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Q58.1160
Q58
How many genes does the drug Docetaxel target and what are they?
There are 15 gene targets for the drug Docetaxel: TUBB4B, TUBB1, TUBA3C, TUBA4A, TUBB3, TUBA1A, TUBB4A, TUBB8, TUBB, TUBA1B, TUBA1C, TUBA3E, TUBB2A, TUBB2B, and TUBB6.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%docetaxel%" OR LOWER(tradeNames_string) LIKE "%d...
[{'UUID': 'DrugGeneTargets_v2_1267', 'drugName': 'Docetaxel', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'TUBB4B (ENSG00000188229), TUBB1 (ENSG00000101162), TUBA3C (ENSG00000198033), TUBA4A (ENSG00000127824), TUBB3 (ENSG00000258947), TUBA1A (ENSG00000167552), TUBB4A (ENSG00000104833), TUBB8 (ENSG...
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Genetic Target
Q58.797
Q58
How many genes does the drug Sapropterin Dihydrochloride target and what are they?
PAH is the only gene target of drug Sapropterin Dihydrochloride.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%sapropterin dihydrochloride%" OR LOWER(tradeName...
[{'UUID': 'DrugGeneTargets_v2_4864', 'drugName': 'Sapropterin Dihydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PAH (ENSG00000171759)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2007, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.119
Q58
How many genes does the drug Benztropine Mesylate target and what are they?
CHRM1 is the only gene target of drug Benztropine Mesylate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%benztropine mesylate%" OR LOWER(tradeNames_strin...
[{'UUID': 'DrugGeneTargets_v2_321', 'drugName': 'Benztropine Mesylate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CHRM1 (ENSG00000168539)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1954, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.747
Q58
How many genes does the drug Cholecalciferol target and what are they?
VDR is the only gene target of drug Cholecalciferol.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%cholecalciferol%" OR LOWER(tradeNames_string) LI...
[{'UUID': 'DrugGeneTargets_v2_4543', 'drugName': 'Alfacalcidol', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'VDR (ENSG00000111424)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_4232', 'drugName': 'Calcitriol...
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Genetic Target
Q58.1691
Q58
How many genes does the drug Gaboxadol target and what are they?
The drug Gaboxadol is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 9 genes: GABRA1, GABRB2, GABRB3, GABRA4, GABRA3, GABRB1, GABRA2, GABRA5, and GABRA6.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%gaboxadol%" OR LOWER(tradeNames_string) LIKE "%g...
[{'UUID': 'DrugGeneTargets_v2_3615', 'drugName': 'Gaboxadol', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRA3 (ENSG00000011677), GABRB1 (ENSG00000163288), GABRA2 (ENSG00000151834), GABRA5 (E...
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Genetic Target
Q58.1090
Q58
How many genes does the drug Pimavanserin Tartrate target and what are they?
HTR2A is the only gene target of drug Pimavanserin Tartrate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%pimavanserin tartrate%" OR LOWER(tradeNames_stri...
[{'UUID': 'DrugGeneTargets_v2_5097', 'drugName': 'Pimavanserin Tartrate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HTR2A (ENSG00000102468)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2016, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.837
Q58
How many genes does the drug Sildenafil Citrate target and what are they?
PDE5A is the only gene target of drug Sildenafil Citrate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%sildenafil citrate%" OR LOWER(tradeNames_string)...
[{'UUID': 'DrugGeneTargets_v2_4134', 'drugName': 'Sildenafil Citrate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PDE5A (ENSG00000138735)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1998, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.122
Q58
How many genes does the drug Proglumide target and what are they?
There are 2 gene targets for the drug Proglumide: CCKBR and CCKAR.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%proglumide%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5575', 'drugName': 'Proglumide', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CCKBR (ENSG00000110148), CCKAR (ENSG00000163394)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.663
Q58
How many genes does the drug Zonisamide target and what are they?
There are 10 gene targets for the drug Zonisamide: SCN1A, SCN5A, SCN4A, SCN7A, SCN2A, SCN9A, SCN3A, SCN11A, SCN8A, and SCN10A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%zonisamide%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_315', 'drugName': 'Zonisamide', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SCN1A (ENSG00000144285), SCN5A (ENSG00000183873), SCN4A (ENSG00000007314), SCN7A (ENSG00000136546), SCN2A (ENSG00000136531), SCN9A (ENSG00000169432), SCN3A (ENSG00000153253), SCN11A (ENSG0000...
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Genetic Target
Q58.1908
Q58
How many genes does the drug Atomoxetine target and what are they?
SLC6A2 is the only gene target of drug Atomoxetine.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%atomoxetine%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_4562', 'drugName': 'Atomoxetine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SLC6A2 (ENSG00000103546)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2002, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_1334', 'drugName': 'Atomo...
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Genetic Target
Q58.642
Q58
How many genes does the drug Indomethacin target and what are they?
There are 2 gene targets for the drug Indomethacin: PTGS2 and PTGS1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%indomethacin%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_3165', 'drugName': 'Indomethacin', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PTGS2 (ENSG00000073756), PTGS1 (ENSG00000095303)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1965, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_...
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Genetic Target
Q58.374
Q58
How many genes does the drug Gsk-2245035 target and what are they?
The drug Gsk-2245035 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene TLR7.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%gsk-2245035%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_4576', 'drugName': 'Gsk-2245035', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'TLR7 (ENSG00000196664)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.271
Q58
How many genes does the drug Deserpidine target and what are they?
