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36
36
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4
873
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19
1.07k
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14
3.37k
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1
581
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1
433
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634 values
catalyst_smiles
large_stringlengths
1
683
solvent_smiles
large_stringlengths
1
245
rxn_insight_class
large_stringclasses
11 values
rxn_insight_name
large_stringclasses
346 values
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large_stringlengths
64
64
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64
64
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5
288
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large_stringlengths
24
2.64k
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float64
-0.8
90,205,160,000B
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large_stringlengths
2
864
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float64
-230
30.1k
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large_stringclasses
3 values
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float64
0
4k
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large_stringclasses
4 values
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1
23.6k
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large_stringclasses
96 values
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large_stringclasses
19 values
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large_stringlengths
3
716
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large_stringlengths
3
539
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large_stringlengths
5
293
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large_stringlengths
5
271
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large_stringlengths
5
271
byproduct_smiles
large_stringclasses
176 values
agent_smiles
large_stringlengths
1
712
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float64
-230
30.1k
reaction_time_hours
float64
0
2.16k
reaction_smiles_with_agents
large_stringlengths
4
882
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-5aec4936e2b14990b36f20c777c7be91
O=C(CCCCl)c1ccc(F)cc1>>O=C(c1ccc(F)cc1)C1CC1
ClCCCC(=O)C1=CC=C(C=C1)F.[OH-].[K+]>>C1(CC1)C(=O)C1=CC=C(C=C1)F
Cl[CH2:11][CH2:12][CH2:10][C:2](=[O:1])[c:3]1[cH:4][cH:5][c:6]([F:7])[cH:8][cH:9]1>>[O:1]=[C:2]([c:3]1[cH:4][cH:5][c:6]([F:7])[cH:8][cH:9]1)[CH:10]1[CH2:11][CH2:12]1
O=C(CCCCl)c1ccc(F)cc1
O=C(c1ccc(F)cc1)C1CC1
null
null
O
Functional Group Interconversion
OtherReaction
ba8a5853cba106ae1f1dcc05bcdfa09e62558319dc12ba5eccf6e53858edaf29
d3448bc803db0fe7d73b7f0b0223b52cbc55d6c3e8733418e0ff66fb97fe6c3c
O=C(c1ccccc1)C1CC1
Cl-[CH2;D2;+0:1]-[C:2]-[CH2;D2;+0:3]-[C:4](=[O;D1;H0:5])-[c:6]>>[O;D1;H0:5]=[C:4](-[c:6])-[CH;D3;+0:3]1-[C:2]-[CH2;D2;+0:1]-1
null
[]
null
null
40
MINUTE
Add 20.0 g (0.10 mole) γ-chloro-p-fluorobutyrophenone dropwise to a methanolic KOH solution (prepared from 9.8 g of 86% KOH pellets and 60 ml of methanol). Stir the mixture at room temperature for 40 minutes and pour into 100 ml of water and then extract with 3×30 ml of methylene chloride. Wash the methylene chloride e...
10.6084/m9.figshare.5104873.v1
null
Primary halide.Ketone
Ketone
null
C1CC1
c1ccccc1.C1CC1
HCl
O
null
0.666667
O=C(CCCCl)c1ccc(F)cc1>O>O=C(c1ccc(F)cc1)C1CC1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-92b0f2861ac34052b60247cb0c8be69d
O=C(Cc1ccc(F)cc1)C1CC1>>OC(c1ccc(F)cc1)C1CC1
C1(CC1)C(=O)CC1=CC=C(C=C1)F.[BH4-].[Na+].C(C)(=O)O>>C1(CC1)C(O)C1=CC=C(C=C1)F
C([C:2](=[O:1])[CH:10]1[CH2:11][CH2:12]1)[c:3]1[cH:4][cH:5][c:6]([F:7])[cH:8][cH:9]1>>[OH:1][CH:2]([c:3]1[cH:4][cH:5][c:6]([F:7])[cH:8][cH:9]1)[CH:10]1[CH2:11][CH2:12]1
O=C(Cc1ccc(F)cc1)C1CC1
OC(c1ccc(F)cc1)C1CC1
null
null
C(C)O
Miscellaneous
OtherReaction
daa987aec145c5852e562241e17e37111eea3b585b24d8bb5f6c658727c519bc
65c0f1e474134afe581396038c9eec1081d3cf2c66a067b33a419661521d5253
c1ccc(CC2CC2)cc1
[O;H0;D1;+0:1]=[C;H0;D3;+0:2](-C-[c;H0;D3;+0:3](:[c:4]:[c:5]):[c:6]:[c:7])-[C:8]1-[C:9]-[C:10]-1>>[OH;D1;+0:1]-[CH;D3;+0:2](-[C:8]1-[C:9]-[C:10]-1)-[c;H0;D3;+0:3](:[c:4]:[c:5]):[c:6]:[c:7]
null
[]
null
null
6
HOUR
Add 3.2 g (0.085 mole) cyclopropyl-4-fluorobenzylmethanone to 80 ml of 3.2 g (0.085 mole) sodium borohydride partially dissolved in absolute ethanol, following the reaction by thin-layer chromatography. After about 6 hours at room temperature, cool the reaction in an ice bath and add acetic acid. Extract the mixture wi...
10.6084/m9.figshare.5104873.v1
null
Ketone
Secondary alcohol
c1ccccc1
c1ccccc1
c1ccccc1.C1CC1
Other
C(C)O
null
6
O=C(Cc1ccc(F)cc1)C1CC1>C(C)O>OC(c1ccc(F)cc1)C1CC1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-e683030b619748749d3b54d0c6f9699e
Cl.OC(c1ccc(F)cc1)C1CC1>>Fc1ccc(/C=C/CCCl)cc1
C1(CC1)C(O)C1=CC=C(C=C1)F.Cl>>ClCC/C=C/C1=CC=C(C=C1)F
[ClH:10].O[CH:6]([c:5]1[cH:4][cH:3][c:2]([F:1])[cH:12][cH:11]1)[CH:7]1[CH2:8][CH2:9]1>>[F:1][c:2]1[cH:3][cH:4][c:5](/[CH:6]=[CH:7]/[CH2:8][CH2:9][Cl:10])[cH:11][cH:12]1
Cl.OC(c1ccc(F)cc1)C1CC1
Fc1ccc(/C=C/CCCl)cc1
null
null
C(Cl)(Cl)Cl
Miscellaneous
OtherReaction
38776c52da3dcee213ec339130f3a6eb8327d8aaa90f172b6e0d73056aef0190
8452b9e7b957d084b8e6296c5c757c325bf3c4bf79ebb0ec829e6b9eb1c76119
c1ccccc1
O-[CH;D3;+0:1](-[CH;D3;+0:2]1-[C:3]-[CH2;D2;+0:4]-1)-[c:5](:[c:6]):[c:7].[ClH;D0;+0:8]>>[Cl;H0;D1;+0:8]-[CH2;D2;+0:4]-[C:3]/[CH;D2;+0:2]=[CH;D2;+0:1]/[c:5](:[c:6]):[c:7]
null
[]
null
null
null
null
Dissolve 12.8 g (0.077 mole) of α-cyclopropyl-4-fluorobenzenemethanol in 60 ml of CHCl3, add 20 ml of concentrated HCl and reflux overnight. Separate the two layers, and extract the aqueous layer with methylene chloride. Combine the methylene chloride extracts with the chloroform layer and wash with saturated aqueous s...
10.6084/m9.figshare.5104873.v1
null
Secondary alcohol
Primary halide
C1CC1
null
c1ccccc1
HO-
C(Cl)(Cl)Cl
null
null
Cl.OC(c1ccc(F)cc1)C1CC1>C(Cl)(Cl)Cl>Fc1ccc(/C=C/CCCl)cc1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-ba9c9b48fdb74de58d6c82f059e70a26
C=C=COC.Clc1ccc(Br)cc1>>C#CCc1ccc(Cl)cc1
BrC1=CC=C(C=C1)Cl.[Cl-].[NH4+].BrC1=CC=C(C=C1)Cl.COC=C=C.[Mg]>>ClC1=CC=C(C=C1)CC#C
CO[CH:1]=[C:2]=[CH2:3].Br[c:4]1[cH:5][cH:6][c:7]([Cl:8])[cH:9][cH:10]1>>[CH:1]#[C:2][CH2:3][c:4]1[cH:5][cH:6][c:7]([Cl:8])[cH:9][cH:10]1
C=C=COC.Clc1ccc(Br)cc1
C#CCc1ccc(Cl)cc1
null
null
CCOCC.OC(CN1C=NC=C1)C1=CC=C(C=C1)NS(=O)(=O)C
C-C Coupling
OtherReaction
d463bef59147a48ffa0bdcc2f2f7a5cbe0a47fb61f5677cff6959b17d4edaee0
959abc43744b7d49d3e4fd04c436d5ff1da10d013edea2fdc4015d8e383fb9c0
c1ccccc1
Br-[c;H0;D3;+0:1](:[c:2]:[c:3]):[c:4]:[c:5].C-O-[CH;D2;+0:6]=[C;H0;D2;+0:7]=[CH2;D1;+0:8]>>[CH;D1;+0:6]#[C;H0;D2;+0:7]-[CH2;D2;+0:8]-[c;H0;D3;+0:1](:[c:2]:[c:3]):[c:4]:[c:5]
null
[]
null
null
null
null
In a flask containing 59 g (2.43 mole) magnesium turnings in 500 ml anhydrous ether under an atmosphere of nitroge add slowly a solution of 465 g (2.43 mole) of 4-bromochlorobenzene in 1 liter 4 anhydrous ether. With caution, once the Grignard has started maintain slow reflux until all 4-bromochlorobenzene has been add...
10.6084/m9.figshare.5104873.v1
null
Aromatic halide.Ether.Allene
Alkyne
c1ccccc1
c1ccccc1
c1ccccc1
HBr
CCOCC.OC(CN1C=NC=C1)C1=CC=C(C=C1)NS(=O)(=O)C
null
null
C=C=COC.Clc1ccc(Br)cc1>CCOCC.OC(CN1C=NC=C1)C1=CC=C(C=C1)NS(=O)(=O)C>C#CCc1ccc(Cl)cc1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-b179caa1edde4d7db85b74b59893ce31
C#CCc1ccc(Cl)cc1.C=O>>CC#CC(O)c1ccc(Cl)cc1
[Cl-].[Na+].ClC1=CC=C(C=C1)CC#C.C(CCC)[Li].C=O>>ClC1=CC=C(C=C1)C(C#CC)O
[CH:2]#[C:3][CH2:4][c:6]1[cH:7][cH:8][c:9]([Cl:10])[cH:11][cH:12]1.[CH2:1]=[O:5]>>[CH3:1][C:2]#[C:3][CH:4]([OH:5])[c:6]1[cH:7][cH:8][c:9]([Cl:10])[cH:11][cH:12]1
C#CCc1ccc(Cl)cc1.C=O
CC#CC(O)c1ccc(Cl)cc1
null
null
CCCCCC.CCOCC
Heteroatom Alkylation and Arylation
OtherReaction
a680c0cf8515532e7e0210252422e861ecf3c6c70d246905f921324730c1f764
28d240c35612efe41f2146d35d9bbe8f29ec1a21f7fa08aecaf86256546f8ff7
c1ccccc1
[CH2;D1;+0:1]=[O;H0;D1;+0:2].[CH;D1;+0:3]#[C:4]-[CH2;D2;+0:5]-[c:6](:[c:7]):[c:8]>>[CH3;D1;+0:1]-[C;H0;D2;+0:3]#[C:4]-[CH;D3;+0:5](-[OH;D1;+0:2])-[c:6](:[c:7]):[c:8]
null
[]
null
null
30
MINUTE
Under nitrogen and with cooling, to a solution of 150.6 g (1.0 mole) 1-chloro-4-(2-propynyl)benzene in 600 ml of anhydrous ether, add dropwise 400 ml of 2.5M n-butyllithium (1.0 mole) in hexane. When addition is complete, stir a further 30 minutes and under N2 add 31 g of para-formaldehyde. Stir the mixture in a dry ic...
10.6084/m9.figshare.5104873.v1
null
Formaldehyde.Alkyne
Secondary alcohol.Alkyne
null
null
c1ccccc1
null
CCCCCC.CCOCC
null
0.5
C#CCc1ccc(Cl)cc1.C=O>CCCCCC.CCOCC>CC#CC(O)c1ccc(Cl)cc1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-93abc6b367ac4c85828867dcc8b49366
CC#CC(O)c1ccc(Cl)cc1>>C/C=C\C(O)c1ccc(Cl)cc1
ClC1=CC=C(C=C1)C(C#CC)O>>ClC1=CC=C(C=C1)C(\C=C/C)O
[CH3:1][C:2]#[C:3][CH:4]([OH:5])[c:6]1[cH:7][cH:8][c:9]([Cl:10])[cH:11][cH:12]1>>[CH3:1]/[CH:2]=[CH:3]\[CH:4]([OH:5])[c:6]1[cH:7][cH:8][c:9]([Cl:10])[cH:11][cH:12]1
CC#CC(O)c1ccc(Cl)cc1
C/C=C\C(O)c1ccc(Cl)cc1
null
[Pd].CC(=O)[O-].CC(=O)[O-].[Pb+2]
null
Reduction
Hydrogenation (triple to double)
2bb8d5b532a2781e0a7c069a5cd3e8a7e8d44660c0ec1d9e17c04d8ba2cb383b
1990560e9c55934bde8ca0feaed9c61d80f37f94f0cf240a9929dc374d0a33aa
c1ccccc1
[C;D1;H3:1]-[C;H0;D2;+0:2]#[C;H0;D2;+0:3]-[C:4](-[O;D1;H1:5])-[c:6]>>[C;D1;H3:1]/[CH;D2;+0:2]=[CH;D2;+0:3]\[C:4](-[O;D1;H1:5])-[c:6]
null
[]
null
null
2
DAY
Under nitrogen, hydrogenate a mixture of 10 g (0.055 mole) of 1-(4-chlorophenyl)-2-butyn-1-ol and 0.6 g Lindlar catalyst. Following the reaction via NMR the reaction is complete in about two days. The hydrogenation is stopped and the reaction stirred under N2 at room temperature overnight. Filter off the catalysts, was...
10.6084/m9.figshare.5104873.v1
null
Alkyne
null
null
null
c1ccccc1
null
[Pd].CC(=O)[O-].CC(=O)[O-].[Pb+2]
null
48
CC#CC(O)c1ccc(Cl)cc1>[Pd].CC(=O)[O-].CC(=O)[O-].[Pb+2]>C/C=C\C(O)c1ccc(Cl)cc1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-0dd86c3f04a44ab8bb79b472f6559150
C/C=C\C(O)c1ccc(Cl)cc1.Cc1ccc(S(=O)(=O)Cl)cc1.[OH-]>>Cc1ccc(S(=O)(=O)[O-])cc1.OC/C=C\Cc1ccc(Cl)cc1
C1(=CC=C(C=C1)S(=O)(=O)Cl)C.ClC1=CC=C(C=C1)C(\C=C/C)O.[OH-].[K+]>>ClC1=CC=C(C=C1)C\C=C/CO.CC1=CC=C(C=C1)S(=O)(=O)[O-]
[OH:12][CH:16](/[CH:15]=[CH:14]\[CH3:13])[c:17]1[cH:18][cH:19][c:20]([Cl:21])[cH:22][cH:23]1.Cl[S:6]([c:5]1[cH:4][cH:3][c:2]([CH3:1])[cH:11][cH:10]1)(=[O:7])=[O:8].[OH-:9]>>[CH3:1][c:2]1[cH:3][cH:4][c:5]([S:6](=[O:7])(=[O:8])[O-:9])[cH:10][cH:11]1.[OH:12][CH2:13]/[CH:14]=[CH:15]\[CH2:16][c:17]1[cH:18][cH:19][c:20]([Cl:...
C/C=C\C(O)c1ccc(Cl)cc1.Cc1ccc(S(=O)(=O)Cl)cc1.[OH-]
Cc1ccc(S(=O)(=O)[O-])cc1.OC/C=C\Cc1ccc(Cl)cc1
null
null
CCOCC
Acylation
OtherReaction
8d4c958d57c5893436aa88ba1f5a74f2b58c73a3b83674dc98a2d1b6d9b25311
5bc8747d49693f36603549f26fda054bb5784c3dcc17d9b54a3a2bf840b3fcaf
c1ccccc1.c1ccccc1
Cl-[S;H0;D4;+0:1](=[O;D1;H0:2])(=[O;D1;H0:3])-[c:4](:[c:5]):[c:6].[CH3;D1;+0:7]/[C:8]=[C:9]\[CH;D3;+0:10](-[OH;D1;+0:11])-[c:12](:[c:13]):[c:14].[OH-;D0:15]>>[O-;H0;D1:15]-[S;H0;D4;+0:1](=[O;D1;H0:2])(=[O;D1;H0:3])-[c:4](:[c:5]):[c:6].[OH;D1;+0:11]-[CH2;D2;+0:7]/[C:8]=[C:9]\[CH2;D2;+0:10]-[c:12](:[c:13]):[c:14]
null
[]
null
null
null
null
Dissolve 6.7 g (0.036 mole) of (Z)-1-(4-chlorophenyl)-2-buten-1-ol in 100 ml of anhydrous ether, add 3.2 g of powdered KOH. Stir the mixture and with cooling add a solution of 7.0 g p-toluenesulfonylchloride in 30 ml of anhydrous ether. Continue to stir with cooling for 30 minutes, then allow to warm to room temperatur...
10.6084/m9.figshare.5104873.v1
null
Tosylate.Secondary alcohol.Sulfonyl halide
Tosylate.Primary alcohol
null
null
c1ccccc1.c1ccccc1
HCl
CCOCC
null
null
C/C=C\C(O)c1ccc(Cl)cc1.Cc1ccc(S(=O)(=O)Cl)cc1.[OH-]>CCOCC>Cc1ccc(S(=O)(=O)[O-])cc1.OC/C=C\Cc1ccc(Cl)cc1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-ba1cfec2e5b445d2b5b9aeef73074f39
CS(=O)(=O)Cl.Nc1ccccc1>>CS(=O)(=O)Nc1ccccc1
NC1=CC=CC=C1.N1=CC=CC=C1.CS(=O)(=O)Cl>>C1(=CC=CC=C1)NS(=O)(=O)C
Cl[S:2]([CH3:1])(=[O:3])=[O:4].[NH2:5][c:6]1[cH:7][cH:8][cH:9][cH:10][cH:11]1>>[CH3:1][S:2](=[O:3])(=[O:4])[NH:5][c:6]1[cH:7][cH:8][cH:9][cH:10][cH:11]1
CS(=O)(=O)Cl.Nc1ccccc1
CS(=O)(=O)Nc1ccccc1
null
null
C(Cl)Cl
Miscellaneous
Sulfonamide synthesis (Schotten-Baumann) primary amine
a86b0632821e188c0a5dc5a5a2aac298ab3eccaee8a52ba46078c3d5975a290d
50f8fbf3d327483c3eeff8f6cbd4065e4c7600bb501fbe08958a5c79a0926428
c1ccccc1
Cl-[S;H0;D4;+0:1](-[C;D1;H3:2])(=[O;D1;H0:3])=[O;D1;H0:4].[NH2;D1;+0:5]-[c:6](:[c:7]):[c:8]>>[C;D1;H3:2]-[S;H0;D4;+0:1](=[O;D1;H0:3])(=[O;D1;H0:4])-[NH;D2;+0:5]-[c:6](:[c:7]):[c:8]
null
[]
0
CELSIUS
30
MINUTE
To a 0° C. solution of 250 g (2.68 mole) of aniline and 233.2 g (2.95 mole) of pyridine in 1.25 L of methylene chloride and 319.6 g (2.79 mole) of methanesulfonyl chloride dropwise. Stir the resulting solution at 0° C. for about 30 minutes then warm to ambient temperature for about 16 hours. Extract the mixture with 2N...
10.6084/m9.figshare.5104873.v1
null
Primary amine.Sulfonyl halide
Sulfonamide
null
null
c1ccccc1
HCl
C(Cl)Cl
0
0.5
CS(=O)(=O)Cl.Nc1ccccc1>C(Cl)Cl>CS(=O)(=O)Nc1ccccc1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-03a078946e734c8a99d29a0b27efcafc
CS(=O)(=O)Nc1ccccc1.O=C(Cl)CCl>>CS(=O)(=O)Nc1ccc(C(=O)CCl)cc1
C1(=CC=CC=C1)NS(=O)(=O)C.ClCC(=O)Cl.Cl.[Cl-].[Al+3].[Cl-].[Cl-]>>ClCC(=O)C1=CC=C(C=C1)NS(=O)(=O)C
[CH3:1][S:2](=[O:3])(=[O:4])[NH:5][c:6]1[cH:7][cH:8][cH:9][cH:14][cH:15]1.Cl[C:10](=[O:11])[CH2:12][Cl:13]>>[CH3:1][S:2](=[O:3])(=[O:4])[NH:5][c:6]1[cH:7][cH:8][c:9]([C:10](=[O:11])[CH2:12][Cl:13])[cH:14][cH:15]1
CS(=O)(=O)Nc1ccccc1.O=C(Cl)CCl
CS(=O)(=O)Nc1ccc(C(=O)CCl)cc1
null
null
C(Cl)Cl
C-C Coupling
Friedel-Crafts acylation
55541449ad4f182ef3dc0497085b282b1dcb76e0fb5ed140dc4eab4973eacb28
fe2a4a0dfbb5b71b9a065e092364c64b22b4eb1ad4d6ba2a1e8edc9d31fce3e4
c1ccccc1
Cl-[C;H0;D3;+0:1](=[O;D1;H0:2])-[C:3]-[Cl;D1;H0:4].[c:5]:[c:6]:[cH;D2;+0:7]:[c:8]:[c:9]>>[Cl;D1;H0:4]-[C:3]-[C;H0;D3;+0:1](=[O;D1;H0:2])-[c;H0;D3;+0:7](:[c:6]:[c:5]):[c:8]:[c:9]
null
[]
-10
CELSIUS
16
HOUR
In a flask containing 128.4 g (0.75 mole) of N-phenylmethanesulfonamide, 169.5 g (1.50 mole) of chloroacetyl chloride in 1 L of methylene chloride under an atmosphere of nitrogen and cooled to about -10° C. add 300 g (2.25 mole) of aluminum chloride. Stir the resulting mixture for about 16 hours. Pour the reaction mixt...
10.6084/m9.figshare.5104873.v1
null
Acyl halide
Ketone
c1ccccc1
c1ccccc1
c1ccccc1
HCl
C(Cl)Cl
-10
16
CS(=O)(=O)Nc1ccccc1.O=C(Cl)CCl>C(Cl)Cl>CS(=O)(=O)Nc1ccc(C(=O)CCl)cc1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-708517c15fa34a6a9187edfc91752e67
COc1ccc(CCCBr)cc1.Cn1ccnc1>>COc1ccc(CCC[n+]2ccn(C)c2)cc1.[Br-]
CN1C=NC=C1.BrCCCC1=CC=C(C=C1)OC>>[Br-].COC1=CC=C(C=C1)CCC[N+]1=CN(C=C1)C
[CH3:1][O:2][c:3]1[cH:4][cH:5][c:6]([CH2:7][CH2:8][CH2:9][Br:18])[cH:16][cH:17]1.[n:10]1[cH:11][cH:12][n:13]([CH3:14])[cH:15]1>>[CH3:1][O:2][c:3]1[cH:4][cH:5][c:6]([CH2:7][CH2:8][CH2:9][n+:10]2[cH:11][cH:12][n:13]([CH3:14])[cH:15]2)[cH:16][cH:17]1.[Br-:18]
COc1ccc(CCCBr)cc1.Cn1ccnc1
COc1ccc(CCC[n+]2ccn(C)c2)cc1.[Br-]
null
null
null
Functional Group Interconversion
OtherReaction
5e72d8623d1d11df3a484f13beed495bb29975189dd55fb2f640a2dac5643123
47a659f5704a5b7ca1b92ff731f18f109c6bde1d45152a3a393eefbd10265508
c1ccc(CCC[n+]2cc[nH]c2)cc1
[Br;H0;D1;+0:1]-[CH2;D2;+0:2]-[C:3]-[C:4].[C;D1;H3:5]-[#7;a:6]1:[c:7]:[c:8]:[n;H0;D2;+0:9]:[c:10]:1>>[Br-;H0;D0:1].[C:4]-[C:3]-[CH2;D2;+0:2]-[n+;H0;D3:9]1:[c:8]:[c:7]:[#7;a:6](-[C;D1;H3:5]):[c:10]:1
null
[]
140
CELSIUS
null
null
A mixture of 2.50 g (0.03 mole) of 1-methyl-1H-imidazole and 6.9 g (0.03 mole) of 1-(3-bromopropyl)-4-methoxybenzene is heated at 140° C. for 1.5 hours. Follow the progress of the reaction by thin-layer chromatography on silica gel (methanol:1M sodium chloride, 95:5). At the completion, the cooled reaction product is t...
10.6084/m9.figshare.5104873.v1
null
Primary halide
null
c1c[nH]cn1
c1c[n+]cn1
c1ccccc1.c1c[n+]cn1
null
null
140
null
COc1ccc(CCCBr)cc1.Cn1ccnc1>>COc1ccc(CCC[n+]2ccn(C)c2)cc1.[Br-]
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-713fc3bc0f894dfc920890737d051b18
CCCCn1ccnc1.COc1ccc(CCCBr)cc1>>CCCC[n+]1ccn(CCCc2ccc(OC)cc2)c1.[Br-]
C(CCC)N1C=NC=C1.BrCCCC1=CC=C(C=C1)OC>>[Br-].C(CCC)[N+]1=CN(C=C1)CCCC1=CC=C(C=C1)OC
[CH3:1][CH2:2][CH2:3][CH2:4][n:5]1[cH:6][cH:7][n:8][cH:20]1.[CH2:9]([CH2:10][CH2:11][c:12]1[cH:13][cH:14][c:15]([O:16][CH3:17])[cH:18][cH:19]1)[Br:21]>>[CH3:1][CH2:2][CH2:3][CH2:4][n+:5]1[cH:6][cH:7][n:8]([CH2:9][CH2:10][CH2:11][c:12]2[cH:13][cH:14][c:15]([O:16][CH3:17])[cH:18][cH:19]2)[cH:20]1.[Br-:21]
CCCCn1ccnc1.COc1ccc(CCCBr)cc1
CCCC[n+]1ccn(CCCc2ccc(OC)cc2)c1.[Br-]
null
null
null
Functional Group Interconversion
OtherReaction
5e72d8623d1d11df3a484f13beed495bb29975189dd55fb2f640a2dac5643123
47a659f5704a5b7ca1b92ff731f18f109c6bde1d45152a3a393eefbd10265508
c1ccc(CCCn2cc[nH+]c2)cc1
[Br;H0;D1;+0:1]-[CH2;D2;+0:2]-[C:3]-[C:4].[C:5]-[C:6]-[n;H0;D3;+0:7]1:[c:8]:[n;H0;D2;+0:9]:[c:10]:[c:11]:1>>[Br-;H0;D0:1].[C:4]-[C:3]-[CH2;D2;+0:2]-[n;H0;D3;+0:9]1:[c:8]:[n+;H0;D3:7](-[C:6]-[C:5]):[c:11]:[c:10]:1
null
[]
140
CELSIUS
null
null
A mixture of 2.5 g (0.02 mole) of 1-butyl-1H-imidazole and 4.61 g (0.02 mole) of 1-(3-bromopropyl)-4-methoxybenzene is heated at 140° C. for about 1.5 hours. Follow the progress of the reaction by thin-layer chromatography on silica gel (methanol: 1M sodium chloride, 95:5). At the completion of the reaction, the cooled...
10.6084/m9.figshare.5104873.v1
null
Primary halide
null
c1c[nH]cn1
c1c[n+]cn1
c1c[n+]cn1.c1ccccc1
null
null
140
null
CCCCn1ccnc1.COc1ccc(CCCBr)cc1>>CCCC[n+]1ccn(CCCc2ccc(OC)cc2)c1.[Br-]
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-0975481c31384d8881e268fde82a7716
CCCCCCCn1ccnc1.COc1ccc(CCCBr)cc1>>CCCCCCC[n+]1ccn(CCCc2ccc(OC)cc2)c1.[Br-]
C(CCCCCC)N1C=NC=C1.BrCCCC1=CC=C(C=C1)OC>>[Br-].C(CCCCCC)[N+]1=CN(C=C1)CCCC1=CC=C(C=C1)OC
[CH3:1][CH2:2][CH2:3][CH2:4][CH2:5][CH2:6][CH2:7][n:8]1[cH:9][cH:10][n:11][cH:23]1.[CH2:12]([CH2:13][CH2:14][c:15]1[cH:16][cH:17][c:18]([O:19][CH3:20])[cH:21][cH:22]1)[Br:24]>>[CH3:1][CH2:2][CH2:3][CH2:4][CH2:5][CH2:6][CH2:7][n+:8]1[cH:9][cH:10][n:11]([CH2:12][CH2:13][CH2:14][c:15]2[cH:16][cH:17][c:18]([O:19][CH3:20])[...
CCCCCCCn1ccnc1.COc1ccc(CCCBr)cc1
CCCCCCC[n+]1ccn(CCCc2ccc(OC)cc2)c1.[Br-]
null
null
null
Functional Group Interconversion
OtherReaction
5e72d8623d1d11df3a484f13beed495bb29975189dd55fb2f640a2dac5643123
47a659f5704a5b7ca1b92ff731f18f109c6bde1d45152a3a393eefbd10265508
c1ccc(CCCn2cc[nH+]c2)cc1
[Br;H0;D1;+0:1]-[CH2;D2;+0:2]-[C:3]-[C:4].[C:5]-[C:6]-[n;H0;D3;+0:7]1:[c:8]:[n;H0;D2;+0:9]:[c:10]:[c:11]:1>>[Br-;H0;D0:1].[C:4]-[C:3]-[CH2;D2;+0:2]-[n;H0;D3;+0:9]1:[c:10]:[c:11]:[n+;H0;D3:7](-[C:6]-[C:5]):[c:8]:1
null
[]
140
CELSIUS
null
null
A mixture of 2.5 g (0.015 mole) of 1-heptyl-1H-imidazole and 3.45 g (0.015 mole) of 1-(3-bromopropyl)-4-methoxybenzene is heated at 140° C. for about 1.5 hours. Follow the progress of the reaction by thin-layer chromatography on silica gel (methanol: 1M sodium chloride, 95:5). At the completion of the reaction, the coo...
10.6084/m9.figshare.5104873.v1
null
Primary halide
null
c1c[nH]cn1
c1c[n+]cn1
c1c[n+]cn1.c1ccccc1
null
null
140
null
CCCCCCCn1ccnc1.COc1ccc(CCCBr)cc1>>CCCCCCC[n+]1ccn(CCCc2ccc(OC)cc2)c1.[Br-]
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-511fd087a3a740b095b9c1e3aec28d32
CCCCCCCn1ccnc1.COc1ccc(CCCCBr)cc1>>CCCCCCC[n+]1ccn(CCCCc2ccc(OC)cc2)c1.[Br-]
C(CCCCCC)N1C=NC=C1.BrCCCCC1=CC=C(C=C1)OC>>[Br-].C(CCCCCC)[N+]1=CN(C=C1)CCCCC1=CC=C(C=C1)OC
[CH3:1][CH2:2][CH2:3][CH2:4][CH2:5][CH2:6][CH2:7][n:8]1[cH:9][cH:10][n:11][cH:24]1.[CH2:12]([CH2:13][CH2:14][CH2:15][c:16]1[cH:17][cH:18][c:19]([O:20][CH3:21])[cH:22][cH:23]1)[Br:25]>>[CH3:1][CH2:2][CH2:3][CH2:4][CH2:5][CH2:6][CH2:7][n+:8]1[cH:9][cH:10][n:11]([CH2:12][CH2:13][CH2:14][CH2:15][c:16]2[cH:17][cH:18][c:19](...
