PDBID
stringlengths
4
4
Resolution
stringlengths
1
13
Year
int64
1.98k
2.02k
Ligand Name
stringlengths
1
7
Ligand Chain
stringclasses
53 values
Ligand Residue Number
stringlengths
1
9
Binding Affinity Measurement
stringclasses
4 values
Binding Affinity Sign
stringclasses
6 values
Binding Affinity Value
float64
0
500M
Binding Affinity Unit
stringclasses
6 values
Log Binding Affinity
float64
-14
2.97
Binding Affinity Source
stringclasses
3 values
Binding Affinity Annotation
stringlengths
6
72
Protein UniProtID
stringlengths
6
55
Protein UniProtName
stringlengths
2
575
Ligand SMILES
stringlengths
4
352
Ligand MW
float64
44
1.82k
Ligand LogP
float64
-23.01
13.7
Ligand TPSA
float64
0
786
Ligand NumRotBond
int64
0
59
Ligand NumHeavyAtoms
int64
3
120
Ligand NumHDon
int64
0
30
Ligand NumHAcc
int64
0
56
Ligand QED
float64
0.01
0.95
1ajn
2.36
1,997
AAN
B
559
ki
=
2.32
mM
-2.634512
MOAD
Ki=2.32mM
P06875,P06875
PENICILLIN AMIDOHYDROLASE,PENICILLIN AMIDOHYDROLASE
O=C([O-])Cc1ccc([N+](=O)[O-])cc1
180.139
-0.1128
83.27
3
13
0
4
0.479409
1ajp
2.31
1,997
OMD
A
210
ki
=
5.85
mM
-2.232844
MOAD
Ki=5.85mM
P06875,P06875
PENICILLIN AMIDOHYDROLASE,PENICILLIN AMIDOHYDROLASE
O=C([O-])Cc1cc(O)ccc1O
167.14
-0.6098
80.59
2
12
2
4
0.575592
1ajq
2.05
1,997
SPA
B
559
ki
=
0.049
mM
-4.309804
MOAD
Ki=0.049mM
P06875,P06875
PENICILLIN AMIDOHYDROLASE,PENICILLIN AMIDOHYDROLASE
O=C([O-])Cc1cccs1
141.171
0.0405
40.13
2
9
0
3
0.58308
1ajv
2.0
1,997
NMB
A
501
ki
=
19.1
nM
-7.718967
MOAD
Ki=19.1nM
P03366,P03366
HIV-1 PROTEASE,HIV-1 PROTEASE
O=S1(=O)N(Cc2ccccc2)[C@H](COc2ccccc2)[C@H](O)[C@@H](O)[C@@H](COc2ccccc2)N1Cc1ccccc1
574.699
3.8662
99.54
10
41
2
6
0.29851
1ajx
2.0
1,997
AH1
A
500
ki
=
12.2
nM
-7.91364
MOAD
Ki=12.2nM
P03366,P03366
HIV-1 PROTEASE,HIV-1 PROTEASE
O=C1N(Cc2ccccc2)[C@H](COc2ccccc2)[C@H](O)[C@@H](O)[C@@H](COc2ccccc2)N1Cc1ccccc1
538.644
4.7414
82.47
10
40
2
5
0.304856
1akq
1.9
1,998
FMN
A
149
kd
=
0.79
nM
-9.102373
MOAD
Kd=0.79nM
P00323
FLAVODOXIN
Cc1cc2nc3c(=O)[nH]c(=O)nc-3n(C[C@H](O)[C@H](O)[C@H](O)COP(=O)([O-])[O-])c2cc1C
454.332
-2.87056
213.75
7
31
4
12
0.210194
1akr
1.58
1,998
FMN
A
149
kd
=
0.82
nM
-9.086186
MOAD
Kd=0.82nM
P00323
FLAVODOXIN
Cc1cc2nc3c(=O)[nH]c(=O)nc-3n(C[C@H](O)[C@H](O)[C@H](O)COP(=O)([O-])[O-])c2cc1C
454.332
-2.87056
213.75
7
31
4
12
0.210194
1akt
1.8
1,998
FMN
A
149
kd
=
3.2
nM
-8.49485
MOAD
Kd=3.2nM
P00323
FLAVODOXIN
Cc1cc2nc3c(=O)[nH]c(=O)nc-3n(C[C@H](O)[C@H](O)[C@H](O)COP(=O)([O-])[O-])c2cc1C
454.332
-2.87056
213.75
7
31
4
12
0.210194
1aku
1.9
1,998
FMN
A
150
kd
=
746
nM
-6.127261
MOAD
Kd=746.0nM
P00323
FLAVODOXIN
Cc1cc2nc3c(=O)[nH]c(=O)nc-3n(C[C@H](O)[C@H](O)[C@H](O)COP(=O)([O-])[O-])c2cc1C
454.332
-2.87056
213.75
7
31
4
12
0.210194
1akv
2.0
1,998
FMN
A
152
kd
=
0.0026
nM
-11.585027
MOAD
Kd=0.0026nM
P00323
FLAVODOXIN