SLC18A2 is the only gene target of drug Deserpidine.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%deserpidine%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_4303', 'drugName': 'Deserpidine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SLC18A2 (ENSG00000165646)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1957, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.662
Q58
How many genes does the drug Norethindrone target and what are they?
PGR is the only gene target of drug Norethindrone.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%norethindrone%" OR LOWER(tradeNames_string) LIKE...
[{'UUID': 'DrugGeneTargets_v2_3759', 'drugName': 'Norethindrone', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PGR (ENSG00000082175)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1962, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_2855', 'drugName': 'Noreth...
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Genetic Target
Q58.944
Q58
How many genes does the drug Alverine target and what are they?
There are 2 gene targets for the drug Alverine: HTR1A and HNF4A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%alverine%" OR LOWER(tradeNames_string) LIKE "%al...
[{'UUID': 'DrugGeneTargets_v2_4846', 'drugName': 'Alverine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HTR1A (ENSG00000178394), HNF4A (ENSG00000101076)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_4847', ...
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Genetic Target
Q58.829
Q58
How many genes does the drug Nusinersen target and what are they?
SMN2 is the only gene target of drug Nusinersen.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%nusinersen%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2674', 'drugName': 'Nusinersen', 'drugMolecularType': 'Oligonucleotide', 'newLinkedTargets_string': 'SMN2 (ENSG00000205571)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_6328', 'drugName': 'Nusinersen...
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Genetic Target
Q58.873
Q58
How many genes does the drug Rontalizumab target and what are they?
The drug Rontalizumab is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 13 genes: IFNA6, IFNA8, IFNA5, IFNA10, IFNA2, IFNA1, IFNA13, IFNA7, IFNA21, IFNA16, IFNA14, IFNA17, and IFNA4.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%rontalizumab%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_4431', 'drugName': 'Rontalizumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'IFNA6 (ENSG00000120235), IFNA8 (ENSG00000120242), IFNA5 (ENSG00000147873), IFNA10 (ENSG00000186803), IFNA2 (ENSG00000188379), IFNA1 (ENSG00000197919), IFNA13 (ENSG00000233816), IFNA7 (ENSG000002...
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Genetic Target
Q58.47
Q58
How many genes does the drug Rolapitant target and what are they?
TACR1 is the only gene target of drug Rolapitant.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%rolapitant%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_3346', 'drugName': 'Rolapitant Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'TACR1 (ENSG00000115353)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2015, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_5768', 'drugN...
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Genetic Target
Q58.1388
Q58
How many genes does the drug Desmopressin target and what are they?
There are 3 gene targets for the drug Desmopressin: AVPR2, AVPR1A, and AVPR1B.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%desmopressin%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_1017', 'drugName': 'Desmopressin', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'AVPR2 (ENSG00000126895), AVPR1A (ENSG00000166148), AVPR1B (ENSG00000198049)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 1978, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': ...
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Q58.1709
Q58
How many genes does the drug Abarelix target and what are they?
GNRHR is the only gene target of drug Abarelix.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%abarelix%" OR LOWER(tradeNames_string) LIKE "%ab...
[{'UUID': 'DrugGeneTargets_v2_4834', 'drugName': 'Abarelix', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'GNRHR (ENSG00000109163)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2003, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.1000
Q58
How many genes does the drug Selexipag target and what are they?
PTGIR is the only gene target of drug Selexipag.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%selexipag%" OR LOWER(tradeNames_string) LIKE "%s...
[{'UUID': 'DrugGeneTargets_v2_5447', 'drugName': 'Selexipag', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PTGIR (ENSG00000160013)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2015, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.883
Q58
How many genes does the drug Coformycin target and what are they?
The drug Coformycin is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene ADA.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%coformycin%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_251', 'drugName': 'Pentostatin', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADA (ENSG00000196839)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1991, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_5186', 'drugName': 'Coformyci...
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Q58.780
Q58
How many genes does the drug Anifrolumab target and what are they?
IFNAR1 is the only gene target of drug Anifrolumab.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%anifrolumab%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_4280', 'drugName': 'Anifrolumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'IFNAR1 (ENSG00000142166)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2021, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1229
Q58
How many genes does the drug Hydrocortisone Acetate target and what are they?
NR3C1 is the only gene target of drug Hydrocortisone Acetate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%hydrocortisone acetate%" OR LOWER(tradeNames_str...
[{'UUID': 'DrugGeneTargets_v2_71', 'drugName': 'Hydrocortisone Acetate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'NR3C1 (ENSG00000113580)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1951, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_1393', 'drugName'...
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Genetic Target
Q58.2000
Q58
How many genes does the drug Fluphenazine Decanoate target and what are they?
DRD2 is the only gene target of drug Fluphenazine Decanoate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%fluphenazine decanoate%" OR LOWER(tradeNames_str...
[{'UUID': 'DrugGeneTargets_v2_432', 'drugName': 'Fluphenazine Decanoate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'DRD2 (ENSG00000149295)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1972, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.5
Q58
How many genes does the drug Decitabine target and what are they?
There are 2 gene targets for the drug Decitabine: DNMT1 and DNMT3A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%decitabine%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2158', 'drugName': 'Decitabine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'DNMT1 (ENSG00000130816), DNMT3A (ENSG00000119772)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2006, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_2...
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Genetic Target
Q58.1012
Q58
How many genes does the drug Ospemifene target and what are they?
