
Q58.267
Q58
How many genes does the drug Propantheline Bromide target and what are they?
There are 3 gene targets for the drug Propantheline Bromide: CHRM3, CHRM1, and CHRM2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%propantheline bromide%" OR LOWER(tradeNames_stri...
[{'UUID': 'DrugGeneTargets_v2_4309', 'drugName': 'Propantheline Bromide', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CHRM3 (ENSG00000133019), CHRM1 (ENSG00000168539), CHRM2 (ENSG00000181072)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 1953, 'maxClinicalTrialPhase': 4, 'drugIsApproved': Tr...
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Genetic Target
Q58.78
Q58
How many genes does the drug Afamelanotide target and what are they?
MC1R is the only gene target of drug Afamelanotide.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%afamelanotide%" OR LOWER(tradeNames_string) LIKE...
[{'UUID': 'DrugGeneTargets_v2_6266', 'drugName': 'Afamelanotide', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'MC1R (ENSG00000258839)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2019, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_5286', 'drugName': 'Afamelanotid...
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Genetic Target
Q58.1785
Q58
How many genes does the drug Relenopride target and what are they?
The drug Relenopride is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene HTR4.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%relenopride%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_3693', 'drugName': 'Relenopride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HTR4 (ENSG00000164270)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.450
Q58
How many genes does the drug Fenoprofen target and what are they?
There are 2 gene targets for the drug Fenoprofen: PTGS2 and PTGS1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%fenoprofen%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_4670', 'drugName': 'Fenoprofen', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PTGS2 (ENSG00000073756), PTGS1 (ENSG00000095303)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1976, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_30...
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Genetic Target
Q58.401
Q58
How many genes does the drug Olodaterol Hydrochloride target and what are they?
ADRB2 is the only gene target of drug Olodaterol Hydrochloride.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%olodaterol hydrochloride%" OR LOWER(tradeNames_s...
[{'UUID': 'DrugGeneTargets_v2_5322', 'drugName': 'Olodaterol Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRB2 (ENSG00000169252)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2014, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.179
Q58
How many genes does the drug Tocainide target and what are they?
There are 10 gene targets for the drug Tocainide: SCN1A, SCN5A, SCN4A, SCN7A, SCN2A, SCN9A, SCN3A, SCN11A, SCN8A, and SCN10A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tocainide%" OR LOWER(tradeNames_string) LIKE "%t...
[{'UUID': 'DrugGeneTargets_v2_5269', 'drugName': 'Tocainide', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SCN1A (ENSG00000144285), SCN5A (ENSG00000183873), SCN4A (ENSG00000007314), SCN7A (ENSG00000136546), SCN2A (ENSG00000136531), SCN9A (ENSG00000169432), SCN3A (ENSG00000153253), SCN11A (ENSG0000...
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Genetic Target
Q58.1051
Q58
How many genes does the drug Sipuleucel-T target and what are they?
ACP3 is the only gene target of drug Sipuleucel-T.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%sipuleucel-t%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_2303', 'drugName': 'Sipuleucel-T', 'drugMolecularType': 'Cell', 'newLinkedTargets_string': 'ACP3 (ENSG00000014257)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1737
Q58
How many genes does the drug Bimagrumab target and what are they?
The drug Bimagrumab is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene ACVR2B.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%bimagrumab%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_299', 'drugName': 'Bimagrumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'ACVR2B (ENSG00000114739)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.1609
Q58
How many genes does the drug Mepolizumab target and what are they?
IL5 is the only gene target of drug Mepolizumab.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%mepolizumab%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_1703', 'drugName': 'Mepolizumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'IL5 (ENSG00000113525)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2015, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1869
Q58
How many genes does the drug Ce-326597 target and what are they?
The drug Ce-326597 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene CCKAR.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ce-326597%" OR LOWER(tradeNames_string) LIKE "%c...
[{'UUID': 'DrugGeneTargets_v2_2827', 'drugName': 'Ce-326597', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CCKAR (ENSG00000163394)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.602
Q58
How many genes does the drug Maraviroc target and what are they?
CCR5 is the only gene target of drug Maraviroc.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%maraviroc%" OR LOWER(tradeNames_string) LIKE "%m...
[{'UUID': 'DrugGeneTargets_v2_3537', 'drugName': 'Maraviroc', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CCR5 (ENSG00000160791)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2007, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.63
Q58
How many genes does the drug Ave-9940 target and what are they?
The drug Ave-9940 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene MAPK14.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ave-9940%" OR LOWER(tradeNames_string) LIKE "%av...
[{'UUID': 'DrugGeneTargets_v2_1974', 'drugName': 'Ave-9940', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'MAPK14 (ENSG00000112062)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drugIsApproved': False}]
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Genetic Target
Q58.1309
Q58
How many genes does the drug Upadacitinib target and what are they?
There are 4 gene targets for the drug Upadacitinib: JAK3, JAK1, JAK2, and TYK2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%upadacitinib%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_4653', 'drugName': 'Upadacitinib', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'JAK3 (ENSG00000105639), JAK1 (ENSG00000162434), JAK2 (ENSG00000096968), TYK2 (ENSG00000105397)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 2019, 'maxClinicalTrialPhase': 4, 'drugIsA...