Cc1cc2nc3c(=O)[nH]c(=O)nc-3n(C[C@H](O)[C@H](O)[C@H](O)COP(=O)([O-])[O-])c2cc1C
454.332
-2.87056
213.75
7
31
4
12
0.210194
1akw
1.75
1,998
FMN
A
149
kd
=
2.6
nM
-8.585027
MOAD
Kd=2.6nM
P00323
FLAVODOXIN
Cc1cc2nc3c(=O)[nH]c(=O)nc-3n(C[C@H](O)[C@H](O)[C@H](O)COP(=O)([O-])[O-])c2cc1C
454.332
-2.87056
213.75
7
31
4
12
0.210194
1al8
2.2
1,997
DHP
A
361
ki
=
4.8
uM
-5.318759
MOAD
Ki=4.8uM
P05414
GLYCOLATE OXIDASE
CCCCCCCCCCC1=C(O)C(=O)NC1=O
253.342
2.9857
66.4
9
18
2
3
0.49012
1alw
2.03
1,998
ISA
A
11
ki
=
0.3
uM
-6.522879
MOAD
Ki=0.3uM
P04574
CALPAIN
O=C([O-])[C@@H](S)Cc1ccc(I)cc1
307.132
0.882
40.13
3
13
1
3
0.665182
1alw
2.03
1,998
ISA
B
12
ki
=
0.3
uM
-6.522879
MOAD
Ki=0.3uM
P04574
CALPAIN
O=C([O-])[C@@H](S)Cc1ccc(I)cc1
307.132
0.882
40.13
3
13
1
3
0.665182
1am1
2.0
1,998
ADP
A
300
kd
=
132
mM
-0.879426
MOAD
Kd=132.0mM
P02829
HEAT SHOCK PROTEIN 90
Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@](=O)([O-])OP(=O)([O-])[O-])[C@@H](O)[C@H]1O
424.179
-3.642
241.09
6
27
3
15
0.378904
1am6
2.0
1,998
HAE
A
555
ic50
=
47
uM
-4.327902
MOAD
ic50=47.0uM
P00918
CARBONIC ANHYDRASE
CC(=O)NO
75.067
-0.4883
49.33
0
5
2
2
0.301333
1amk
1.83
1,997
PGA
A
600
ki
=
0.05
mM
-4.30103
MOAD
Ki=0.05mM
P48499
TRIOSE PHOSPHATE ISOMERASE
O=C([O-])COP(=O)([O-])[O-]
153.006
-3.4184
112.55
3
9
0
6
0.389879
1amw
1.85
1,998
ADP
A
300
kd
=
29
uM
-4.537602
MOAD
Kd=29.0uM
P02829
HEAT SHOCK PROTEIN 90
Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@](=O)([O-])OP(=O)([O-])[O-])[C@@H](O)[C@H]1O
424.179
-3.642
241.09
6
27
3
15
0.378904
1anf
1.67
1,997
GLC-GLC
B
1-2
ki
=
3.5
uM
-5.455932
MOAD
Ki=3.5uM
P0AEX9
MALTODEXTRIN-BINDING PROTEIN
OC[C@H]1O[C@H](O[C@H]2[C@H](O)[C@@H](O)[C@@H](O)O[C@@H]2CO)[C@H](O)[C@@H](O)[C@@H]1O
342.297
-5.3972
189.53
4
23
8
11
0.243258
1ao8
NMR
1,998
MTX
A
170
ki
=
0.004
nM
-11.39794
BindingDB
IC50=16nM,Ki=0.004000nM
P00381
DIHYDROFOLATE REDUCTASE
CN(Cc1cnc2nc(N)nc(N)c2n1)c1ccc(C(=O)N[C@@H](CCC(=O)[O-])C(=O)[O-])cc1
452.431
-2.401
216.2
9
33
3
12
0.30942
1aoe
1.6
1,998
GW3
A
194
ki
=
0.22
nM
-9.657577
MOAD
Ki=0.22nM
P22906
DIHYDROFOLATE REDUCTASE
CCC(CC)n1ccc2c3c(N)nc(N)nc3ccc21
269.352
3.11
82.75
3
20
2
5
0.764936
1aoe
1.6
1,998
GW3
B
194
ki
=
0.22
nM
-9.657577
MOAD
Ki=0.22nM
P22906
DIHYDROFOLATE REDUCTASE
CCC(CC)n1ccc2c3c(N)nc(N)nc3ccc21
269.352
3.11
82.75
3
20
2
5
0.764936
1apb
1.76
1,992
FCA
A
307
kd
=
1.51
uM
-5.821023
MOAD
Kd=1.51uM
P02924
L-ARABINOSE-BINDING PROTEIN
C[C@H]1O[C@H](O)[C@H](O)[C@@H](O)[C@H]1O
164.157
-2.1938
90.15
0
11
4
5
0.326216
1apb
1.76
1,992
FCB
A
308
kd
=
1.51
uM
-5.821023
MOAD
Kd=1.51uM
P02924
L-ARABINOSE-BINDING PROTEIN
C[C@H]1O[C@@H](O)[C@H](O)[C@@H](O)[C@H]1O
164.157
-2.1938
90.15
0
11
4
5
0.326216
1apu
1.8
1,994
IVA-32L
I
4-1
ki
=
1.6
nM
-8.79588
MOAD
Ki=1.6nM
P00798
PROTEIN (PENICILLOPEPSIN)
CCOC(=O)C[C@H](O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)CC(C)C)C(C)C)C(C)C