There are 2 gene targets for the drug Ospemifene: ESR2 and ESR1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ospemifene%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_3057', 'drugName': 'Ospemifene', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ESR2 (ENSG00000140009), ESR1 (ENSG00000091831)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2013, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1724
Q58
How many genes does the drug Fruquintinib target and what are they?
The drug Fruquintinib is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 3 genes: FLT1, FLT4, and KDR.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%fruquintinib%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_1715', 'drugName': 'Fruquintinib', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'FLT1 (ENSG00000102755), FLT4 (ENSG00000037280), KDR (ENSG00000128052)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.266
Q58
How many genes does the drug Insm-18 target and what are they?
The drug Insm-18 is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 2 genes: ERBB2 and IGF1R.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%insm-18%" OR LOWER(tradeNames_string) LIKE "%ins...
[{'UUID': 'DrugGeneTargets_v2_12', 'drugName': 'Insm-18', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ERBB2 (ENSG00000141736), IGF1R (ENSG00000140443)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}, {'UUID': 'DrugGeneTargets_v2_13', 'dru...
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Genetic Target
Q58.1570
Q58
How many genes does the drug Miglustat target and what are they?
UGCG is the only gene target of drug Miglustat.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%miglustat%" OR LOWER(tradeNames_string) LIKE "%m...
[{'UUID': 'DrugGeneTargets_v2_5675', 'drugName': 'Miglustat', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'UGCG (ENSG00000148154)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2003, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1832
Q58
How many genes does the drug Azd1981 target and what are they?
The drug Azd1981 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene PTGDR2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%azd1981%" OR LOWER(tradeNames_string) LIKE "%azd...
[{'UUID': 'DrugGeneTargets_v2_3608', 'drugName': 'Azd1981', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PTGDR2 (ENSG00000183134)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.449
Q58
How many genes does the drug Dyclonine Hydrochloride target and what are they?
There are 10 gene targets for the drug Dyclonine Hydrochloride: SCN1A, SCN5A, SCN4A, SCN7A, SCN2A, SCN9A, SCN3A, SCN11A, SCN8A, and SCN10A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%dyclonine hydrochloride%" OR LOWER(tradeNames_st...
[{'UUID': 'DrugGeneTargets_v2_5439', 'drugName': 'Dyclonine Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SCN1A (ENSG00000144285), SCN5A (ENSG00000183873), SCN4A (ENSG00000007314), SCN7A (ENSG00000136546), SCN2A (ENSG00000136531), SCN9A (ENSG00000169432), SCN3A (ENSG00000153253), SC...
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Genetic Target
Q58.1011
Q58
How many genes does the drug Carbenoxolone target and what are they?
There are 2 gene targets for the drug Carbenoxolone: HSD11B2 and HSD11B1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%carbenoxolone%" OR LOWER(tradeNames_string) LIKE...
[{'UUID': 'DrugGeneTargets_v2_5312', 'drugName': 'Carbenoxolone', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HSD11B2 (ENSG00000176387), HSD11B1 (ENSG00000117594)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1086
Q58
How many genes does the drug Macimorelin target and what are they?
GHSR is the only gene target of drug Macimorelin.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%macimorelin%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_5129', 'drugName': 'Macimorelin', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GHSR (ENSG00000121853)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2017, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_942', 'drugName': 'Macimore...
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Genetic Target
Q58.844
Q58
How many genes does the drug Naloxone target and what are they?
There are 3 gene targets for the drug Naloxone: OPRK1, OPRD1, and OPRM1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%naloxone%" OR LOWER(tradeNames_string) LIKE "%na...
[{'UUID': 'DrugGeneTargets_v2_3927', 'drugName': 'Naloxone Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'OPRK1 (ENSG00000082556), OPRD1 (ENSG00000116329), OPRM1 (ENSG00000112038)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 1971, 'maxClinicalTrialPhase': 4, 'drugIsApproved': T...
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Genetic Target
Q58.1792
Q58
How many genes does the drug Metformin Hydrochloride target and what are they?
There are 51 gene targets for the drug Metformin Hydrochloride: GPD2, MT-ND6, NDUFA10, NDUFS8, MT-ND4L, NDUFA6, MT-ND1, NDUFB6, NDUFA4, NDUFA11, NDUFB7, MT-ND2, NDUFS2, MT-ND5, NDUFA8, NDUFB5, MT-ND4, MT-ND3, NDUFAB1, NDUFA1, NDUFS4, NDUFB3, NDUFC1, NDUFA2, NDUFS5, NDUFS7, NDUFS6, NDUFB1, NDUFS3, NDUFA3, NDUFB4, NDUFB8...
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%metformin hydrochloride%" OR LOWER(tradeNames_st...
[{'UUID': 'DrugGeneTargets_v2_1887', 'drugName': 'Metformin Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG000001988...
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Genetic Target
Q58.308
Q58
How many genes does the drug Tipiracil Hydrochloride target and what are they?
TYMP is the only gene target of drug Tipiracil Hydrochloride.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tipiracil hydrochloride%" OR LOWER(tradeNames_st...
[{'UUID': 'DrugGeneTargets_v2_4740', 'drugName': 'Tipiracil Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'TYMP (ENSG00000025708)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2015, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1380
Q58
How many genes does the drug Imaradenant target and what are they?