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Genetic Target
Q58.879
Q58
How many genes does the drug Pegvisomant target and what are they?
GHR is the only gene target of drug Pegvisomant.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%pegvisomant%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_1805', 'drugName': 'Pegvisomant', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'GHR (ENSG00000112964)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2003, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1491
Q58
How many genes does the drug Volanesorsen target and what are they?
APOC3 is the only gene target of drug Volanesorsen.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%volanesorsen%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_2601', 'drugName': 'Volanesorsen', 'drugMolecularType': 'Oligonucleotide', 'newLinkedTargets_string': 'APOC3 (ENSG00000110245)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_3223', 'drugName': 'Volanes...
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Genetic Target
Q58.1880
Q58
How many genes does the drug Insulin Pork target and what are they?
INSR is the only gene target of drug Insulin Pork.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%insulin pork%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_5466', 'drugName': 'Insulin Pork', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'INSR (ENSG00000171105)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1966, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.282
Q58
How many genes does the drug Echothiophate Iodide target and what are they?
ACHE is the only gene target of drug Echothiophate Iodide.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%echothiophate iodide%" OR LOWER(tradeNames_strin...
[{'UUID': 'DrugGeneTargets_v2_2129', 'drugName': 'Echothiophate Iodide', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ACHE (ENSG00000087085)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1960, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.37
Q58
How many genes does the drug Elinogrel target and what are they?
The drug Elinogrel is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene P2RY12.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%elinogrel%" OR LOWER(tradeNames_string) LIKE "%e...
[{'UUID': 'DrugGeneTargets_v2_3842', 'drugName': 'Elinogrel', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'P2RY12 (ENSG00000169313)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1517
Q58
How many genes does the drug Amlodipine Benzoate target and what are they?
There are 4 gene targets for the drug Amlodipine Benzoate: CACNA1C, CACNA1S, CACNA1D, and CACNA1F.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%amlodipine benzoate%" OR LOWER(tradeNames_string...
[{'UUID': 'DrugGeneTargets_v2_5167', 'drugName': 'Amlodipine Benzoate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CACNA1C (ENSG00000151067), CACNA1S (ENSG00000081248), CACNA1D (ENSG00000157388), CACNA1F (ENSG00000102001)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 2019, 'maxClinicalTrial...
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Genetic Target
Q58.669
Q58
How many genes does the drug Codeine Polistirex target and what are they?
There are 3 gene targets for the drug Codeine Polistirex: OPRK1, OPRD1, and OPRM1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%codeine polistirex%" OR LOWER(tradeNames_string)...
[{'UUID': 'DrugGeneTargets_v2_494', 'drugName': 'Codeine Polistirex', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'OPRK1 (ENSG00000082556), OPRD1 (ENSG00000116329), OPRM1 (ENSG00000112038)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 1985, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1829
Q58
How many genes does the drug Atezolizumab target and what are they?
CD274 is the only gene target of drug Atezolizumab.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%atezolizumab%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_449', 'drugName': 'Atezolizumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'CD274 (ENSG00000120217)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2016, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1446
Q58
How many genes does the drug Ketorolac Tromethamine target and what are they?
There are 2 gene targets for the drug Ketorolac Tromethamine: PTGS2 and PTGS1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ketorolac tromethamine%" OR LOWER(tradeNames_str...
[{'UUID': 'DrugGeneTargets_v2_2258', 'drugName': 'Ketorolac Tromethamine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PTGS2 (ENSG00000073756), PTGS1 (ENSG00000095303)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1989, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.986
Q58
How many genes does the drug Tafamidis target and what are they?
TTR is the only gene target of drug Tafamidis.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tafamidis%" OR LOWER(tradeNames_string) LIKE "%t...
[{'UUID': 'DrugGeneTargets_v2_8', 'drugName': 'Tafamidis Meglumine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'TTR (ENSG00000118271)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2019, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_3770', 'drugName': 'Taf...
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Genetic Target
Q58.1572
Q58
How many genes does the drug Vantictumab target and what are they?
The drug Vantictumab is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 5 genes: FZD2, FZD7, FZD1, FZD5, and FZD8.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%vantictumab%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_5828', 'drugName': 'Vantictumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'FZD2 (ENSG00000180340), FZD7 (ENSG00000155760), FZD1 (ENSG00000157240), FZD5 (ENSG00000163251), FZD8 (ENSG00000177283)', 'numberLinkedTargets': 5, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase...
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Genetic Target
Q58.745
Q58
How many genes does the drug Prabotulinumtoxin A target and what are they?
SNAP25 is the only gene target of drug Prabotulinumtoxin A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%prabotulinumtoxin a%" OR LOWER(tradeNames_string...
[{'UUID': 'DrugGeneTargets_v2_2511', 'drugName': 'Prabotulinumtoxin A', 'drugMolecularType': 'Unknown', 'newLinkedTargets_string': 'SNAP25 (ENSG00000132639)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2019, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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