485.666
2.1591
133.83
15
34
4
6
0.262716
1apz
2.3
1,996
ASP
D
552
ki
=
600,000
nM
-3.221849
BindingDB
Ki=600000nM
P20933,P20933,P20933
ASPARTYLGLUCOSAMINIDASE,ASPARTYLGLUCOSAMINIDASE,ASPARTYLGLUCOSAMINIDASE
[NH3+][C@@H](CC(=O)[O-])C(=O)[O-]
132.095
-4.5132
107.9
3
9
1
4
0.416966
1apz
2.3
1,996
ASP
B
551
ki
=
600,000
nM
-3.221849
BindingDB
Ki=600000nM
P20933,P20933,P20933
ASPARTYLGLUCOSAMINIDASE,ASPARTYLGLUCOSAMINIDASE,ASPARTYLGLUCOSAMINIDASE
[NH3+][C@@H](CC(=O)[O-])C(=O)[O-]
132.095
-4.5132
107.9
3
9
1
4
0.416966
1aq7
2.2
1,998
34H-AG2
B
1-4
ic50
=
0.9
uM
-6.045757
MOAD
ic50=0.9uM
P00760
TRYPSIN
CC[C@@H](C)[C@@H](NC(=O)[C@H](O)Cc1ccc(O)cc1)C(=O)N1[C@H](C(=O)NCCCCNC(N)=[NH2+])C[C@@H]2CC[C@@H](OS(=O)(=O)[O-])C[C@@H]21
654.787
-1.9987
249.04
15
45
7
9
0.035819
1atl
1.8
1,995
0QI
A
301
ki
=
0.52
uM
-6.283997
MOAD
Ki=0.52uM
P15167
Snake venom metalloproteinase atrolysin-D
COc1ccc(C[C@H](NC(=O)[C@@H](CS)CC(C)C)C(=O)[O-])cc1
338.449
1.0645
78.46
9
23
2
5
0.660228
1atl
1.8
1,995
0QI
B
311
ki
=
0.52
uM
-6.283997
MOAD
Ki=0.52uM
P15167
Snake venom metalloproteinase atrolysin-D
COc1ccc(C[C@H](NC(=O)[C@@H](CS)CC(C)C)C(=O)[O-])cc1
338.449
1.0645
78.46
9
23
2
5
0.660228
1atp
2.2
1,993
ATP
E
355
kd
=
60
nM
-7.221849
MOAD
Kd=60.0nM
P05132,P63248
cAMP-DEPENDENT PROTEIN KINASE,PEPTIDE INHIBITOR PKI(5-24)
Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@](=O)([O-])O[P@@](=O)([O-])OP(=O)([O-])[O-])[C@@H](O)[C@H]1O
503.15
-4.157
290.45
8
31
3
18
0.28788
1avn
2.0
1,997
HSM
A
264
kd
=
0.125
mM
-3.90309
MOAD
Kd=0.125mM
P00918
CARBONIC ANHYDRASE II
[NH3+]CCc1c[nH]cn1
112.156
-0.8059
56.32
2
8
2
1
0.516436
1awf
2.2
1,998
ASP-LEU
I
55-64
ki
=
0.97
uM
-6.013228
MOAD
Ki=0.97uM
P00734,P00734
ALPHA THROMBIN,ALPHA THROMBIN
CC[C@H](C)[C@H](NC(=O)[C@H](CCC(=O)[O-])NC(=O)[C@H](CCC(=O)[O-])NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H]([NH3+])CC(=O)[O-])C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCC(=O)[O-])C(=O)N[C@@H](CCC(=O)[O-])C(=O)N[C@@H](Cc1ccc(OS(=O)(=O)[O-])cc1)C(=O)N[C@@H](CC(C)C)C(=O)[O-]
1,357.369
-11.1068
587.96
42
95
9
25
0.022011
1awi
2.2
1,998
PRO-PRO
P
1-10
kd
=
90
uM
-4.045757
MOAD
Kd=90.0uM
P07737,P07737
PROFILIN,PROFILIN
O=C([O-])[C@@H]1CCCN1C(=O)[C@@H]1CCCN1C(=O)[C@@H]1CCCN1C(=O)[C@@H]1CCCN1C(=O)[C@@H]1CCCN1C(=O)[C@@H]1CCCN1C(=O)[C@@H]1CCCN1C(=O)[C@@H]1CCCN1C(=O)[C@@H]1CCCN1C(=O)[C@@H]1CCC[NH2+]1
989.185
-2.6189
239.53
10
71
1
11
0.237919
1ax0
1.9
1,998
A2G
A
401
kd
=
0.000746
M
-3.127105
MOAD
Ka=1340.0M^-1
P16404
LECTIN
CC(=O)N[C@@H]1[C@@H](O)[C@@H](O)[C@@H](CO)O[C@@H]1O
221.209
-3.0776
119.25
2
15
5
6
0.337239
1ax1
1.95
1,998
BGC-GAL
C
1-2
kd
=
0.000515
M
-3.287802
MOAD
Ka=1940.0M^-1
P16404
LECTIN
OC[C@H]1O[C@@H](O[C@H]2[C@H](O)[C@@H](O)[C@H](O)O[C@@H]2CO)[C@H](O)[C@@H](O)[C@H]1O
342.297
-5.3972
189.53
4
23
8
11
0.243258