The drug Imaradenant is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene ADORA2A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%imaradenant%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_373', 'drugName': 'Imaradenant', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADORA2A (ENSG00000128271)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1558
Q58
How many genes does the drug Irbesartan target and what are they?
AGTR1 is the only gene target of drug Irbesartan.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%irbesartan%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_355', 'drugName': 'Irbesartan', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'AGTR1 (ENSG00000144891)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1997, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.317
Q58
How many genes does the drug Levilimab target and what are they?
The drug Levilimab is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene IL6R.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%levilimab%" OR LOWER(tradeNames_string) LIKE "%l...
[{'UUID': 'DrugGeneTargets_v2_947', 'drugName': 'Levilimab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'IL6R (ENSG00000160712)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.152
Q58
How many genes does the drug Propiomazine Hydrochloride target and what are they?
HRH1 is the only gene target of drug Propiomazine Hydrochloride.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%propiomazine hydrochloride%" OR LOWER(tradeNames...
[{'UUID': 'DrugGeneTargets_v2_3422', 'drugName': 'Propiomazine Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HRH1 (ENSG00000196639)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1960, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1158
Q58
How many genes does the drug Larotrectinib target and what are they?
There are 3 gene targets for the drug Larotrectinib: NTRK1, NTRK2, and NTRK3.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%larotrectinib%" OR LOWER(tradeNames_string) LIKE...
[{'UUID': 'DrugGeneTargets_v2_894', 'drugName': 'Larotrectinib', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'NTRK1 (ENSG00000198400), NTRK2 (ENSG00000148053), NTRK3 (ENSG00000140538)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 2018, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UU...
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Genetic Target
Q58.1223
Q58
How many genes does the drug Talazoparib Tosylate target and what are they?
There are 2 gene targets for the drug Talazoparib Tosylate: PARP2 and PARP1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%talazoparib tosylate%" OR LOWER(tradeNames_strin...
[{'UUID': 'DrugGeneTargets_v2_2224', 'drugName': 'Talazoparib Tosylate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PARP2 (ENSG00000129484), PARP1 (ENSG00000143799)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2018, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTar...
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Genetic Target
Q58.580
Q58
How many genes does the drug Tasosartan target and what are they?
The drug Tasosartan is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene AGTR1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tasosartan%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_3109', 'drugName': 'Tasosartan', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'AGTR1 (ENSG00000144891)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': -1, 'drugIsApproved': False}]
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Genetic Target
Q58.51
Q58
How many genes does the drug Rpr749 target and what are they?
The drug Rpr749 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene ADORA1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%rpr749%" OR LOWER(tradeNames_string) LIKE "%rpr7...
[{'UUID': 'DrugGeneTargets_v2_5693', 'drugName': 'Rpr749', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADORA1 (ENSG00000163485)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drugIsApproved': False}]
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Genetic Target
Q58.1553
Q58
How many genes does the drug Articaine target and what are they?
There are 10 gene targets for the drug Articaine: SCN1A, SCN5A, SCN4A, SCN7A, SCN2A, SCN9A, SCN3A, SCN11A, SCN8A, and SCN10A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%articaine%" OR LOWER(tradeNames_string) LIKE "%a...
[{'UUID': 'DrugGeneTargets_v2_3040', 'drugName': 'Articaine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SCN1A (ENSG00000144285), SCN5A (ENSG00000183873), SCN4A (ENSG00000007314), SCN7A (ENSG00000136546), SCN2A (ENSG00000136531), SCN9A (ENSG00000169432), SCN3A (ENSG00000153253), SCN11A (ENSG0000...
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Genetic Target
Q58.733
Q58
How many genes does the drug Silodosin target and what are they?
ADRA1A is the only gene target of drug Silodosin.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%silodosin%" OR LOWER(tradeNames_string) LIKE "%s...
[{'UUID': 'DrugGeneTargets_v2_557', 'drugName': 'Silodosin', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRA1A (ENSG00000120907)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2008, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.840
Q58
How many genes does the drug Dacomitinib target and what are they?
There are 3 gene targets for the drug Dacomitinib: ERBB4, ERBB2, and EGFR.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%dacomitinib%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_3948', 'drugName': 'Dacomitinib', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ERBB4 (ENSG00000178568), ERBB2 (ENSG00000141736), EGFR (ENSG00000146648)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 2018, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID...
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Genetic Target
Q58.1392
Q58
How many genes does the drug Netoglitazone target and what are they?
The drug Netoglitazone is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene PPARG.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%netoglitazone%" OR LOWER(tradeNames_string) LIKE...
[{'UUID': 'DrugGeneTargets_v2_1686', 'drugName': 'Netoglitazone', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PPARG (ENSG00000132170)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1125
Q58
How many genes does the drug Iferanserin target and what are they?
The drug Iferanserin is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene HTR2A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%iferanserin%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_1280', 'drugName': 'Iferanserin', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HTR2A (ENSG00000102468)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.1176
Q58
How many genes does the drug Linifanib target and what are they?
The drug Linifanib is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 7 genes: FLT3, PDGFRB, PDGFRA, CSF1R, FLT1, FLT4, and KDR.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%linifanib%" OR LOWER(tradeNames_string) LIKE "%l...
[{'UUID': 'DrugGeneTargets_v2_1027', 'drugName': 'Linifanib', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'FLT3 (ENSG00000122025), PDGFRB (ENSG00000113721), PDGFRA (ENSG00000134853), CSF1R (ENSG00000182578), FLT1 (ENSG00000102755), FLT4 (ENSG00000037280), KDR (ENSG00000128052)', 'numberLinkedTarge...