CCCCCCCn1ccnc1.COc1ccc(CCCCBr)cc1
CCCCCCC[n+]1ccn(CCCCc2ccc(OC)cc2)c1.[Br-]
null
null
null
Functional Group Interconversion
OtherReaction
5e72d8623d1d11df3a484f13beed495bb29975189dd55fb2f640a2dac5643123
47a659f5704a5b7ca1b92ff731f18f109c6bde1d45152a3a393eefbd10265508
c1ccc(CCCCn2cc[nH+]c2)cc1
[Br;H0;D1;+0:1]-[CH2;D2;+0:2]-[C:3]-[C:4].[C:5]-[C:6]-[n;H0;D3;+0:7]1:[c:8]:[n;H0;D2;+0:9]:[c:10]:[c:11]:1>>[Br-;H0;D0:1].[C:4]-[C:3]-[CH2;D2;+0:2]-[n;H0;D3;+0:9]1:[c:10]:[c:11]:[n+;H0;D3:7](-[C:6]-[C:5]):[c:8]:1
null
[]
140
CELSIUS
null
null
A mixture of 2.5 g (0.015 mole) of 1-heptyl-1H-imidazole and 3.66 g (0.015 mole) of 1-(4-bromobutyl)-4-methoxybenzene is heated at 140° C. for about 2 hours. Follow the progress of the reaction by thin-layer chromatography on silica gel (methanol: 1M sodium chloride, 95:5). At the completion of the reaction, the cooled...
10.6084/m9.figshare.5104873.v1
null
Primary halide
null
c1c[nH]cn1
c1c[n+]cn1
c1c[n+]cn1.c1ccccc1
null
null
140
null
CCCCCCCn1ccnc1.COc1ccc(CCCCBr)cc1>>CCCCCCC[n+]1ccn(CCCCc2ccc(OC)cc2)c1.[Br-]
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-31255a6f17e14a98850eb525acf68772
CCCCCCCn1ccnc1C.COc1ccc(CCCCBr)cc1>>CCCCCCC[n+]1ccn(CCCCc2ccc(OC)cc2)c1C.[Br-]
C(CCCCCC)N1C(=NC=C1)C.BrCCCCC1=CC=C(C=C1)OC>>[Br-].C(CCCCCC)[N+]1=C(N(C=C1)CCCCC1=CC=C(C=C1)OC)C
[CH3:1][CH2:2][CH2:3][CH2:4][CH2:5][CH2:6][CH2:7][n:8]1[cH:9][cH:10][n:11][c:24]1[CH3:25].[CH2:12]([CH2:13][CH2:14][CH2:15][c:16]1[cH:17][cH:18][c:19]([O:20][CH3:21])[cH:22][cH:23]1)[Br:26]>>[CH3:1][CH2:2][CH2:3][CH2:4][CH2:5][CH2:6][CH2:7][n+:8]1[cH:9][cH:10][n:11]([CH2:12][CH2:13][CH2:14][CH2:15][c:16]2[cH:17][cH:18]...
CCCCCCCn1ccnc1C.COc1ccc(CCCCBr)cc1
CCCCCCC[n+]1ccn(CCCCc2ccc(OC)cc2)c1C.[Br-]
null
null
null
Functional Group Interconversion
OtherReaction
f4daa7bb824cdaa37f41c90ce9b52b8d64e0bc7c78bf6b7cb7ce4ccad42f806e
47a659f5704a5b7ca1b92ff731f18f109c6bde1d45152a3a393eefbd10265508
c1ccc(CCCCn2cc[nH+]c2)cc1
[Br;H0;D1;+0:1]-[CH2;D2;+0:2]-[C:3]-[C:4].[C:5]-[C:6]-[n;H0;D3;+0:7]1:[c:8]:[c:9]:[n;H0;D2;+0:10]:[c:11]:1-[C;D1;H3:12]>>[Br-;H0;D0:1].[C:4]-[C:3]-[CH2;D2;+0:2]-[n;H0;D3;+0:10]1:[c:9]:[c:8]:[n+;H0;D3:7](-[C:6]-[C:5]):[c:11]:1-[C;D1;H3:12]
null
[]
140
CELSIUS
null
null
A mixture of 2.50 g (0.0139 mole) of 1-heptyl-2-methyl-1H-imidazole and 3.37 g (0.0139 mole) of 1-(4-bromobutyl)-4-methoxybenzene is heated at 140° C. for about 2 hours. Follow the progress of the reaction by thin-layer chromatography on silica gel (methanol:1M sodium chloride, 95:5). At the completion of the reaction,...
10.6084/m9.figshare.5104873.v1
null
Primary halide
null
c1ncc[nH]1
c1ncc[n+]1
c1ncc[n+]1.c1ccccc1
null
null
140
null
CCCCCCCn1ccnc1C.COc1ccc(CCCCBr)cc1>>CCCCCCC[n+]1ccn(CCCCc2ccc(OC)cc2)c1C.[Br-]
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-4ca4ceb16eef4cdaa4b6731e37e52fb8
CCCCCCCn1ccnc1.Cc1cccc(C)c1NS(=O)(=O)CCCCl>>CCCCCCCn1cc[n+](CCCS(=O)(=O)Nc2c(C)cccc2C)c1.[Cl-]
C(CCCCCC)N1C=NC=C1.ClCCCS(=O)(=O)NC1=C(C=CC=C1C)C>>[Cl-].CC1=C(C(=CC=C1)C)NS(=O)(=O)CCC[N+]1=CN(C=C1)CCCCCCC
[CH3:1][CH2:2][CH2:3][CH2:4][CH2:5][CH2:6][CH2:7][n:8]1[cH:9][cH:10][n:11][cH:27]1.[CH2:12]([CH2:13][CH2:14][S:15](=[O:16])(=[O:17])[NH:18][c:19]1[c:20]([CH3:21])[cH:22][cH:23][cH:24][c:25]1[CH3:26])[Cl:28]>>[CH3:1][CH2:2][CH2:3][CH2:4][CH2:5][CH2:6][CH2:7][n:8]1[cH:9][cH:10][n+:11]([CH2:12][CH2:13][CH2:14][S:15](=[O:1...
CCCCCCCn1ccnc1.Cc1cccc(C)c1NS(=O)(=O)CCCCl
CCCCCCCn1cc[n+](CCCS(=O)(=O)Nc2c(C)cccc2C)c1.[Cl-]
null
null
O
Functional Group Interconversion
OtherReaction
af9372efd0d4cbb040a1d2fa469660cc7709681c6c0eb3b6dabfb715f74188ec
47a659f5704a5b7ca1b92ff731f18f109c6bde1d45152a3a393eefbd10265508
O=S(=O)(CCC[n+]1cc[nH]c1)Nc1ccccc1
[C:1]-[#7;a:2]1:[c:3]:[n;H0;D2;+0:4]:[c:5]:[c:6]:1.[C:7]-[C:8]-[CH2;D2;+0:9]-[Cl;H0;D1;+0:10]>>[C:7]-[C:8]-[CH2;D2;+0:9]-[n+;H0;D3:4]1:[c:5]:[c:6]:[#7;a:2](-[C:1]):[c:3]:1.[Cl-;H0;D0:10]
null
[]
null
null
null
null
Combine 15.0 g (0.0919 mole) 1-heptyl-1H-imidazole and 25.5 g (0.0974 mole) 3-chloro-N-(2,6-dimethylphenyl)propanesulfonamide and heat for about 24 hours at 130° C. Follow the progress of the reaction by thin-layer chromatography on silica gel (acetonitrile: ammonium hydroxide, 9:1). At the completion of the reaction, ...
10.6084/m9.figshare.5104873.v1
null
Primary halide
null
c1c[nH]cn1
c1c[nH]c[n+]1
c1c[nH]c[n+]1.c1ccccc1
null
O
null
null
CCCCCCCn1ccnc1.Cc1cccc(C)c1NS(=O)(=O)CCCCl>O>CCCCCCCn1cc[n+](CCCS(=O)(=O)Nc2c(C)cccc2C)c1.[Cl-]
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-755407445f384b12b9268816db7e0b34
CCCCCCCn1ccnc1.ClCCCCc1ccccc1>>CCCCCCC[n+]1ccn(CCCCc2ccccc2)c1.[Cl-]
ClCCCCC1=CC=CC=C1.C(CCCCCC)N1C=NC=C1>>[Cl-].C(CCCCCC)[N+]1=CN(C=C1)CCCCC1=CC=CC=C1
[CH3:1][CH2:2][CH2:3][CH2:4][CH2:5][CH2:6][CH2:7][n:8]1[cH:9][cH:10][n:11][cH:22]1.[CH2:12]([CH2:13][CH2:14][CH2:15][c:16]1[cH:17][cH:18][cH:19][cH:20][cH:21]1)[Cl:23]>>[CH3:1][CH2:2][CH2:3][CH2:4][CH2:5][CH2:6][CH2:7][n+:8]1[cH:9][cH:10][n:11]([CH2:12][CH2:13][CH2:14][CH2:15][c:16]2[cH:17][cH:18][cH:19][cH:20][cH:21]2...
CCCCCCCn1ccnc1.ClCCCCc1ccccc1
CCCCCCC[n+]1ccn(CCCCc2ccccc2)c1.[Cl-]
null
null
CO
Functional Group Interconversion
OtherReaction
5e72d8623d1d11df3a484f13beed495bb29975189dd55fb2f640a2dac5643123
47a659f5704a5b7ca1b92ff731f18f109c6bde1d45152a3a393eefbd10265508
c1ccc(CCCCn2cc[nH+]c2)cc1
[C:1]-[C:2]-[CH2;D2;+0:3]-[Cl;H0;D1;+0:4].[C:5]-[C:6]-[n;H0;D3;+0:7]1:[c:8]:[n;H0;D2;+0:9]:[c:10]:[c:11]:1>>[C:1]-[C:2]-[CH2;D2;+0:3]-[n;H0;D3;+0:9]1:[c:10]:[c:11]:[n+;H0;D3:7](-[C:6]-[C:5]):[c:8]:1.[Cl-;H0;D0:4]
null
[]
null
null
null
null
Combine 5.35 g (0.32 mole) of (4-chlorobutyl)benzene and 5.27 g (0.32 mole) 1-heptyl-1H-imidazole, stir the mixture at approximately 145° C. for about 30 hours. Follow the progress of the reaction by thin-layer chromatography on silica gel (acetonitrile:ammonium hydroxide 9:1). At the completion of the reaction, dissol...
10.6084/m9.figshare.5104873.v1
null
Primary halide
null
c1c[nH]cn1
c1c[n+]cn1
c1c[n+]cn1.c1ccccc1
null
CO
null
null
CCCCCCCn1ccnc1.ClCCCCc1ccccc1>CO>CCCCCCC[n+]1ccn(CCCCc2ccccc2)c1.[Cl-]
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-65a238fbcc58467ca44415ceb2512a3b
CC(=O)Nc1ccc(CCCCOS(=O)(=O)c2ccc(C)cc2)cc1.CCCCCCCn1ccnc1>>CCCCCCCn1cc[n+](CCCCc2ccc(NC(C)=O)cc2)c1.Cc1ccc(S(=O)(=O)[O-])cc1
C(C)(=O)NC1=CC=C(C=C1)CCCCOS(=O)(=O)C1=CC=C(C=C1)C.C(CCCCCC)N1C=NC=C1>>CC1=CC=C(C=C1)S(=O)(=O)[O-].C(C)(=O)NC1=CC=C(C=C1)CCCC[N+]1=CN(C=C1)CCCCCCC
[CH2:12]([CH2:13][CH2:14][CH2:15][c:16]1[cH:17][cH:18][c:19]([NH:20][C:21]([CH3:22])=[O:23])[cH:24][cH:25]1)[O:35][S:32]([c:31]1[cH:30][cH:29][c:28]([CH3:27])[cH:37][cH:36]1)(=[O:33])=[O:34].[CH3:1][CH2:2][CH2:3][CH2:4][CH2:5][CH2:6][CH2:7][n:8]1[cH:9][cH:10][n:11][cH:26]1>>[CH3:1][CH2:2][CH2:3][CH2:4][CH2:5][CH2:6][CH...
CC(=O)Nc1ccc(CCCCOS(=O)(=O)c2ccc(C)cc2)cc1.CCCCCCCn1ccnc1
CCCCCCCn1cc[n+](CCCCc2ccc(NC(C)=O)cc2)c1.Cc1ccc(S(=O)(=O)[O-])cc1
null
null
null
Functional Group Interconversion
OtherReaction
f6336a3ca2c058a82dc422254532a6256a33456d0cf2f851f353d7a1b3fa3922
f1bbf9aa3c82f5e49be9f6d53533b6bb152f359232b6d32090c168949766aa71
c1ccc(CCCC[n+]2cc[nH]c2)cc1.c1ccccc1
[C:1]-[#7;a:2]1:[c:3]:[n;H0;D2;+0:4]:[c:5]:[c:6]:1.[C:7]-[C:8]-[CH2;D2;+0:9]-[O;H0;D2;+0:10]-[#16:11](=[O;D1;H0:12])(=[O;D1;H0:13])-[c:14]1:[c:15]:[c:16]:[c:17](-[C;D1;H3:18]):[c:19]:[c:20]:1>>[C;D1;H3:18]-[c:17]1:[c:16]:[c:15]:[c:14](-[#16:11](-[O-;H0;D1:10])(=[O;D1;H0:12])=[O;D1;H0:13]):[c:20]:[c:19]:1.[C:7]-[C:8]-[C...
null
[]
null
null
5
HOUR
Heat a mixture of 6.23 g (0.017 mole) 4-methylbenzenesulfonic acid 4-(4-acetylaminophenyl)butyl ester and 2.9 g (0.017 mole) 1-heptyl-1H-imidazole to 80° C., for 5 hours, following the reaction by thin-layer chromatography on silica gel (acetonitrile: ammonium hydroxide, 90:10). At the completion of the reaction, tritu...
10.6084/m9.figshare.5104873.v1
null
null
null
c1c[nH]cn1
c1c[nH]c[n+]1
c1c[nH]c[n+]1.c1ccccc1.c1ccccc1
null
null
null
5
CC(=O)Nc1ccc(CCCCOS(=O)(=O)c2ccc(C)cc2)cc1.CCCCCCCn1ccnc1>>CCCCCCCn1cc[n+](CCCCc2ccc(NC(C)=O)cc2)c1.Cc1ccc(S(=O)(=O)[O-])cc1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-179c26676e05430697577cc67e854849
Cc1nccn1C.ClCCCCc1ccc(Cl)cc1>>Cc1n(C)cc[n+]1CCCCc1ccc(Cl)cc1.[Cl-]
ClC1=CC=C(C=C1)CCCCCl.CN1C(=NC=C1)C>>[Cl-].ClC1=CC=C(C=C1)CCCC[N+]1=C(N(C=C1)C)C
[CH3:1][c:2]1[n:3]([CH3:4])[cH:5][cH:6][n:7]1.[CH2:8]([CH2:9][CH2:10][CH2:11][c:12]1[cH:13][cH:14][c:15]([Cl:16])[cH:17][cH:18]1)[Cl:19]>>[CH3:1][c:2]1[n:3]([CH3:4])[cH:5][cH:6][n+:7]1[CH2:8][CH2:9][CH2:10][CH2:11][c:12]1[cH:13][cH:14][c:15]([Cl:16])[cH:17][cH:18]1.[Cl-:19]
Cc1nccn1C.ClCCCCc1ccc(Cl)cc1
Cc1n(C)cc[n+]1CCCCc1ccc(Cl)cc1.[Cl-]
null
null
null
Functional Group Interconversion
OtherReaction
3d5d015c2046556debcf6aeafac05350e91208eeb74adef0cc21fd56e7fc95e0
47a659f5704a5b7ca1b92ff731f18f109c6bde1d45152a3a393eefbd10265508
c1ccc(CCCC[n+]2cc[nH]c2)cc1
[C;D1;H3:1]-[c:2]1:[n;H0;D2;+0:3]:[c:4]:[c:5]:[#7;a:6]:1-[C;D1;H3:7].[C:8]-[C:9]-[CH2;D2;+0:10]-[Cl;H0;D1;+0:11]>>[C:8]-[C:9]-[CH2;D2;+0:10]-[n+;H0;D3:3]1:[c:4]:[c:5]:[#7;a:6](-[C;D1;H3:7]):[c:2]:1-[C;D1;H3:1].[Cl-;H0;D0:11]
null
[]
115
CELSIUS
3
HOUR
To 4.77 g (0.023 mole) 1-chloro-4-(4-chlorobutyl)benzene add 2.23 g (0.023 mole) 1,2-dimethyl-1H-imidazole. Stir the solution for three hours at about 115° C. Follow the progress of the reaction by thin-layer chromatography on silica gel (MeOH:NaCl(1M), 92:8). At the completion of the reaction, cool to obtain an oil. T...
10.6084/m9.figshare.5104873.v1
null
Primary halide
null
c1ncc[nH]1
c1[n+]cc[nH]1
c1[n+]cc[nH]1.c1ccccc1
null
null
115
3
Cc1nccn1C.ClCCCCc1ccc(Cl)cc1>>Cc1n(C)cc[n+]1CCCCc1ccc(Cl)cc1.[Cl-]
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-c554592c9b37465fa73f99fc04d02e8d
CCCCCCCBr.Cc1cccc(C)c1NS(=O)(=O)CCn1ccnc1>>CCCCCCCn1cc[n+](CCS(=O)(=O)Nc2c(C)cccc2C)c1.[Br-]
BrCCCCCCC.CC1=C(C(=CC=C1)C)NS(=O)(=O)CCN1C=NC=C1.O>>[Br-].CC1=C(C(=CC=C1)C)NS(=O)(=O)CC[N+]1=CN(C=C1)CCCCCCC
[CH3:1][CH2:2][CH2:3][CH2:4][CH2:5][CH2:6][CH2:7][Br:27].[n:8]1[cH:9][cH:10][n:11]([CH2:12][CH2:13][S:14](=[O:15])(=[O:16])[NH:17][c:18]2[c:19]([CH3:20])[cH:21][cH:22][cH:23][c:24]2[CH3:25])[cH:26]1>>[CH3:1][CH2:2][CH2:3][CH2:4][CH2:5][CH2:6][CH2:7][n:8]1[cH:9][cH:10][n+:11]([CH2:12][CH2:13][S:14](=[O:15])(=[O:16])[NH:...
CCCCCCCBr.Cc1cccc(C)c1NS(=O)(=O)CCn1ccnc1
CCCCCCCn1cc[n+](CCS(=O)(=O)Nc2c(C)cccc2C)c1.[Br-]
null
null
CN(C)C=O
Functional Group Interconversion
OtherReaction
af9372efd0d4cbb040a1d2fa469660cc7709681c6c0eb3b6dabfb715f74188ec
47a659f5704a5b7ca1b92ff731f18f109c6bde1d45152a3a393eefbd10265508
O=S(=O)(CC[n+]1cc[nH]c1)Nc1ccccc1
[Br;H0;D1;+0:1]-[CH2;D2;+0:2]-[C:3]-[C:4].[C:5]-[C:6]-[n;H0;D3;+0:7]1:[c:8]:[c:9]:[n;H0;D2;+0:10]:[c:11]:1>>[Br-;H0;D0:1].[C:5]-[C:6]-[n+;H0;D3:7]1:[c:8]:[c:9]:[n;H0;D3;+0:10](-[CH2;D2;+0:2]-[C:3]-[C:4]):[c:11]:1
null
[]
null
null
10
HOUR
Combine 3.46 g (0.019 mole) 1-bromoheptane and 5.16 g (0.018 mole) N-(2,6-dimethylphenyl)-2-[1H-imidazol-1-yl]ethane sulfonamide in 10 ml DMF and heat to 100° C. Follow progress of reaction by TLC on silica gel (acetonitrile:ammonium hydroxide, 9:1). After about 10 hours, allow reaction mixture to cool to room temperat...
10.6084/m9.figshare.5104873.v1
null
Primary halide
null
c1c[nH]cn1
c1c[nH]c[n+]1
c1c[nH]c[n+]1.c1ccccc1
null
CN(C)C=O
null
10
CCCCCCCBr.Cc1cccc(C)c1NS(=O)(=O)CCn1ccnc1>CN(C)C=O>CCCCCCCn1cc[n+](CCS(=O)(=O)Nc2c(C)cccc2C)c1.[Br-]
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-560edb78e0de42889fc1ab50fda17b06
CCCn1ccnc1.ClCCCCc1ccc(Cl)cc1>>CCCn1cc[n+](CCCCc2ccc(Cl)cc2)c1.[Cl-]
ClC1=CC=C(C=C1)CCCCCl.C(CC)N1C=NC=C1>>[Cl-].ClC1=CC=C(C=C1)CCCC[N+]1=CN(C=C1)CCC
[CH3:1][CH2:2][CH2:3][n:4]1[cH:5][cH:6][n:7][cH:19]1.[CH2:8]([CH2:9][CH2:10][CH2:11][c:12]1[cH:13][cH:14][c:15]([Cl:16])[cH:17][cH:18]1)[Cl:20]>>[CH3:1][CH2:2][CH2:3][n:4]1[cH:5][cH:6][n+:7]([CH2:8][CH2:9][CH2:10][CH2:11][c:12]2[cH:13][cH:14][c:15]([Cl:16])[cH:17][cH:18]2)[cH:19]1.[Cl-:20]
CCCn1ccnc1.ClCCCCc1ccc(Cl)cc1
CCCn1cc[n+](CCCCc2ccc(Cl)cc2)c1.[Cl-]
null
null
null
Functional Group Interconversion
OtherReaction
af9372efd0d4cbb040a1d2fa469660cc7709681c6c0eb3b6dabfb715f74188ec
47a659f5704a5b7ca1b92ff731f18f109c6bde1d45152a3a393eefbd10265508
c1ccc(CCCC[n+]2cc[nH]c2)cc1
[C:1]-[#7;a:2]1:[c:3]:[n;H0;D2;+0:4]:[c:5]:[c:6]:1.[C:7]-[C:8]-[CH2;D2;+0:9]-[Cl;H0;D1;+0:10]>>[C:7]-[C:8]-[CH2;D2;+0:9]-[n+;H0;D3:4]1:[c:3]:[#7;a:2](-[C:1]):[c:6]:[c:5]:1.[Cl-;H0;D0:10]
null
[]
130
CELSIUS
null
null
Add 7.13 g (0.035 mole) of 1-chloro-4-(4-chlorobutyl)benzene to 3.52 g (0.032 mole) of 1-propyl-1H-imidazole and heat to 130° C. for 18 hours. Follow the progress of reaction by NMR (CDCl3). At the completion of the reaction, cool to room temperature to obtain the title compound. Conditions: See reaction.notes.procedur...
10.6084/m9.figshare.5104873.v1
null
Primary halide
null
c1c[nH]cn1
c1c[nH]c[n+]1
c1c[nH]c[n+]1.c1ccccc1
null
null
130
null
CCCn1ccnc1.ClCCCCc1ccc(Cl)cc1>>CCCn1cc[n+](CCCCc2ccc(Cl)cc2)c1.[Cl-]
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-ca23741c01464b8fb8b22ddafe07b27d
ClCCCCc1ccc(Cl)cc1.c1cn(CC2CCCCC2)cn1>>Clc1ccc(CCCCn2cc[n+](CC3CCCCC3)c2)cc1.[Cl-]
ClC1=CC=C(C=C1)CCCCCl.C1(CCCCC1)CN1C=NC=C1>>[Cl-].C1(CCCCC1)C[N+]1=CN(C=C1)CCCCC1=CC=C(C=C1)Cl
[Cl:1][c:2]1[cH:3][cH:4][c:5]([CH2:6][CH2:7][CH2:8][CH2:9][Cl:24])[cH:22][cH:23]1.[n:10]1[cH:11][cH:12][n:13]([CH2:14][CH:15]2[CH2:16][CH2:17][CH2:18][CH2:19][CH2:20]2)[cH:21]1>>[Cl:1][c:2]1[cH:3][cH:4][c:5]([CH2:6][CH2:7][CH2:8][CH2:9][n:10]2[cH:11][cH:12][n+:13]([CH2:14][CH:15]3[CH2:16][CH2:17][CH2:18][CH2:19][CH2:20...
ClCCCCc1ccc(Cl)cc1.c1cn(CC2CCCCC2)cn1
Clc1ccc(CCCCn2cc[n+](CC3CCCCC3)c2)cc1.[Cl-]
null
null
null
Functional Group Interconversion
OtherReaction
af9372efd0d4cbb040a1d2fa469660cc7709681c6c0eb3b6dabfb715f74188ec
47a659f5704a5b7ca1b92ff731f18f109c6bde1d45152a3a393eefbd10265508
c1ccc(CCCCn2cc[n+](CC3CCCCC3)c2)cc1
[C:1]-[C:2]-[CH2;D2;+0:3]-[Cl;H0;D1;+0:4].[C:5]-[C:6]-[n;H0;D3;+0:7]1:[c:8]:[c:9]:[n;H0;D2;+0:10]:[c:11]:1>>[C:5]-[C:6]-[n+;H0;D3:7]1:[c:8]:[c:9]:[n;H0;D3;+0:10](-[CH2;D2;+0:3]-[C:2]-[C:1]):[c:11]:1.[Cl-;H0;D0:4]
null
[]
130
CELSIUS
null
null
Add 6.55 g (0.03 mole) of 1-chloro-4-(4-chlorobutyl)benzene to 4.81 g (0.293 mole) of 1-cyclohexylmethyl-1H-imidazole and heat at 130° C. for 18 hours. Conditions: See reaction.notes.procedure_details.
10.6084/m9.figshare.5104873.v1
null
Primary halide
null
c1c[nH]cn1
c1c[nH]c[n+]1
c1ccccc1.c1c[nH]c[n+]1.C1CCCCC1
null
null
130
null
ClCCCCc1ccc(Cl)cc1.c1cn(CC2CCCCC2)cn1>>Clc1ccc(CCCCn2cc[n+](CC3CCCCC3)c2)cc1.[Cl-]
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-d30bd7fa8b074e34af76c288efa5a890
CCCCCCCn1c(C)nc(C)c1C.COc1ccc(CCCCBr)cc1>>CCCCCCC[n+]1c(C)c(C)n(CCCCc2ccc(OC)cc2)c1C.[Br-]
BrCCCCC1=CC=C(C=C1)OC.C(CCCCCC)N1C(=NC(=C1C)C)C>>[Br-].C(CCCCCC)[N+]1=C(N(C(=C1C)C)CCCCC1=CC=C(C=C1)OC)C
[CH3:1][CH2:2][CH2:3][CH2:4][CH2:5][CH2:6][CH2:7][n:8]1[c:9]([CH3:10])[c:11]([CH3:12])[n:13][c:26]1[CH3:27].[CH2:14]([CH2:15][CH2:16][CH2:17][c:18]1[cH:19][cH:20][c:21]([O:22][CH3:23])[cH:24][cH:25]1)[Br:28]>>[CH3:1][CH2:2][CH2:3][CH2:4][CH2:5][CH2:6][CH2:7][n+:8]1[c:9]([CH3:10])[c:11]([CH3:12])[n:13]([CH2:14][CH2:15][...
CCCCCCCn1c(C)nc(C)c1C.COc1ccc(CCCCBr)cc1
CCCCCCC[n+]1c(C)c(C)n(CCCCc2ccc(OC)cc2)c1C.[Br-]
null
null
O
Functional Group Interconversion
OtherReaction
5e72d8623d1d11df3a484f13beed495bb29975189dd55fb2f640a2dac5643123
47a659f5704a5b7ca1b92ff731f18f109c6bde1d45152a3a393eefbd10265508
c1ccc(CCCCn2cc[nH+]c2)cc1
[Br;H0;D1;+0:1]-[CH2;D2;+0:2]-[C:3]-[C:4].[C:5]-[C:6]-[n;H0;D3;+0:7]1:[c:8](-[C;D1;H3:9]):[n;H0;D2;+0:10]:[c:11](-[C;D1;H3:12]):[c:13]:1-[C;D1;H3:14]>>[Br-;H0;D0:1].[C:4]-[C:3]-[CH2;D2;+0:2]-[n;H0;D3;+0:10]1:[c:11](-[C;D1;H3:12]):[c:13](-[C;D1;H3:14]):[n+;H0;D3:7](-[C:6]-[C:5]):[c:8]:1-[C;D1;H3:9]
null
[]
125
CELSIUS
null
null
Add 3.23 g (0.0133 mole) of 1-(4-bromobutyl)-4-methoxybenzene to 2.77 g (0.0133 mole) of 1-heptyl-2,4,5-trimethyl-1H-imidazole and heat at 125° C. for two hours. Follow the progress of the reaction by thin-layer chromatography on silica gel (methanol: 1M sodium chloride, 95:5). At the completion of the reaction, dissol...
10.6084/m9.figshare.5104873.v1
null
Primary halide
null
c1c[nH]cn1
c1c[n+]cn1
c1c[n+]cn1.c1ccccc1
null
O
125
null
CCCCCCCn1c(C)nc(C)c1C.COc1ccc(CCCCBr)cc1>O>CCCCCCC[n+]1c(C)c(C)n(CCCCc2ccc(OC)cc2)c1C.[Br-]
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-902acbb33e034967a63b13b5cc75a2c2
ClCCCCc1ccc(Cl)cc1.Cn1ccnc1>>Cn1cc[n+](CCCCc2ccc(Cl)cc2)c1.[Cl-]
ClC1=CC=C(C=C1)CCCCCl.CN1C=NC=C1>>[Cl-].ClC1=CC=C(C=C1)CCCC[N+]1=CN(C=C1)C
[CH2:6]([CH2:7][CH2:8][CH2:9][c:10]1[cH:11][cH:12][c:13]([Cl:14])[cH:15][cH:16]1)[Cl:18].[CH3:1][n:2]1[cH:3][cH:4][n:5][cH:17]1>>[CH3:1][n:2]1[cH:3][cH:4][n+:5]([CH2:6][CH2:7][CH2:8][CH2:9][c:10]2[cH:11][cH:12][c:13]([Cl:14])[cH:15][cH:16]2)[cH:17]1.[Cl-:18]
ClCCCCc1ccc(Cl)cc1.Cn1ccnc1
Cn1cc[n+](CCCCc2ccc(Cl)cc2)c1.[Cl-]
null
null
null
Functional Group Interconversion
OtherReaction
af9372efd0d4cbb040a1d2fa469660cc7709681c6c0eb3b6dabfb715f74188ec
47a659f5704a5b7ca1b92ff731f18f109c6bde1d45152a3a393eefbd10265508
c1ccc(CCCC[n+]2cc[nH]c2)cc1
[C;D1;H3:1]-[#7;a:2]1:[c:3]:[n;H0;D2;+0:4]:[c:5]:[c:6]:1.[C:7]-[C:8]-[CH2;D2;+0:9]-[Cl;H0;D1;+0:10]>>[C:7]-[C:8]-[CH2;D2;+0:9]-[n+;H0;D3:4]1:[c:3]:[#7;a:2](-[C;D1;H3:1]):[c:6]:[c:5]:1.[Cl-;H0;D0:10]
null
[]
null
null
null
null
Combine 6.1 g (0.03 mole) 1-chloro-4-(4-chlorobutyl)benzene with 2.5 g (0.03 mole) 1-methyl-1H-imidazole and heat at 120° C., following the course of the reaction by thin-layer chromatography on silica gel (methanol:1M sodium chloride, 95:5). At the completion of the reaction, cool and triturate with ether, collect the...
10.6084/m9.figshare.5104873.v1
null
Primary halide
null
c1c[nH]cn1
c1c[nH]c[n+]1
c1c[nH]c[n+]1.c1ccccc1
null
null
null
null
ClCCCCc1ccc(Cl)cc1.Cn1ccnc1>>Cn1cc[n+](CCCCc2ccc(Cl)cc2)c1.[Cl-]
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-057cda30ba974403950321e96ed564fa
CI.CS(=O)(=O)Nc1ccc(C(O)Cn2ccnc2)cc1>>Cn1cc[n+](CC(O)c2ccc(NS(C)(=O)=O)cc2)c1.[I-]
OC(CN1C=NC=C1)C1=CC=C(C=C1)NS(=O)(=O)C.IC>>[I-].OC(C[N+]1=CN(C=C1)C)C1=CC=C(C=C1)NS(=O)(=O)C
[CH3:1][I:21].[n:2]1[cH:3][cH:4][n:5]([CH2:6][CH:7]([OH:8])[c:9]2[cH:10][cH:11][c:12]([NH:13][S:14]([CH3:15])(=[O:16])=[O:17])[cH:18][cH:19]2)[cH:20]1>>[CH3:1][n:2]1[cH:3][cH:4][n+:5]([CH2:6][CH:7]([OH:8])[c:9]2[cH:10][cH:11][c:12]([NH:13][S:14]([CH3:15])(=[O:16])=[O:17])[cH:18][cH:19]2)[cH:20]1.[I-:21]
CI.CS(=O)(=O)Nc1ccc(C(O)Cn2ccnc2)cc1
Cn1cc[n+](CC(O)c2ccc(NS(C)(=O)=O)cc2)c1.[I-]
null
null
CO
Functional Group Interconversion
OtherReaction
f6336a3ca2c058a82dc422254532a6256a33456d0cf2f851f353d7a1b3fa3922
f1bbf9aa3c82f5e49be9f6d53533b6bb152f359232b6d32090c168949766aa71
c1ccc(CC[n+]2cc[nH]c2)cc1
[CH3;D1;+0:1]-[I;H0;D1;+0:2].[C:3]-[C:4]-[n;H0;D3;+0:5]1:[c:6]:[n;H0;D2;+0:7]:[c:8]:[c:9]:1>>[C:3]-[C:4]-[n+;H0;D3:5]1:[c:6]:[n;H0;D3;+0:7](-[CH3;D1;+0:1]):[c:8]:[c:9]:1.[I-;H0;D0:2]
null
[]
null
null
null
null
Heat a solution of 4.0 g (14.2 mmole) of (±)-N-[4-[1-hydroxy-2-(1H-imidazol-1-yl)ethyl]phenyl]methanesulfonamide, 2 ml (32.1 mmole) of iodomethane and 50 ml methanol in a glass pressure tube to 80° C. for 24 hours. Remove the solvent in vacuo. Crystallize the residue from acetone. Recrystallize from acetone to provide ...