1ax2
1.95
1,998
NDG-GAL
C
1-2
kd
=
0.000103
M
-3.988113
MOAD
Ka=9730.0M^-1
P16404
LECTIN
CC(=O)N[C@@H]1[C@@H](O)[C@H](O[C@@H]2O[C@H](CO)[C@H](O)[C@H](O)[C@H]2O)[C@@H](CO)O[C@@H]1O
383.35
-5.2534
198.4
5
26
8
11
0.225556
1axr
2.3
1,998
HTP
A
998
ki
=
540
uM
-3.267606
MOAD
Ki=540.0uM
P00489
GLYCOGEN PHOSPHORYLASE
OC[C@@H]1[C@@H](O)[C@H](O)[C@@H](O)c2cn[nH][n+]21
202.19
-3.0006
113.48
1
14
5
5
0.311377
1axz
1.95
1,998
GLA
A
401
kd
=
0.000637
M
-3.1959
MOAD
Ka=1570.0M^-1
P16404
LECTIN
OC[C@H]1O[C@H](O)[C@H](O)[C@@H](O)[C@H]1O
180.156
-3.2214
110.38
1
12
5
6
0.290153
1axz
1.95
1,998
GAL
A
402
kd
=
0.000637
M
-3.1959
MOAD
Ka=1570.0M^-1
P16404
LECTIN
OC[C@H]1O[C@@H](O)[C@H](O)[C@@H](O)[C@H]1O
180.156
-3.2214
110.38
1
12
5
6
0.290153
1az1
1.8
1,998
ALR
A
318
ki
=
2,000
nM
-5.69897
BindingDB
IC50=79000nM,Ki=2000nM
P15121
ALDOSE REDUCTASE
O=C([O-])CN1C(=O)c2cccc3cccc(c23)C1=O
254.221
0.1857
77.51
2
19
0
4
0.716407
1az1
1.8
1,998
ALR
A
317
ki
=
2,000
nM
-5.69897
BindingDB
IC50=79000nM,Ki=2000nM
P15121
ALDOSE REDUCTASE
O=C([O-])CN1C(=O)c2cccc3cccc(c23)C1=O
254.221
0.1857
77.51
2
19
0
4
0.716407
1azl
1.8
1,998
FMN
A
149
kd
=
2.4
nM
-8.619789
MOAD
Kd=2.4nM
P00323
FLAVODOXIN
Cc1cc2nc3c(=O)[nH]c(=O)nc-3n(C[C@H](O)[C@H](O)[C@H](O)COP(=O)([O-])[O-])c2cc1C
454.332
-2.87056
213.75
7
31
4
12
0.210194
1azm
2.0
1,994
AZM
A
262
kd
=
1,400
nM
-5.853872
BindingDB
Ki=250nM,Kd=1400nM,IC50=5.8nM
P00915
CARBONIC ANHYDRASE I
CC(=O)Nc1nnc(S(N)(=O)=O)s1
222.251
-0.8561
115.04
2
13
2
6
0.631859
1b05
2.0
1,998
LYS-LYS
B
1-3
kd
=
75
nM
-7.124939
MOAD
Kd=75.0nM
P06202
PERIPLASMIC OLIGOPEPTIDE-BINDING PROTEIN
[NH3+]CCCC[C@H](NC(=O)[C@H](CS)NC(=O)[C@@H]([NH3+])CCCC[NH3+])C(=O)[O-]
379.527
-4.9294
181.25
14
25
6
5
0.130667
1b0h
1.9
1,998
LYS-LYS
B
601-603
kd
=
0.2
uM
-6.69897
MOAD
Kd=0.2uM
P06202
PERIPLASMIC OLIGOPEPTIDE-BINDING PROTEIN
[NH3+]CCCC[C@H](NC(=O)[C@H](Cc1cccc2ccccc12)NC(=O)[C@@H]([NH3+])CCCC[NH3+])C(=O)[O-]
473.618
-2.4633
181.25
15
34
5
4
0.179954
1b1h
1.8
1,998
LYS-LYS
B
1-3
kd
=
0.093
uM
-7.031517
MOAD
Kd=0.093uM
P06202
PROTEIN (OLIGO-PEPTIDE BINDING PROTEIN)
[NH3+]CCCC[C@H](NC(=O)[C@H](CCc1ccccc1)NC(=O)[C@@H]([NH3+])CCCC[NH3+])C(=O)[O-]
437.585
-3.2264
181.25
16
31
5
4
0.170617
1b2h
1.9
1,998
LYS-LYS
B
1-3
kd
=
29
uM
-4.537602
MOAD
Kd=29.0uM
P06202
PERIPLASMIC OLIGOPEPTIDE-BINDING PROTEIN
[NH3+]CCCC[C@H](NC(=O)[C@H](CCC[NH3+])NC(=O)[C@@H]([NH3+])CCCC[NH3+])C(=O)[O-]
391.537
-5.8371
208.89
16
27
6
4
0.14191
1b2i
NMR
1,999
AMH
A
84
kd
=
1,100
nM
-5.958607
BindingDB
Kd=1100nM,IC50=3100nM,Ki=25000000nM
P00747
PROTEIN (PLASMINOGEN)
[NH3+]C[C@H]1CC[C@H](C(=O)[O-])CC1
157.213
-1.2154
67.77
2
11
1
2
0.5459
1b32
1.75
1,998
LYS-LYS
B
1-3
kd
=
79
nM
-7.102373
MOAD
Kd=79.0nM
P06202
PROTEIN (OLIGO-PEPTIDE BINDING PROTEIN)
CSCC[C@H](NC(=O)[C@@H]([NH3+])CCCC[NH3+])C(=O)N[C@@H](CCCC[NH3+])C(=O)[O-]