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Genetic Target
Q58.476
Q58
How many genes does the drug Meclofenamate Sodium target and what are they?
There are 3 gene targets for the drug Meclofenamate Sodium: ALOX5, PTGS2, and PTGS1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%meclofenamate sodium%" OR LOWER(tradeNames_strin...
[{'UUID': 'DrugGeneTargets_v2_3724', 'drugName': 'Meclofenamate Sodium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ALOX5 (ENSG00000012779), PTGS2 (ENSG00000073756), PTGS1 (ENSG00000095303)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 1980, 'maxClinicalTrialPhase': 4, 'drugIsApproved': Tru...
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Genetic Target
Q58.980
Q58
How many genes does the drug Butamben target and what are they?
There are 2 gene targets for the drug Butamben: TRPA1 and TRPV4.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%butamben%" OR LOWER(tradeNames_string) LIKE "%bu...
[{'UUID': 'DrugGeneTargets_v2_269', 'drugName': 'Butamben Picrate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'TRPV4 (ENSG00000111199), TRPA1 (ENSG00000104321)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_...
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Genetic Target
Q58.660
Q58
How many genes does the drug Vilanterol target and what are they?
ADRB2 is the only gene target of drug Vilanterol.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%vilanterol%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_837', 'drugName': 'Vilanterol Trifenatate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRB2 (ENSG00000169252)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2013, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_4124', 'drugName...
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Genetic Target
Q58.405
Q58
How many genes does the drug Riluzole target and what are they?
There are 10 gene targets for the drug Riluzole: SCN1A, SCN5A, SCN4A, SCN7A, SCN2A, SCN9A, SCN3A, SCN11A, SCN8A, and SCN10A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%riluzole%" OR LOWER(tradeNames_string) LIKE "%ri...
[{'UUID': 'DrugGeneTargets_v2_2334', 'drugName': 'Riluzole', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SCN1A (ENSG00000144285), SCN5A (ENSG00000183873), SCN4A (ENSG00000007314), SCN7A (ENSG00000136546), SCN2A (ENSG00000136531), SCN9A (ENSG00000169432), SCN3A (ENSG00000153253), SCN11A (ENSG00000...
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Genetic Target
Q58.517
Q58
How many genes does the drug Parathyroid Hormone target and what are they?
PTH1R is the only gene target of drug Parathyroid Hormone.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%parathyroid hormone%" OR LOWER(tradeNames_string...
[{'UUID': 'DrugGeneTargets_v2_2407', 'drugName': 'Teriparatide', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'PTH1R (ENSG00000160801)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2002, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_499', 'drugName': 'Parathyroid H...
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Genetic Target
Q58.324
Q58
How many genes does the drug Lovastatin target and what are they?
HMGCR is the only gene target of drug Lovastatin.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%lovastatin%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_4581', 'drugName': 'Lovastatin', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HMGCR (ENSG00000113161)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1987, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.20
Q58
How many genes does the drug Tofersen target and what are they?
The drug Tofersen is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene SOD1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tofersen%" OR LOWER(tradeNames_string) LIKE "%to...
[{'UUID': 'DrugGeneTargets_v2_651', 'drugName': 'Tofersen', 'drugMolecularType': 'Oligonucleotide', 'newLinkedTargets_string': 'SOD1 (ENSG00000142168)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.691
Q58
How many genes does the drug Alpidem target and what are they?
TSPO is the only gene target of drug Alpidem.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%alpidem%" OR LOWER(tradeNames_string) LIKE "%alp...
[{'UUID': 'DrugGeneTargets_v2_4038', 'drugName': 'Alpidem', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'TSPO (ENSG00000100300)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.36
Q58
How many genes does the drug Trifluoperazine target and what are they?
There are 5 gene targets for the drug Trifluoperazine: HTR2C, DRD2, DRD3, DRD4, and HTR2A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%trifluoperazine%" OR LOWER(tradeNames_string) LI...
[{'UUID': 'DrugGeneTargets_v2_5160', 'drugName': 'Trifluoperazine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HTR2C (ENSG00000147246), DRD2 (ENSG00000149295), DRD3 (ENSG00000151577), DRD4 (ENSG00000069696), HTR2A (ENSG00000102468)', 'numberLinkedTargets': 5, 'yearOfFirstApproval': 1959, 'maxCli...
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Genetic Target
Q58.910
Q58
How many genes does the drug Trastuzumab target and what are they?
ERBB2 is the only gene target of drug Trastuzumab.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%trastuzumab%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_3205', 'drugName': 'Trastuzumab Deruxtecan', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'TOP1 (ENSG00000198900), ERBB2 (ENSG00000141736)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2019, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_...
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Genetic Target
Q58.834
Q58
How many genes does the drug Escitalopram target and what are they?
SLC6A4 is the only gene target of drug Escitalopram.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%escitalopram%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_4125', 'drugName': 'Escitalopram Oxalate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SLC6A4 (ENSG00000108576)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2002, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_767', 'drugName'...
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Genetic Target
Q58.1798
Q58
How many genes does the drug Teclistamab target and what are they?