10.6084/m9.figshare.5104873.v1
null
null
null
c1c[nH]cn1
c1c[nH]c[n+]1
c1c[nH]c[n+]1.c1ccccc1
null
CO
null
null
CI.CS(=O)(=O)Nc1ccc(C(O)Cn2ccnc2)cc1>CO>Cn1cc[n+](CC(O)c2ccc(NS(C)(=O)=O)cc2)c1.[I-]
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-d7be8a0b10e1453c9251730ccc298a72
CS(=O)(=O)Nc1ccc(C(=O)CCl)cc1.Cn1ccnc1>>CN1C=C[NH+](CC(=O)c2ccc(NS(C)(=O)=O)cc2)C1.[Cl-]
ClCC(=O)C1=CC=C(C=C1)NS(=O)(=O)C.CN1C=NC=C1>>[Cl-].CN1C[NH+](C=C1)CC(=O)C1=CC=C(C=C1)NS(=O)(=O)C
[CH2:6]([C:7](=[O:8])[c:9]1[cH:10][cH:11][c:12]([NH:13][S:14]([CH3:15])(=[O:16])=[O:17])[cH:18][cH:19]1)[Cl:21].[CH3:1][n:2]1[cH:3][cH:4][n:5][cH:20]1>>[CH3:1][N:2]1[CH:3]=[CH:4][NH+:5]([CH2:6][C:7](=[O:8])[c:9]2[cH:10][cH:11][c:12]([NH:13][S:14]([CH3:15])(=[O:16])=[O:17])[cH:18][cH:19]2)[CH2:20]1.[Cl-:21]
CS(=O)(=O)Nc1ccc(C(=O)CCl)cc1.Cn1ccnc1
CN1C=C[NH+](CC(=O)c2ccc(NS(C)(=O)=O)cc2)C1.[Cl-]
null
null
C(C)#N
Heteroatom Alkylation and Arylation
OtherReaction
b8a36c115de439e42d925db9132e5b213bced5e9293ac4627b21408663bd0ea9
26d4750eaad79ede0d7168e363193f9b045f95289d4a8e5e240badd96495d35b
O=C(C[NH+]1C=CNC1)c1ccccc1
[C;D1;H3:1]-[n;H0;D3;+0:2]1:[cH;D2;+0:3]:[n;H0;D2;+0:4]:[cH;D2;+0:5]:[cH;D2;+0:6]:1.[Cl;H0;D1;+0:7]-[CH2;D2;+0:8]-[C:9](=[O;D1;H0:10])-[c:11]>>[C;D1;H3:1]-[N;H0;D3;+0:2]1-[CH2;D2;+0:3]-[NH+;D3:4](-[CH2;D2;+0:8]-[C:9](=[O;D1;H0:10])-[c:11])-[CH;D2;+0:5]=[CH;D2;+0:6]-1.[Cl-;H0;D0:7]
null
[]
null
null
null
null
Heat a mixture of 160 g (0.646 mole) of N-[4-(2-chloro-1-oxoethyl)phenyl]methanesulfonamide, 55.7 g (0.678 mole) of 1-methyl-1H-imidazole and 2.1 L of acetonitrile at reflux for about 16 hours. Cool the mixture to room temperature and collect the solid and wash with 2 L of acetonitrile. Drying provides the title compou...
10.6084/m9.figshare.5104873.v1
null
Primary halide.Ketone
Enamine.Ketone
c1c[nH]cn1
C1=C[NH+]C[NH]1
C1=C[NH+]C[NH]1.c1ccccc1
null
C(C)#N
null
null
CS(=O)(=O)Nc1ccc(C(=O)CCl)cc1.Cn1ccnc1>C(C)#N>CN1C=C[NH+](CC(=O)c2ccc(NS(C)(=O)=O)cc2)C1.[Cl-]
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-04d3b9ce6ec74a958e6dc71bb1716b03
CN1C=C[NH+](CC(=O)c2ccc(NS(C)(=O)=O)cc2)C1>>CN1C=C[NH+](CC(O)c2ccc(NS(C)(=O)=O)cc2)C1
[Cl-].CN1C[NH+](C=C1)CC(=O)C1=CC=C(C=C1)NS(=O)(=O)C>>[Cl-].OC(C[NH+]1CN(C=C1)C)C1=CC=C(C=C1)NS(=O)(=O)C
[CH3:1][N:2]1[CH:3]=[CH:4][NH+:5]([CH2:6][C:7](=[O:8])[c:9]2[cH:10][cH:11][c:12]([NH:13][S:14]([CH3:15])(=[O:16])=[O:17])[cH:18][cH:19]2)[CH2:20]1>>[CH3:1][N:2]1[CH:3]=[CH:4][NH+:5]([CH2:6][CH:7]([OH:8])[c:9]2[cH:10][cH:11][c:12]([NH:13][S:14]([CH3:15])(=[O:16])=[O:17])[cH:18][cH:19]2)[CH2:20]1
CN1C=C[NH+](CC(=O)c2ccc(NS(C)(=O)=O)cc2)C1
CN1C=C[NH+](CC(O)c2ccc(NS(C)(=O)=O)cc2)C1
null
[Pd]
O
Reduction
Reduction of ketone to secondary alcohol
02790ac194d8bf7ccb13d6247c59412024d87f77d2c906ef7804f021f57d5070
1bd3cd74b454139c0a0068ac0135836499926b274bff569df163210c6c944a89
C1=C[NH+](CCc2ccccc2)CN1
[C:1]=[C:2]-[#7;+:3]-[C:4]-[C;H0;D3;+0:5](=[O;H0;D1;+0:6])-[c:7](:[c:8]):[c:9]>>[C:1]=[C:2]-[#7;+:3]-[C:4]-[CH;D3;+0:5](-[OH;D1;+0:6])-[c:7](:[c:8]):[c:9]
null
[]
null
null
null
null
A solution of 152.3 g (0.463 mole) of 3-methyl-1[2-[4-((methylsulfonyl)amino)phenyl]-2-oxoethyl]-1H-imidazolium chloride in 1 L of distilled water and 7.62 g 10% Pd/C catalyst are placed in a 2 L Parr bottle and hydrogenated at 50 psi pressure for ca. 5 hours. Conditions: See reaction.notes.procedure_details.
10.6084/m9.figshare.5104873.v1
null
Ketone
Secondary alcohol
null
null
C1=C[NH+]C[NH]1.c1ccccc1
null
[Pd].O
null
null
CN1C=C[NH+](CC(=O)c2ccc(NS(C)(=O)=O)cc2)C1>[Pd].O>CN1C=C[NH+](CC(O)c2ccc(NS(C)(=O)=O)cc2)C1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-8942f05ad9b44f1aa6ee60dbe5607694
O=[N+]([O-])c1ccc(CCn2ccnc2)cc1>>Nc1ccc(CCn2ccnc2)cc1
[N+](=O)([O-])C1=CC=C(C=C1)CCN1C=NC=C1>>NC1=CC=C(C=C1)CCN1C=NC=C1
O=[N+:1]([O-])[c:2]1[cH:3][cH:4][c:5]([CH2:6][CH2:7][n:8]2[cH:9][cH:10][n:11][cH:12]2)[cH:13][cH:14]1>>[NH2:1][c:2]1[cH:3][cH:4][c:5]([CH2:6][CH2:7][n:8]2[cH:9][cH:10][n:11][cH:12]2)[cH:13][cH:14]1
O=[N+]([O-])c1ccc(CCn2ccnc2)cc1
Nc1ccc(CCn2ccnc2)cc1
null
[Pd]
Cl.C(C)O
Reduction
Reduction of nitro groups to amines
bbc242b150a51e69d3ad1caaa391f4422710431b398dcb880555f476706790be
7b0317532ea57a4fcedc1efc3e3c22eb5238d1c8330da53d4f9801fc2391f567
c1ccc(CCn2ccnc2)cc1
O=[N+;H0;D3:1](-[O-])-[c:2](:[c:3]):[c:4]>>[NH2;D1;+0:1]-[c:2](:[c:3]):[c:4]
null
[]
null
null
null
null
A solution of 10 g (0.046 mole) of 1-[2-(4-nitrophenyl)ethyl]-1H-imidazole in 100 mL of ethanol, 50 mL of 10% aqueous hydrochloric acid and 1.0 g of 5% Pd/C catalyst are placed in a small Parr bottle and hydrogenated at 50 psi pressure for about 24 hours. Additional H2 is added as needed to maintain 50 psi pressure. Th...
10.6084/m9.figshare.5104873.v1
null
Nitro group
Primary amine
null
null
c1ccccc1.c1c[nH]cn1
Other
[Pd].Cl.C(C)O
null
null
O=[N+]([O-])c1ccc(CCn2ccnc2)cc1>[Pd].Cl.C(C)O>Nc1ccc(CCn2ccnc2)cc1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-cd66aca946ca4ec298c6a1d5a5a8d280
CS(=O)(=O)Cl.Nc1ccc(CCn2ccnc2)cc1>>CS(=O)(=O)Nc1ccc(CCn2ccnc2)cc1
NC1=CC=C(C=C1)CCN1C=NC=C1.C(C)N(CC)CC.CS(=O)(=O)Cl>>CS(=O)(=O)NC1=CC=C(C=C1)CCN1C=NC=C1
Cl[S:2]([CH3:1])(=[O:3])=[O:4].[NH2:5][c:6]1[cH:7][cH:8][c:9]([CH2:10][CH2:11][n:12]2[cH:13][cH:14][n:15][cH:16]2)[cH:17][cH:18]1>>[CH3:1][S:2](=[O:3])(=[O:4])[NH:5][c:6]1[cH:7][cH:8][c:9]([CH2:10][CH2:11][n:12]2[cH:13][cH:14][n:15][cH:16]2)[cH:17][cH:18]1
CS(=O)(=O)Cl.Nc1ccc(CCn2ccnc2)cc1
CS(=O)(=O)Nc1ccc(CCn2ccnc2)cc1
null
null
C(Cl)Cl
Miscellaneous
Sulfonamide synthesis (Schotten-Baumann) primary amine
a86b0632821e188c0a5dc5a5a2aac298ab3eccaee8a52ba46078c3d5975a290d
50f8fbf3d327483c3eeff8f6cbd4065e4c7600bb501fbe08958a5c79a0926428
c1ccc(CCn2ccnc2)cc1
Cl-[S;H0;D4;+0:1](-[C;D1;H3:2])(=[O;D1;H0:3])=[O;D1;H0:4].[NH2;D1;+0:5]-[c:6](:[c:7]):[c:8]>>[C;D1;H3:2]-[S;H0;D4;+0:1](=[O;D1;H0:3])(=[O;D1;H0:4])-[NH;D2;+0:5]-[c:6](:[c:7]):[c:8]
null
[]
-10
CELSIUS
30
MINUTE
To a -10° C. solution of 8 g (0.064 mole) of 1-[2-(4-aminophenyl)ethyl]-1H-imidazole and 10 mL triethylamine in 200 mL of methylene chloride add 5 mL of methanesulfonyl chloride dropwise. Stir the resulting solution at -10° C. for about 30 minutes then warm to ambient temperature for about 30 minutes. Wash the reaction...
10.6084/m9.figshare.5104873.v1
null
Primary amine.Sulfonyl halide
Sulfonamide
null
null
c1ccccc1.c1c[nH]cn1
HCl
C(Cl)Cl
-10
0.5
CS(=O)(=O)Cl.Nc1ccc(CCn2ccnc2)cc1>C(Cl)Cl>CS(=O)(=O)Nc1ccc(CCn2ccnc2)cc1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-fe6bc469579849c190d98ec39f6d6c77
CI.CS(=O)(=O)Nc1ccc(CCn2ccnc2)cc1>>CN1C=C[NH+](CCc2ccc(NS(C)(=O)=O)cc2)C1.[I-]
N1(C=NC=C1)CCC1=CC=C(C=C1)NS(=O)(=O)C.IC>>[I-].CN1C[NH+](C=C1)CCC1=CC=C(C=C1)NS(=O)(=O)C
[CH3:1][I:20].[n:2]1[cH:3][cH:4][n:5]([CH2:6][CH2:7][c:8]2[cH:9][cH:10][c:11]([NH:12][S:13]([CH3:14])(=[O:15])=[O:16])[cH:17][cH:18]2)[cH:19]1>>[CH3:1][N:2]1[CH:3]=[CH:4][NH+:5]([CH2:6][CH2:7][c:8]2[cH:9][cH:10][c:11]([NH:12][S:13]([CH3:14])(=[O:15])=[O:16])[cH:17][cH:18]2)[CH2:19]1.[I-:20]
CI.CS(=O)(=O)Nc1ccc(CCn2ccnc2)cc1
CN1C=C[NH+](CCc2ccc(NS(C)(=O)=O)cc2)C1.[I-]
null
null
CO
Heteroatom Alkylation and Arylation
OtherReaction
32965ddc6bb6823ee266c09a6be2c69531f43f0c3e42e160da364d8852910592
0e973515f9f7e54073d059763104290284f0f6fd900e82ab9e6c66160ee2e711
C1=C[NH+](CCc2ccccc2)CN1
[CH3;D1;+0:1]-[I;H0;D1;+0:2].[C:3]-[C:4]-[n;H0;D3;+0:5]1:[cH;D2;+0:6]:[n;H0;D2;+0:7]:[cH;D2;+0:8]:[cH;D2;+0:9]:1>>[C:3]-[C:4]-[NH+;D3:5]1-[CH2;D2;+0:6]-[N;H0;D3;+0:7](-[CH3;D1;+0:1])-[CH;D2;+0:8]=[CH;D2;+0:9]-1.[I-;H0;D0:2]
null
[]
null
null
null
null
Heat a mixture of 5 g (0.019 mole) of N-[4-[2-(1H-imidazol-1-yl)ethyl]phenyl]methanesulfonamide, 5 mL of iodomethane and 25 mL of methanol in a pressure tube at 75° C. for about 24 hours. Cool the mixture to room temperature and remove the solvents in vacuo. Slurry the residue in acetone (50 mL) and filter and wash wit...
10.6084/m9.figshare.5104873.v1
null
null
Enamine
c1c[nH]cn1
C1=C[NH+]C[NH]1
C1=C[NH+]C[NH]1.c1ccccc1
null
CO
null
null
CI.CS(=O)(=O)Nc1ccc(CCn2ccnc2)cc1>CO>CN1C=C[NH+](CCc2ccc(NS(C)(=O)=O)cc2)C1.[I-]
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-9c952c876e5e4332a35b6f1b55bcb233
CS(=O)(=O)Nc1ccc(CCn2ccnc2O)cc1>>CS(=O)(=O)Nc1ccc(C(O)Cn2ccnc2)cc1
Cl.OC=1N(C=CN1)CCC1=CC=C(C=C1)NS(=O)(=O)C.C[O-].[Na+]>>OC(CN1C=NC=C1)C1=CC=C(C=C1)NS(=O)(=O)C
[CH3:1][S:2](=[O:3])(=[O:4])[NH:5][c:6]1[cH:7][cH:8][c:9]([CH2:10][CH2:12][n:13]2[cH:14][cH:15][n:16][c:17]2[OH:11])[cH:18][cH:19]1>>[CH3:1][S:2](=[O:3])(=[O:4])[NH:5][c:6]1[cH:7][cH:8][c:9]([CH:10]([OH:11])[CH2:12][n:13]2[cH:14][cH:15][n:16][cH:17]2)[cH:18][cH:19]1
CS(=O)(=O)Nc1ccc(CCn2ccnc2O)cc1
CS(=O)(=O)Nc1ccc(C(O)Cn2ccnc2)cc1
null
null
CO
Miscellaneous
OtherReaction
1763e158f5b6b8a342399a42bad5f4eb7bc3f82e5bebcc25b957a7ea5a15f932
061968087242247210331763a175366f5365580fa41e03eed87c9ba3d167230a
c1ccc(CCn2ccnc2)cc1
[OH;D1;+0:1]-[c;H0;D3;+0:2]1:[#7;a:3]:[c:4]:[c:5]:[#7;a:6]:1-[C:7]-[CH2;D2;+0:8]-[c:9](:[c:10]):[c:11]>>[OH;D1;+0:1]-[CH;D3;+0:8](-[C:7]-[#7;a:6]1:[c:5]:[c:4]:[#7;a:3]:[cH;D2;+0:2]:1)-[c:9](:[c:10]):[c:11]
null
[]
null
null
null
null
Heat a mixture of 30.83 g (0.097 mole) of (±)-1-[2-hydroxy-2-[4-((methylsulfonyl)amino)phenyl]ethyl-1H-imidazole hydrochloride and 5.24 g (0.097 mole) of sodium methylate in 100 mL of methanol and filter hot through 300 g of alumina (Fisher, neutral, activity III). Wash the alumina with 20% methanol in methylene chlori...
10.6084/m9.figshare.5104873.v1
null
Aromatic alcohol
Secondary alcohol
c1ncc[nH]1
c1c[nH]cn1
c1ccccc1.c1c[nH]cn1
null
CO
null
null
CS(=O)(=O)Nc1ccc(CCn2ccnc2O)cc1>CO>CS(=O)(=O)Nc1ccc(C(O)Cn2ccnc2)cc1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-0ca5c9efb5e24a3793181b1d509ee238
CCOC(=O)C(C(=O)OCC)C(C)(C)CCCCCCCCCCC(C)(C)C(C(=O)OCC)C(=O)OCC>>CC(C)(CCCCCCCCCCC(C)(C)CC(=O)O)CC(=O)O
C(C)OC(=O)C(C(CCCCCCCCCCC(C(C(=O)OCC)C(=O)OCC)(C)C)(C)C)C(=O)OCC.[OH-].[K+]>>CC(CC(=O)O)(CCCCCCCCCCC(CC(=O)O)(C)C)C
CCOC(=O)[CH:17]([C:14]([CH2:13][CH2:12][CH2:11][CH2:10][CH2:9][CH2:8][CH2:7][CH2:6][CH2:5][CH2:4][C:2]([CH3:1])([CH3:3])[CH:21](C(=O)OCC)[C:22](=[O:23])[O:24]CC)([CH3:15])[CH3:16])[C:18](=[O:19])[O:20]CC>>[CH3:1][C:2]([CH3:3])([CH2:4][CH2:5][CH2:6][CH2:7][CH2:8][CH2:9][CH2:10][CH2:11][CH2:12][CH2:13][C:14]([CH3:15])([C...
CCOC(=O)C(C(=O)OCC)C(C)(C)CCCCCCCCCCC(C)(C)C(C(=O)OCC)C(=O)OCC
CC(C)(CCCCCCCCCCC(C)(C)CC(=O)O)CC(=O)O
null
null
C(C)OCC
Reduction
OtherReaction
c66b299b40f3bbe41ba1575d603bfa618c1cfd61a8332cce6a45cf083197b05c
710ca63f65f20afd2d083b70f6465deae8116e1dce84a7e30ca74e667dfb146a
null
C-C-O-C(=O)-[CH;D3;+0:1](-[C:2](=[O;D1;H0:3])-[O;H0;D2;+0:4]-C-C)-[C:5](-[C:6])(-[C;D1;H3:7])-[C;D1;H3:8].C-C-O-C(=O)-[CH;D3;+0:9](-[C:10](=[O;D1;H0:11])-[O;H0;D2;+0:12]-C-C)-[C:13](-[C:14])(-[C;D1;H3:15])-[C;D1;H3:16]>>[C:6]-[C:5](-[C;D1;H3:7])(-[C;D1;H3:8])-[CH2;D2;+0:1]-[C:2](=[O;D1;H0:3])-[OH;D1;+0:4].[C:14]-[C:13]...
null
[]
null
null
null
null
A mixture of 17.0 g of the tetra-ester of Example 1 and 300 ml of a 25% aqueous KOH solution was heated in an oil bath to reflux temperature and the mixture was refluxed until the organic phase has completely disappeared (about 48 hours). The aqueous solution was then cooled to room temperature, extracted with ether, f...
10.6084/m9.figshare.5104873.v1
null
Ester.Ester.Ester.Ester
Carboxylic acid.Carboxylic acid
null
null
null
HO-
C(C)OCC
null
null
CCOC(=O)C(C(=O)OCC)C(C)(C)CCCCCCCCCCC(C)(C)C(C(=O)OCC)C(=O)OCC>C(C)OCC>CC(C)(CCCCCCCCCCC(C)(C)CC(=O)O)CC(=O)O
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-145fe5702635444bbf4bf1aa20451280
O=C(O)CC(CCC(=O)CCCCC(=O)CCC(CC(=O)O)(c1ccccc1)c1ccccc1)(c1ccccc1)c1ccccc1>>O=C(O)CC(CCCCCCCCCCC(CC(=O)O)(c1ccccc1)c1ccccc1)(c1ccccc1)c1ccccc1
C1(=CC=CC=C1)C(CC(=O)O)(CCC(CCCCC(CCC(CC(=O)O)(C1=CC=CC=C1)C1=CC=CC=C1)=O)=O)C1=CC=CC=C1.O.NN.[OH-].[K+]>>C1(=CC=CC=C1)C(CC(=O)O)(CCCCCCCCCCC(CC(=O)O)(C1=CC=CC=C1)C1=CC=CC=C1)C1=CC=CC=C1
O=[C:8]([CH2:7][CH2:6][C:5]([CH2:4][C:2](=[O:1])[OH:3])([c:33]1[cH:34][cH:35][cH:36][cH:37][cH:38]1)[c:39]1[cH:40][cH:41][cH:42][cH:43][cH:44]1)[CH2:9][CH2:10][CH2:11][CH2:12][C:13](=O)[CH2:14][CH2:15][C:16]([CH2:17][C:18](=[O:19])[OH:20])([c:21]1[cH:22][cH:23][cH:24][cH:25][cH:26]1)[c:27]1[cH:28][cH:29][cH:30][cH:31][...
O=C(O)CC(CCC(=O)CCCCC(=O)CCC(CC(=O)O)(c1ccccc1)c1ccccc1)(c1ccccc1)c1ccccc1
O=C(O)CC(CCCCCCCCCCC(CC(=O)O)(c1ccccc1)c1ccccc1)(c1ccccc1)c1ccccc1
null
null
O.C(COCCOCCO)O
Reduction
OtherReaction
3437f16d0dd3b11b660197591cbb75aa04be8c11f375001f94aed07467d803aa
6649363095331d33ffc4a587081bd0362ca141cb8f6a811c996a9356e6f05344
c1ccc(C(CCCCCCCCCCC(c2ccccc2)c2ccccc2)c2ccccc2)cc1
O=[C;H0;D3;+0:1](-[C:2]-[C:3]-[C:4]-[C:5]-[C;H0;D3;+0:6](=O)-[C:7]-[C:8])-[C:9]-[C:10]>>[C:10]-[C:9]-[CH2;D2;+0:1]-[C:2]-[C:3]-[C:4]-[C:5]-[CH2;D2;+0:6]-[C:7]-[C:8]
58
[{"value": 58.0, "product": "C1(=CC=CC=C1)C(CC(=O)O)(CCCCCCCCCCC(CC(=O)O)(C1=CC=CC=C1)C1=CC=CC=C1)C1=CC=CC=C1", "details": "PERCENTYIELD", "is_desired": false}]
120
CELSIUS
null
null
0.27 g of 3,3,14,14-tetraphenyl-6,11-diketohexadecane-1,16-dioic acid prepared as described in Example 23 and 0.23 ml of 85% hydrazine hydrate were added to a solution of 0.4 g KOH in 10 ml of triethyleneglycol. The mixture was heated at 120° C. for 24 h, then heated to 195° C. with the evaporation of water followed by...
10.6084/m9.figshare.5104873.v1
null
Ketone.Ketone
null
null
null
c1ccccc1.c1ccccc1.c1ccccc1.c1ccccc1
Other
O.C(COCCOCCO)O
120
null
O=C(O)CC(CCC(=O)CCCCC(=O)CCC(CC(=O)O)(c1ccccc1)c1ccccc1)(c1ccccc1)c1ccccc1>O.C(COCCOCCO)O>O=C(O)CC(CCCCCCCCCCC(CC(=O)O)(c1ccccc1)c1ccccc1)(c1ccccc1)c1ccccc1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-78276eeaba744eaabcd654099a62e06f
COC(=O)N1CCC(=O)C(C)C1.C[N+](=O)[O-]>>COC(=O)N1CC=C(C[N+](=O)[O-])C(C)C1
CC1CN(CCC1=O)C(=O)OC.C(CN)N.[N+](=O)([O-])C>>CC1CN(CC=C1C[N+](=O)[O-])C(=O)OC
O=[C:8]1[CH2:7][CH2:6][N:5]([C:3]([O:2][CH3:1])=[O:4])[CH2:15][CH:13]1[CH3:14].[CH3:9][N+:10](=[O:11])[O-:12]>>[CH3:1][O:2][C:3](=[O:4])[N:5]1[CH2:6][CH:7]=[C:8]([CH2:9][N+:10](=[O:11])[O-:12])[CH:13]([CH3:14])[CH2:15]1
COC(=O)N1CCC(=O)C(C)C1.C[N+](=O)[O-]
COC(=O)N1CC=C(C[N+](=O)[O-])C(C)C1
null
null
null
C-C Coupling
OtherReaction
2d30abe5d929ae968f04050cad94efe1d8c00104f747873587301c7d85c7b868
04707d47c6d6b8f2f7722c07a7f221fd5b5734d3345e34e53c95ebad5e4e59e3
C1=CCNCC1
O=[C;H0;D3;+0:1]1-[CH2;D2;+0:2]-[C:3]-[#7:4](-[C:5](-[#8:6])=[O;D1;H0:7])-[C:8]-[C:9]-1-[C;D1;H3:10].[CH3;D1;+0:11]-[#7;+:12](-[O;-;D1;H0:13])=[O;D1;H0:14]>>[#8:6]-[C:5](=[O;D1;H0:7])-[#7:4]1-[C:8]-[C:9](-[C;D1;H3:10])-[C;H0;D3;+0:1](-[CH2;D2;+0:11]-[#7;+:12](-[O;-;D1;H0:13])=[O;D1;H0:14])=[CH;D2;+0:2]-[C:3]-1
87.2
[{"value": 87.2, "product": "CC1CN(CC=C1C[N+](=O)[O-])C(=O)OC", "details": "PERCENTYIELD", "is_desired": false}]
null
null
null
null
A mixture of 64 parts of methyl 3-methyl-4-oxo-1-piperidinecarboxylate, 305 parts of nitromethane and 3.02 parts of 1,2-ethanediamine was stirred and refluxed for 4 hours. The reaction mixture was evaporated. The residue was taken up in trichloromethane. The solution was washed twice with a dilute hydrochloric acid sol...
10.6084/m9.figshare.5104873.v1
null
Ketone.Nitro group
Nitro group
C1CC[NH]CC1
C1=CC[NH]CC1
C1=CC[NH]CC1
HO-
null
null
null
COC(=O)N1CCC(=O)C(C)C1.C[N+](=O)[O-]>>COC(=O)N1CC=C(C[N+](=O)[O-])C(C)C1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-72abaa3c2d9c442991cf635fc70be709
CCOC(=O)N1CCC(=O)CC1.C[N+](=O)[O-]>>CCOC(=O)N1CCC(O)(C[N+](=O)[O-])CC1
O=C1CCN(CC1)C(=O)OCC.[N+](=O)([O-])C.C[O-].[Na+]>>OC1(CCN(CC1)C(=O)OCC)C[N+](=O)[O-]
[CH3:1][CH2:2][O:3][C:4](=[O:5])[N:6]1[CH2:7][CH2:8][C:9](=[O:10])[CH2:15][CH2:16]1.[CH3:11][N+:12](=[O:13])[O-:14]>>[CH3:1][CH2:2][O:3][C:4](=[O:5])[N:6]1[CH2:7][CH2:8][C:9]([OH:10])([CH2:11][N+:12](=[O:13])[O-:14])[CH2:15][CH2:16]1
CCOC(=O)N1CCC(=O)CC1.C[N+](=O)[O-]
CCOC(=O)N1CCC(O)(C[N+](=O)[O-])CC1
null
null
CO
C-C Coupling
Henry Reaction
b4bc771a3c4b2ab61f0ff05eb4e9a10f23529852e8464d6fe5f008137056d647
b784cb10b22de077efeecdc9f77dadffa83c0aad754bce89e06fd63e3bb6c28a
C1CCNCC1
[CH3;D1;+0:1]-[#7;+:2](-[O;-;D1;H0:3])=[O;D1;H0:4].[O;H0;D1;+0:5]=[C;H0;D3;+0:6]1-[C:7]-[C:8]-[#7:9]-[C:10]-[C:11]-1>>[O;-;D1;H0:3]-[#7;+:2](=[O;D1;H0:4])-[CH2;D2;+0:1]-[C;H0;D4;+0:6]1(-[OH;D1;+0:5])-[C:7]-[C:8]-[#7:9]-[C:10]-[C:11]-1
null
[]
null
null
8
HOUR
To a stirred and cooled mixture of 85.5 parts of ethyl 4-oxo-1-piperidinecarboxylate, 33.6 parts of nitromethane and 240 parts of methanol were added dropwise 10 parts of a sodium methoxide solution 30% at 10°~15° C. Upon completion, stirring was continued first for 2 hours at about 10° C. and further overnight at room...
10.6084/m9.figshare.5104873.v1
null
Ketone.Nitro group
Nitro group.Tertiary alcohol
C1CC[NH]CC1
C1CC[NH]CC1
C1CC[NH]CC1
null
CO
null
8
CCOC(=O)N1CCC(=O)CC1.C[N+](=O)[O-]>CO>CCOC(=O)N1CCC(O)(C[N+](=O)[O-])CC1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-5ff753d9df04493ba4054e7e71de4b30
CCOC(=O)N1CC=C(C[N+](=O)[O-])CC1>>CCOC(=O)N1CCC(CN)CC1
N.[N+](=O)([O-])CC=1CCN(CC1)C(=O)OCC.[H][H]>>NCC1CCN(CC1)C(=O)OCC
O=[N+:11]([O-])[CH2:10][C:9]1=[CH:8][CH2:7][N:6]([C:4]([O:3][CH2:2][CH3:1])=[O:5])[CH2:13][CH2:12]1>>[CH3:1][CH2:2][O:3][C:4](=[O:5])[N:6]1[CH2:7][CH2:8][CH:9]([CH2:10][NH2:11])[CH2:12][CH2:13]1
CCOC(=O)N1CC=C(C[N+](=O)[O-])CC1
CCOC(=O)N1CCC(CN)CC1
null
[Ni]
CO
Reduction
OtherReaction
5889e730401aed00e40fafd9b46e5746f82f14df365183900a6f8d37eff473dc
7b0317532ea57a4fcedc1efc3e3c22eb5238d1c8330da53d4f9801fc2391f567
C1CCNCC1
O=[N+;H0;D3:1](-[O-])-[C:2]-[C;H0;D3;+0:3]1=[CH;D2;+0:4]-[C:5]-[#7:6](-[C:7](-[#8:8])=[O;D1;H0:9])-[C:10]-[C:11]-1>>[#8:8]-[C:7](=[O;D1;H0:9])-[#7:6]1-[C:10]-[C:11]-[CH;D3;+0:3](-[C:2]-[NH2;D1;+0:1])-[CH2;D2;+0:4]-[C:5]-1
98.9
[{"value": 98.9, "product": "NCC1CCN(CC1)C(=O)OCC", "details": "PERCENTYIELD", "is_desired": false}]
null
null
null
null
A mixture of 41 parts of ethyl 3,6-dihydro-4-(nitromethyl)-1(2H)-pyridinecarboxylate and 400 parts of methanol, saturated with ammonia, was hydrogenated at normal pressure and at room temperature with 6 parts of Raney-nickel catalyst. After the calculated amount of hydrogen was taken up, the catalyst was filtered off a...