407.581
-4.1061
181.25
16
27
5
5
0.162686
1b38
2.0
1,998
ATP
A
381
kd
=
0.254
uM
-6.595166
MOAD
Kd=0.254uM
P24941
PROTEIN (CELL DIVISION PROTEIN KINASE 2)
Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@](=O)([O-])O[P@](=O)([O-])OP(=O)([O-])[O-])[C@@H](O)[C@H]1O
503.15
-4.157
290.45
8
31
3
18
0.28788
1b39
2.1
1,998
ATP
A
381
kd
=
0.12
uM
-6.920819
MOAD
Kd=0.12uM
P24941
PROTEIN (CELL DIVISION PROTEIN KINASE 2)
Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@](=O)([O-])O[P@](=O)([O-])OP(=O)([O-])[O-])[C@@H](O)[C@H]1O
503.15
-4.157
290.45
8
31
3
18
0.28788
1b3d
2.3
1,999
S27
B
401
ic50
=
24
nM
-7.619789
BindingDB
IC50=24nM
P08254
STROMELYSIN-1
CC(C)C[C@H](C(=O)NO)N(Cc1ccccc1)[P@](C)(=O)c1ccccc1
374.421
3.6421
69.64
8
26
2
3
0.420465
1b3f
1.8
1,998
LYS-LYS
B
1-3
kd
=
130
nM
-6.886057
MOAD
Kd=130.0nM
P06202
PROTEIN (OLIGO-PEPTIDE BINDING PROTEIN)
[NH3+]CCCC[C@H](NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@@H]([NH3+])CCCC[NH3+])C(=O)[O-]
413.523
-4.8934
209.93
15
29
6
5
0.155651
1b3g
2.0
1,998
LYS-LYS
B
1-3
kd
=
200
nM
-6.69897
MOAD
Kd=200.0nM
P06202
PROTEIN (OLIGO-PEPTIDE BINDING PROTEIN)
CC[C@H](C)[C@H](NC(=O)[C@@H]([NH3+])CCCC[NH3+])C(=O)N[C@@H](CCCC[NH3+])C(=O)[O-]
389.541
-3.8131
181.25
15
27
5
4
0.180082
1b3h
2.0
1,998
LYS-LYS
B
1-3
kd
=
0.62
uM
-6.207608
MOAD
Kd=0.62uM
P06202
PERIPLASMIC OLIGOPEPTIDE-BINDING PROTEIN
[NH3+]CCCC[C@H](NC(=O)[C@H](CC1CCCCC1)NC(=O)[C@@H]([NH3+])CCCC[NH3+])C(=O)[O-]
429.606
-2.8888
181.25
15
30
5
4
0.175302
1b3l
2.0
1,998
LYS-LYS
D
1-3
kd
=
1,300
nM
-5.886057
MOAD
Kd=1300.0nM
P06202
PROTEIN (OLIGO-PEPTIDE BINDING PROTEIN)
[NH3+]CCCC[C@H](NC(=O)CNC(=O)[C@@H]([NH3+])CCCC[NH3+])C(=O)[O-]
333.433
-5.2278
181.25
13
23
5
4
0.211237
1b3l
2.0
1,998
LYS-LYS
B
1-3
kd
=
1,300
nM
-5.886057
MOAD
Kd=1300.0nM
P06202
PROTEIN (OLIGO-PEPTIDE BINDING PROTEIN)
[NH3+]CCCC[C@H](NC(=O)CNC(=O)[C@@H]([NH3+])CCCC[NH3+])C(=O)[O-]
333.433
-5.2278
181.25
13
23
5
4
0.211237
1b42
2.2
1,999
M1A
A
600
kd
=
97.9
uM
-4.009217
MOAD
Kd=97.9uM
P07617
VP39
C[n+]1cnc2[nH]cnc2c1N
150.165
-0.6354
71.47
0
11
2
3
0.490764
1b46
1.8
1,999
LYS-LYS
B
1-3
kd
=
5,200
nM
-5.283997
MOAD
Kd=5200.0nM
P06202
PROTEIN (OLIGO-PEPTIDE BINDING PROTEIN)
[NH3+]CCCC[C@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H]([NH3+])CCCC[NH3+])C(=O)[O-]
373.498
-4.353
172.46
12
26
4
4
0.25327
1b4d
2.0
1,998
CRA
A
998
ki
=
15.6
uM
-4.806875
MOAD
Ki=15.6uM
P00489
PROTEIN (GLYCOGEN PHOSPHORYLASE B)
COC(=O)N[C@]1(C(N)=O)O[C@H](CO)[C@@H](O)[C@H](O)[C@H]1O
280.233
-4.0022
171.57
3
19
6
8
0.303273
1b4h
1.9
1,998
LYS-LYS
B
1-3
kd
=
3.44
uM
-5.463442
MOAD
Kd=3.44uM
P06202
PERIPLASMIC OLIGO-PEPTIDE BINDING PROTEIN
[NH3+]CCCC[C@H](NC(=O)[C@H](CC[NH3+])NC(=O)[C@@H]([NH3+])CCCC[NH3+])C(=O)[O-]
377.51
-6.2272
208.89
15
26
6
4
0.153743
1b4z
1.75
1,999
LYS-LYS
B
1-3