There are 4 gene targets for the drug Teclistamab: CD3E, CD3G, CD3D, and TNFRSF17.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%teclistamab%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_6102', 'drugName': 'Teclistamab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'CD3E (ENSG00000198851), CD3G (ENSG00000160654), CD3D (ENSG00000167286), TNFRSF17 (ENSG00000048462)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 2022, 'maxClinicalTrialPhase': 4, 'drugIsAppr...
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Genetic Target
Q58.413
Q58
How many genes does the drug Lanoteplase target and what are they?
The drug Lanoteplase is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene PLG.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%lanoteplase%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_5822', 'drugName': 'Lanoteplase', 'drugMolecularType': 'Enzyme', 'newLinkedTargets_string': 'PLG (ENSG00000122194)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': -1, 'drugIsApproved': False}]
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Genetic Target
Q58.928
Q58
How many genes does the drug Sotorasib target and what are they?
KRAS is the only gene target of drug Sotorasib.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%sotorasib%" OR LOWER(tradeNames_string) LIKE "%s...
[{'UUID': 'DrugGeneTargets_v2_1834', 'drugName': 'Sotorasib', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'KRAS (ENSG00000133703)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2021, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.543
Q58
How many genes does the drug Romiplostim target and what are they?
MPL is the only gene target of drug Romiplostim.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%romiplostim%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_4980', 'drugName': 'Romiplostim', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'MPL (ENSG00000117400)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2008, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.765
Q58
How many genes does the drug Verubulin target and what are they?
The drug Verubulin is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 15 genes: TUBB4B, TUBB1, TUBA3C, TUBA4A, TUBB3, TUBA1A, TUBB4A, TUBB8, TUBB, TUBA1B, TUBA1C, TUBA3E, TUBB2A, TUBB2B, and TUBB6.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%verubulin%" OR LOWER(tradeNames_string) LIKE "%v...
[{'UUID': 'DrugGeneTargets_v2_4227', 'drugName': 'Verubulin', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'TUBB4B (ENSG00000188229), TUBB1 (ENSG00000101162), TUBA3C (ENSG00000198033), TUBA4A (ENSG00000127824), TUBB3 (ENSG00000258947), TUBA1A (ENSG00000167552), TUBB4A (ENSG00000104833), TUBB8 (ENSG...
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Genetic Target
Q58.1905
Q58
How many genes does the drug Tlc-388 target and what are they?
The drug Tlc-388 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene TOP1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tlc-388%" OR LOWER(tradeNames_string) LIKE "%tlc...
[{'UUID': 'DrugGeneTargets_v2_1007', 'drugName': 'Tlc-388', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'TOP1 (ENSG00000198900)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1071
Q58
How many genes does the drug Interferon Alfa-N3 target and what are they?
There are 2 gene targets for the drug Interferon Alfa-N3: IFNAR1 and IFNAR2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%interferon alfa-n3%" OR LOWER(tradeNames_string)...
[{'UUID': 'DrugGeneTargets_v2_404', 'drugName': 'Interferon Alfa-N3', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'IFNAR1 (ENSG00000142166), IFNAR2 (ENSG00000159110)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1989, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1209
Q58
How many genes does the drug Cisatracurium Besylate target and what are they?
There are 5 gene targets for the drug Cisatracurium Besylate: CHRNA1, CHRNG, CHRNB1, CHRND, and CHRNE.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%cisatracurium besylate%" OR LOWER(tradeNames_str...
[{'UUID': 'DrugGeneTargets_v2_3676', 'drugName': 'Cisatracurium Besylate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CHRNA1 (ENSG00000138435), CHRNG (ENSG00000196811), CHRNB1 (ENSG00000170175), CHRND (ENSG00000135902), CHRNE (ENSG00000108556)', 'numberLinkedTargets': 5, 'yearOfFirstApproval': 1...
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Genetic Target
Q58.248
Q58
How many genes does the drug Ttp-607 target and what are they?
The drug Ttp-607 is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 3 genes: AURKB, AURKC, and AURKA.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ttp-607%" OR LOWER(tradeNames_string) LIKE "%ttp...
[{'UUID': 'DrugGeneTargets_v2_4902', 'drugName': 'Ttp-607', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'AURKB (ENSG00000178999), AURKC (ENSG00000105146), AURKA (ENSG00000087586)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drugIsApproved': False}]
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Genetic Target
Q58.1431
Q58
How many genes does the drug Methotrexate target and what are they?
DHFR is the only gene target of drug Methotrexate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%methotrexate%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_2797', 'drugName': 'Methotrexate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'DHFR (ENSG00000228716)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1953, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_1736', 'drugName': 'Methot...
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Genetic Target
Q58.1137
Q58
How many genes does the drug Diphenidol target and what are they?
CHRM1 is the only gene target of drug Diphenidol.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%diphenidol%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1476', 'drugName': 'Diphenidol Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CHRM1 (ENSG00000168539)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1967, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_4667', 'drugN...
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Genetic Target
Q58.791
Q58
How many genes does the drug Pentaerythritol Tetranitrate target and what are they?
There are 4 gene targets for the drug Pentaerythritol Tetranitrate: GUCY1B1, GUCY1B2, GUCY1A2, and GUCY1A1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%pentaerythritol tetranitrate%" OR LOWER(tradeNam...
[{'UUID': 'DrugGeneTargets_v2_31', 'drugName': 'Pentaerythritol Tetranitrate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GUCY1B1 (ENSG00000061918), GUCY1B2 (ENSG00000123201), GUCY1A2 (ENSG00000152402), GUCY1A1 (ENSG00000164116)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 0, 'maxClinicalT...