10.6084/m9.figshare.5104873.v1
null
Nitro group
Primary amine
C1=CC[NH]CC1
C1CC[NH]CC1
C1CC[NH]CC1
Other
[Ni].CO
null
null
CCOC(=O)N1CC=C(C[N+](=O)[O-])CC1>[Ni].CO>CCOC(=O)N1CCC(CN)CC1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-446a94c66a0c4158844c2afd4599238d
CCOC(=O)N1CCC(O)(C[N+](=O)[O-])CC1>>CCOC(=O)N1CCC(O)(CN)CC1
OC1(CCN(CC1)C(=O)OCC)C[N+](=O)[O-].CO.[H][H]>>NCC1(CCN(CC1)C(=O)OCC)O
O=[N+:12]([O-])[CH2:11][C:9]1([OH:10])[CH2:8][CH2:7][N:6]([C:4]([O:3][CH2:2][CH3:1])=[O:5])[CH2:14][CH2:13]1>>[CH3:1][CH2:2][O:3][C:4](=[O:5])[N:6]1[CH2:7][CH2:8][C:9]([OH:10])([CH2:11][NH2:12])[CH2:13][CH2:14]1
CCOC(=O)N1CCC(O)(C[N+](=O)[O-])CC1
CCOC(=O)N1CCC(O)(CN)CC1
null
[Pd]
C(C)(=O)O
Reduction
Reduction of nitro groups to amines
bbc242b150a51e69d3ad1caaa391f4422710431b398dcb880555f476706790be
7b0317532ea57a4fcedc1efc3e3c22eb5238d1c8330da53d4f9801fc2391f567
C1CCNCC1
O=[N+;H0;D3:1](-[O-])-[C:2]-[C:3]>>[C:3]-[C:2]-[NH2;D1;+0:1]
null
[]
null
null
null
null
A mixture of 73 parts of ethyl 4-hydroxy-4-(nitromethyl)-1-piperidinecarboxylate, 400 parts of methanol and 150 parts of acetic acid was hydrogenated in the Parr-apparatus with 5 parts of palladium-on-charcoal catalyst 10%. After the calculated amount of hydrogen was taken up, the catalyst was filtered off and the filt...
10.6084/m9.figshare.5104873.v1
null
Nitro group
Primary amine
null
null
C1CC[NH]CC1
Other
[Pd].C(C)(=O)O
null
null
CCOC(=O)N1CCC(O)(C[N+](=O)[O-])CC1>[Pd].C(C)(=O)O>CCOC(=O)N1CCC(O)(CN)CC1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-e93f204559cf4920afe9669d4b4737e9
CC(=O)N1CCC(CN)CC1.S=C=S>>CC(=O)N1CCC(CN=C=S)CC1
C(=S)=S.C(C)(=O)N1CCC(CC1)CN>>C(C)(=O)N1CCC(CC1)CN=C=S
[CH3:1][C:2](=[O:3])[N:4]1[CH2:5][CH2:6][CH:7]([CH2:8][NH2:9])[CH2:12][CH2:13]1.S=[C:10]=[S:11]>>[CH3:1][C:2](=[O:3])[N:4]1[CH2:5][CH2:6][CH:7]([CH2:8][N:9]=[C:10]=[S:11])[CH2:12][CH2:13]1
CC(=O)N1CCC(CN)CC1.S=C=S
CC(=O)N1CCC(CN=C=S)CC1
null
null
O1CCCC1
Heteroatom Alkylation and Arylation
OtherReaction
99faaca01b29bb4aacdf8b5dd838744c8a4a0ba5e793c41d71f6ab61fd987eaa
b4d1d5962cf9cde357eea1a492f332beb32c18a22c0b29a341204737bdcfdaa7
C1CCNCC1
S=[C;H0;D2;+0:1]=[S;D1;H0:2].[C:3]-[C:4]-[NH2;D1;+0:5]>>[C:3]-[C:4]-[N;H0;D2;+0:5]=[C;H0;D2;+0:1]=[S;D1;H0:2]
100
[{"value": 100.0, "product": "C(C)(=O)N1CCC(CC1)CN=C=S", "details": "PERCENTYIELD", "is_desired": false}]
null
null
8
HOUR
To a stirred and cooled (-10° C.) mixture of 41.6 parts of N,N'-methanetetraylbis[cyclohexanamine], 101 parts of carbon disulfide and 450 parts of tetrahydrofuran was added dropwise a solution of 31.2 parts of 1-acetyl-4-piperidinmethanamine in 90 parts of tetrahydrofuran. Upon completion, stirring was continued overni...
10.6084/m9.figshare.5104873.v1
null
Primary amine
Isothiocyanate
null
null
C1CC[NH]CC1
Other
O1CCCC1
null
8
CC(=O)N1CCC(CN)CC1.S=C=S>O1CCCC1>CC(=O)N1CCC(CN=C=S)CC1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-1ab8dde909e448d38b66977ecfbc2c78
CC(=O)N1CCC(CN=C=S)CC1.Nc1ccc(F)cc1>>CC(=O)N1CCC(CNC(=S)Nc2ccc(F)cc2)CC1
C(C)(=O)N1CCC(CC1)CN=C=S.FC1=CC=C(C=C1)N>>C(C)(=O)N1CCC(CC1)CNC(=S)NC1=CC=C(C=C1)F
[CH3:1][C:2](=[O:3])[N:4]1[CH2:5][CH2:6][CH:7]([CH2:8][N:9]=[C:10]=[S:11])[CH2:20][CH2:21]1.[NH2:12][c:13]1[cH:14][cH:15][c:16]([F:17])[cH:18][cH:19]1>>[CH3:1][C:2](=[O:3])[N:4]1[CH2:5][CH2:6][CH:7]([CH2:8][NH:9][C:10](=[S:11])[NH:12][c:13]2[cH:14][cH:15][c:16]([F:17])[cH:18][cH:19]2)[CH2:20][CH2:21]1
CC(=O)N1CCC(CN=C=S)CC1.Nc1ccc(F)cc1
CC(=O)N1CCC(CNC(=S)Nc2ccc(F)cc2)CC1
null
null
O1CCCC1
Heteroatom Alkylation and Arylation
thiourea
9037f368cdf8e91fcd9f93f4d9cf27991f85fa921c9d19c7875d3a77561f439b
0fbf3d6c8cd704ac451c2cf111f32090de5e76a9d41cce326e212c758f4ed46f
S=C(NCC1CCNCC1)Nc1ccccc1
[C:1]-[C:2]-[N;H0;D2;+0:3]=[C;H0;D2;+0:4]=[S;D1;H0:5].[NH2;D1;+0:6]-[c:7](:[c:8]):[c:9]>>[C:1]-[C:2]-[NH;D2;+0:3]-[C;H0;D3;+0:4](=[S;D1;H0:5])-[NH;D2;+0:6]-[c:7](:[c:8]):[c:9]
100
[{"value": 100.0, "product": "C(C)(=O)N1CCC(CC1)CNC(=S)NC1=CC=C(C=C1)F", "details": "PERCENTYIELD", "is_desired": false}]
null
null
8
HOUR
A mixture of 4 parts of 1-acetyl-4-(isothiocyanatomethyl)piperidine, 2.2 parts of 4-fluorobenzenamine and 90 parts of tetrahydrofuran was stirred overnight at reflux temperature. The reaction mixture was evaporated, yielding 6.2 parts (100%) of N-[(1-acetyl-4-piperidinyl)methyl]-N'-(4-fluorophenyl)thiourea as a residue...
10.6084/m9.figshare.5104873.v1
null
Primary amine.Isothiocyanate
Thiourea
null
null
C1CC[NH]CC1.c1ccccc1
null
O1CCCC1
null
8
CC(=O)N1CCC(CN=C=S)CC1.Nc1ccc(F)cc1>O1CCCC1>CC(=O)N1CCC(CNC(=S)Nc2ccc(F)cc2)CC1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-b8d469ec02df442d9a9d4e4733d2e923
CC(=O)N1CCC(CN)CC1.S=C=Nc1ccc(Cl)cc1>>CC(=O)N1CCC(CNC(=S)Nc2ccc(Cl)cc2)CC1
C(C)(=O)N1CCC(CC1)CN.ClC1=CC=C(C=C1)N=C=S>>C(C)(=O)N1CCC(CC1)CNC(=S)NC1=CC=C(C=C1)Cl
[CH3:1][C:2](=[O:3])[N:4]1[CH2:5][CH2:6][CH:7]([CH2:8][NH2:9])[CH2:20][CH2:21]1.[C:10](=[S:11])=[N:12][c:13]1[cH:14][cH:15][c:16]([Cl:17])[cH:18][cH:19]1>>[CH3:1][C:2](=[O:3])[N:4]1[CH2:5][CH2:6][CH:7]([CH2:8][NH:9][C:10](=[S:11])[NH:12][c:13]2[cH:14][cH:15][c:16]([Cl:17])[cH:18][cH:19]2)[CH2:20][CH2:21]1
CC(=O)N1CCC(CN)CC1.S=C=Nc1ccc(Cl)cc1
CC(=O)N1CCC(CNC(=S)Nc2ccc(Cl)cc2)CC1
null
null
O1CCCC1
Heteroatom Alkylation and Arylation
thiourea
9037f368cdf8e91fcd9f93f4d9cf27991f85fa921c9d19c7875d3a77561f439b
0fbf3d6c8cd704ac451c2cf111f32090de5e76a9d41cce326e212c758f4ed46f
S=C(NCC1CCNCC1)Nc1ccccc1
[C:1]-[C:2]-[NH2;D1;+0:3].[S;D1;H0:4]=[C;H0;D2;+0:5]=[N;H0;D2;+0:6]-[c:7](:[c:8]):[c:9]>>[C:1]-[C:2]-[NH;D2;+0:3]-[C;H0;D3;+0:5](=[S;D1;H0:4])-[NH;D2;+0:6]-[c:7](:[c:8]):[c:9]
99.7
[{"value": 99.7, "product": "C(C)(=O)N1CCC(CC1)CNC(=S)NC1=CC=C(C=C1)Cl", "details": "PERCENTYIELD", "is_desired": false}]
null
null
3
HOUR
A mixture of 3.1 parts of 1-acetyl-4-piperidinemethanamine, 3.4 parts of 1-chloro-4-isothiocyanatobenzene and 90 parts of tetrahydrofuran was stirred for 3 hours at room temperature. The reaction mixture was evaporated, yielding 6.5 parts (99.7%) of N-[(1-acetyl-4-piperidinyl)methyl]-N'-(4-chlorophenyl)thiourea as a re...
10.6084/m9.figshare.5104873.v1
null
Primary amine.Isothiocyanate
Thiourea
null
null
C1CC[NH]CC1.c1ccccc1
null
O1CCCC1
null
3
CC(=O)N1CCC(CN)CC1.S=C=Nc1ccc(Cl)cc1>O1CCCC1>CC(=O)N1CCC(CNC(=S)Nc2ccc(Cl)cc2)CC1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-ee56261ae4364f3eb952ade8c36ca8dd
CC(=O)N1CCC(CNC(=S)Nc2ccccc2)CC1>>CC(=O)N1CCC(CNc2nc3ccccc3s2)CC1
C(C)O.C(C)(=O)N1CCC(CC1)CNC(=S)NC1=CC=CC=C1.ClC(Cl)(Cl)Cl.BrBr>>C(C)(=O)N1CCC(CC1)CNC=1SC2=C(N1)C=CC=C2
[CH3:1][C:2](=[O:3])[N:4]1[CH2:5][CH2:6][CH:7]([CH2:8][NH:9][C:10]([NH:11][c:12]2[cH:13][cH:14][cH:15][cH:16][cH:17]2)=[S:18])[CH2:19][CH2:20]1>>[CH3:1][C:2](=[O:3])[N:4]1[CH2:5][CH2:6][CH:7]([CH2:8][NH:9][c:10]2[n:11][c:12]3[cH:13][cH:14][cH:15][cH:16][c:17]3[s:18]2)[CH2:19][CH2:20]1
CC(=O)N1CCC(CNC(=S)Nc2ccccc2)CC1
CC(=O)N1CCC(CNc2nc3ccccc3s2)CC1
null
null
C(C)#N
Aromatic Heterocycle Formation
OtherReaction
9fc354848fb2fb52ac9a677ec08efbe70faac27defb4ee4a070dc3814d93a73c
01ff041a21adca51a94f69a62115e81e604cce12edd47d529ec3eedb88c39f4c
c1ccc2sc(NCC3CCNCC3)nc2c1
[C:1]-[#7:2]-[C;H0;D3;+0:3](=[S;H0;D1;+0:4])-[NH;D2;+0:5]-[c:6](:[c:7]):[cH;D2;+0:8]:[c:9]:[c:10]>>[C:1]-[#7:2]-[c;H0;D3;+0:3]1:[n;H0;D2;+0:5]:[c:6](:[c:7]):[c;H0;D3;+0:8](:[c:9]:[c:10]):[s;H0;D2;+0:4]:1
null
[]
null
null
null
null
To a stirred mixture of 5.8 parts of N-[(1-acetyl-4-piperidinyl)methyl]-N'-phenylthiourea and 160 parts of tetrachloromethane were added 3.7 parts of bromine. The whole was stirred and refluxed for 15 minutes. After the additions of 16 parts of ethanol and 16 parts of acetonitrile, the reaction mixture was cooled. The ...
10.6084/m9.figshare.5104873.v1
null
Thiourea
null
c1ccccc1
c1ccc2scnc2c1
C1CC[NH]CC1.c1ccc2scnc2c1
null
C(C)#N
null
null
CC(=O)N1CCC(CNC(=S)Nc2ccccc2)CC1>C(C)#N>CC(=O)N1CCC(CNc2nc3ccccc3s2)CC1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-1d5e504cf6ef4230b04acc78d845b3d1
BrBr.CC(=O)N1CCC(CNC(=S)Nc2ccc3c(c2)OCO3)CC1>>Br.c1c2c(cc3sc(NCC4CCNCC4)nc13)OCO2
C(C)(=O)N1CCC(CC1)CNC(=S)NC1=CC2=C(OCO2)C=C1.Br.BrBr>>Br.Br.N1CCC(CC1)CNC=1SC2=C(N1)C=C1C(=C2)OCO1
Br[Br:2].CC(=O)[N:15]1[CH2:14][CH2:13][CH:12]([CH2:11][NH:10][C:9](=[S:8])[NH:18][c:19]2[cH:3][c:4]3[c:5]([cH:6][cH:7]2)[O:20][CH2:21][O:22]3)[CH2:17][CH2:16]1>>[BrH:2].[cH:3]1[c:4]2[c:5]([cH:6][c:7]3[s:8][c:9]([NH:10][CH2:11][CH:12]4[CH2:13][CH2:14][NH:15][CH2:16][CH2:17]4)[n:18][c:19]13)[O:20][CH2:21][O:22]2
BrBr.CC(=O)N1CCC(CNC(=S)Nc2ccc3c(c2)OCO3)CC1
Br.c1c2c(cc3sc(NCC4CCNCC4)nc13)OCO2
null
null
O
Aromatic Heterocycle Formation
OtherReaction
b21aac40b9fa5db102a5f0ced2b27c262361293cdbbfa875470bd435c685e345
91b316de46b0059d06bca8c45d016b409246fcf8be4d5e8a003be4245d82d8e4
c1c2c(cc3sc(NCC4CCNCC4)nc13)OCO2
Br-[Br;H0;D1;+0:1].C-C(=O)-[N;H0;D3;+0:2](-[C:3]-[C:4])-[C:5]-[C:6].[#8:7]-[c:8]:[c:9]:[cH;D2;+0:10]:[c:11](-[NH;D2;+0:12]-[C;H0;D3;+0:13](=[S;H0;D1;+0:14])-[#7:15]-[C:16]):[c:17]>>[#8:7]-[c:8]:[c:9]:[c;H0;D3;+0:10]1:[s;H0;D2;+0:14]:[c;H0;D3;+0:13](-[#7:15]-[C:16]):[n;H0;D2;+0:12]:[c:11]:1:[c:17].[C:4]-[C:3]-[NH;D2;+0:...
58.4
[{"value": 58.4, "product": "Br.Br.N1CCC(CC1)CNC=1SC2=C(N1)C=C1C(=C2)OCO1", "details": "PERCENTYIELD", "is_desired": false}]
null
null
8
HOUR
A mixture of 33.3 parts of N-[(1-acetyl-4-piperidinyl)methyl]-N'-(1,3-benzodioxol-5-yl)thiourea, 112.5 parts of a hydrobromic acid solution 48% in water and 75 parts of water was stirred till all solid entered the solution. Then there were added 16 parts of bromine and stirring was continued overnight at reflux. After ...
10.6084/m9.figshare.5104873.v1
null
Thiourea.Tertiary amide
Secondary amine
C1CC[NH]CC1.c1ccc2c(c1)OCO2
C1CCNCC1.c1nc2cc3c(cc2s1)OCO3
C1CCNCC1.c1nc2cc3c(cc2s1)OCO3
HBr
O
null
8
BrBr.CC(=O)N1CCC(CNC(=S)Nc2ccc3c(c2)OCO3)CC1>O>Br.c1c2c(cc3sc(NCC4CCNCC4)nc13)OCO2
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-e394f3d7b4114983b64b840292c23c89
CI.Nc1ncnc2sc(S)nc12>>CSc1nc2c(N)ncnc2s1
[H-].[Na+].NC=1C2=C(N=CN1)SC(=N2)S.CN(C=O)C.IC>>CSC=1SC=2N=CN=C(C2N1)N
I[CH3:1].[SH:2][c:3]1[n:4][c:5]2[c:6]([NH2:7])[n:8][cH:9][n:10][c:11]2[s:12]1>>[CH3:1][S:2][c:3]1[n:4][c:5]2[c:6]([NH2:7])[n:8][cH:9][n:10][c:11]2[s:12]1
CI.Nc1ncnc2sc(S)nc12
CSc1nc2c(N)ncnc2s1
null
null
O
Heteroatom Alkylation and Arylation
thioether_nucl_sub
cbeef1e4b9250d05ec80fbfc2f139c184e610b2c8de8aec4214044a1d69bd441
a20e50d7df818b91ffc2e826d304ad74f6246978a284c599e867e2d806b7437e
c1ncc2ncsc2n1
I-[CH3;D1;+0:1].[#7;a:2]:[c:3]1:[#16;a:4]:[c:5](-[SH;D1;+0:6]):[#7;a:7]:[c:8]:1:[c:9]:[#7;a:10]>>[#7;a:2]:[c:3]1:[#16;a:4]:[c:5](-[S;H0;D2;+0:6]-[CH3;D1;+0:1]):[#7;a:7]:[c:8]:1:[c:9]:[#7;a:10]
null
[]
null
null
4
HOUR
To a stirred and cooled (below 25° C.) mixture of 13.9 parts of 7-aminothiazolo[5,4-d]pyrimidin-2-thiol and 180 parts of N,N-dimethylformamide were added portionwise 4.3 parts of a sodium hydride dispersion 50% while cooling. After stirring for 1 hour, 11.5 parts of iodomethane were added dropwise at a temperature belo...
10.6084/m9.figshare.5104873.v1
null
Aromatic thiol
Monosulfide
null
null
c1ncc2ncsc2n1
HI
O
null
4
CI.Nc1ncnc2sc(S)nc12>O>CSc1nc2c(N)ncnc2s1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-9e71969e97bc4104b9560ff69314f6e6
CC(=O)N1CCC(CN)CC1.CSc1nc2cccnc2s1>>CC(=O)N1CCC(CNc2nc3cccnc3s2)CC1
C(C)(=O)N1CCC(CC1)CN.CSC=1SC2=NC=CC=C2N1>>C(C)(=O)N1CCC(CC1)CNC=1SC2=NC=CC=C2N1
[CH3:1][C:2](=[O:3])[N:4]1[CH2:5][CH2:6][CH:7]([CH2:8][NH2:9])[CH2:19][CH2:20]1.CS[c:10]1[n:11][c:12]2[cH:13][cH:14][cH:15][n:16][c:17]2[s:18]1>>[CH3:1][C:2](=[O:3])[N:4]1[CH2:5][CH2:6][CH:7]([CH2:8][NH:9][c:10]2[n:11][c:12]3[cH:13][cH:14][cH:15][n:16][c:17]3[s:18]2)[CH2:19][CH2:20]1
CC(=O)N1CCC(CN)CC1.CSc1nc2cccnc2s1
CC(=O)N1CCC(CNc2nc3cccnc3s2)CC1
null
null
null
Heteroatom Alkylation and Arylation
OtherReaction
23be8ab067f9bcd8ca31730b1ce864559d67359a071482ff9cb09b381b50c384
88e0224d19b2dce8f9987d52554afb32090d36ff7ee19e89dc5bf66d30974ec4
c1cnc2sc(NCC3CCNCC3)nc2c1
C-S-[c;H0;D3;+0:1]1:[#16;a:2]:[c:3](:[#7;a:4]:[c:5]):[c:6]:[#7;a:7]:1.[C:8]-[C:9]-[NH2;D1;+0:10]>>[C:8]-[C:9]-[NH;D2;+0:10]-[c;H0;D3;+0:1]1:[#16;a:2]:[c:3](:[#7;a:4]:[c:5]):[c:6]:[#7;a:7]:1
93
[{"value": 93.0, "product": "C(C)(=O)N1CCC(CC1)CNC=1SC2=NC=CC=C2N1", "details": "PERCENTYIELD", "is_desired": false}]
140
CELSIUS
null
null
A mixture of 11 parts of 1-acetyl-4-piperidinemethanamine and 9 parts of 2-(methylthio)thiazolo[5,4-b]pyridine was stirred and heated for 20 hours at 140° C. The whole was purified by column chromatography over silica gel using a mixture of trichloromethane and methanol (95:5 by volume) as eluent. The pure fractions we...
10.6084/m9.figshare.5104873.v1
null
Primary amine.Monosulfide
Secondary amine
c1cnc2scnc2c1
c1cnc2scnc2c1
C1CC[NH]CC1.c1cnc2scnc2c1
Other
null
140
null
CC(=O)N1CCC(CN)CC1.CSc1nc2cccnc2s1>>CC(=O)N1CCC(CNc2nc3cccnc3s2)CC1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-8ac978557b4942dd8db7d2fbfc8ff579
CC(=O)N1CCC(CNc2nc3ccccc3s2)CC1.CI>>CC(=O)N1CCC(CN(C)c2nc3ccccc3s2)CC1
IC.C(C)(=O)N1CCC(CC1)CNC=1SC2=C(N1)C=CC=C2.[H-].[Na+].CN(C=O)C>>C(C)(=O)N1CCC(CC1)CN(C)C=1SC2=C(N1)C=CC=C2
[CH3:1][C:2](=[O:3])[N:4]1[CH2:5][CH2:6][CH:7]([CH2:8][NH:9][c:11]2[n:12][c:13]3[cH:14][cH:15][cH:16][cH:17][c:18]3[s:19]2)[CH2:20][CH2:21]1.I[CH3:10]>>[CH3:1][C:2](=[O:3])[N:4]1[CH2:5][CH2:6][CH:7]([CH2:8][N:9]([CH3:10])[c:11]2[n:12][c:13]3[cH:14][cH:15][cH:16][cH:17][c:18]3[s:19]2)[CH2:20][CH2:21]1
CC(=O)N1CCC(CNc2nc3ccccc3s2)CC1.CI
CC(=O)N1CCC(CN(C)c2nc3ccccc3s2)CC1
null
null
O
Heteroatom Alkylation and Arylation
N-alkylation of secondary amines with alkyl halides
e1587a52a1bca6a80c6048d43276d8bccf8d3e94e692e6b210e5fd3b22494187
7cc25fba33369069673bac5bd8fc404dc064da8d6c8cf4a77f21f4df0a617fe3
c1ccc2sc(NCC3CCNCC3)nc2c1
I-[CH3;D1;+0:1].[C:2]-[C:3]-[NH;D2;+0:4]-[c:5]1:[#16;a:6]:[c:7]:[c:8]:[#7;a:9]:1>>[C:2]-[C:3]-[N;H0;D3;+0:4](-[CH3;D1;+0:1])-[c:5]1:[#16;a:6]:[c:7]:[c:8]:[#7;a:9]:1
84
[{"value": 84.0, "product": "C(C)(=O)N1CCC(CC1)CN(C)C=1SC2=C(N1)C=CC=C2", "details": "PERCENTYIELD", "is_desired": false}]
null
null
1
HOUR
A mixture of 8.7 parts of 1-acetyl-N-(2-benzothiazolyl)-4-piperidinemethanamine, 1.44 parts of a sodium hydride dispersion 60% and 270 parts of N,N-dimethylformamide was stirred for 1 hour at room temperature. 5.48 Parts of iodomethane were added dropwise slowly. Upon completion, stirring was continued overnight at roo...
10.6084/m9.figshare.5104873.v1
null
Secondary amine
Tertiary amine
null
null
C1CC[NH]CC1.c1ccc2scnc2c1
HI
O
null
1
CC(=O)N1CCC(CNc2nc3ccccc3s2)CC1.CI>O>CC(=O)N1CCC(CN(C)c2nc3ccccc3s2)CC1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-c9b16aa6f74749a99eb7aab43a37c592
CC(=O)N1CCC(CNc2nc3ccccc3s2)CC1>>Br.c1ccc2sc(NCC3CCNCC3)nc2c1
C(C)(=O)N1CCC(CC1)CNC=1SC2=C(N1)C=CC=C2.Br>>Br.Br.N1CCC(CC1)CNC=1SC2=C(N1)C=CC=C2
CC(=O)[N:14]1[CH2:13][CH2:12][CH:11]([CH2:10][NH:9][c:8]2[s:7][c:6]3[cH:5][cH:4][cH:3][cH:19][c:18]3[n:17]2)[CH2:16][CH2:15]1>>[BrH:2].[cH:3]1[cH:4][cH:5][c:6]2[s:7][c:8]([NH:9][CH2:10][CH:11]3[CH2:12][CH2:13][NH:14][CH2:15][CH2:16]3)[n:17][c:18]2[cH:19]1
CC(=O)N1CCC(CNc2nc3ccccc3s2)CC1
Br.c1ccc2sc(NCC3CCNCC3)nc2c1
null
null
O
Miscellaneous
Hydrogenolysis of tertiary amines
9b929ebabc9d56e2ac499595af1f340b21610b5f71874bd02f1d8f46a982605e
5ba542a97dd3ca917dd84dc29c99ae9b05b6ca96dbd806e22774484cf1a34b59
c1ccc2sc(NCC3CCNCC3)nc2c1
C-C(=O)-[N;H0;D3;+0:1](-[C:2]-[C:3])-[C:4]-[C:5]>>[C:3]-[C:2]-[NH;D2;+0:1]-[C:4]-[C:5]
79
[{"value": 79.0, "product": "Br.Br.N1CCC(CC1)CNC=1SC2=C(N1)C=CC=C2", "details": "PERCENTYIELD", "is_desired": false}]
null
null
null
null
A mixture of 140 parts of 1-acetyl-N-(2-benzothiazolyl)-4-piperidinemethanamine and 1500 parts of a hydrobromic acid solution 24% in water was stirred and refluxed for 5 hours. The reaction mixture was evaporated and the residue was suspended in boiling ethanol. After cooling, the product was filtered off and dried, yi...
10.6084/m9.figshare.5104873.v1
null
Tertiary amide
Secondary amine
C1CC[NH]CC1
C1CCNCC1
c1ccc2scnc2c1.C1CCNCC1
HO-
O
null
null
CC(=O)N1CCC(CNc2nc3ccccc3s2)CC1>O>Br.c1ccc2sc(NCC3CCNCC3)nc2c1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-75690f0a653d4186828de4ecee7463a7
Nc1ccccc1O.S=C=NCc1ccncc1>>Oc1ccccc1NC(=S)NCc1ccncc1
N(=C=S)CC1=CC=NC=C1.NC1=C(C=CC=C1)O>>OC1=C(C=CC=C1)NC(=S)NCC1=CC=NC=C1
[OH:1][c:2]1[cH:3][cH:4][cH:5][cH:6][c:7]1[NH2:8].[C:9](=[S:10])=[N:11][CH2:12][c:13]1[cH:14][cH:15][n:16][cH:17][cH:18]1>>[OH:1][c:2]1[cH:3][cH:4][cH:5][cH:6][c:7]1[NH:8][C:9](=[S:10])[NH:11][CH2:12][c:13]1[cH:14][cH:15][n:16][cH:17][cH:18]1
Nc1ccccc1O.S=C=NCc1ccncc1
Oc1ccccc1NC(=S)NCc1ccncc1
null
null
C(C)#N
Heteroatom Alkylation and Arylation
thiourea
9037f368cdf8e91fcd9f93f4d9cf27991f85fa921c9d19c7875d3a77561f439b
0fbf3d6c8cd704ac451c2cf111f32090de5e76a9d41cce326e212c758f4ed46f
S=C(NCc1ccncc1)Nc1ccccc1
[NH2;D1;+0:1]-[c:2](:[c:3]):[c:4].[S;D1;H0:5]=[C;H0;D2;+0:6]=[N;H0;D2;+0:7]-[C:8]-[c:9]>>[S;D1;H0:5]=[C;H0;D3;+0:6](-[NH;D2;+0:7]-[C:8]-[c:9])-[NH;D2;+0:1]-[c:2](:[c:3]):[c:4]
null
[]
null
null
3
HOUR
A mixture of 15 parts of 4-(isothiocyanatomethyl)pyridine, 9.5 parts of 2-aminophenol and 160 parts of acetonitrile was stirred for 3 hours at room temperature. The precipitated product was filtered off, washed with 2,2'-oxybispropane and crystallized from acetonitrile, yielding 8.22 parts of N-(2-hydroxyphenyl)-N'-(4-...
10.6084/m9.figshare.5104873.v1
null
Primary amine.Isothiocyanate
Thiourea
null
null
c1ccccc1.c1ccncc1
null
C(C)#N
null
3
Nc1ccccc1O.S=C=NCc1ccncc1>C(C)#N>Oc1ccccc1NC(=S)NCc1ccncc1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-1f8d4057264749fe934f5d65ae0c3eaf
Oc1ccccc1NC(=S)NCc1ccncc1>>c1ccc2oc(NCc3ccncc3)nc2c1
OC1=C(C=CC=C1)NC(=S)NCC1=CC=NC=C1.[S].CC(C)O>>N1=CC=C(C=C1)CNC=1OC2=C(N1)C=CC=C2
S=[C:6]([NH:7][CH2:8][c:9]1[cH:10][cH:11][n:12][cH:13][cH:14]1)[NH:15][c:16]1[c:4]([OH:5])[cH:3][cH:2][cH:1][cH:17]1>>[cH:1]1[cH:2][cH:3][c:4]2[o:5][c:6]([NH:7][CH2:8][c:9]3[cH:10][cH:11][n:12][cH:13][cH:14]3)[n:15][c:16]2[cH:17]1
Oc1ccccc1NC(=S)NCc1ccncc1
c1ccc2oc(NCc3ccncc3)nc2c1
null
[Hg]=O
C(C)#N
Aromatic Heterocycle Formation
OtherReaction
e5161dad16ba0de611bb88bf71727cf43a1a35a2554fa1428c27f381c2392622
5b50b5990b44a3b8932dd42e9875f76813cd6ae8ffd0db2c3ea135be28fae54d
c1ccc2oc(NCc3ccncc3)nc2c1
S=[C;H0;D3;+0:1](-[#7:2]-[C:3])-[NH;D2;+0:4]-[c:5](:[c:6]):[c:7](-[OH;D1;+0:8]):[c:9]>>[C:3]-[#7:2]-[c;H0;D3;+0:1]1:[n;H0;D2;+0:4]:[c:5](:[c:6]):[c:7](:[c:9]):[o;H0;D2;+0:8]:1
56
[{"value": 56.0, "product": "N1=CC=C(C=C1)CNC=1OC2=C(N1)C=CC=C2", "details": "PERCENTYIELD", "is_desired": false}]
null
null
null
null
A mixture of 14 parts of N-(2-hydroxyphenyl)-N'-(4-pyridinylmethyl)thiourea, 20 parts of mercury(II) oxide, 1 part of sulfur, 160 parts of 2-propanol and 160 parts of acetonitrile was stirred and refluxed for 14 hours. The reaction mixture was filtered over diatomaceous earth and the filtrate was evaporated. The oily r...