kd
=
5,900
nM
-5.229148
MOAD
Kd=5900.0nM
P06202
PROTEIN (OLIGO-PEPTIDE BINDING PROTEIN)
[NH3+]CCCC[C@H](NC(=O)[C@H](CC(=O)[O-])NC(=O)[C@@H]([NH3+])CCCC[NH3+])C(=O)[O-]
390.461
-6.7192
221.38
15
27
5
6
0.170736
1b51
1.8
1,999
LYS-LYS
B
1-3
kd
=
43
nM
-7.366532
MOAD
Kd=43.0nM
P06202
PROTEIN (OLIGO-PEPTIDE BINDING PROTEIN)
[NH3+]CCCC[C@H](NC(=O)[C@H](CO)NC(=O)[C@@H]([NH3+])CCCC[NH3+])C(=O)[O-]
363.459
-5.8669
201.48
14
25
6
5
0.16644
1b52
2.3
1,999
LYS-LYS
B
1-3
kd
=
76
nM
-7.119186
MOAD
Kd=76.0nM
P06202
PROTEIN (OLIGO-PEPTIDE BINDING PROTEIN)
C[C@@H](O)[C@H](NC(=O)[C@@H]([NH3+])CCCC[NH3+])C(=O)N[C@@H](CCCC[NH3+])C(=O)[O-]
377.486
-5.4784
201.48
14
26
6
5
0.163552
1b55
2.4
1,999
4IP
B
172
kd
=
40
nM
-7.39794
MOAD
Kd=40.0nM
Q06187,Q06187
TYROSINE-PROTEIN KINASE BTK,TYROSINE-PROTEIN KINASE BTK
O=P([O-])([O-])O[C@H]1[C@H](O)[C@@H](OP(=O)([O-])[O-])[C@H](OP(=O)([O-])[O-])[C@@H](OP(=O)([O-])[O-])[C@H]1O
492.008
-8.4226
330.14
8
28
2
18
0.296895
1b55
2.4
1,999
4IP
A
171
kd
=
40
nM
-7.39794
MOAD
Kd=40.0nM
Q06187,Q06187
TYROSINE-PROTEIN KINASE BTK,TYROSINE-PROTEIN KINASE BTK
O=P([O-])([O-])O[C@H]1[C@H](O)[C@@H](OP(=O)([O-])[O-])[C@H](OP(=O)([O-])[O-])[C@@H](OP(=O)([O-])[O-])[C@H]1O
492.008
-8.4226
330.14
8
28
2
18
0.296895
1b58
1.8
1,999
LYS-LYS
B
1-3
kd
=
260
nM
-6.585027
MOAD
Kd=260.0nM
P06202
PROTEIN (OLIGO-PEPTIDE BINDING PROTEIN)
[NH3+]CCCC[C@H](NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@@H]([NH3+])CCCC[NH3+])C(=O)[O-]
439.557
-3.9109
201.48
15
31
6
5
0.151257
1b5h
1.9
1,998
LYS-LYS
B
1-3
kd
=
0.97
uM
-6.013228
MOAD
Kd=0.97uM
P06202
OLIGO-PEPTIDE BINDING PROTEIN
[NH3+]CCCC[C@H](NC(=O)[C@H](C[NH3+])NC(=O)[C@@H]([NH3+])CCCC[NH3+])C(=O)[O-]
363.483
-6.6173
208.89
14
25
6
4
0.166131
1b5i
1.9
1,999
LYS-LYS
B
1-3
kd
=
90
nM
-7.045757
MOAD
Kd=90.0nM
P06202
PROTEIN (OLIGO-PEPTIDE BINDING PROTEIN)
NC(=O)C[C@H](NC(=O)[C@@H]([NH3+])CCCC[NH3+])C(=O)N[C@@H](CCCC[NH3+])C(=O)[O-]
390.485
-5.9838
224.34
15
27
6
5
0.149662
1b5j
1.8
1,999
LYS-LYS
B
1-3
kd
=
37
nM
-7.431798
MOAD
Kd=37.0nM
P06202
PROTEIN (OLIGO-PEPTIDE BINDING PROTEIN)
NC(=O)CC[C@H](NC(=O)[C@@H]([NH3+])CCCC[NH3+])C(=O)N[C@@H](CCCC[NH3+])C(=O)[O-]
404.512
-5.5937
224.34
16
28
6
5
0.137908
1b6h
1.8
1,998
LYS-LYS
B
1-3
kd
=
0.015
uM
-7.823909
MOAD
Kd=0.015uM
P06202
Periplasmic oligopeptide-binding protein
CCC[C@H](NC(=O)[C@@H]([NH3+])CCCC[NH3+])C(=O)N[C@@H](CCCC[NH3+])C(=O)[O-]
375.514
-4.0591
181.25
15
26
5
4
0.182674
1b6k
1.85
2,000
PI5
A
201
ki
=
1.8
nM
-8.744727
MOAD
Ki=1.8nM
P03369,P03369
RETROPEPSIN,RETROPEPSIN
CC[C@H](C)[C@@H]1NC(=O)[C@@H]([NH2+]C[C@@H](O)[C@H](Cc2ccc(O)cc2)NC(=O)[C@H](C(C)C)N2CCCC2=O)Cc2ccc(cc2)OCCCNC1=O
680.867
1.0317
173.91
12
49
6
7
0.194296
1b6l
1.75
2,000
PI4
A
201
ki
=
5
nM
-8.30103
MOAD
Ki=5.0nM
P03369,P03369
RETROPEPSIN,RETROPEPSIN