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Genetic Target
Q58.1744
Q58
How many genes does the drug Adriforant target and what are they?
The drug Adriforant is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene HRH4.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%adriforant%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1729', 'drugName': 'Adriforant', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HRH4 (ENSG00000134489)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.495
Q58
How many genes does the drug Denileukin Diftitox target and what are they?
There are 4 gene targets for the drug Denileukin Diftitox: IL2RA, IL2RG, IL2RB, and EEF2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%denileukin diftitox%" OR LOWER(tradeNames_string...
[{'UUID': 'DrugGeneTargets_v2_5633', 'drugName': 'Denileukin Diftitox', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'IL2RA (ENSG00000134460), IL2RG (ENSG00000147168), IL2RB (ENSG00000100385), EEF2 (ENSG00000167658)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 1999, 'maxClinicalTrialPhase': 4, 'drug...
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Genetic Target
Q58.157
Q58
How many genes does the drug Gilteritinib Fumarate target and what are they?
There are 2 gene targets for the drug Gilteritinib Fumarate: FLT3 and AXL.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%gilteritinib fumarate%" OR LOWER(tradeNames_stri...
[{'UUID': 'DrugGeneTargets_v2_3307', 'drugName': 'Gilteritinib Fumarate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'FLT3 (ENSG00000122025), AXL (ENSG00000167601)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2018, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTarge...
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Genetic Target
Q58.970
Q58
How many genes does the drug Pentazocine target and what are they?
SIGMAR1 is the only gene target of drug Pentazocine.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%pentazocine%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_1542', 'drugName': 'Pentazocine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SIGMAR1 (ENSG00000147955)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1967, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_652', 'drugName': 'Penta...
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Genetic Target
Q58.860
Q58
How many genes does the drug Darusentan target and what are they?
The drug Darusentan is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 2 genes: EDNRA and EDNRB.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%darusentan%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_4363', 'drugName': 'Darusentan', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'EDNRA (ENSG00000151617), EDNRB (ENSG00000136160)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}, {'UUID': 'DrugGeneTargets_v2_4364...
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Genetic Target
Q58.1325
Q58
How many genes does the drug Amsacrine target and what are they?
There are 2 gene targets for the drug Amsacrine: TOP2A and TOP2B.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%amsacrine%" OR LOWER(tradeNames_string) LIKE "%a...
[{'UUID': 'DrugGeneTargets_v2_3938', 'drugName': 'Amsacrine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'TOP2A (ENSG00000131747), TOP2B (ENSG00000077097)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.632
Q58
How many genes does the drug Difamilast target and what are they?
The drug Difamilast is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 4 genes: PDE4A, PDE4D, PDE4B, and PDE4C.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%difamilast%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_4073', 'drugName': 'Difamilast', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PDE4A (ENSG00000065989), PDE4D (ENSG00000113448), PDE4B (ENSG00000184588), PDE4C (ENSG00000105650)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsAp...
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Genetic Target
Q58.692
Q58
How many genes does the drug Methylergonovine Maleate target and what are they?
There are 2 gene targets for the drug Methylergonovine Maleate: DRD1 and HTR2B.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%methylergonovine maleate%" OR LOWER(tradeNames_s...
[{'UUID': 'DrugGeneTargets_v2_2336', 'drugName': 'Methylergonovine Maleate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'DRD1 (ENSG00000184845), HTR2B (ENSG00000135914)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1946, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGene...
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Genetic Target
Q58.1562
Q58
How many genes does the drug Butorphanol target and what are they?
There are 2 gene targets for the drug Butorphanol: OPRM1 and OPRK1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%butorphanol%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_750', 'drugName': 'Butorphanol', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'OPRM1 (ENSG00000112038), OPRK1 (ENSG00000082556)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1978, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_74...
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Genetic Target
Q58.575
Q58
How many genes does the drug Golimumab target and what are they?
TNF is the only gene target of drug Golimumab.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%golimumab%" OR LOWER(tradeNames_string) LIKE "%g...
[{'UUID': 'DrugGeneTargets_v2_393', 'drugName': 'Golimumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'TNF (ENSG00000232810)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2009, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1909
Q58
How many genes does the drug Levobupivacaine target and what are they?
SCN4A is the only gene target of drug Levobupivacaine.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%levobupivacaine%" OR LOWER(tradeNames_string) LI...
[{'UUID': 'DrugGeneTargets_v2_4768', 'drugName': 'Levobupivacaine Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SCN4A (ENSG00000007314)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1999, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_3325', '...
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Genetic Target
Q58.18
Q58
How many genes does the drug Phenoxypropazine target and what are they?
There are 2 gene targets for the drug Phenoxypropazine: MAOA and MAOB.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%phenoxypropazine%" OR LOWER(tradeNames_string) L...
[{'UUID': 'DrugGeneTargets_v2_4642', 'drugName': 'Phenoxypropazine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'MAOA (ENSG00000189221), MAOB (ENSG00000069535)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.130
Q58
How many genes does the drug Siltuximab target and what are they?
IL6 is the only gene target of drug Siltuximab.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%siltuximab%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2074', 'drugName': 'Siltuximab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'IL6 (ENSG00000136244)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2014, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1361
Q58
How many genes does the drug Degarelix Acetate target and what are they?
GNRHR is the only gene target of drug Degarelix Acetate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%degarelix acetate%" OR LOWER(tradeNames_string) ...