10.6084/m9.figshare.5104873.v1
null
Thiourea.Aromatic alcohol
null
c1ccccc1
c1ccc2ocnc2c1
c1ccc2ocnc2c1.c1ccncc1
Other
[Hg]=O.C(C)#N
null
null
Oc1ccccc1NC(=S)NCc1ccncc1>[Hg]=O.C(C)#N>c1ccc2oc(NCc3ccncc3)nc2c1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-e920b357190a42caa0fed114a232849c
c1ccc2oc(NCc3ccncc3)nc2c1>>c1ccc2oc(NCC3CCNCC3)nc2c1
N1=CC=C(C=C1)CNC=1OC2=C(N1)C=CC=C2.[H][H]>>N1CCC(CC1)CNC=1OC2=C(N1)C=CC=C2
[cH:1]1[cH:2][cH:3][c:4]2[o:5][c:6]([NH:7][CH2:8][c:9]3[cH:10][cH:11][n:12][cH:13][cH:14]3)[n:15][c:16]2[cH:17]1>>[cH:1]1[cH:2][cH:3][c:4]2[o:5][c:6]([NH:7][CH2:8][CH:9]3[CH2:10][CH2:11][NH:12][CH2:13][CH2:14]3)[n:15][c:16]2[cH:17]1
c1ccc2oc(NCc3ccncc3)nc2c1
c1ccc2oc(NCC3CCNCC3)nc2c1
null
null
CO
Reduction
OtherReaction
8a6c78a63989dd47e282eb33ae5ce6bfcead5defaa210963e9125c31297ee886
2b7f370a519e29b4dede190aa36b37f30822496e32f2c8bfa9736e631bde52e2
c1ccc2oc(NCC3CCNCC3)nc2c1
[#7:1]-[C:2]-[c;H0;D3;+0:3]1:[cH;D2;+0:4]:[cH;D2;+0:5]:[n;H0;D2;+0:6]:[cH;D2;+0:7]:[cH;D2;+0:8]:1>>[#7:1]-[C:2]-[CH;D3;+0:3]1-[CH2;D2;+0:4]-[CH2;D2;+0:5]-[NH;D2;+0:6]-[CH2;D2;+0:7]-[CH2;D2;+0:8]-1
null
[]
null
null
null
null
A mixture of 4.5 parts of N-(4-pyridinylmethyl)-2-benzoxazolamine and 120 parts of methanol was hydrogenated at normal pressure at about 50° C. with 2 parts of rhodium-on-charcoal catalyst 5%. After the calculated amount of hydrogen was taken up, the catalyst was filtered off and the filtrate was evaporated, yielding 4...
10.6084/m9.figshare.5104873.v1
null
null
Secondary amine
c1ccncc1
C1CCNCC1
c1ccc2ocnc2c1.C1CCNCC1
null
CO
null
null
c1ccc2oc(NCc3ccncc3)nc2c1>CO>c1ccc2oc(NCC3CCNCC3)nc2c1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-254beb3cf13148c9862feb5a4f049125
CC(=O)c1ccc(F)cc1O.ClCc1ccccc1>>CC(=O)c1ccc(F)cc1OCc1ccccc1
FC1=CC(=C(C=C1)C(C)=O)O.ClCC1=CC=CC=C1.C([O-])([O-])=O.[K+].[K+].[I-].[K+]>>FC1=CC(=C(C=C1)C(C)=O)OCC1=CC=CC=C1
[CH3:1][C:2](=[O:3])[c:4]1[cH:5][cH:6][c:7]([F:8])[cH:9][c:10]1[OH:11].Cl[CH2:12][c:13]1[cH:14][cH:15][cH:16][cH:17][cH:18]1>>[CH3:1][C:2](=[O:3])[c:4]1[cH:5][cH:6][c:7]([F:8])[cH:9][c:10]1[O:11][CH2:12][c:13]1[cH:14][cH:15][cH:16][cH:17][cH:18]1
CC(=O)c1ccc(F)cc1O.ClCc1ccccc1
CC(=O)c1ccc(F)cc1OCc1ccccc1
null
null
CC(C)=O
Heteroatom Alkylation and Arylation
Williamson Ether Synthesis
7e1040116e3a4cf0e8ec5cc7865388d9cd0efabce6d320a1c25a36e411018d8b
d5f4610d46ccc0478471c5bc0fb862644eaf764bbc5d93badb39d54f6ec8e0a5
c1ccc(COc2ccccc2)cc1
Cl-[CH2;D2;+0:1]-[c:2](:[c:3]):[c:4].[C;D1;H3:5]-[C:6](=[O;D1;H0:7])-[c:8]:[c:9](-[OH;D1;+0:10]):[c:11]>>[C;D1;H3:5]-[C:6](=[O;D1;H0:7])-[c:8]:[c:9](-[O;H0;D2;+0:10]-[CH2;D2;+0:1]-[c:2](:[c:3]):[c:4]):[c:11]
58
[{"value": 58.0, "product": "FC1=CC(=C(C=C1)C(C)=O)OCC1=CC=CC=C1", "details": "PERCENTYIELD", "is_desired": false}]
null
null
8
HOUR
A mixture of 13 parts of 1-(4-fluoro-2-hydroxyphenyl)ethanone, 14.9 parts of (chloromethyl)benzene, 16.4 parts of potassium carbonate, 0.1 parts of potassium iodide and 120 parts of 2-propanone was stirred overnight at reflux temperature. The reaction mixture was evaporated. The reaction mixture was poured into water. ...
10.6084/m9.figshare.5104873.v1
null
Primary halide.Aromatic alcohol
Ether
null
null
c1ccccc1.c1ccccc1
HCl
CC(C)=O
null
8
CC(=O)c1ccc(F)cc1O.ClCc1ccccc1>CC(C)=O>CC(=O)c1ccc(F)cc1OCc1ccccc1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-0d9543b504514c609d822aa97a645569
ClCCCBr.Oc1ccc(F)cc1OCc1ccccc1>>Fc1ccc(OCCCCl)c(OCc2ccccc2)c1
[OH-].[Na+].FC1=CC(=C(C=C1)O)OCC1=CC=CC=C1.BrCCCCl>>ClCCCOC1=C(C=C(C=C1)F)OCC1=CC=CC=C1
Br[CH2:7][CH2:8][CH2:9][Cl:10].[F:1][c:2]1[cH:3][cH:4][c:5]([OH:6])[c:11]([O:12][CH2:13][c:14]2[cH:15][cH:16][cH:17][cH:18][cH:19]2)[cH:20]1>>[F:1][c:2]1[cH:3][cH:4][c:5]([O:6][CH2:7][CH2:8][CH2:9][Cl:10])[c:11]([O:12][CH2:13][c:14]2[cH:15][cH:16][cH:17][cH:18][cH:19]2)[cH:20]1
ClCCCBr.Oc1ccc(F)cc1OCc1ccccc1
Fc1ccc(OCCCCl)c(OCc2ccccc2)c1
null
S(=O)(=O)(O)[O-].C(CCC)[N+](CCCC)(CCCC)CCCC
O
Heteroatom Alkylation and Arylation
Williamson Ether Synthesis
7e1040116e3a4cf0e8ec5cc7865388d9cd0efabce6d320a1c25a36e411018d8b
d5f4610d46ccc0478471c5bc0fb862644eaf764bbc5d93badb39d54f6ec8e0a5
c1ccc(COc2ccccc2)cc1
Br-[CH2;D2;+0:1]-[C:2]-[C:3].[OH;D1;+0:4]-[c:5](:[c:6]):[c:7]>>[C:3]-[C:2]-[CH2;D2;+0:1]-[O;H0;D2;+0:4]-[c:5](:[c:6]):[c:7]
100
[{"value": 100.0, "product": "ClCCCOC1=C(C=C(C=C1)F)OCC1=CC=CC=C1", "details": "PERCENTYIELD", "is_desired": false}]
70
CELSIUS
2
HOUR
To a stirred mixture of 2.5 parts of 4-fluoro-2-(phenylmethoxy)phenol, 2.3 parts of 1-bromo-3-chloropropane, 10 parts of water and 0.39 parts of tetrabutylammonium hydrogen sulfate was added dropwise a solution of 0.7 parts of sodium hydroxide in 5 parts of D at 60° C. (exothermic reaction: temperature rose to 70°). Th...
10.6084/m9.figshare.5104873.v1
null
Primary halide.Aromatic alcohol
Ether
null
null
c1ccccc1.c1ccccc1
HBr
S(=O)(=O)(O)[O-].C(CCC)[N+](CCCC)(CCCC)CCCC.O
70
2
ClCCCBr.Oc1ccc(F)cc1OCc1ccccc1>S(=O)(=O)(O)[O-].C(CCC)[N+](CCCC)(CCCC)CCCC.O>Fc1ccc(OCCCCl)c(OCc2ccccc2)c1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-8dcd6c4737cf4236a7025063f5be88e5
NCC1CCN(CC2COc3ccccc3O2)CC1.O=Cc1ccc(F)cc1>>Fc1ccc(CNCC2CCN(CC3COc4ccccc4O3)CC2)cc1
[H][H].Br.Br.O1C(COC2=C1C=CC=C2)CN2CCC(CC2)CN.FC1=CC=C(C=O)C=C1.S1C=CC=C1.[O-2].[Ca+2]>>O1C(COC2=C1C=CC=C2)CN2CCC(CC2)CNCC2=CC=C(C=C2)F
[NH2:7][CH2:8][CH:9]1[CH2:10][CH2:11][N:12]([CH2:13][CH:14]2[CH2:15][O:16][c:17]3[cH:18][cH:19][cH:20][cH:21][c:22]3[O:23]2)[CH2:24][CH2:25]1.O=[CH:6][c:5]1[cH:4][cH:3][c:2]([F:1])[cH:27][cH:26]1>>[F:1][c:2]1[cH:3][cH:4][c:5]([CH2:6][NH:7][CH2:8][CH:9]2[CH2:10][CH2:11][N:12]([CH2:13][CH:14]3[CH2:15][O:16][c:17]4[cH:18]...
NCC1CCN(CC2COc3ccccc3O2)CC1.O=Cc1ccc(F)cc1
Fc1ccc(CNCC2CCN(CC3COc4ccccc4O3)CC2)cc1
null
[Pd]
CO
Heteroatom Alkylation and Arylation
Reductive amination with aldehyde
422be648aea52bce28ccc8fb32ec3178aaa47bbd624f063874619362f075b5f2
7915721a3e395aed85e3c40dc4d725c571a931ac517c6a0da16f2a2b0bb5eac7
c1ccc(CNCC2CCN(CC3COc4ccccc4O3)CC2)cc1
O=[CH;D2;+0:1]-[c:2](:[c:3]):[c:4].[C:5]-[C:6]-[NH2;D1;+0:7]>>[C:5]-[C:6]-[NH;D2;+0:7]-[CH2;D2;+0:1]-[c:2](:[c:3]):[c:4]
98.3
[{"value": 98.3, "product": "O1C(COC2=C1C=CC=C2)CN2CCC(CC2)CNCC2=CC=C(C=C2)F", "details": "PERCENTYIELD", "is_desired": false}]
null
null
null
null
A mixture of 5 parts of 1-[(2,3-dihydro-1,4-benzodioxin-2-yl)methyl]-4-piperidinmethanamine dihydrobromide, 1.6 parts of 4-fluorobenzaldehyde, 3 parts of a solution of thiophene in methanol 4%, 200 parts of methanol and 4 parts of calcium oxide was hydrogenated at normal pressure and at room temperature with 2 parts of...
10.6084/m9.figshare.5104873.v1
null
Aldehyde.Primary amine
Secondary amine
null
null
c1ccccc1.C1CC[NH]CC1.c1ccc2c(c1)OCCO2
Other
[Pd].CO
null
null
NCC1CCN(CC2COc3ccccc3O2)CC1.O=Cc1ccc(F)cc1>[Pd].CO>Fc1ccc(CNCC2CCN(CC3COc4ccccc4O3)CC2)cc1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-b827a6a6c42e4114b2f5cab02191890a
CC(NCc1ccccc1)C1CCN(CC2COc3ccccc3O2)CC1>>CC(N)C1CCN(CC2COc3ccccc3O2)CC1
[H][H].O1C(COC2=C1C=CC=C2)CN2CCC(CC2)C(NCC2=CC=CC=C2)C>>O1C(COC2=C1C=CC=C2)CN2CCC(CC2)C(N)C
c1ccc(C[NH:3][CH:2]([CH3:1])[CH:4]2[CH2:5][CH2:6][N:7]([CH2:8][CH:9]3[CH2:10][O:11][c:12]4[cH:13][cH:14][cH:15][cH:16][c:17]4[O:18]3)[CH2:19][CH2:20]2)cc1>>[CH3:1][CH:2]([NH2:3])[CH:4]1[CH2:5][CH2:6][N:7]([CH2:8][CH:9]2[CH2:10][O:11][c:12]3[cH:13][cH:14][cH:15][cH:16][c:17]3[O:18]2)[CH2:19][CH2:20]1
CC(NCc1ccccc1)C1CCN(CC2COc3ccccc3O2)CC1
CC(N)C1CCN(CC2COc3ccccc3O2)CC1
null
[Pd]
CO
Deprotection
OtherReaction
93c46c2f9981b731115295839d7158a8a73faedd00707b7604ace2fa5f580cbc
f6571fb5b7780a2b467937abfba91ba7d787f19d503265f299ff4a25a08963bd
c1ccc2c(c1)OCC(CN1CCCCC1)O2
[C:1]-[C:2](-[C;D1;H3:3])-[NH;D2;+0:4]-C-c1:c:c:c:c:c:1>>[C:1]-[C:2](-[C;D1;H3:3])-[NH2;D1;+0:4]
80.4
[{"value": 80.4, "product": "O1C(COC2=C1C=CC=C2)CN2CCC(CC2)C(N)C", "details": "PERCENTYIELD", "is_desired": false}]
null
null
null
null
A mixture of 13.2 parts of 1-[(2,3-dihydro-1,4-benzodioxin-2-yl)methyl]-α-methyl-N-(phenylmethyl)-4-piperidinemethanamine and 160 parts of methanol was hydrogenated at normal pressure and at 50° C. with 2 parts of palladium-on-charcoal catalyst 10%. After the calculated amount of hydrogen was taken up, the catalyst was...
10.6084/m9.figshare.5104873.v1
null
Secondary amine
Primary amine
c1ccccc1
null
C1CC[NH]CC1.c1ccc2c(c1)OCCO2
Other
[Pd].CO
null
null
CC(NCc1ccccc1)C1CCN(CC2COc3ccccc3O2)CC1>[Pd].CO>CC(N)C1CCN(CC2COc3ccccc3O2)CC1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-ce4481d3c1e949b698e956653885160d
CC1(C2CCNCC2)OCCO1.OCC1COc2ccccc2O1>>CC1(C2CCN(CC3COc4ccccc4O3)CC2)OCCO1
O1C(COC2=C1C=CC=C2)CO.CC1=CC=C(C=C1)S(=O)(=O)[O-].CC1(OCCO1)C1CCNCC1.C([O-])([O-])=O.[Na+].[Na+].CN(C(C)=O)C>>O1C(COC2=C1C=CC=C2)CN2CCC(CC2)C2(OCCO2)C
[CH3:1][C:2]1([CH:3]2[CH2:4][CH2:5][NH:6][CH2:18][CH2:19]2)[O:20][CH2:21][CH2:22][O:23]1.O[CH2:7][CH:8]1[CH2:9][O:10][c:11]2[cH:12][cH:13][cH:14][cH:15][c:16]2[O:17]1>>[CH3:1][C:2]1([CH:3]2[CH2:4][CH2:5][N:6]([CH2:7][CH:8]3[CH2:9][O:10][c:11]4[cH:12][cH:13][cH:14][cH:15][c:16]4[O:17]3)[CH2:18][CH2:19]2)[O:20][CH2:21][C...
CC1(C2CCNCC2)OCCO1.OCC1COc2ccccc2O1
CC1(C2CCN(CC3COc4ccccc4O3)CC2)OCCO1
null
null
O
Heteroatom Alkylation and Arylation
OtherReaction
511913fc601efdcc18555347fcfe0c2354215793b65f509995496ee3f61c9425
87693a475e46c41583976158ec46dcaf8be8cc05c5635654a6a68033770f8d5c
c1ccc2c(c1)OCC(CN1CCC(C3OCCO3)CC1)O2
O-[CH2;D2;+0:1]-[C:2](-[#8:3]-[c:4])-[C:5]-[#8:6].[C:7]-[C:8]-[NH;D2;+0:9]-[C:10]-[C:11]>>[#8:6]-[C:5]-[C:2](-[CH2;D2;+0:1]-[N;H0;D3;+0:9](-[C:8]-[C:7])-[C:10]-[C:11])-[#8:3]-[c:4]
100
[{"value": 100.0, "product": "O1C(COC2=C1C=CC=C2)CN2CCC(CC2)C2(OCCO2)C", "details": "PERCENTYIELD", "is_desired": false}]
75
CELSIUS
8
HOUR
A mixture of 22.5 parts of 2,3-dihydro-1,4-benzodioxin-2-methanol 4-methylbenzenesulfonate (ester), 11.1 parts of 4-(2-methyl-1,3-dioxolan-2-yl)piperidine, 15 parts of sodium carbonate and 135 parts of N,N-dimethylacetamide was stirred overnight at 75° C. Water was added. The product was extracted with 4-methyl-2-penta...
10.6084/m9.figshare.5104873.v1
null
Primary alcohol.Secondary amine
Tertiary amine
C1CCNCC1
C1CC[NH]CC1
C1CC[NH]CC1.c1ccc2c(c1)OCCO2.C1COCO1
HO-
O
75
8
CC1(C2CCNCC2)OCCO1.OCC1COc2ccccc2O1>O>CC1(C2CCN(CC3COc4ccccc4O3)CC2)OCCO1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-6e6cbc22abe547e39f9456ddca12ca59
CC1(C2CCN(CC3COc4ccccc4O3)CC2)OCCO1>>CC(=O)C1CCN(CC2COc3ccccc3O2)CC1
[OH-].[Na+].O1C(COC2=C1C=CC=C2)CN2CCC(CC2)C2(OCCO2)C.Cl>>O1C(COC2=C1C=CC=C2)CN2CCC(CC2)C(C)=O
C1C[O:3][C:2]([CH3:1])([CH:4]2[CH2:5][CH2:6][N:7]([CH2:8][CH:9]3[CH2:10][O:11][c:12]4[cH:13][cH:14][cH:15][cH:16][c:17]4[O:18]3)[CH2:19][CH2:20]2)O1>>[CH3:1][C:2](=[O:3])[CH:4]1[CH2:5][CH2:6][N:7]([CH2:8][CH:9]2[CH2:10][O:11][c:12]3[cH:13][cH:14][cH:15][cH:16][c:17]3[O:18]2)[CH2:19][CH2:20]1
CC1(C2CCN(CC3COc4ccccc4O3)CC2)OCCO1
CC(=O)C1CCN(CC2COc3ccccc3O2)CC1
null
null
null
Miscellaneous
Ketal hydrolysis to ketone
bc99a45944d6d67c8bd263755d04463b42623d20ce36570ebfd14e405f44ca50
547697208447432e865290cf95eed8e4fcddc12f59856b7ddbf24dc1accb1210
c1ccc2c(c1)OCC(CN1CCCCC1)O2
[C:1]-[C:2](-[C;H0;D4;+0:3]1(-[C;D1;H3:4])-O-C-C-[O;H0;D2;+0:5]-1)-[C:6]>>[C:1]-[C:2](-[C;H0;D3;+0:3](-[C;D1;H3:4])=[O;H0;D1;+0:5])-[C:6]
55.8
[{"value": 55.8, "product": "O1C(COC2=C1C=CC=C2)CN2CCC(CC2)C(C)=O", "details": "PERCENTYIELD", "is_desired": false}]
null
null
null
null
A mixture of 20.6 parts of 1-[(2,3-dihydro-1,4-benzodioxin-2-yl)methyl]-4-(2-methyl-1,3-dioxolan-2-yl)piperidine and 200 parts of a hydrochloric acid solution 2N was stirred and refluxed for 15 hours. After cooling, crushed ice was added. The whole was treated with a sodium hydroxide solution. The product was extracted...
10.6084/m9.figshare.5104873.v1
null
Ether.Ether
Ketone
C1COCO1
null
C1CC[NH]CC1.c1ccc2c(c1)OCCO2
HO-
null
null
null
CC1(C2CCN(CC3COc4ccccc4O3)CC2)OCCO1>>CC(=O)C1CCN(CC2COc3ccccc3O2)CC1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-9ef0208a4e5b43b2b7f150bae866db41
CC(=O)C1CCN(CC2COc3ccccc3O2)CC1.NCc1ccccc1>>CC(NCc1ccccc1)C1CCN(CC2COc3ccccc3O2)CC1
[H][H].O1C(COC2=C1C=CC=C2)CN2CCC(CC2)C(C)=O.C1(=CC=CC=C1)CN.S1C=CC=C1>>O1C(COC2=C1C=CC=C2)CN2CCC(CC2)C(NCC2=CC=CC=C2)C
O=[C:2]([CH3:1])[CH:11]1[CH2:12][CH2:13][N:14]([CH2:15][CH:16]2[CH2:17][O:18][c:19]3[cH:20][cH:21][cH:22][cH:23][c:24]3[O:25]2)[CH2:26][CH2:27]1.[NH2:3][CH2:4][c:5]1[cH:6][cH:7][cH:8][cH:9][cH:10]1>>[CH3:1][CH:2]([NH:3][CH2:4][c:5]1[cH:6][cH:7][cH:8][cH:9][cH:10]1)[CH:11]1[CH2:12][CH2:13][N:14]([CH2:15][CH:16]2[CH2:17]...
CC(=O)C1CCN(CC2COc3ccccc3O2)CC1.NCc1ccccc1
CC(NCc1ccccc1)C1CCN(CC2COc3ccccc3O2)CC1
null
[Pd]
CO
Heteroatom Alkylation and Arylation
Reductive amination with ketone
4940e8ed9a0db9bde699fdcdc3aff2cff0409c19478aa0ed1acfd98213338adf
07faf85ffe990e88a1de7fd04a339bf226f78d8bfae9712ea59eebd76bb54b9f
c1ccc(CNCC2CCN(CC3COc4ccccc4O3)CC2)cc1
O=[C;H0;D3;+0:1](-[C;D1;H3:2])-[C:3](-[C:4])-[C:5].[NH2;D1;+0:6]-[C:7]-[c:8]>>[C:4]-[C:3](-[CH;D3;+0:1](-[C;D1;H3:2])-[NH;D2;+0:6]-[C:7]-[c:8])-[C:5]
100
[{"value": 100.0, "product": "O1C(COC2=C1C=CC=C2)CN2CCC(CC2)C(NCC2=CC=CC=C2)C", "details": "PERCENTYIELD", "is_desired": false}]
null
null
null
null
A mixture of 10 parts of 1-[1-[(2,3-dihydro-1,4-benzodioxin-2-yl)methyl]-4-piperidinyl]ethanone, 3.8 part of benzenemethanamine, 1 part of a solution of thiophene in methanol 4% and 160 parts of methanol was hydrogenated at normal pressure and at 50° C. with 2 parts of palladium-on-charcoal catalyst 10%. After the calc...
10.6084/m9.figshare.5104873.v1
null
Ketone.Primary amine
Secondary amine
null
null
c1ccccc1.C1CC[NH]CC1.c1ccc2c(c1)OCCO2
Other
[Pd].CO
null
null
CC(=O)C1CCN(CC2COc3ccccc3O2)CC1.NCc1ccccc1>[Pd].CO>CC(NCc1ccccc1)C1CCN(CC2COc3ccccc3O2)CC1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-c88b668ea68341bc8637a8183b3a01fe
BrCC1COc2ccccc2O1.CC(=O)NCC1CCNCC1>>CC(=O)NCC1CCN(CC2COc3ccccc3O2)CC1
BrCC1COC2=C(O1)C=CC=C2.C(C)(=O)O.N1CCC(CC1)CNC(C)=O.C([O-])([O-])=O.[Na+].[Na+].[I-].[Na+]>>O1C(COC2=C1C=CC=C2)CN2CCC(CC2)CNC(C)=O
Br[CH2:10][CH:11]1[CH2:12][O:13][c:14]2[cH:15][cH:16][cH:17][cH:18][c:19]2[O:20]1.[CH3:1][C:2](=[O:3])[NH:4][CH2:5][CH:6]1[CH2:7][CH2:8][NH:9][CH2:21][CH2:22]1>>[CH3:1][C:2](=[O:3])[NH:4][CH2:5][CH:6]1[CH2:7][CH2:8][N:9]([CH2:10][CH:11]2[CH2:12][O:13][c:14]3[cH:15][cH:16][cH:17][cH:18][c:19]3[O:20]2)[CH2:21][CH2:22]1
BrCC1COc2ccccc2O1.CC(=O)NCC1CCNCC1
CC(=O)NCC1CCN(CC2COc3ccccc3O2)CC1
null
null
O.CN(C(C)=O)C
Heteroatom Alkylation and Arylation
N-alkylation of secondary amines with alkyl halides
0240b8450ff2c489d02f5f0d90bc953079d7a3ab239d35a03f26392fc248b4ef
523d37155b42c8dc851abeddadebb241cdd90bdf649ba750c35e13c8c752d7b0
c1ccc2c(c1)OCC(CN1CCCCC1)O2
Br-[CH2;D2;+0:1]-[C:2](-[#8:3]-[c:4])-[C:5]-[#8:6].[C:7]-[C:8]-[NH;D2;+0:9]-[C:10]-[C:11]>>[#8:6]-[C:5]-[C:2](-[CH2;D2;+0:1]-[N;H0;D3;+0:9](-[C:8]-[C:7])-[C:10]-[C:11])-[#8:3]-[c:4]
21
[{"value": 21.0, "product": "O1C(COC2=C1C=CC=C2)CN2CCC(CC2)CNC(C)=O", "details": "PERCENTYIELD", "is_desired": false}]
75
CELSIUS
8
HOUR
A mixture of 12.6 parts of 2-(bromomethyl)-2,3-dihydro-1,4-benzodioxin, 11 parts of N-(4-piperidinylmethyl)acetamide acetate (1:1), 15 parts of sodium carbonate, 0.1 parts of sodium iodide and 135 parts of N,N-dimethylacetamide was stirred overnight at 75° C. The reaction mixture was poured into water. The product was ...
10.6084/m9.figshare.5104873.v1
null
Primary halide.Secondary amine
Tertiary amine
C1CCNCC1
C1CC[NH]CC1
C1CC[NH]CC1.c1ccc2c(c1)OCCO2
HBr
O.CN(C(C)=O)C
75
8
BrCC1COc2ccccc2O1.CC(=O)NCC1CCNCC1>O.CN(C(C)=O)C>CC(=O)NCC1CCN(CC2COc3ccccc3O2)CC1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-665d6e5a8cd442d9a9c1be826d85823b
CC(=O)NCC1CCN(CC2COc3ccccc3O2)CC1>>Br.NCC1CCN(CC2COc3ccccc3O2)CC1
O1C(COC2=C1C=CC=C2)CN2CCC(CC2)CNC(C)=O.Br>>Br.Br.O1C(COC2=C1C=CC=C2)CN2CCC(CC2)CN
CC(=O)[NH:3][CH2:4][CH:5]1[CH2:6][CH2:7][N:8]([CH2:9][CH:10]2[CH2:11][O:12][c:13]3[cH:14][cH:15][cH:16][cH:17][c:18]3[O:19]2)[CH2:20][CH2:21]1>>[BrH:2].[NH2:3][CH2:4][CH:5]1[CH2:6][CH2:7][N:8]([CH2:9][CH:10]2[CH2:11][O:12][c:13]3[cH:14][cH:15][cH:16][cH:17][c:18]3[O:19]2)[CH2:20][CH2:21]1
CC(=O)NCC1CCN(CC2COc3ccccc3O2)CC1
Br.NCC1CCN(CC2COc3ccccc3O2)CC1
null
null
O
Miscellaneous
Hydrogenolysis of amides/imides/carbamates
707d862673494df308d0498876d0cad3507dbc14401d385dbef5e48e25cb04ab
9a852660e38a73253f286565bb98edc48afeded5895ee8b4d0c2bc8a5eeae729
c1ccc2c(c1)OCC(CN1CCCCC1)O2
C-C(=O)-[NH;D2;+0:1]-[C:2]-[C:3]>>[C:3]-[C:2]-[NH2;D1;+0:1]
null
[]
null
null
4
HOUR
A mixture of 2 parts of N-[[1-[(2,3-dihydro-1,4-benzodioxin-2-yl)methyl]-4-piperidinyl]methyl]acetamide, 15 parts of a hydrobromic acid solution 48% in water and 10 parts of water was stirred for 4 hours at reflux temperature. The reaction mixture was evaporated. The residue was crystallized from a mixture of ethanol a...
10.6084/m9.figshare.5104873.v1
null
Secondary amide
Primary amine
null
null
C1CC[NH]CC1.c1ccc2c(c1)OCCO2
HO-
O
null
4
CC(=O)NCC1CCN(CC2COc3ccccc3O2)CC1>O>Br.NCC1CCN(CC2COc3ccccc3O2)CC1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-14205214171c4d26b4456f89ea25af7d
COc1ccc(N=C=S)cc1.NCC1CCN(CC2COc3ccccc3O2)CC1>>COc1ccc(NC(=S)NCC2CCN(CC3COc4ccccc4O3)CC2)cc1
Br.Br.O1C(COC2=C1C=CC=C2)CN2CCC(CC2)CN.[O-2].[Ca+2].N(=C=S)C1=CC=C(C=C1)OC>>O1C(COC2=C1C=CC=C2)CN2CCC(CC2)CNC(=S)NC2=CC=C(C=C2)OC
[CH3:1][O:2][c:3]1[cH:4][cH:5][c:6]([N:7]=[C:8]=[S:9])[cH:29][cH:30]1.[NH2:10][CH2:11][CH:12]1[CH2:13][CH2:14][N:15]([CH2:16][CH:17]2[CH2:18][O:19][c:20]3[cH:21][cH:22][cH:23][cH:24][c:25]3[O:26]2)[CH2:27][CH2:28]1>>[CH3:1][O:2][c:3]1[cH:4][cH:5][c:6]([NH:7][C:8](=[S:9])[NH:10][CH2:11][CH:12]2[CH2:13][CH2:14][N:15]([CH...
COc1ccc(N=C=S)cc1.NCC1CCN(CC2COc3ccccc3O2)CC1
COc1ccc(NC(=S)NCC2CCN(CC3COc4ccccc4O3)CC2)cc1
null
null
CO
Heteroatom Alkylation and Arylation
thiourea
9037f368cdf8e91fcd9f93f4d9cf27991f85fa921c9d19c7875d3a77561f439b
0fbf3d6c8cd704ac451c2cf111f32090de5e76a9d41cce326e212c758f4ed46f
S=C(NCC1CCN(CC2COc3ccccc3O2)CC1)Nc1ccccc1
[C:1]-[C:2]-[NH2;D1;+0:3].[S;D1;H0:4]=[C;H0;D2;+0:5]=[N;H0;D2;+0:6]-[c:7](:[c:8]):[c:9]>>[C:1]-[C:2]-[NH;D2;+0:3]-[C;H0;D3;+0:5](=[S;D1;H0:4])-[NH;D2;+0:6]-[c:7](:[c:8]):[c:9]
null
[]
null
null
3
HOUR
A mixture of 6.4 parts of (1-[(2,3-dihydro-1,4-benzodioxin-2-yl)methyl]-4-piperidinemethanamine dihydrobromide, 4 parts of calcium oxide and 80 parts of methanol was stirred for 3 hours at room temperature. Then there were added 5 parts of 1-isothiocyanato-4-methoxybenzene and the whole was stirred for 3 hours at room ...