CC(C)(C)NC(=O)[C@@H]1CCCC[N@H+]1C[C@@H](O)[C@@H]1Cc2ccc(cc2)OCCCC(=O)N[C@@H](CC(N)=O)C(=O)N1
546.689
-1.0403
164.29
6
39
6
6
0.266852
1b6m
1.85
2,000
PI6
B
201
ki
=
4
nM
-8.39794
MOAD
Ki=4.0nM
P03369,P03369
RETROPEPSIN,RETROPEPSIN
CC[C@H](C)[C@@H]1NC(=O)[C@@H]([NH2+]C[C@@H](O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)Cc2ccc(cc2)OCCCNC1=O
597.777
2.0876
142.6
9
43
5
6
0.299739
1b6p
2.0
2,000
PI7
A
201
ki
=
3
nM
-8.522879
MOAD
Ki=3.0nM
P03369,P03369
RETROPEPSIN,RETROPEPSIN
CCC(=O)N[C@H](C(=O)N[C@@H](Cc1ccc(O)cc1)[C@H](O)C[NH2+][C@H]1Cc2ccc(cc2)OCCCNC(=O)[C@H]([C@@H](C)CC)NC1=O)C(C)C
668.856
0.9355
182.7
13
48
7
7
0.165764
1b74
2.3
2,000
DGN
A
538
ki
=
50
mM
-1.30103
MOAD
Ki=50.0mM
P56868
GLUTAMATE RACEMASE
NC(=O)CC[C@@H]([NH3+])C(=O)[O-]
146.146
-3.3877
110.86
4
10
2
3
0.431057
1b7h
2.0
1,998
LYS-LYS
B
1-3
kd
=
0.0095
uM
-8.022276
MOAD
Kd=0.0095uM
P06202
Periplasmic oligopeptide-binding protein
CCCC[C@H](NC(=O)[C@@H]([NH3+])CCCC[NH3+])C(=O)N[C@@H](CCCC[NH3+])C(=O)[O-]
389.541
-3.669
181.25
16
27
5
4
0.170609
1b8n
2.0
1,999
IMG
A
600
ki
=
30
pM
-10.522879
MOAD
Ki=30.0pM
P55859
PURINE NUCLEOSIDE PHOSPHORYLASE
Nc1nc2c([C@@H]3[NH2+][C@H](CO)[C@@H](O)[C@H]3O)c[nH]c2c(=O)[nH]1
282.28
-3.4658
164.86
2
20
7
6
0.302195
1b8o
1.5
1,999
IMH
A
600
ki
=
23
pM
-10.638272
MOAD
Ki=23.0pM
P55859
PURINE NUCLEOSIDE PHOSPHORYLASE
O=c1[nH]cnc2c([C@@H]3[NH2+][C@H](CO)[C@@H](O)[C@H]3O)c[nH]c12
267.265
-3.048
138.84
2
19
6
5
0.343065
1b8y
2.0
1,999
IN7
A
502
ki
=
14
nM
-7.853872
MOAD
Ki=14.0nM
P08254
PROTEIN (STROMELYSIN-1)
O=C([O-])CNS(=O)(=O)c1ccc(N2CCC(c3ccccc3)CC2)cc1
373.454
1.0988
89.54
6
26
1
5
0.818956
1b9j
1.8
1,999
LYS-LYS
B
1-3
kd
=
1,100
nM
-5.958607
MOAD
Kd=1100.0nM
P06202
PROTEIN (OLIGO-PEPTIDE BINDING PROTEIN)
CC(C)C[C@H](NC(=O)[C@@H]([NH3+])CCCC[NH3+])C(=O)N[C@@H](CCCC[NH3+])C(=O)[O-]
389.541
-3.8131
181.25
15
27
5
4
0.180082
1b9s
2.5
1,999
FDI
A
468
ic50
>
667
uM
-3.175874
MOAD
ic50>667.0uM
P03474
PROTEIN (NEURAMINIDASE)
CCC(CC)C(=O)Nc1cc(C(=O)[O-])ccc1NC(C)=O
291.327
1.3832
98.33
6
21
2
4
0.82687
1b9t
2.4
1,999
RAI
A
468
ic50
=
8
uM
-5.09691
MOAD
ic50=8.0uM
P03474
PROTEIN (NEURAMINIDASE)
NC(=[NH2+])Nc1cc(C(=O)[O-])ccc1N1C(=O)CCC1(CO)CO
322.321
-3.614
164.54
5
23
5
5
0.275671
1b9v
2.35
1,999
RA2
A
468
ic50
=
224
uM
-3.649752
MOAD
ic50=224.0uM
P03474
PROTEIN (NEURAMINIDASE)
CCC(CC)Nc1cc(C(=O)[O-])ccc1N1C(=O)CCC1(CO)CO
349.407
0.5008
112.93
8
25
3
6
0.629882
1bai
2.4
1,999
0Q4
A
125
ki
=
20
nM
-7.69897
MOAD
Ki=20.0nM
P03322,P03322
PROTEASE,PROTEASE
CCCC[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CCC(=O)[O-])NC(=O)[C@H](Cc1ccccc1)[NH2+]C[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@@H]([NH3+])CCCNC(N)=[NH2+])C(C)C)C(N)=O
834.077
-5.4332
336.61
29
59
11
8
0.020677
1bap
1.75
1,992
ARA
A
307
kd
=
0.14
uM
-6.853872
MOAD
Kd=0.14uM
P02924
L-ARABINOSE-BINDING PROTEIN