[{'UUID': 'DrugGeneTargets_v2_6054', 'drugName': 'Degarelix Acetate', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'GNRHR (ENSG00000109163)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2008, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1291
Q58
How many genes does the drug Biciromab Brallobarbital target and what are they?
The drug Biciromab Brallobarbital is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene FGB.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%biciromab brallobarbital%" OR LOWER(tradeNames_s...
[{'UUID': 'DrugGeneTargets_v2_5505', 'drugName': 'Biciromab Brallobarbital', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'FGB (ENSG00000171564)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drugIsApproved': False}]
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Genetic Target
Q58.1969
Q58
How many genes does the drug Insulin Purified Pork target and what are they?
INSR is the only gene target of drug Insulin Purified Pork.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%insulin purified pork%" OR LOWER(tradeNames_stri...
[{'UUID': 'DrugGeneTargets_v2_1882', 'drugName': 'Insulin Purified Pork', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'INSR (ENSG00000171105)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1979, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.935
Q58
How many genes does the drug Halazepam target and what are they?
There are 16 gene targets for the drug Halazepam: GABRA1, GABRB2, GABRG2, GABRB3, GABRA4, GABRG3, GABRQ, GABRA3, GABRP, GABRD, GABRG1, GABRB1, GABRE, GABRA2, GABRA5, and GABRA6.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%halazepam%" OR LOWER(tradeNames_string) LIKE "%h...
[{'UUID': 'DrugGeneTargets_v2_4122', 'drugName': 'Halazepam', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089), GABRA3 (EN...
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Genetic Target
Q58.989
Q58
How many genes does the drug Insulin Zinc Susp Prompt Beef target and what are they?
INSR is the only gene target of drug Insulin Zinc Susp Prompt Beef.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%insulin zinc susp prompt beef%" OR LOWER(tradeNa...
[{'UUID': 'DrugGeneTargets_v2_3871', 'drugName': 'Insulin Zinc Susp Prompt Beef', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'INSR (ENSG00000171105)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1982, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1965
Q58
How many genes does the drug Eliglustat target and what are they?
UGCG is the only gene target of drug Eliglustat.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%eliglustat%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_4249', 'drugName': 'Eliglustat', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'UGCG (ENSG00000148154)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2014, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_5337', 'drugName': 'Eliglust...
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Genetic Target
Q58.193
Q58
How many genes does the drug Dimethyl Fumarate target and what are they?
KEAP1 is the only gene target of drug Dimethyl Fumarate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%dimethyl fumarate%" OR LOWER(tradeNames_string) ...
[{'UUID': 'DrugGeneTargets_v2_3182', 'drugName': 'Dimethyl Fumarate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'KEAP1 (ENSG00000079999)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2013, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1149
Q58
How many genes does the drug Oxybutynin Chloride target and what are they?
There are 2 gene targets for the drug Oxybutynin Chloride: CHRM3 and CHRM2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%oxybutynin chloride%" OR LOWER(tradeNames_string...
[{'UUID': 'DrugGeneTargets_v2_871', 'drugName': 'Oxybutynin Chloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CHRM3 (ENSG00000133019), CHRM2 (ENSG00000181072)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1975, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTarge...
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Genetic Target
Q58.1001
Q58
How many genes does the drug Yttrium Y 90 Ibritumomab Tiuxetan target and what are they?
MS4A1 is the only gene target of drug Yttrium Y 90 Ibritumomab Tiuxetan.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%yttrium y 90 ibritumomab tiuxetan%" OR LOWER(tra...
[{'UUID': 'DrugGeneTargets_v2_1480', 'drugName': 'Yttrium Y 90 Ibritumomab Tiuxetan', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'MS4A1 (ENSG00000156738)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2002, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1956
Q58
How many genes does the drug Blinatumomab target and what are they?
There are 4 gene targets for the drug Blinatumomab: CD3E, CD3G, CD3D, and CD19.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%blinatumomab%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_4607', 'drugName': 'Blinatumomab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'CD3E (ENSG00000198851), CD3G (ENSG00000160654), CD3D (ENSG00000167286), CD19 (ENSG00000177455)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 2014, 'maxClinicalTrialPhase': 4, 'drugIsApprove...
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Genetic Target
Q58.1657
Q58
How many genes does the drug Abiraterone target and what are they?
There are 5 gene targets for the drug Abiraterone: AR, CYP17A1, SRD5A1, SRD5A2, and SRD5A3.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%abiraterone%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_6320', 'drugName': 'Abiraterone', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'AR (ENSG00000169083), CYP17A1 (ENSG00000148795), SRD5A1 (ENSG00000145545), SRD5A2 (ENSG00000277893), SRD5A3 (ENSG00000128039)', 'numberLinkedTargets': 5, 'yearOfFirstApproval': 0, 'maxClini...
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Genetic Target
Q58.613
Q58
How many genes does the drug Picotamide target and what are they?
There are 2 gene targets for the drug Picotamide: TBXAS1 and TBXA2R.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%picotamide%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_4429', 'drugName': 'Picotamide', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'TBXAS1 (ENSG00000059377), TBXA2R (ENSG00000006638)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_443...
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Genetic Target
Q58.183
Q58
How many genes does the drug Ritobegron target and what are they?
The drug Ritobegron is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene ADRB3.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ritobegron%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_3401', 'drugName': 'Ritobegron', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRB3 (ENSG00000188778)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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