10.6084/m9.figshare.5104873.v1
null
Primary amine.Isothiocyanate
Thiourea
null
null
c1ccccc1.C1CC[NH]CC1.c1ccc2c(c1)OCCO2
null
CO
null
3
COc1ccc(N=C=S)cc1.NCC1CCN(CC2COc3ccccc3O2)CC1>CO>COc1ccc(NC(=S)NCC2CCN(CC3COc4ccccc4O3)CC2)cc1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-cedeedf2881343c2aac2758f88e3644b
BrCC1COc2ccccc2O1.c1ccc2sc(NCC3CCNCC3)nc2c1>>c1ccc2c(c1)OCC(CN1CCC(CNc3nc4ccccc4s3)CC1)O2
BrCC1COC2=C(O1)C=CC=C2.Br.Br.N1CCC(CC1)CNC=1SC2=C(N1)C=CC=C2.C([O-])([O-])=O.[Na+].[Na+].[I-].[Na+]>>O1C(COC2=C1C=CC=C2)CN2CCC(CC2)CNC=2SC1=C(N2)C=CC=C1
Br[CH2:10][CH:9]1[CH2:8][O:7][c:5]2[c:4]([cH:3][cH:2][cH:1][cH:6]2)[O:28]1.[NH:11]1[CH2:12][CH2:13][CH:14]([CH2:15][NH:16][c:17]2[n:18][c:19]3[cH:20][cH:21][cH:22][cH:23][c:24]3[s:25]2)[CH2:26][CH2:27]1>>[cH:1]1[cH:2][cH:3][c:4]2[c:5]([cH:6]1)[O:7][CH2:8][CH:9]([CH2:10][N:11]1[CH2:12][CH2:13][CH:14]([CH2:15][NH:16][c:1...
BrCC1COc2ccccc2O1.c1ccc2sc(NCC3CCNCC3)nc2c1
c1ccc2c(c1)OCC(CN1CCC(CNc3nc4ccccc4s3)CC1)O2
null
null
O.CN(C=O)C
Heteroatom Alkylation and Arylation
N-alkylation of secondary amines with alkyl halides
0240b8450ff2c489d02f5f0d90bc953079d7a3ab239d35a03f26392fc248b4ef
523d37155b42c8dc851abeddadebb241cdd90bdf649ba750c35e13c8c752d7b0
c1ccc2c(c1)OCC(CN1CCC(CNc3nc4ccccc4s3)CC1)O2
Br-[CH2;D2;+0:1]-[C:2](-[#8:3]-[c:4])-[C:5]-[#8:6].[C:7]-[C:8]-[NH;D2;+0:9]-[C:10]-[C:11]>>[#8:6]-[C:5]-[C:2](-[CH2;D2;+0:1]-[N;H0;D3;+0:9](-[C:8]-[C:7])-[C:10]-[C:11])-[#8:3]-[c:4]
null
[]
70
CELSIUS
48
HOUR
A mixture of 3.8 parts of 2-(bromomethyl)-2,3-dihydro-1,4-benzodioxin, 6.3 parts of N-(4-piperidinylmethyl)-2-benzothiazolamine dihydrobromide, 10 parts of sodium carbonate, 0.1 parts of sodium iodide and 68 parts of N,N-dimethylformamide was stirred for 48 hours at 70° C. The reaction mixture was poured into water and...
10.6084/m9.figshare.5104873.v1
null
Primary halide.Secondary amine
Tertiary amine
C1CCNCC1
C1CC[NH]CC1
c1ccc2c(c1)OCCO2.C1CC[NH]CC1.c1ccc2scnc2c1
HBr
O.CN(C=O)C
70
48
BrCC1COc2ccccc2O1.c1ccc2sc(NCC3CCNCC3)nc2c1>O.CN(C=O)C>c1ccc2c(c1)OCC(CN1CCC(CNc3nc4ccccc4s3)CC1)O2
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-29a97bcfac644df88361595b25c59427
BrCC1COc2ccccc2O1.Clc1ccc2nc(NCC3CCNCC3)sc2c1>>Clc1ccc2nc(NCC3CCN(CC4COc5ccccc5O4)CC3)sc2c1
BrCC1COC2=C(O1)C=CC=C2.Br.Br.ClC1=CC2=C(N=C(S2)NCC2CCNCC2)C=C1.C([O-])([O-])=O.[Na+].[Na+].[I-].[Na+]>>ClC1=CC2=C(N=C(S2)NCC2CCN(CC2)CC2COC3=C(O2)C=CC=C3)C=C1
Br[CH2:14][CH:15]1[CH2:16][O:17][c:18]2[cH:19][cH:20][cH:21][cH:22][c:23]2[O:24]1.[Cl:1][c:2]1[cH:3][cH:4][c:5]2[n:6][c:7]([NH:8][CH2:9][CH:10]3[CH2:11][CH2:12][NH:13][CH2:25][CH2:26]3)[s:27][c:28]2[cH:29]1>>[Cl:1][c:2]1[cH:3][cH:4][c:5]2[n:6][c:7]([NH:8][CH2:9][CH:10]3[CH2:11][CH2:12][N:13]([CH2:14][CH:15]4[CH2:16][O:...
BrCC1COc2ccccc2O1.Clc1ccc2nc(NCC3CCNCC3)sc2c1
Clc1ccc2nc(NCC3CCN(CC4COc5ccccc5O4)CC3)sc2c1
null
null
CN(C(C)=O)C.O
Heteroatom Alkylation and Arylation
N-alkylation of secondary amines with alkyl halides
0240b8450ff2c489d02f5f0d90bc953079d7a3ab239d35a03f26392fc248b4ef
523d37155b42c8dc851abeddadebb241cdd90bdf649ba750c35e13c8c752d7b0
c1ccc2c(c1)OCC(CN1CCC(CNc3nc4ccccc4s3)CC1)O2
Br-[CH2;D2;+0:1]-[C:2](-[#8:3]-[c:4])-[C:5]-[#8:6].[C:7]-[C:8]-[NH;D2;+0:9]-[C:10]-[C:11]>>[#8:6]-[C:5]-[C:2](-[CH2;D2;+0:1]-[N;H0;D3;+0:9](-[C:8]-[C:7])-[C:10]-[C:11])-[#8:3]-[c:4]
59.8
[{"value": 59.8, "product": "ClC1=CC2=C(N=C(S2)NCC2CCN(CC2)CC2COC3=C(O2)C=CC=C3)C=C1", "details": "PERCENTYIELD", "is_desired": false}]
75
CELSIUS
8
HOUR
A mixture of 1.9 parts of 2-(bromomethyl)-2,3-dihydro-1,4-benzodioxin, 3.3 parts of 6-chloro-N-(4-piperidinylmethyl)-2-benzothiazolamine dihydrobromide, 5 parts of sodium carbonate, 0.1 parts of sodium iodide and 67.5 parts of N,N-dimethylacetamide was stirred overnight at about 75° C. Water was added to the reaction m...
10.6084/m9.figshare.5104873.v1
null
Primary halide.Secondary amine
Tertiary amine
C1CCNCC1
C1CC[NH]CC1
c1ccc2scnc2c1.C1CC[NH]CC1.c1ccc2c(c1)OCCO2
HBr
CN(C(C)=O)C.O
75
8
BrCC1COc2ccccc2O1.Clc1ccc2nc(NCC3CCNCC3)sc2c1>CN(C(C)=O)C.O>Clc1ccc2nc(NCC3CCN(CC4COc5ccccc5O4)CC3)sc2c1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-b15535aa13964aff82f7738b038b6fa8
Fc1ccc(OCCCCl)c(OCc2ccccc2)c1.c1ccc2sc(NCC3CCNCC3)nc2c1>>Fc1ccc(OCCCN2CCC(CNc3nc4ccccc4s3)CC2)c(OCc2ccccc2)c1
ClCCCOC1=C(C=C(C=C1)F)OCC1=CC=CC=C1.Br.Br.N1CCC(CC1)CNC=1SC2=C(N1)C=CC=C2.C([O-])([O-])=O.[Na+].[Na+].[I-].[Na+]>>FC1=CC(=C(OCCCN2CCC(CC2)CNC=2SC3=C(N2)C=CC=C3)C=C1)OCC1=CC=CC=C1
Cl[CH2:9][CH2:8][CH2:7][O:6][c:5]1[cH:4][cH:3][c:2]([F:1])[cH:36][c:27]1[O:28][CH2:29][c:30]1[cH:31][cH:32][cH:33][cH:34][cH:35]1.[NH:10]1[CH2:11][CH2:12][CH:13]([CH2:14][NH:15][c:16]2[n:17][c:18]3[cH:19][cH:20][cH:21][cH:22][c:23]3[s:24]2)[CH2:25][CH2:26]1>>[F:1][c:2]1[cH:3][cH:4][c:5]([O:6][CH2:7][CH2:8][CH2:9][N:10]...
Fc1ccc(OCCCCl)c(OCc2ccccc2)c1.c1ccc2sc(NCC3CCNCC3)nc2c1
Fc1ccc(OCCCN2CCC(CNc3nc4ccccc4s3)CC2)c(OCc2ccccc2)c1
null
null
CN(C(C)=O)C.O
Heteroatom Alkylation and Arylation
N-alkylation of secondary amines with alkyl halides
0240b8450ff2c489d02f5f0d90bc953079d7a3ab239d35a03f26392fc248b4ef
523d37155b42c8dc851abeddadebb241cdd90bdf649ba750c35e13c8c752d7b0
c1ccc(COc2ccccc2OCCCN2CCC(CNc3nc4ccccc4s3)CC2)cc1
Cl-[CH2;D2;+0:1]-[C:2]-[C:3].[C:4]-[C:5]-[NH;D2;+0:6]-[C:7]-[C:8]>>[C:4]-[C:5]-[N;H0;D3;+0:6](-[CH2;D2;+0:1]-[C:2]-[C:3])-[C:7]-[C:8]
65.2
[{"value": 65.2, "product": "FC1=CC(=C(OCCCN2CCC(CC2)CNC=2SC3=C(N2)C=CC=C3)C=C1)OCC1=CC=CC=C1", "details": "PERCENTYIELD", "is_desired": false}]
75
CELSIUS
8
HOUR
A mixture of 3.2 parts of 1-(3-chloropropoxy)-4-fluoro-2-(phenylmethoxy)benzene, 4.1 parts of N-(4-piperidinylmethyl)-2-benzothiazolamine dihydrobromide, 6 parts of sodium carbonate, 0.1 parts of sodium iodide and 67.5 parts of N,N-dimethylacetamide was stirred overnight at 75° C. Water was added and the product was ex...
10.6084/m9.figshare.5104873.v1
null
Primary halide.Secondary amine
Tertiary amine
C1CCNCC1
C1CC[NH]CC1
c1ccccc1.C1CC[NH]CC1.c1ccc2scnc2c1.c1ccccc1
HCl
CN(C(C)=O)C.O
75
8
Fc1ccc(OCCCCl)c(OCc2ccccc2)c1.c1ccc2sc(NCC3CCNCC3)nc2c1>CN(C(C)=O)C.O>Fc1ccc(OCCCN2CCC(CNc3nc4ccccc4s3)CC2)c(OCc2ccccc2)c1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-e5b173451e7142968c31ab748f8e6b09
CC(=O)N(C)C.COc1cc2nc(NCC3CCNCC3)sc2c(OC)c1OC.CS(=O)(=O)OCC1COc2ccccc2O1.O=C([O-])[O-]>>COc1cc2nc(NCC3CCN(CC4COc5ccccc5O4)CC3)sc2c(OC)c1OC.O=C(O)/C=C/C(=O)O
CS(=O)(=O)OCC1COC2=C(O1)C=CC=C2.COC=1C(=C(C2=C(N=C(S2)NCC2CCNCC2)C1)OC)OC.C([O-])([O-])=O.[Na+].[Na+].CN(C(C)=O)C>>C(\C=C\C(=O)O)(=O)O.O1C(COC2=C1C=CC=C2)CN2CCC(CC2)CNC=2SC1=C(N2)C=C(C(=C1OC)OC)OC
CN(C)[C:40]([CH3:39])=[O:41].[CH3:1][O:2][c:3]1[cH:4][c:5]2[n:6][c:7]([NH:8][CH2:9][CH:10]3[CH2:11][CH2:12][NH:13][CH2:25][CH2:26]3)[s:27][c:28]2[c:29]([O:30][CH3:31])[c:32]1[O:33][CH3:34].O=S(=O)([CH3:38])[O:42][CH2:14][CH:15]1[CH2:16][O:17][c:18]2[cH:19][cH:20][cH:21][cH:22][c:23]2[O:24]1.[O-][C:36](=[O:35])[O-:37]>>...
CC(=O)N(C)C.COc1cc2nc(NCC3CCNCC3)sc2c(OC)c1OC.CS(=O)(=O)OCC1COc2ccccc2O1.O=C([O-])[O-]
COc1cc2nc(NCC3CCN(CC4COc5ccccc5O4)CC3)sc2c(OC)c1OC.O=C(O)/C=C/C(=O)O
null
null
O
C-C Coupling
OtherReaction
c0b9b32cc0d0e92c4a163b6990a02d376ad04552d535ae7e12787c7251090f66
fc8c326d38ab0e2894800f133c978339a31cf8467e0f147ca1c863a787660d0f
c1ccc2c(c1)OCC(CN1CCC(CNc3nc4ccccc4s3)CC1)O2
C-N(-C)-[C;H0;D3;+0:1](-[CH3;D1;+0:2])=[O;D1;H0:3].O=S(=O)(-[CH3;D1;+0:4])-[O;H0;D2;+0:5]-[CH2;D2;+0:6]-[C:7](-[#8:8]-[c:9])-[C:10]-[#8:11].[C:12]-[C:13]-[NH;D2;+0:14]-[C:15]-[C:16].[O-;H0;D1:17]-[C;H0;D3;+0:18](-[O-])=[O;D1;H0:19]>>[#8:11]-[C:10]-[C:7](-[CH2;D2;+0:6]-[N;H0;D3;+0:14](-[C:13]-[C:12])-[C:15]-[C:16])-[#8:...
48.5
[{"value": 48.5, "product": "C(\\C=C\\C(=O)O)(=O)O.O1C(COC2=C1C=CC=C2)CN2CCC(CC2)CNC=2SC1=C(N2)C=C(C(=C1OC)OC)OC", "details": "PERCENTYIELD", "is_desired": false}]
75
CELSIUS
8
HOUR
A mixture of 2.8 parts of 2,3-dihydro-1,4-benzodioxin-2-methanol methanesulfonate (ester), 3.4 parts of 5,6,7-trimethoxy-N-(4-piperidinylmethyl)-2-benzothiazolamine, 3 parts of sodium carbonate and 67.5 parts of N,N-dimethylacetamide was stirred overnight at about 75° C. Water was added. The product was extracted with ...
10.6084/m9.figshare.5104873.v1
null
Mesylate.Tertiary amide.Secondary amine
Carboxylic acid.Carboxylic acid.Tertiary amine
C1CCNCC1
C1CC[NH]CC1
c1ccc2scnc2c1.C1CC[NH]CC1.c1ccc2c(c1)OCCO2
MsOH.HO-
O
75
8
CC(=O)N(C)C.COc1cc2nc(NCC3CCNCC3)sc2c(OC)c1OC.CS(=O)(=O)OCC1COc2ccccc2O1.O=C([O-])[O-]>O>COc1cc2nc(NCC3CCN(CC4COc5ccccc5O4)CC3)sc2c(OC)c1OC.O=C(O)/C=C/C(=O)O
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-0701af8e90954ddcb99b613811caad29
CS(=O)(=O)c1nc2cnccc2s1.NCC1CCN(CC2COc3ccccc3O2)CC1>>c1ccc2c(c1)OCC(CN1CCC(CNc3nc4cnccc4s3)CC1)O2
Br.Br.O1C(COC2=C1C=CC=C2)CN2CCC(CC2)CN.CS(=O)(=O)C=1SC2=C(C=NC=C2)N1.C([O-])([O-])=O.[Na+].[Na+]>>O1C(COC2=C1C=CC=C2)CN2CCC(CC2)CNC=2SC1=C(C=NC=C1)N2
CS(=O)(=O)[c:17]1[n:18][c:19]2[cH:20][n:21][cH:22][cH:23][c:24]2[s:25]1.[cH:1]1[cH:2][cH:3][c:4]2[c:5]([cH:6]1)[O:7][CH2:8][CH:9]([CH2:10][N:11]1[CH2:12][CH2:13][CH:14]([CH2:15][NH2:16])[CH2:26][CH2:27]1)[O:28]2>>[cH:1]1[cH:2][cH:3][c:4]2[c:5]([cH:6]1)[O:7][CH2:8][CH:9]([CH2:10][N:11]1[CH2:12][CH2:13][CH:14]([CH2:15][N...
CS(=O)(=O)c1nc2cnccc2s1.NCC1CCN(CC2COc3ccccc3O2)CC1
c1ccc2c(c1)OCC(CN1CCC(CNc3nc4cnccc4s3)CC1)O2
null
null
CN(C(C)=O)C
Heteroatom Alkylation and Arylation
OtherReaction
66df03e7c79caa9950bf46712c3292329d3797faeace235d09531e13fa57c7e8
f263fb011eaf2f85af25e2af9b0908fb2797226f3495a5d6be9230bf229d4fae
c1ccc2c(c1)OCC(CN1CCC(CNc3nc4cnccc4s3)CC1)O2
C-S(=O)(=O)-[c;H0;D3;+0:1]1:[#16;a:2]:[c:3]:[c:4](:[#7;a:5]:1):[c:6]:[#7;a:7].[C:8]-[C:9]-[NH2;D1;+0:10]>>[#7;a:7]:[c:6]:[c:4]1:[#7;a:5]:[c;H0;D3;+0:1](-[NH;D2;+0:10]-[C:9]-[C:8]):[#16;a:2]:[c:3]:1
20
[{"value": 20.0, "product": "O1C(COC2=C1C=CC=C2)CN2CCC(CC2)CNC=2SC1=C(C=NC=C1)N2", "details": "PERCENTYIELD", "is_desired": false}]
150
CELSIUS
2
HOUR
A mixture of 6.7 parts of 1-[(2,3-dihydro-1,4-benzodioxin-2-yl)methyl]-4-piperidinemethanamine dihydrobromide, 3.26 parts of 2-(methylsulfonyl)thiazolo[4,5-c]pyridine, 4.25 parts of sodium carbonate and 18 parts of N,N-dimethylacetamide was stirred for 2 hours at 150° C. The reaction mixture was poured into ice water. ...
10.6084/m9.figshare.5104873.v1
null
Primary amine.Sulfone
Secondary amine
c1cc2scnc2cn1
c1cc2scnc2cn1
c1ccc2c(c1)OCCO2.C1CC[NH]CC1.c1cc2scnc2cn1
HO-
CN(C(C)=O)C
150
2
CS(=O)(=O)c1nc2cnccc2s1.NCC1CCN(CC2COc3ccccc3O2)CC1>CN(C(C)=O)C>c1ccc2c(c1)OCC(CN1CCC(CNc3nc4cnccc4s3)CC1)O2
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-45b8253e9c01479cbece5ecd18a962aa
CC(=O)N(C)C.CC(N)C1CCN(CC2COc3ccccc3O2)CC1.Clc1nc2ccccc2s1.[O-2]>>CC(Nc1nc2ccccc2s1)C1CCN(CC2COc3ccccc3O2)CC1.O=C(O)C(=O)O
O1C(COC2=C1C=CC=C2)CN2CCC(CC2)C(N)C.ClC=1SC2=C(N1)C=CC=C2.[O-2].[Ca+2].CN(C(C)=O)C>>C(C(=O)O)(=O)O.O1C(COC2=C1C=CC=C2)CN2CCC(CC2)C(C)NC=2SC1=C(N2)C=CC=C1
CN(C)[C:33]([CH3:31])=[O:34].[CH3:1][CH:2]([NH2:3])[CH:13]1[CH2:14][CH2:15][N:16]([CH2:17][CH:18]2[CH2:19][O:20][c:21]3[cH:22][cH:23][cH:24][cH:25][c:26]3[O:27]2)[CH2:28][CH2:29]1.Cl[c:4]1[n:5][c:6]2[cH:7][cH:8][cH:9][cH:10][c:11]2[s:12]1.[O-2:30]>>[CH3:1][CH:2]([NH:3][c:4]1[n:5][c:6]2[cH:7][cH:8][cH:9][cH:10][c:11]2[s...
CC(=O)N(C)C.CC(N)C1CCN(CC2COc3ccccc3O2)CC1.Clc1nc2ccccc2s1.[O-2]
CC(Nc1nc2ccccc2s1)C1CCN(CC2COc3ccccc3O2)CC1.O=C(O)C(=O)O
null
null
null
Acylation
OtherReaction
0c8075d2d1fe29c7f41c41bf76a14390f86cda55b48fbbc231d49ce5c010f6d7
ea2fa6358c9b24db3f2c985013e3a1847fb8d9c8a280d7bd27f4a04a4b83c055
c1ccc2c(c1)OCC(CN1CCC(CNc3nc4ccccc4s3)CC1)O2
C-N(-C)-[C;H0;D3;+0:1](-[CH3;D1;+0:2])=[O;D1;H0:3].Cl-[c;H0;D3;+0:4]1:[#16;a:5]:[c:6]:[c:7]:[#7;a:8]:1.[C:9]-[C:10](-[C;D1;H3:11])-[NH2;D1;+0:12].[O-2;H0;D0:13]>>[C:9]-[C:10](-[C;D1;H3:11])-[NH;D2;+0:12]-[c;H0;D3;+0:4]1:[#16;a:5]:[c:6]:[c:7]:[#7;a:8]:1.[O;D1;H0:3]=[C;H0;D3;+0:1](-[O;D1;H1:14])-[C;H0;D3;+0:2](-[O;D1;H1:...
39.7
[{"value": 39.7, "product": "C(C(=O)O)(=O)O.O1C(COC2=C1C=CC=C2)CN2CCC(CC2)C(C)NC=2SC1=C(N2)C=CC=C1", "details": "PERCENTYIELD", "is_desired": false}]
140
CELSIUS
4
HOUR
A mixture of 4 parts of 1-[(2,3-dihydro-1,4-benzodioxin-2-yl)methyl]-α-methyl-4-piperidinemethanamine, 2.7 parts of 2-chlorobenzothiazole, 1.5 parts of calcium oxide and 18 parts of N,N-dimethylacetamide was stirred for 4 hours at 140° C. The whole was filtered and to the filtrate was added 4-methyl-2-pentanone. The wh...
10.6084/m9.figshare.5104873.v1
null
Aromatic halide.Tertiary amide.Primary amine
Carboxylic acid.Carboxylic acid.Secondary amine
c1ccc2scnc2c1
c1ccc2scnc2c1
c1ccc2scnc2c1.C1CC[NH]CC1.c1ccc2c(c1)OCCO2
HCl
null
140
4
CC(=O)N(C)C.CC(N)C1CCN(CC2COc3ccccc3O2)CC1.Clc1nc2ccccc2s1.[O-2]>>CC(Nc1nc2ccccc2s1)C1CCN(CC2COc3ccccc3O2)CC1.O=C(O)C(=O)O
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-8448f9365305453fbaf740a187d7bdeb
CI.c1ccc2c(c1)OCC(CN1CCC(CNc3nc4ccccc4s3)CC1)O2>>CN(CC1CCN(CC2COc3ccccc3O2)CC1)c1nc2ccccc2s1
IC.CN(C=O)C.O1C(COC2=C1C=CC=C2)CN2CCC(CC2)CNC=2SC1=C(N2)C=CC=C1.CN(C=O)C.[H-].[Na+]>>O1C(COC2=C1C=CC=C2)CN2CCC(CC2)CN(C=2SC1=C(N2)C=CC=C1)C
I[CH3:1].[NH:2]([CH2:3][CH:4]1[CH2:5][CH2:6][N:7]([CH2:8][CH:9]2[CH2:10][O:11][c:12]3[cH:13][cH:14][cH:15][cH:16][c:17]3[O:18]2)[CH2:19][CH2:20]1)[c:21]1[n:22][c:23]2[cH:24][cH:25][cH:26][cH:27][c:28]2[s:29]1>>[CH3:1][N:2]([CH2:3][CH:4]1[CH2:5][CH2:6][N:7]([CH2:8][CH:9]2[CH2:10][O:11][c:12]3[cH:13][cH:14][cH:15][cH:16]...
CI.c1ccc2c(c1)OCC(CN1CCC(CNc3nc4ccccc4s3)CC1)O2
CN(CC1CCN(CC2COc3ccccc3O2)CC1)c1nc2ccccc2s1
null
null
O
Heteroatom Alkylation and Arylation
N-alkylation of secondary amines with alkyl halides
e1587a52a1bca6a80c6048d43276d8bccf8d3e94e692e6b210e5fd3b22494187
7cc25fba33369069673bac5bd8fc404dc064da8d6c8cf4a77f21f4df0a617fe3
c1ccc2c(c1)OCC(CN1CCC(CNc3nc4ccccc4s3)CC1)O2
I-[CH3;D1;+0:1].[C:2]-[C:3]-[NH;D2;+0:4]-[c:5]1:[#16;a:6]:[c:7]:[c:8]:[#7;a:9]:1>>[C:2]-[C:3]-[N;H0;D3;+0:4](-[CH3;D1;+0:1])-[c:5]1:[#16;a:6]:[c:7]:[c:8]:[#7;a:9]:1
null
[]
null
null
30
MINUTE
To a stirred solution of 11.85 parts of N-[1-[(2,3-dihydro-1,4-benzodioxin-2-yl)methyl]-4-piperidinylmethyl]-2-benzothiazolamine in 72 parts of N,N-dimethylformamide were added portionwise 1.5 parts of a sodium hydride dispersion 50%. Upon completion, stirring was continued for 30 minutes. A solution of 4.6 parts of io...
10.6084/m9.figshare.5104873.v1
null
Secondary amine
Tertiary amine
null
null
C1CC[NH]CC1.c1ccc2c(c1)OCCO2.c1ccc2scnc2c1
HI
O
null
0.5
CI.c1ccc2c(c1)OCC(CN1CCC(CNc3nc4ccccc4s3)CC1)O2>O>CN(CC1CCN(CC2COc3ccccc3O2)CC1)c1nc2ccccc2s1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-3c011460876e45b6b5bb44988893edcf
O=C(O)c1ccco1.c1ccc2c(c1)OCC(CN1CCC(CNc3nc4ccccc4s3)CC1)O2>>Cl.O=C(c1ccco1)N(CC1CCN(CC2COc3ccccc3O2)CC1)c1nc2ccccc2s1
O1C(=CC=C1)C(=O)O.C(C)N(CC)CC.O1C(COC2=C1C=CC=C2)CN2CCC(CC2)CNC=2SC1=C(N2)C=CC=C1.[I-].ClC1=[N+](C=CC=C1)C>>Cl.S1C(=NC2=C1C=CC=C2)N(C(=O)C=2OC=CC2)CC2CCN(CC2)CC2COC1=C(O2)C=CC=C1
O[C:3](=[O:2])[c:4]1[cH:5][cH:6][cH:7][o:8]1.[NH:9]([CH2:10][CH:11]1[CH2:12][CH2:13][N:14]([CH2:15][CH:16]2[CH2:17][O:18][c:19]3[cH:20][cH:21][cH:22][cH:23][c:24]3[O:25]2)[CH2:26][CH2:27]1)[c:28]1[n:29][c:30]2[cH:31][cH:32][cH:33][cH:34][c:35]2[s:36]1>>[ClH:1].[O:2]=[C:3]([c:4]1[cH:5][cH:6][cH:7][o:8]1)[N:9]([CH2:10][C...
O=C(O)c1ccco1.c1ccc2c(c1)OCC(CN1CCC(CNc3nc4ccccc4s3)CC1)O2
Cl.O=C(c1ccco1)N(CC1CCN(CC2COc3ccccc3O2)CC1)c1nc2ccccc2s1
null
null
ClCCl.O.O1CCCC1
Acylation
Acylation of Nitrogen Nucleophiles by Carboxylic Acids
ac72df6259d5d7baee7abdbd4706ef4b4627f86ead9dc94f0cefcfcb37c21def
c5e4172490b2731ba9322b68af56376edadc31ce0bb9a3dfdea23a1817a852fd
O=C(c1ccco1)N(CC1CCN(CC2COc3ccccc3O2)CC1)c1nc2ccccc2s1
O-[C;H0;D3;+0:1](=[O;D1;H0:2])-[c:3](:[c:4]):[#8;a:5]:[c:6].[C:7]-[C:8]-[NH;D2;+0:9]-[c:10]1:[#16;a:11]:[c:12]:[c:13]:[#7;a:14]:1>>[C:7]-[C:8]-[N;H0;D3;+0:9](-[C;H0;D3;+0:1](=[O;D1;H0:2])-[c:3](:[c:4]):[#8;a:5]:[c:6])-[c:10]1:[#16;a:11]:[c:12]:[c:13]:[#7;a:14]:1
41.8
[{"value": 41.8, "product": "Cl.S1C(=NC2=C1C=CC=C2)N(C(=O)C=2OC=CC2)CC2CCN(CC2)CC2COC1=C(O2)C=CC=C1", "details": "PERCENTYIELD", "is_desired": false}]
null
null
30
MINUTE
To a stirred mixture of 1.12 parts of 2-furancarboxylic acid, 2.02 parts of N,N-diethylethanamine and 195 parts of dichloromethane were added 2.55 parts of 2-chloro-1-methylpyridinium iodide. Stirring was continued for 30 minutes at room temperature. A solution of 3.93 parts of N-[1-[(2,3-dihydro-1,4-benzodioxin-2-yl)m...
10.6084/m9.figshare.5104873.v1
null
Carboxylic acid.Secondary amine
Tertiary amide
null
null
c1ccoc1.C1CC[NH]CC1.c1ccc2c(c1)OCCO2.c1ccc2scnc2c1
null
ClCCl.O.O1CCCC1
null
0.5
O=C(O)c1ccco1.c1ccc2c(c1)OCC(CN1CCC(CNc3nc4ccccc4s3)CC1)O2>ClCCl.O.O1CCCC1>Cl.O=C(c1ccco1)N(CC1CCN(CC2COc3ccccc3O2)CC1)c1nc2ccccc2s1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-d2176593c0e7446f81b8b594876307c6
COc1ccc(NC(=S)NCC2CCN(CC3COc4ccccc4O3)CC2)cc1>>COc1ccc2nc(NCC3CCN(CC4COc5ccccc5O4)CC3)sc2c1
[OH-].[Na+].O1C(COC2=C1C=CC=C2)CN2CCC(CC2)CNC(=S)NC2=CC=C(C=C2)OC.ClC(Cl)Cl.BrBr>>O1C(COC2=C1C=CC=C2)CN2CCC(CC2)CNC=2SC1=C(N2)C=CC(=C1)OC
[CH3:1][O:2][c:3]1[cH:4][cH:5][c:6]([NH:7][C:8]([NH:9][CH2:10][CH:11]2[CH2:12][CH2:13][N:14]([CH2:15][CH:16]3[CH2:17][O:18][c:19]4[cH:20][cH:21][cH:22][cH:23][c:24]4[O:25]3)[CH2:26][CH2:27]2)=[S:28])[cH:29][cH:30]1>>[CH3:1][O:2][c:3]1[cH:4][cH:5][c:6]2[n:7][c:8]([NH:9][CH2:10][CH:11]3[CH2:12][CH2:13][N:14]([CH2:15][CH:...
COc1ccc(NC(=S)NCC2CCN(CC3COc4ccccc4O3)CC2)cc1
COc1ccc2nc(NCC3CCN(CC4COc5ccccc5O4)CC3)sc2c1
null
null
ClC(Cl)(Cl)Cl
Aromatic Heterocycle Formation
OtherReaction
9fc354848fb2fb52ac9a677ec08efbe70faac27defb4ee4a070dc3814d93a73c
01ff041a21adca51a94f69a62115e81e604cce12edd47d529ec3eedb88c39f4c
c1ccc2c(c1)OCC(CN1CCC(CNc3nc4ccccc4s3)CC1)O2
[C:1]-[#7:2]-[C;H0;D3;+0:3](=[S;H0;D1;+0:4])-[NH;D2;+0:5]-[c:6](:[c:7]):[cH;D2;+0:8]:[c:9]:[c:10]>>[C:1]-[#7:2]-[c;H0;D3;+0:3]1:[n;H0;D2;+0:5]:[c:6](:[c:7]):[c;H0;D3;+0:8](:[c:9]:[c:10]):[s;H0;D2;+0:4]:1
21
[{"value": 21.0, "product": "O1C(COC2=C1C=CC=C2)CN2CCC(CC2)CNC=2SC1=C(N2)C=CC(=C1)OC", "details": "PERCENTYIELD", "is_desired": false}]
null
null
null
null
To a stirred mixture of 8.3 parts of N-[[1-[(2,3-dihydro-1,4-benzodioxin-2-yl)methyl]-4-piperidinyl]methyl]-N'-(4-methoxyphenyl)thiourea, 60 parts of trichloromethane and 240 parts of tetrachloromethane were added at once 3.1 parts of bromine. The whole was stirred and refluxed for 1 hour. After cooling, the reaction m...