O[C@@H]1[C@@H](O)[C@@H](O)CO[C@H]1O
150.13
-2.5823
90.15
0
10
4
5
0.30425
1bap
1.75
1,992
ARB
A
308
kd
=
0.14
uM
-6.853872
MOAD
Kd=0.14uM
P02924
L-ARABINOSE-BINDING PROTEIN
O[C@@H]1[C@@H](O)[C@@H](O)OC[C@@H]1O
150.13
-2.5823
90.15
0
10
4
5
0.30425
1bb6
2.0
1,999
UMG
A
130
kd
=
0.000002
M
-5.69897
MOAD
Ka=500000.0M^-1
P11941
LYSOZYME
CC(=O)N[C@H]1[C@@H](Oc2ccc3c(C)cc(=O)oc3c2)O[C@H](CO)[C@@H](O[C@@H]2O[C@H](CO)[C@@H](O[C@@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@H]3NC(C)=O)[C@H](O)[C@H]2NC(C)=O)[C@@H]1O
785.753
-4.64008
314.5
12
55
10
18
0.090496
1bb7
2.0
1,999
GUM
A
130
kd
=
0.000067
M
-4.176091
MOAD
Ka=15000.0M^-1
P11941
LYSOZYME
CC(=O)N[C@H]1[C@H](Oc2ccc3c(C)cc(=O)oc3c2)O[C@H](CO)[C@@H](O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2NC(C)=O)[C@@H]1O
582.559
-2.60808
226.48
8
41
7
13
0.158614
1bcd
1.9
1,993
FMS
A
500
kd
=
2
nM
-8.69897
MOAD
Kd=2.0nM
P00918
CARBONIC ANHYDRASE II
NS(=O)(=O)C(F)(F)F
149.093
-0.2053
60.16
0
8
1
2
0.517815
1bcj
2.1
1,998
NGA
1
1
kd
=
0.2
mM
-3.69897
MOAD
Kd=0.2mM
P19999
MANNOSE-BINDING PROTEIN-A
CC(=O)N[C@@H]1[C@@H](O)[C@@H](O)[C@@H](CO)O[C@H]1O
221.209
-3.0776
119.25
2
15
5
6
0.337239
1bcj
2.1
1,998
NGA
2
1
kd
=
0.2
mM
-3.69897
MOAD
Kd=0.2mM
P19999
MANNOSE-BINDING PROTEIN-A
CC(=O)N[C@@H]1[C@@H](O)[C@@H](O)[C@@H](CO)O[C@H]1O
221.209
-3.0776
119.25
2
15
5
6
0.337239
1bcj
2.1
1,998
NGA
3
1
kd
=
0.2
mM
-3.69897
MOAD
Kd=0.2mM
P19999
MANNOSE-BINDING PROTEIN-A
CC(=O)N[C@@H]1[C@@H](O)[C@@H](O)[C@@H](CO)O[C@H]1O
221.209
-3.0776
119.25
2
15
5
6
0.337239
1bcu
2.0
1,998
PRL
H
280
kd
=
0.53
mM
-3.275724
MOAD
Kd=0.53mM
P00734,P00734
ALPHA-THROMBIN,ALPHA-THROMBIN
Nc1ccc2cc3ccc(N)cc3nc2c1
209.252
2.5524
64.93
0
16
2
3
0.441447
1bf3
2.2
1,998
PHB
A
396
kd
=
120
uM
-3.920819
MOAD
Kd=120.0uM
P00438
P-HYDROXYBENZOATE HYDROXYLASE
O=C([O-])c1ccc(O)cc1
137.114
-0.2443
60.36
1
10
1
3
0.580454
1bfv
2.1
1,997
STG
H
200
kd
~
0
M
-7
MOAD
Ka~10000000.0M^-1
P18529,P01631
FV4155,FV4155
C[C@]12CC[C@@H]3c4ccc(O[C@@H]5O[C@H](C(=O)[O-])[C@@H](O)[C@H](O)[C@H]5O)cc4CC[C@H]3[C@@H]1C[C@@H](O)[C@@H]2O
463.503
-1.1893
159.74
3
33
5
9
0.371375
1bgq
2.5
1,999
RDC
A
300
kd
=
2.7
nM
-8.568636
MOAD
Kd=2.7nM
P02829
HEAT SHOCK PROTEIN 90
C[C@@H]1C[C@H]2O[C@@H]2/C=C\C=C\C(=O)Cc2c(Cl)c(O)cc(O)c2C(=O)O1
364.781
2.6916
96.36
0
25
2
6
0.542437
1bhf
1.8
1,998
ACE-ILE
I
251-255
kd
=
42
uM
-4.376751
MOAD
Kd=42.0uM
P06239
T-LYMPHOCYTE-SPECIFIC PROTEIN TYROSINE KINASE P56LCK
CC[C@H](C)[C@H](NC(=O)[C@H](CCC(=O)[O-])NC(=O)[C@H](CCC(=O)[O-])NC(=O)[C@H](Cc1ccc(CC(=O)[O-])cc1)NC(C)=O)C(=O)[O-]
632.623
-5.6632
276.92
20
45
4
12
0.104675
1bhx
2.3
1,998
R56
F
1
ki
=
0.145
uM
-6.838632
MOAD
Ki=0.145uM
P00734,P00734,P00734
ALPHA THROMBIN,ALPHA THROMBIN,ALPHA THROMBIN
NC(=[NH2+])NCCCNC(=O)[C@@H]1CS[C@H]2CC[C@@H](NS(=O)(=O)Cc3ccccc3)C(=O)N21
469.613
-2.2918
159.22
9
31
5
5
0.15457