10.6084/m9.figshare.5104873.v1
null
Thiourea
null
c1ccccc1
c1ccc2scnc2c1
c1ccc2scnc2c1.C1CC[NH]CC1.c1ccc2c(c1)OCCO2
null
ClC(Cl)(Cl)Cl
null
null
COc1ccc(NC(=S)NCC2CCN(CC3COc4ccccc4O3)CC2)cc1>ClC(Cl)(Cl)Cl>COc1ccc2nc(NCC3CCN(CC4COc5ccccc5O4)CC3)sc2c1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-0786b25dde1d411a93033313798ab033
CCC(CCCCCl)OC.ClC1C=CCC1>>CCC(CCCCC1C=CCC1)OC
ClC1C=CCC1.[Cl-].[NH4+].[Mg].ClCCCCC(CC)OC>>COC(CCCCC1C=CCC1)CC
Cl[CH2:7][CH2:6][CH2:5][CH2:4][CH:3]([CH2:2][CH3:1])[O:13][CH3:14].Cl[CH:8]1[CH:9]=[CH:10][CH2:11][CH2:12]1>>[CH3:1][CH2:2][CH:3]([CH2:4][CH2:5][CH2:6][CH2:7][CH:8]1[CH:9]=[CH:10][CH2:11][CH2:12]1)[O:13][CH3:14]
CCC(CCCCCl)OC.ClC1C=CCC1
CCC(CCCCC1C=CCC1)OC
null
null
O1CCCC1
C-C Coupling
Negishi
9a6bf7e2b45e73e51c658250a4e70cb08f6a32ab7a16b4f9f48c368b31fb4ddc
d4cf29bb0f2586f258c9eb5d3edb710b86094a4be60be4638a5468606055dcb5
C1=CCCC1
Cl-[CH2;D2;+0:1]-[C:2]-[C:3].Cl-[CH;D3;+0:4]1-[C:5]-[C:6]-[C:7]=[C:8]-1>>[C:3]-[C:2]-[CH2;D2;+0:1]-[CH;D3;+0:4]1-[C:5]-[C:6]-[C:7]=[C:8]-1
null
[]
-25
CELSIUS
null
null
Magnesium metal turnings (7.2 g, 0.299 moles) are added to a three-necked, round-bottomed flask equipped with a Friedrich condenser and kept under nitrogen gas. Tetrahydrofuran (300 ml) is transferred to the flask and the contents stirred. A clear, colorless solution of 1-chloro-5-methoxyheptane (48.1 g, 0.292 moles) i...
10.6084/m9.figshare.5104873.v1
null
Secondary halide.Primary halide
null
C1=CCCC1
C1=CCCC1
C1=CCCC1
Other
O1CCCC1
-25
null
CCC(CCCCCl)OC.ClC1C=CCC1>O1CCCC1>CCC(CCCCC1C=CCC1)OC
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-c21ededa198241be8bfe0a31117ca8c5
CCC(CCCCC1C=CCC1)OC.CCCCCC.CCCCCC.CCN(CC)CC.O=C(Cl)C(Cl)Cl>>CCC(CCC(C)C12CCCC1C(=O)C2(Cl)Cl)OC.CCC(CCCCC1CCC2C(=O)C(Cl)(Cl)C12)OC.CCC(CCCCC1CCC2C1C(=O)C2(Cl)Cl)OC
ClC(C(=O)Cl)Cl.COC(CCCCC1C=CCC1)CC.CCCCCC.C(C)N(CC)CC.CCCCCC>>ClC1(C2CCC(C2C1=O)CCCCC(CC)OC)Cl.ClC1(C(C2CCCC12C(C)CCC(CC)OC)=O)Cl.ClC1(C(C2CCC(C12)CCCCC(CC)OC)=O)Cl
[CH3:39][CH2:40][CH:41]([CH2:42][CH2:43][CH2:44][CH2:45][CH:46]1[CH2:47][CH2:48][CH:49]=[CH:50]1)[O:56][CH3:57].[CH2:3]([CH2:4][CH2:5][CH2:6][CH3:7])[CH3:12].[CH3:20][CH2:21][CH2:22][CH2:23][CH2:24][CH3:25].N([CH2:2][CH3:1])([CH2:26][CH3:27])[CH2:53][CH3:51].[C:13](=[O:14])([CH:15]([Cl:16])[Cl:17])[Cl:34]>>[CH3:1][CH2:...
CCC(CCCCC1C=CCC1)OC.CCCCCC.CCCCCC.CCN(CC)CC.O=C(Cl)C(Cl)Cl
CCC(CCC(C)C12CCCC1C(=O)C2(Cl)Cl)OC.CCC(CCCCC1CCC2C(=O)C(Cl)(Cl)C12)OC.CCC(CCCCC1CCC2C1C(=O)C2(Cl)Cl)OC
null
null
null
C-C Coupling
OtherReaction
9f73c275c1d2644e37d7ac436393a1d4820702c5ea292d9ac31e9749814026ce
619721e0a1ae47aa4c59b8686b40ef843f5a95b0374e4d345c70e6b8b4761eae
O=C1CC2CCCC12.O=C1CC2CCCC12.O=C1CC2CCCC12
[C;D1;H3:1]-[CH2;D2;+0:2]-N(-[CH2;D2;+0:3]-[CH3;D1;+0:4])-[CH2;D2;+0:5]-[CH3;D1;+0:6].[C;D1;H3:7]-[CH2;D2;+0:8]-[C:9]-[C:10]-[CH2;D2;+0:11]-[CH3;D1;+0:12].[C;D1;H3:13]-[C:14]-[CH2;D2;+0:15]-[C:16]-[C:17]-[CH3;D1;+0:18].[C:19]-[C:20]1-[C:21]-[C:22]-[CH;D2;+0:23]=[CH;D2;+0:24]-1.[Cl;D1;H0:25]-[CH;D3;+0:26](-[Cl;D1;H0:27]...
null
[]
null
null
null
null
To a 1,000 ml three-necked, round-bottomed flask, equipped with a reflux condenser containing 3-(5-methoxyhept-1-yl)cyclopentene {3-(5-methoxyheptyl)cyclopentene} (15.0 g, 0.076 moles) in 300 ml of hexane, freshly distilled dichloroacetyl chloride (35.1 g, 0.240 moles) is added and the solution is stirred by a mechanic...
10.6084/m9.figshare.5104873.v1
null
Acyl halide.Secondary halide.Secondary halide.Tertiary amine
Tertiary halide.Tertiary halide.Tertiary halide.Tertiary halide.Tertiary halide.Tertiary halide.Ketone.Ketone.Ketone.Ether.Ether
C1=CCCC1
C1CC2CCC2C1.C1CC2CCC2C1.C1CC2CCC2C1
C1CC2CCC2C1.C1CC2CCC2C1.C1CC2CCC2C1
null
null
null
null
CCC(CCCCC1C=CCC1)OC.CCCCCC.CCCCCC.CCN(CC)CC.O=C(Cl)C(Cl)Cl>>CCC(CCC(C)C12CCCC1C(=O)C2(Cl)Cl)OC.CCC(CCCCC1CCC2C(=O)C(Cl)(Cl)C12)OC.CCC(CCCCC1CCC2C1C(=O)C2(Cl)Cl)OC
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-f0be817ce3d042319adc6ba51ba5d29c
CCC(O)CCCC(=O)O.CCOC(OCC)OCC>>CCOC(=O)CCCC(CC)OCC
OC(CCCC(=O)O)CC.C(C)C1CCCC(O1)=O.[OH-].[Na+].Cl(=O)(=O)(=O)O.S(O)(O)(=O)=O.C(C)OC(OCC)OCC.C(C)OC(OCC)OCC>>C(C)OC(CCCC(=O)OCC)CC
[OH:3][C:4](=[O:5])[CH2:6][CH2:7][CH2:8][CH:9]([CH2:10][CH3:11])[OH:12].CCOC(O[CH2:2][CH3:1])O[CH2:13][CH3:14]>>[CH3:1][CH2:2][O:3][C:4](=[O:5])[CH2:6][CH2:7][CH2:8][CH:9]([CH2:10][CH3:11])[O:12][CH2:13][CH3:14]
CCC(O)CCCC(=O)O.CCOC(OCC)OCC
CCOC(=O)CCCC(CC)OCC
null
null
C(C)O
Heteroatom Alkylation and Arylation
OtherReaction
a367edd36e7a6d4fc8bcf7d6eeb3291b269bea15b3edbb95c515f2124c66dff5
bcb571b9242e6612bdc8f209381b773bf471f4584cc3238291f772a3f2b72931
null
C-C-O-C(-O-[CH2;D2;+0:1]-[C;D1;H3:2])-O-[CH2;D2;+0:3]-[C;D1;H3:4].[C:5]-[C:6](-[C:7])-[OH;D1;+0:8].[C:9]-[C:10](=[O;D1;H0:11])-[OH;D1;+0:12]>>[C:5]-[C:6](-[C:7])-[O;H0;D2;+0:8]-[CH2;D2;+0:1]-[C;D1;H3:2].[C:9]-[C:10](=[O;D1;H0:11])-[O;H0;D2;+0:12]-[CH2;D2;+0:3]-[C;D1;H3:4]
null
[]
null
null
4
HOUR
A mixture of 400 g 5-hydroxyheptanoic acid and 6-ethyltetrahydro-2H-pyran-2-one (400 g) is added to the reaction vessel containing ethanol (4000 ml) and triethylorthoformate (4000 ml). Perchloric acid (160 ml) is slowly added. The mixture is stirred at room temperature for 4 hours, after which time sodium hydroxide pel...
10.6084/m9.figshare.5104873.v1
null
Carboxylic acid.Ether.Ether.Ether.Secondary alcohol
Ester.Ether
null
null
null
HO-
C(C)O
null
4
CCC(O)CCCC(=O)O.CCOC(OCC)OCC>C(C)O>CCOC(=O)CCCC(CC)OCC
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-4e55915b9af54cf3b59fbf584e4c51f2
CCOC(=O)CCCC(CC)OCC>>CCOC(CC)CCCCO
C(C)OC(CCCC(=O)OCC)CC.[H-].[Al+3].[Li+].[H-].[H-].[H-]>>C(C)OC(CCCCO)CC
CCO[C:10]([CH2:9][CH2:8][CH2:7][CH:4]([O:3][CH2:2][CH3:1])[CH2:5][CH3:6])=[O:11]>>[CH3:1][CH2:2][O:3][CH:4]([CH2:5][CH3:6])[CH2:7][CH2:8][CH2:9][CH2:10][OH:11]
CCOC(=O)CCCC(CC)OCC
CCOC(CC)CCCCO
null
null
O1CCCC1
Reduction
Reduction of ester to primary alcohol
21d61543c6ec8a8cebe1b3ef55ef3dd20acbf79a4f1c12a7fb51e32be7a3248a
1fbcd628a0426673c5d10aa49a977cd2d1ae02a8cdf57bbb10d94aa03a94e937
null
C-C-O-[C;H0;D3;+0:1](=[O;H0;D1;+0:2])-[C:3]-[C:4]>>[C:4]-[C:3]-[CH2;D2;+0:1]-[OH;D1;+0:2]
null
[]
-60
CELSIUS
null
null
A solution of tetrahydrofuran (2000 ml) containing lithium aluminum hydride (46 g, 1.21 moles) is cooled in a -60° C. dry ice/ethanol bath. Ethyl 5-ethoxyheptanoate (302 g, 1.49 moles) is diluted in tetrahydrofuran (300 ml) and added dropwise to the stirring reaction. After the addition is complete the reaction is warm...
10.6084/m9.figshare.5104873.v1
null
Ester
Primary alcohol
null
null
null
HO-
O1CCCC1
-60
null
CCOC(=O)CCCC(CC)OCC>O1CCCC1>CCOC(CC)CCCCO
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-848bac7c24cc4261bb2073abefd468c5
CCOC(CC)CCCCO.O=S(Cl)Cl>>CCOC(CC)CCCCCl
C(C)OC(CCCCO)CC.N1=CC=CC=C1.S(=O)(Cl)Cl>>ClCCCCC(CC)OCC
O[CH2:10][CH2:9][CH2:8][CH2:7][CH:4]([O:3][CH2:2][CH3:1])[CH2:5][CH3:6].O=S(Cl)[Cl:11]>>[CH3:1][CH2:2][O:3][CH:4]([CH2:5][CH3:6])[CH2:7][CH2:8][CH2:9][CH2:10][Cl:11]
CCOC(CC)CCCCO.O=S(Cl)Cl
CCOC(CC)CCCCCl
null
null
O
Functional Group Interconversion
Alcohol to chloride_SOCl2
bb752b9027dc4488ba075e5955118a819f80cabd751a7497b67c2eeb1db6b071
cbf41c7cf9fe6b47a243b1674d74ed5bf46a151f7f3a71d206e23176e158facf
null
Cl-S(=O)-[Cl;H0;D1;+0:1].O-[CH2;D2;+0:2]-[C:3]-[C:4]>>[C:4]-[C:3]-[CH2;D2;+0:2]-[Cl;H0;D1;+0:1]
75.8
[{"value": 75.8, "product": "ClCCCCC(CC)OCC", "details": "CALCULATEDPERCENTYIELD", "is_desired": false}]
null
null
null
null
5-Ethoxyheptanol (238 g, 1.49 moles) is diluted in pyridine (128 g, 1.62 moles). The solution is stirred at room temperature and thionyl chloride (388 g, 3.22 moles) is added dropwise over 2 hours. After this time the mixture is heated in a 70° C. water bath for 2 additional hours. Water (700 ml) is added to the reacti...
10.6084/m9.figshare.5104873.v1
null
Primary alcohol
Primary halide
null
null
null
HCl
O
null
null
CCOC(CC)CCCCO.O=S(Cl)Cl>O>CCOC(CC)CCCCCl
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-40763d3e96f8401aa86089cd7aca46a8
CCCCCCCBr.ClC1C=CCC1>>CCCCCCCC1C=CCC1
[Mg].ClC1C=CCC1.BrCCCCCCC>>C(CCCCCC)C1C=CCC1
Br[CH2:7][CH2:6][CH2:5][CH2:4][CH2:3][CH2:2][CH3:1].Cl[CH:8]1[CH:9]=[CH:10][CH2:11][CH2:12]1>>[CH3:1][CH2:2][CH2:3][CH2:4][CH2:5][CH2:6][CH2:7][CH:8]1[CH:9]=[CH:10][CH2:11][CH2:12]1
CCCCCCCBr.ClC1C=CCC1
CCCCCCCC1C=CCC1
null
null
O1CCCC1
C-C Coupling
Negishi
9a6bf7e2b45e73e51c658250a4e70cb08f6a32ab7a16b4f9f48c368b31fb4ddc
d4cf29bb0f2586f258c9eb5d3edb710b86094a4be60be4638a5468606055dcb5
C1=CCCC1
Br-[CH2;D2;+0:1]-[C:2]-[C:3].Cl-[CH;D3;+0:4]1-[C:5]-[C:6]-[C:7]=[C:8]-1>>[C:3]-[C:2]-[CH2;D2;+0:1]-[CH;D3;+0:4]1-[C:5]-[C:6]-[C:7]=[C:8]-1
51.8
[{"value": 51.8, "product": "C(CCCCCC)C1C=CCC1", "details": "CALCULATEDPERCENTYIELD", "is_desired": false}]
null
null
null
null
The procedure followed is the same as that described in Example 20 substituting 1-bromoheptane (100 g, 0.56 moles) diluted in tetrahydrofuran (100 ml), granular magnesium (25 g) in tetrahydrofuran (100 ml), 0.1 M solution of Li2CuCl4 (1.7 mmoles), and 3-chlorocyclopentene (57 g, 0.56 moles) diluted in tetrahydrofuran (...
10.6084/m9.figshare.5104873.v1
null
Secondary halide.Primary halide
null
C1=CCCC1
C1=CCCC1
C1=CCCC1
Br-
O1CCCC1
null
null
CCCCCCCBr.ClC1C=CCC1>O1CCCC1>CCCCCCCC1C=CCC1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-829aaf2fa95e4efd9138f91fff56f06b
CC(C)(C)[Si](C)(C)Cl.CCC(O)CCCl>>CCC(CCCl)O[Si](C)(C)CC(C)C
CN(C=O)C.ClCCC(CC)O.[Si](C)(C)(C(C)(C)C)Cl.N1C=NC=C1>>ClCCC(CC)O[Si](C)(C)CC(C)C
Cl[Si:8]([CH3:9])([CH3:10])[C:12]([CH3:11])([CH3:13])[CH3:14].[CH3:1][CH2:2][CH:3]([CH2:4][CH2:5][Cl:6])[OH:7]>>[CH3:1][CH2:2][CH:3]([CH2:4][CH2:5][Cl:6])[O:7][Si:8]([CH3:9])([CH3:10])[CH2:11][CH:12]([CH3:13])[CH3:14]
CC(C)(C)[Si](C)(C)Cl.CCC(O)CCCl
CCC(CCCl)O[Si](C)(C)CC(C)C
null
null
null
Protection
OtherReaction
ea139b3cb6171a748fbc881d815cc598a14c6b8245b87168b4a15a10e325f24c
1e2a25dd539d267852f3b05b92dd4080ece1d4c7abb9db1b6fd2b64d2b33a864
null
Cl-[Si;H0;D4;+0:1](-[C;D1;H3:2])(-[C;D1;H3:3])-[C;H0;D4;+0:4](-[C;D1;H3:5])(-[C;D1;H3:6])-[CH3;D1;+0:7].[C:8]-[C:9](-[C:10])-[OH;D1;+0:11]>>[C:8]-[C:9](-[C:10])-[O;H0;D2;+0:11]-[Si;H0;D4;+0:1](-[C;D1;H3:2])(-[C;D1;H3:3])-[CH2;D2;+0:7]-[CH;D3;+0:4](-[C;D1;H3:5])-[C;D1;H3:6]
null
[]
null
null
null
null
The procedure followed is the same as that described in Example 19 substituting 5-chloropentan-3-ol (1-chloro-3-pentanol) (50 g, 0.41 moles), tert-butyldimethylsilyl chloride (71 g, 0.47 moles), imidazole (32.6 g, 0.48 moles), and dimethylformamide (150 ml). The crude product is fractionally distilled under vacuum leav...
10.6084/m9.figshare.5104873.v1
null
Secondary alcohol.Silyl protective group
Silyl protective group
null
null
null
HCl
null
null
null
CC(C)(C)[Si](C)(C)Cl.CCC(O)CCCl>>CCC(CCCl)O[Si](C)(C)CC(C)C
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-12c3c2d8e2cb4fb682b0b5844f5c681d
CCC(CCCl)O[Si](C)(C)C(C)(C)C.CCC(CCCl)O[Si](C)(C)CC(C)C.ClC1C=CCC1>>CCC(CCC1C=CCC1)O[Si](C)(C)C(C)(C)C.CCC(CCC1C=CCC1)O[Si](C)(C)C(C)(C)C
[Mg].ClC1C=CCC1.ClCCC(O[Si](C)(C)C(C)(C)C)CC.ClCCC(CC)O[Si](C)(C)CC(C)C>>C1(C=CCC1)CCC(O[Si](C)(C)C(C)(C)C)CC.CC(C)(C)[Si](OC(CCC1C=CCC1)CC)(C)C
Cl[CH2:5][CH2:4][CH:3]([CH2:2][CH3:1])[O:11][Si:12]([CH3:13])([CH3:14])[C:15]([CH3:16])([CH3:18])[CH3:36].Cl[CH2:23][CH2:22][CH:21]([CH2:20][CH3:19])[O:29][Si:30]([CH3:17])([CH3:28])[CH2:33][CH:35]([CH3:26])[CH3:27].Cl[CH:6]1[CH:7]=[CH:8][CH2:9][CH2:10]1>>[CH3:1][CH2:2][CH:3]([CH2:4][CH2:5][CH:6]1[CH:7]=[CH:8][CH2:9][C...
CCC(CCCl)O[Si](C)(C)C(C)(C)C.CCC(CCCl)O[Si](C)(C)CC(C)C.ClC1C=CCC1
CCC(CCC1C=CCC1)O[Si](C)(C)C(C)(C)C.CCC(CCC1C=CCC1)O[Si](C)(C)C(C)(C)C
null
null
O1CCCC1
Functional Group Addition
OtherReaction
f7fbeb208eeb150a59a3d1aaf4d167c0f98de0c3a124ab5c5e2cdd448e417190
0dd17fb8382e7be43ae3d3a371180bc22450eab508f050be2cb0fdda2faeb419
C1=CCCC1.C1=CCCC1
Cl-[CH2;D2;+0:1]-[C:2]-[C:3]-[#8:4]-[#14:5](-[C;D1;H3:6])(-[C;D1;H3:7])-[C;H0;D4;+0:8](-[C;D1;H3:9])(-[C;D1;H3:10])-[CH3;D1;+0:11].Cl-[CH2;D2;+0:12]-[C:13]-[C:14]-[#8:15]-[Si;H0;D4;+0:16](-[CH3;D1;+0:17])(-[CH3;D1;+0:18])-[CH2;D2;+0:19]-[CH;D3;+0:20](-[CH3;D1;+0:21])-[CH3;D1;+0:22].Cl-[CH;D3;+0:23]1-[C:24]-[C:25]-[C:26...
null
[]
null
null
null
null
The procedure followed is the same as that described in Example 20 substituting (5-chloro-3-pentyloxy)(2,2-dimethylethyl)dimethylsilane {3-chloro-1-ethylpropoxy)(1,1-dimethylethyl) dimethylsilane,} (78 g, 0.33 moles) diluted in tetrahydrofuran (100 ml), granular magnesium (24 g, 1.00 moles) in tetrahydrofuran (100 ml),...
10.6084/m9.figshare.5104873.v1
null
Secondary halide.Primary halide.Primary halide.TMS ether protective group.Silyl protective group
TMS ether protective group.TMS ether protective group
C1=CCCC1
C1=CCCC1.C1=CCCC1
C1=CCCC1.C1=CCCC1
null
O1CCCC1
null
null
CCC(CCCl)O[Si](C)(C)C(C)(C)C.CCC(CCCl)O[Si](C)(C)CC(C)C.ClC1C=CCC1>O1CCCC1>CCC(CCC1C=CCC1)O[Si](C)(C)C(C)(C)C.CCC(CCC1C=CCC1)O[Si](C)(C)C(C)(C)C
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-70d1a100986c414c97318dea1fbc40ac
CC(C)(C)[Si](C)(C)Cl.CN(C)C=O.OCCCCCCl.c1c[nH]cn1>>CC(C)(C)[Si](C)(C)OCCCCCCl.CC(C)C[Si](C)(C)OCCCCCCl
N1C=NC=C1.ClCCCCCO.[Si](C)(C)(C(C)(C)C)Cl.CN(C=O)C>>ClCCCCCO[Si](C)(C)C(C)(C)C.ClCCCCCO[Si](C)(C)CC(C)C
[CH3:1][C:2]([CH3:3])([Si:5]([CH3:6])([CH3:7])[Cl:28])[CH3:17].N([CH3:4])([CH:23]=[O:22])[CH3:26].[OH:8][CH2:9][CH2:10][CH2:11][CH2:12][CH2:13][Cl:14].n1[cH:24][cH:25][nH][cH:27]1>>[CH3:1][C:2]([CH3:3])([CH3:4])[Si:5]([CH3:6])([CH3:7])[O:8][CH2:9][CH2:10][CH2:11][CH2:12][CH2:13][Cl:14].[CH3:15][CH:16]([CH3:17])[CH2:18]...
CC(C)(C)[Si](C)(C)Cl.CN(C)C=O.OCCCCCCl.c1c[nH]cn1
CC(C)(C)[Si](C)(C)OCCCCCCl.CC(C)C[Si](C)(C)OCCCCCCl
null
null
O
C-C Coupling
OtherReaction
362b97bd308e1674d119f00f7193eb661001ec8b391ea68feb0fdd105b74f0a6
41459d5f85371d21209ad2e99e4133e1a13552dd3bfaa7e9511c73964195a9b6
null
[C;D1;H3:1]-[C;H0;D4;+0:2](-[C;D1;H3:3])(-[CH3;D1;+0:4])-[Si;H0;D4;+0:5](-[C;D1;H3:6])(-[C;D1;H3:7])-[Cl;H0;D1;+0:8].[CH3;D1;+0:9]-N(-[CH3;D1;+0:10])-[CH;D2;+0:11]=[O;H0;D1;+0:12].[C:13]-[C:14]-[OH;D1;+0:15].[cH;D2;+0:16]1:[cH;D2;+0:17]:[nH]:[cH;D2;+0:18]:n:1>>[C;D1;H3:19]-[C:20](-[CH3;D1;+0:4])-[C:21]-[#14:22](-[C;D1;...
null
[]
null
null
6
HOUR
5-Chloropentanol (325 g, 2.65 moles) is added to a solution containing tert-butyldimethylsilyl chloride (439 g, 2.91 moles) and dimethylformamide (1.625 liters). Imidazole (199 g, 2.91 moles) is added in one portion and the solution is stirred at room temperature for 6 hours, after which time water (1 liter) is added a...
10.6084/m9.figshare.5104873.v1
null
Tertiary amide.Primary alcohol.Silyl protective group
Primary halide.TMS ether protective group.Silyl protective group
c1c[nH]cn1
null
null
null
O
null
6
CC(C)(C)[Si](C)(C)Cl.CN(C)C=O.OCCCCCCl.c1c[nH]cn1>O>CC(C)(C)[Si](C)(C)OCCCCCCl.CC(C)C[Si](C)(C)OCCCCCCl
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-572be6f88f034fd7920d4ba2775bac75
CCC(CC=O)C1CC=CC1.O=CCCCCC1C=CCC1>>CCC(O)CCCCC1C=CCC1
C=1CC(CC1)C(CC=O)CC.C(C)[Mg]Br.S(O)(O)(=O)=O.C1(C=CCC1)CCCCC=O>>OC(CCCCC1C=CCC1)CC
O=CCC(C1CC=CC1)[CH2:2][CH3:1].[CH:3](=[O:4])[CH2:5][CH2:6][CH2:7][CH2:8][CH:9]1[CH:10]=[CH:11][CH2:12][CH2:13]1>>[CH3:1][CH2:2][CH:3]([OH:4])[CH2:5][CH2:6][CH2:7][CH2:8][CH:9]1[CH:10]=[CH:11][CH2:12][CH2:13]1
CCC(CC=O)C1CC=CC1.O=CCCCCC1C=CCC1
CCC(O)CCCCC1C=CCC1
null
null
O1CCCC1.O
C-C Coupling
OtherReaction
f5b623078728746259c96d8d7e10451b72e36bdaf1d0f607dd894f0c133668e9
a8a096ebbde9746ae0a48228da6e8add5c1838f16988a8681e93e688f2c97cf9
C1=CCCC1
O=C-C-C(-[CH2;D2;+0:1]-[C;D1;H3:2])-C1-C-C=C-C-1.[C:3]-[C:4]-[CH;D2;+0:5]=[O;H0;D1;+0:6]>>[C:3]-[C:4]-[CH;D3;+0:5](-[OH;D1;+0:6])-[CH2;D2;+0:1]-[C;D1;H3:2]
null
[]
-30
CELSIUS
null
null
All work is performed an inert atmosphere using anhydrous tetrahydrofuran. The starting material, 3-(5-cyclopenten-3-yl) valeraldehyde {2-cyclopentene-1-pentanal} (75 g, 0.493 moles) is diluted in tetrahydrofurar (750 ml) and cooled in a -30° C. ethanol/dry ice bath. Ethyl magnesium bromide (0.493 moles) is added dropw...
10.6084/m9.figshare.5104873.v1
null
Aldehyde.Aldehyde
Secondary alcohol
C1=CCCC1
null
C1=CCCC1
HO-
O1CCCC1.O
-30
null
CCC(CC=O)C1CC=CC1.O=CCCCCC1C=CCC1>O1CCCC1.O>CCC(O)CCCCC1C=CCC1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-ff888ae3a7c44055b46ba6e76b9b5081
CC(C)(C)[Si](C)(C)Cl.OCCCCCl>>CC(C)C[Si](C)(C)OCCCCCl
CN(C=O)C.ClCCCCO.[Si](C)(C)(C(C)(C)C)Cl.N1C=NC=C1>>ClCCCCO[Si](C)(C)CC(C)C
Cl[Si:5]([C:2]([CH3:1])([CH3:3])[CH3:4])([CH3:6])[CH3:7].[OH:8][CH2:9][CH2:10][CH2:11][CH2:12][Cl:13]>>[CH3:1][CH:2]([CH3:3])[CH2:4][Si:5]([CH3:6])([CH3:7])[O:8][CH2:9][CH2:10][CH2:11][CH2:12][Cl:13]
CC(C)(C)[Si](C)(C)Cl.OCCCCCl
CC(C)C[Si](C)(C)OCCCCCl
null
null
null
Protection
OtherReaction
16b089e75ae0faeb6299d6901714a961ddf80ba40eb5191df04d4efe8b4a1af5
a12fb6ee4294c877f426f603ce64d893e39b302f1553f4ca246c599e7a8e7068
null
Cl-[Si;H0;D4;+0:1](-[C;D1;H3:2])(-[C;D1;H3:3])-[C;H0;D4;+0:4](-[C;D1;H3:5])(-[C;D1;H3:6])-[CH3;D1;+0:7].[C:8]-[C:9]-[OH;D1;+0:10]>>[C:8]-[C:9]-[O;H0;D2;+0:10]-[Si;H0;D4;+0:1](-[C;D1;H3:2])(-[C;D1;H3:3])-[CH2;D2;+0:7]-[CH;D3;+0:4](-[C;D1;H3:5])-[C;D1;H3:6]
null
[]
null
null
null
null
The procedure followed is the same as that described in Example 19 substituting 4-chlorobutanol (326 g, 3.00 moles), tert-butyldimethylsilyl chloride (500 g, 3.31 moles), imidazole (225 g, 3.30 mmoles), and dimethylformamide (1600 ml). The crude product is fractionally distilled under reduced vacuum leaving a clear, co...
10.6084/m9.figshare.5104873.v1
null
Primary alcohol.Silyl protective group
Silyl protective group
null
null
null
HCl
null
null
null
CC(C)(C)[Si](C)(C)Cl.OCCCCCl>>CC(C)C[Si](C)(C)OCCCCCl
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-7706b324198043e6ac6221284bfb46e7
CC(C)(C)[Si](C)(C)OCCCCC1C=CCC1>>OCCCCC1C=CCC1
C1(C=CCC1)CCCCO[Si](C)(C)C(C)(C)C.F>>OCCCCC1C=CCC1
CC(C)(C)[Si](C)(C)[O:1][CH2:2][CH2:3][CH2:4][CH2:5][CH:6]1[CH:7]=[CH:8][CH2:9][CH2:10]1>>[OH:1][CH2:2][CH2:3][CH2:4][CH2:5][CH:6]1[CH:7]=[CH:8][CH2:9][CH2:10]1
CC(C)(C)[Si](C)(C)OCCCCC1C=CCC1
OCCCCC1C=CCC1
null
null
C(C)#N
Deprotection
Alcohol deprotection from silyl ethers
6ff8c9c41093ab5237b871dd4689ba6431022d615e227d3774901a983c846e4b
84d9f5b4e7757c58e584c26c7d52c9a3f594fbcb0c0d22f34765a93a932fcd5b
C1=CCCC1
C-C(-C)(-C)-[Si](-C)(-C)-[O;H0;D2;+0:1]-[C:2]-[C:3]>>[C:3]-[C:2]-[OH;D1;+0:1]
null
[]
null
null
null
null
The procedure followed is the same as that described in Example 23 substituting 3-(5-[(1,1-dimethylethyl)dimethylsiloxyl]but-1-yl)cyclopentene {[4-(2-cyclopenten-1-yl)butoxy](1,1-dimethylethyl)dimethylsilane} (100 g, 0.407 moles), 5% hydrofluoric acid (78 ml), and acetonitrile (1500 ml). The crude product is kugelrohre...
10.6084/m9.figshare.5104873.v1
null
TMS ether protective group
Primary alcohol
null
null
C1=CCCC1
Other
C(C)#N
null
null
CC(C)(C)[Si](C)(C)OCCCCC1C=CCC1>C(C)#N>OCCCCC1C=CCC1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-4312836202594ea2b2a1aafcadb9333b
CS(=O)(=O)Cl.OCCCCC1C=CCC1>>ClCCCCC1C=CCC1
OCCCCC1C=CCC1.N1=CC=CC=C1.CS(=O)(=O)Cl>>ClCCCCC1C=CCC1
CS(=O)(=O)[Cl:1].O[CH2:2][CH2:3][CH2:4][CH2:5][CH:6]1[CH:7]=[CH:8][CH2:9][CH2:10]1>>[Cl:1][CH2:2][CH2:3][CH2:4][CH2:5][CH:6]1[CH:7]=[CH:8][CH2:9][CH2:10]1
CS(=O)(=O)Cl.OCCCCC1C=CCC1
ClCCCCC1C=CCC1
null
null
CN(C=O)C
Functional Group Interconversion
Alcohol to chloride_sulfonyl chloride
58d25ddf86b8daa38762ecb08ed922faa2d01716f69924f9b8413703fe1b3fc7
d5d71bad4297b1f4f93dd1d1d9cddf0bb6fadb3f4dca1f84369c4074a39097d6
C1=CCCC1
C-S(=O)(=O)-[Cl;H0;D1;+0:1].O-[CH2;D2;+0:2]-[C:3]-[C:4]>>[C:4]-[C:3]-[CH2;D2;+0:2]-[Cl;H0;D1;+0:1]
null
[]
null
null
null
null
3-(4-Hydroxybut-1-yl)cyclopentene {2-cyclopentene-1-butanol} (51 g, 0.37 moles) is diluted in dimethylformamide (100 ml) and added to pyridine (38 g, 0.40 moles). The solution is stirred and methanesulfonyl chloride (46 g, 0.40 moles) is added dropwise over 10 minutes. The reaction is partitioned between hexane (500 ml...
10.6084/m9.figshare.5104873.v1
null
Primary alcohol.Sulfonyl halide
Primary halide
null
null
C1=CCCC1
HO-
CN(C=O)C
null
null
CS(=O)(=O)Cl.OCCCCC1C=CCC1>CN(C=O)C>ClCCCCC1C=CCC1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-1925490ceb67467592872507621e072d
CCC=O.ClCCCCC1C=CCC1>>CCC(O)CCCCC1C=CCC1
C(CC)=O.ClCCCCC1C=CCC1.[Mg].O.ClCCCCC1C=CCC1>>OC(CCCCC1C=CCC1)CC
[CH3:1][CH2:2][CH:3]=[O:4].Cl[CH2:5][CH2:6][CH2:7][CH2:8][CH:9]1[CH:10]=[CH:11][CH2:12][CH2:13]1>>[CH3:1][CH2:2][CH:3]([OH:4])[CH2:5][CH2:6][CH2:7][CH2:8][CH:9]1[CH:10]=[CH:11][CH2:12][CH2:13]1
CCC=O.ClCCCCC1C=CCC1
CCC(O)CCCCC1C=CCC1
null
null
O1CCCC1
C-C Coupling
Grignard_alcohol
983d8b8e9b89ba290d93feeffe843caf411eba49bd1aefb21a784058d86f3a30
3e80fe0b4a87df3724831714de4ab23fef101254d00d9b3074e300e6e8f4b9ea
C1=CCCC1
Cl-[CH2;D2;+0:1]-[C:2]-[C:3].[C;D1;H3:4]-[C:5]-[CH;D2;+0:6]=[O;H0;D1;+0:7]>>[C:3]-[C:2]-[CH2;D2;+0:1]-[CH;D3;+0:6](-[OH;D1;+0:7])-[C:5]-[C;D1;H3:4]
null
[]
0
CELSIUS
null
null
All reactions are carried out under an inert atmosphere. 3-(4-Chlorobut-1-yl)cyclopentene {3-(4-chlorobutyl)cyclopentene} (43 g, 0.27 moles) is diluted in tetrahydrofuran (50 ml) and added dropwise to a stirred, refluxing solution of tetrahydrofuran (200 ml) containing granular magnesium (30 g, 1.25 moles). After the a...
10.6084/m9.figshare.5104873.v1
null
Primary halide.Aldehyde
Secondary alcohol
null
null
C1=CCCC1
Other
O1CCCC1
0
null
CCC=O.ClCCCCC1C=CCC1>O1CCCC1>CCC(O)CCCCC1C=CCC1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-658d441f736741cb9c772b3cd708c096
CCC(CCCCC1CCC2C1CC(=O)C2(Cl)Cl)OC>>CCC(CCCCC1CCC2CC(=O)CC12)OC
ClC1(C2CCC(C2CC1=O)CCCCC(CC)OC)Cl>>COC(CCCCC1C2CC(CC2CC1)=O)CC
Cl[C:12]1(Cl)[CH:11]2[CH2:10][CH2:9][CH:8]([CH2:7][CH2:6][CH2:5][CH2:4][CH:3]([CH2:2][CH3:1])[O:17][CH3:18])[CH:16]2[CH2:15][C:13]1=[O:14]>>[CH3:1][CH2:2][CH:3]([CH2:4][CH2:5][CH2:6][CH2:7][CH:8]1[CH2:9][CH2:10][CH:11]2[CH2:12][C:13](=[O:14])[CH2:15][CH:16]12)[O:17][CH3:18]
CCC(CCCCC1CCC2C1CC(=O)C2(Cl)Cl)OC
CCC(CCCCC1CCC2CC(=O)CC12)OC
null
[Zn].[Cl-].[Cl-].[Zn+2]
C(C)(=O)O
Functional Group Interconversion
OtherReaction
96adc8577184d4d7f9d08648c84f095e8cfcbb983c5ca7b6ef569e3540d5d72d
1a16202f689fbcf4c49583e05a4736360fc884dbe7bf9b78f3063aeae48ae6e3
O=C1CC2CCCC2C1
Cl-[C;H0;D4;+0:1]1(-Cl)-[C:2](-[C:3])-[C:4]-[C:5]-[C:6]-1=[O;D1;H0:7]>>[C:3]-[C:2]1-[C:4]-[C:5]-[C:6](=[O;D1;H0:7])-[CH2;D2;+0:1]-1
null
[]
null
null
null
null
6,6-dichloro-2-(5-methoxyhept-1-yl)bicyclo[3.3.0]octan-7-one {1,1-dichlorohexahydro-4-(5-methoxyheptyl)-2(lH)-pentalenone} or the isomer (45.9 g) are added to a single-neck 100 ml, round-bottom flask equipped with a condenser. The solution is stirred by a magnetic stirrer and powdered zinc metal (92 g) and glacial acet...
10.6084/m9.figshare.5104873.v1
null
Tertiary halide.Tertiary halide
Ketone
C1CC2CCCC2C1
C1CC2CCCC2C1
C1CC2CCCC2C1
Other
[Zn].[Cl-].[Cl-].[Zn+2].C(C)(=O)O
null
null
CCC(CCCCC1CCC2C1CC(=O)C2(Cl)Cl)OC>[Zn].[Cl-].[Cl-].[Zn+2].C(C)(=O)O>CCC(CCCCC1CCC2CC(=O)CC12)OC
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-a0fb30ee3b2c41b0b02c77836884e130
CCC(CCCCC1CCC2C1C(=O)C2(Cl)Cl)OC>>CCC(CCCCC1CCC2CC(=O)C12)OC
ClC1(C2CCC(C2C1=O)CCCCC(CC)OC)Cl>>COC(CCCCC1C2C(CC2CC1)=O)CC
Cl[C:12]1(Cl)[CH:11]2[CH2:10][CH2:9][CH:8]([CH2:7][CH2:6][CH2:5][CH2:4][CH:3]([CH2:2][CH3:1])[O:16][CH3:17])[CH:15]2[C:13]1=[O:14]>>[CH3:1][CH2:2][CH:3]([CH2:4][CH2:5][CH2:6][CH2:7][CH:8]1[CH2:9][CH2:10][CH:11]2[CH2:12][C:13](=[O:14])[CH:15]12)[O:16][CH3:17]
CCC(CCCCC1CCC2C1C(=O)C2(Cl)Cl)OC
CCC(CCCCC1CCC2CC(=O)C12)OC
null
[Zn]
C(C)(=O)O
Functional Group Interconversion
OtherReaction
bfc3e020573e20351ad68954934065203460bc52bee5735cde0606376ab375d3
1a16202f689fbcf4c49583e05a4736360fc884dbe7bf9b78f3063aeae48ae6e3
O=C1CC2CCCC12
Cl-[C;H0;D4;+0:1]1(-Cl)-[C:2](-[C:3])-[C:4]-[C:5]-1=[O;D1;H0:6]>>[C:3]-[C:2]1-[C:4]-[C:5](=[O;D1;H0:6])-[CH2;D2;+0:1]-1
null
[]
null
null
1
HOUR
Zinc (3 g) is added to a stirred solution of 6,6-dichloro-2(5-methoxyhept-1-yl)bicyclo[3.2.0]heptan-7-one {7,7-dichloro-4(5-methoxyheptyl)bicyclo[3.2.0]heptan-6-one} (2 g, 6 moles) in acetic acid (100 ml) under a nitrogen atmosphere. The solution is stirred at room temperature for one hour, then refluxed for 13 hours, ...
10.6084/m9.figshare.5104873.v1
null
Tertiary halide.Tertiary halide
Ketone
C1CC2CCC2C1
C1CC2CCC2C1
C1CC2CCC2C1
Other
[Zn].C(C)(=O)O
null
1
CCC(CCCCC1CCC2C1C(=O)C2(Cl)Cl)OC>[Zn].C(C)(=O)O>CCC(CCCCC1CCC2CC(=O)C12)OC
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-3b4f3d8c616a4a45ba2bbc193e565046
CCC(CCCCC1CCC2CC(=O)CC12)OC>>CCC(CCCCC1CCC2CC(C)(O)CC12)OC
COC(CCCCC1C2CC(CC2CC1)=O)CC.COC(CCCCC1C2CC(CC2CC1)=O)CC.C(C)[Mg]Br>>COC(CCCCC1C2CC(CC2CC1)(O)C)CC
[CH3:1][CH2:2][CH:3]([CH2:4][CH2:5][CH2:6][CH2:7][CH:8]1[CH2:9][CH2:10][CH:11]2[CH2:12][C:13](=[O:15])[CH2:16][CH:17]12)[O:18][CH3:19]>>[CH3:1][CH2:2][CH:3]([CH2:4][CH2:5][CH2:6][CH2:7][CH:8]1[CH2:9][CH2:10][CH:11]2[CH2:12][C:13]([CH3:14])([OH:15])[CH2:16][CH:17]12)[O:18][CH3:19]
CCC(CCCCC1CCC2CC(=O)CC12)OC
CCC(CCCCC1CCC2CC(C)(O)CC12)OC
null
null
CCOCC.C(C)OCC
Miscellaneous
OtherReaction
1ecd181abde8298e671a9f4f1de0a680fd98e618629b4139d000f7403ddf00cd
8811b4d793f7cfa9f0f1f47a008648edabb54f371f76dfa680dd5b2e1564c6c5
C1CC2CCCC2C1
[O;H0;D1;+0:1]=[C;H0;D3;+0:2]1-[C:3]-[C:4]-[C:5]-[C:6]-1>>[C;D1;H3:7]-[C;H0;D4;+0:2]1(-[OH;D1;+0:1])-[C:3]-[C:4]-[C:5]-[C:6]-1
39.9
[{"value": 39.9, "product": "COC(CCCCC1C2CC(CC2CC1)(O)C)CC", "details": "CALCULATEDPERCENTYIELD", "is_desired": false}]
null
null
null
null
2-(5-Methoxyhept-1-yl)bicyclo[3.3.0]octan-7-one hexahydro-4-(5-methoxyheptyl)-2(1H)-pentalenone, (4 g, 0.0158 moles) diluted in ether is added dropwise to a stirring solution of ethyl magnesium bromide (0.0158 moles) dissolved with diethyl ether. The mixture is cooled in an ice bath during the addition. The ice bath is...
10.6084/m9.figshare.5104873.v1
null
Ketone
Tertiary alcohol
C1CC2CCCC2C1
C1CC2CCCC2C1
C1CC2CCCC2C1
Other
CCOCC.C(C)OCC
null
null
CCC(CCCCC1CCC2CC(=O)CC12)OC>CCOCC.C(C)OCC>CCC(CCCCC1CCC2CC(C)(O)CC12)OC
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-59112f48b25e446cb302058979b54590
CCC(CCCCCl)OC.ClC1C=CCC1>>CCC(CCCCC1C=CCC1)OC
ClCCCCC(CC)OC.[Cl-].[NH4+].[Mg].ClC1C=CCC1>>COC(CCCCC1C=CCC1)CC
Cl[CH2:7][CH2:6][CH2:5][CH2:4][CH:3]([CH2:2][CH3:1])[O:13][CH3:14].Cl[CH:8]1[CH:9]=[CH:10][CH2:11][CH2:12]1>>[CH3:1][CH2:2][CH:3]([CH2:4][CH2:5][CH2:6][CH2:7][CH:8]1[CH:9]=[CH:10][CH2:11][CH2:12]1)[O:13][CH3:14]
CCC(CCCCCl)OC.ClC1C=CCC1
CCC(CCCCC1C=CCC1)OC
null
null
O1CCCC1
C-C Coupling
Negishi
9a6bf7e2b45e73e51c658250a4e70cb08f6a32ab7a16b4f9f48c368b31fb4ddc
d4cf29bb0f2586f258c9eb5d3edb710b86094a4be60be4638a5468606055dcb5
C1=CCCC1
Cl-[CH2;D2;+0:1]-[C:2]-[C:3].Cl-[CH;D3;+0:4]1-[C:5]-[C:6]-[C:7]=[C:8]-1>>[C:3]-[C:2]-[CH2;D2;+0:1]-[CH;D3;+0:4]1-[C:5]-[C:6]-[C:7]=[C:8]-1
null
[]
-25
CELSIUS
null
null
A three-neck, round-bottomed flask containing magnesium metal turnings (7.2 g, 0.299 moles), is equipped with a Friedrich condenser and kept under a nitrogen atmosphere. Tetrahydrofuran (300 ml) is added and the contents are allowed to stir. A solution of 1-chloro-5-methoxyheptane (48.1 g, 0.292 moles) is added in smal...
10.6084/m9.figshare.5104873.v1
null
Secondary halide.Primary halide
null
C1=CCCC1
C1=CCCC1
C1=CCCC1
Other
O1CCCC1
-25
null
CCC(CCCCCl)OC.ClC1C=CCC1>O1CCCC1>CCC(CCCCC1C=CCC1)OC
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-463df9a7378c4be6b53eb256f879c341
CCC(CCCCC1CCC2C1C(=O)C2(Cl)Cl)OC>>CCC(CCCCC1CCC2C1CC(=O)C2(Cl)Cl)OC
ClC1(C2CCC(C2C1=O)CCCCC(CC)OC)Cl.[OH-].[K+].[N+](=[N-])=C.CN(S(=O)(=O)C1=CC=C(C=C1)C)N=O.[N+](=[N-])=C.ClC1(C(C2C(CCC12)CCCCC(CC)OC)=O)Cl>>ClC1(C2CCC(C2CC1=O)CCCCC(CC)OC)Cl
[CH3:1][CH2:2][CH:3]([CH2:4][CH2:5][CH2:6][CH2:7][CH:8]1[CH2:9][CH2:10][CH:11]2[CH:12]1[C:14](=[O:15])[C:16]2([Cl:17])[Cl:18])[O:19][CH3:20]>>[CH3:1][CH2:2][CH:3]([CH2:4][CH2:5][CH2:6][CH2:7][CH:8]1[CH2:9][CH2:10][CH:11]2[CH:12]1[CH2:13][C:14](=[O:15])[C:16]2([Cl:17])[Cl:18])[O:19][CH3:20]
CCC(CCCCC1CCC2C1C(=O)C2(Cl)Cl)OC
CCC(CCCCC1CCC2C1CC(=O)C2(Cl)Cl)OC
null
null
CCOCC.C(C)(=O)O.C(C)O
Miscellaneous
OtherReaction
97d98f33c73f2831bc5bd487ce5dea0447a55d13adc3d8dc0ef940f61adf4799
f394080031812a9c0cde55fa330311dfe42bea38dbdf0b4621700859838ffa32
O=C1CC2CCCC2C1
[C:1]-[C:2]1-[C:3]-[C:4]-[C:5]2-[CH;D3;+0:6]-1-[C;H0;D3;+0:7](=[O;D1;H0:8])-[C:9]-2(-[Cl;D1;H0:10])-[Cl;D1;H0:11]>>[C:1]-[C:2]1-[C:3]-[C:4]-[C:5]2-[CH;D3;+0:6]-1-[C:12]-[C;H0;D3;+0:7](=[O;D1;H0:8])-[C:9]-2(-[Cl;D1;H0:10])-[Cl;D1;H0:11]
null
[]
null
null
null
null
The starting material, 6,6-dichloro-2-(5-methoxyhept-1-yl) bicyclo[3.2.0]heptan-7-one {7,7-dichloro-4-(5-methoxyheptyl)bicyclo [3.2.0]heptan-6-one} (5 g), is dissolved in 100 ml of ether and transferred to a 500 ml, round-bottomed flask. An excess of diazomethane is generated in situ by reacting N-methyl-N-nitroso-p-to...
10.6084/m9.figshare.5104873.v1
null
Ketone
Ketone
C1CC2CCC2C1
C1CC2CCCC2C1
C1CC2CCCC2C1
Other
CCOCC.C(C)(=O)O.C(C)O
null
null
CCC(CCCCC1CCC2C1C(=O)C2(Cl)Cl)OC>CCOCC.C(C)(=O)O.C(C)O>CCC(CCCCC1CCC2C1CC(=O)C2(Cl)Cl)OC
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-7f3ea532b31d44c58d8e70e3fda794e9
CCC(CCCCC1CCC2C1CC(=O)C2(Cl)Cl)OC>>CCC(CCCCC1CCC2CC(=O)CC12)OC
ClC1(C2CCC(C2CC1=O)CCCCC(CC)OC)Cl>>COC(CCCCC1C2CC(CC2CC1)=O)CC
Cl[C:12]1(Cl)[CH:11]2[CH2:10][CH2:9][CH:8]([CH2:7][CH2:6][CH2:5][CH2:4][CH:3]([CH2:2][CH3:1])[O:17][CH3:18])[CH:16]2[CH2:15][C:13]1=[O:14]>>[CH3:1][CH2:2][CH:3]([CH2:4][CH2:5][CH2:6][CH2:7][CH:8]1[CH2:9][CH2:10][CH:11]2[CH2:12][C:13](=[O:14])[CH2:15][CH:16]12)[O:17][CH3:18]
CCC(CCCCC1CCC2C1CC(=O)C2(Cl)Cl)OC
CCC(CCCCC1CCC2CC(=O)CC12)OC
null
[Zn]
C(C)(=O)O
Functional Group Interconversion
OtherReaction
96adc8577184d4d7f9d08648c84f095e8cfcbb983c5ca7b6ef569e3540d5d72d
1a16202f689fbcf4c49583e05a4736360fc884dbe7bf9b78f3063aeae48ae6e3
O=C1CC2CCCC2C1
Cl-[C;H0;D4;+0:1]1(-Cl)-[C:2](-[C:3])-[C:4]-[C:5]-[C:6]-1=[O;D1;H0:7]>>[C:3]-[C:2]1-[C:4]-[C:5]-[C:6](=[O;D1;H0:7])-[CH2;D2;+0:1]-1
null
[]
null
null
null
null
6,6-Dichloro-2-(5-methoxyhept-1-yl)bicyclo[3.3.0]octan-7-one {1,1-dichlorohexahydro-4-(5-methoxyheptyl)-2(1H)-pentalenone} (45.9 g) is added to a 100 ml, round-bottomed flask fitted with a condenser. Powdered zinc metal (92 g) and glacial acetic acid (312 ml) are added to the flask and the solution allowed to reflux fo...
10.6084/m9.figshare.5104873.v1
null
Tertiary halide.Tertiary halide
Ketone
C1CC2CCCC2C1
C1CC2CCCC2C1
C1CC2CCCC2C1
Other
[Zn].C(C)(=O)O
null
null
CCC(CCCCC1CCC2C1CC(=O)C2(Cl)Cl)OC>[Zn].C(C)(=O)O>CCC(CCCCC1CCC2CC(=O)CC12)OC
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-cc943bb8137844e696e7511318aca43f
CCOC(CC)CCCCC1CCC2C1C(=O)C2(Cl)Cl>>CCOC(CC)CCCCC1CCC2C1CC(=O)C2(Cl)Cl
ClC1(C2CCC(C2C1=O)CCCCC(CC)OCC)Cl.C(C)OC(CCCCC1C=CCC1)CC.ClC1(C(C2C(CCC12)CCCCC(CC)OCC)=O)Cl.[N+](=[N-])=C.ClCCCCC(CC)OCC>>ClC1(C2CCC(C2CC1=O)CCCCC(CC)OCC)Cl
[CH3:1][CH2:2][O:3][CH:4]([CH2:5][CH3:6])[CH2:7][CH2:8][CH2:9][CH2:10][CH:11]1[CH2:12][CH2:13][CH:14]2[CH:15]1[C:17](=[O:18])[C:19]2([Cl:20])[Cl:21]>>[CH3:1][CH2:2][O:3][CH:4]([CH2:5][CH3:6])[CH2:7][CH2:8][CH2:9][CH2:10][CH:11]1[CH2:12][CH2:13][CH:14]2[CH:15]1[CH2:16][C:17](=[O:18])[C:19]2([Cl:20])[Cl:21]
CCOC(CC)CCCCC1CCC2C1C(=O)C2(Cl)Cl
CCOC(CC)CCCCC1CCC2C1CC(=O)C2(Cl)Cl
null
null
null
Miscellaneous
OtherReaction
97d98f33c73f2831bc5bd487ce5dea0447a55d13adc3d8dc0ef940f61adf4799
f394080031812a9c0cde55fa330311dfe42bea38dbdf0b4621700859838ffa32
O=C1CC2CCCC2C1
[C:1]-[C:2]1-[C:3]-[C:4]-[C:5]2-[CH;D3;+0:6]-1-[C;H0;D3;+0:7](=[O;D1;H0:8])-[C:9]-2(-[Cl;D1;H0:10])-[Cl;D1;H0:11]>>[C:1]-[C:2]1-[C:3]-[C:4]-[C:5]2-[CH;D3;+0:6]-1-[C:12]-[C;H0;D3;+0:7](=[O;D1;H0:8])-[C:9]-2(-[Cl;D1;H0:10])-[Cl;D1;H0:11]
null
[]
null
null
null
null
The corresponding 2-(5-ethoxyhept-1-yl) homologs are prepared by substituting an equivalent amount of 1-chloro-5-ethoxyheptane in the Grignard reaction of Example 1 in place of the 5-methoxy homolog and using the reaction sequence shown above to prepare first the 3-(5-ethoxyhept-1-yl)cyclopentene, which is then convert...
10.6084/m9.figshare.5104873.v1
null
Ketone
Ketone
C1CC2CCC2C1
C1CC2CCCC2C1
C1CC2CCCC2C1
Other
null
null
null
CCOC(CC)CCCCC1CCC2C1C(=O)C2(Cl)Cl>>CCOC(CC)CCCCC1CCC2C1CC(=O)C2(Cl)Cl
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-f7eb1d9de728438c9f42db028e332833
CCC(CCCCC1CCC2CC(=O)CC12)OC>>CCC(CCCCC1CCC2CC(C)(O)CC12)OC
COC(CCCCC1C2CC(CC2CC1)=O)CC.C(C)[Mg]Br>>COC(CCCCC1C2CC(CC2CC1)(O)C)CC
[CH3:1][CH2:2][CH:3]([CH2:4][CH2:5][CH2:6][CH2:7][CH:8]1[CH2:9][CH2:10][CH:11]2[CH2:12][C:13](=[O:15])[CH2:16][CH:17]12)[O:18][CH3:19]>>[CH3:1][CH2:2][CH:3]([CH2:4][CH2:5][CH2:6][CH2:7][CH:8]1[CH2:9][CH2:10][CH:11]2[CH2:12][C:13]([CH3:14])([OH:15])[CH2:16][CH:17]12)[O:18][CH3:19]
CCC(CCCCC1CCC2CC(=O)CC12)OC
CCC(CCCCC1CCC2CC(C)(O)CC12)OC
null
null
CCOCC.C(C)OCC
Miscellaneous
OtherReaction
1ecd181abde8298e671a9f4f1de0a680fd98e618629b4139d000f7403ddf00cd
8811b4d793f7cfa9f0f1f47a008648edabb54f371f76dfa680dd5b2e1564c6c5
C1CC2CCCC2C1
[O;H0;D1;+0:1]=[C;H0;D3;+0:2]1-[C:3]-[C:4]-[C:5]-[C:6]-1>>[C;D1;H3:7]-[C;H0;D4;+0:2]1(-[OH;D1;+0:1])-[C:3]-[C:4]-[C:5]-[C:6]-1
null
[]
null
null
null
null
2-(5-Methoxyhept-1-yl)bicyclo[3.3.0]octan-7-one {hexahydro-4-(5-methoxyheptyl)-2(1H)-pentalenone} (4 g, 0.0158 moles) diluted in ether is added dropwise to a stirring solution of ethyl magnesium bromide (0.0158 moles) dissolved with diethyl ether. The mixture is cooled in an ice bath during the addition. The ice bath i...
10.6084/m9.figshare.5104873.v1
null
Ketone
Tertiary alcohol
C1CC2CCCC2C1
C1CC2CCCC2C1
C1CC2CCCC2C1
Other
CCOCC.C(C)OCC
null
null
CCC(CCCCC1CCC2CC(=O)CC12)OC>CCOCC.C(C)OCC>CCC(CCCCC1CCC2CC(C)(O)CC12)OC
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-bed3dee93a03496f83549f0ad35d1929
CCC(CCCCC1CCC2C1CC(=O)C2(Cl)Cl)OC>>CCC(CCCCC1CCC2CC(O)CC12)OC
ClC1(C2CCC(C2CC1=O)CCCCC(CC)OC)Cl.ClC1(C2CCC(C2CC1O)CCCCC(CC)OC)Cl>>COC(CCCCC1C2CC(CC2CC1)O)CC
Cl[C:12]1(Cl)[CH:11]2[CH2:10][CH2:9][CH:8]([CH2:7][CH2:6][CH2:5][CH2:4][CH:3]([CH2:2][CH3:1])[O:17][CH3:18])[CH:16]2[CH2:15][C:13]1=[O:14]>>[CH3:1][CH2:2][CH:3]([CH2:4][CH2:5][CH2:6][CH2:7][CH:8]1[CH2:9][CH2:10][CH:11]2[CH2:12][CH:13]([OH:14])[CH2:15][CH:16]12)[O:17][CH3:18]
CCC(CCCCC1CCC2C1CC(=O)C2(Cl)Cl)OC
CCC(CCCCC1CCC2CC(O)CC12)OC
null
[Zn]
C(C)(=O)O
Reduction
OtherReaction
351c9b612406ce72847eab727b7250c3b9dbfef2aaf513caea6ec04764d30901
842aa4ebb60cfc8e76502bd50f3e0d33e0dc5566b03c89a81de612990dca6c8c
C1CC2CCCC2C1
Cl-[C;H0;D4;+0:1]1(-Cl)-[C:2](-[C:3])-[C:4]-[C:5]-[C;H0;D3;+0:6]-1=[O;H0;D1;+0:7]>>[C:3]-[C:2]1-[C:4]-[C:5]-[CH;D3;+0:6](-[OH;D1;+0:7])-[CH2;D2;+0:1]-1
null
[]
null
null
null
null
The reactions of this example can also be conducted using an equivalent amount of 6,6-dichloro-2-(5-methoxyhept-1-yl)bicyclo [3.3.0]octan-7-one {1-1-dichlorohexahydro-4-(5-methoxyheptyl)-2 (1H)-pentalenone} to first prepare 6,6-dichloro-2-(5-methoxyhept-1-yl) bicyclo[3.3.0]octan-7-ol {1,1-dichlorooctahydro-4-(5-methoxy...
10.6084/m9.figshare.5104873.v1
null
Tertiary halide.Tertiary halide.Ketone
Secondary alcohol
C1CC2CCCC2C1
C1CC2CCCC2C1
C1CC2CCCC2C1
Other
[Zn].C(C)(=O)O
null
null
CCC(CCCCC1CCC2C1CC(=O)C2(Cl)Cl)OC>[Zn].C(C)(=O)O>CCC(CCCCC1CCC2CC(O)CC12)OC
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-642222c817f14c568dd170c84ef8109c
CC(C)(C)[Si](C)(C)Cl.OCCCCCCl>>CC(C)C[Si](C)(C)OCCCCCCl
N1C=NC=C1.ClCCCCCO.[Si](C)(C)(C(C)(C)C)Cl.CN(C=O)C>>ClCCCCCO[Si](C)(C)CC(C)C
Cl[Si:5]([C:2]([CH3:1])([CH3:3])[CH3:4])([CH3:6])[CH3:7].[OH:8][CH2:9][CH2:10][CH2:11][CH2:12][CH2:13][Cl:14]>>[CH3:1][CH:2]([CH3:3])[CH2:4][Si:5]([CH3:6])([CH3:7])[O:8][CH2:9][CH2:10][CH2:11][CH2:12][CH2:13][Cl:14]
CC(C)(C)[Si](C)(C)Cl.OCCCCCCl
CC(C)C[Si](C)(C)OCCCCCCl
null
null
O
Protection
OtherReaction
16b089e75ae0faeb6299d6901714a961ddf80ba40eb5191df04d4efe8b4a1af5
a12fb6ee4294c877f426f603ce64d893e39b302f1553f4ca246c599e7a8e7068
null
Cl-[Si;H0;D4;+0:1](-[C;D1;H3:2])(-[C;D1;H3:3])-[C;H0;D4;+0:4](-[C;D1;H3:5])(-[C;D1;H3:6])-[CH3;D1;+0:7].[C:8]-[C:9]-[OH;D1;+0:10]>>[C:8]-[C:9]-[O;H0;D2;+0:10]-[Si;H0;D4;+0:1](-[C;D1;H3:2])(-[C;D1;H3:3])-[CH2;D2;+0:7]-[CH;D3;+0:4](-[C;D1;H3:5])-[C;D1;H3:6]
null
[]
null
null
null
null
5-Chloropentanol (325 g, 2.65 moles) is added to a solution containing tert-butyldimethylsilyl chloride (439 g, 2.91 moles) and dimethylformamide (1.625 liters). The solution is stirred and imidazole (199 g, 2.91 moles) is added at once. The solution is stirred at room temperature for 6 hours, after which time water (1...
10.6084/m9.figshare.5104873.v1
null
Primary alcohol.Silyl protective group
Silyl protective group
null
null
null
HCl
O
null
null
CC(C)(C)[Si](C)(C)Cl.OCCCCCCl>O>CC(C)C[Si](C)(C)OCCCCCCl
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-44a89d079e1d4521b5a9c6a109d06cd9
CC(C)(C)[Si](C)(C)OCCCCCCl.ClC1C=CCC1>>CC(C)(C)[Si](C)(C)OCCCCCC1C=CCC1
[Mg].ClCCCCCO[Si](C)(C)CC(C)C.ClC1C=CCC1.ClCCCCCO[Si](C)(C)C(C)(C)C>>CC(C)(C)[Si](OCCCCCC1C=CCC1)(C)C
Cl[CH2:13][CH2:12][CH2:11][CH2:10][CH2:9][O:8][Si:5]([C:2]([CH3:1])([CH3:3])[CH3:4])([CH3:6])[CH3:7].Cl[CH:14]1[CH:15]=[CH:16][CH2:17][CH2:18]1>>[CH3:1][C:2]([CH3:3])([CH3:4])[Si:5]([CH3:6])([CH3:7])[O:8][CH2:9][CH2:10][CH2:11][CH2:12][CH2:13][CH:14]1[CH:15]=[CH:16][CH2:17][CH2:18]1
CC(C)(C)[Si](C)(C)OCCCCCCl.ClC1C=CCC1
CC(C)(C)[Si](C)(C)OCCCCCC1C=CCC1
null
null
O1CCCC1.O
C-C Coupling
Negishi
9a6bf7e2b45e73e51c658250a4e70cb08f6a32ab7a16b4f9f48c368b31fb4ddc
d4cf29bb0f2586f258c9eb5d3edb710b86094a4be60be4638a5468606055dcb5
C1=CCCC1
Cl-[CH2;D2;+0:1]-[C:2]-[C:3].Cl-[CH;D3;+0:4]1-[C:5]=[C:6]-[C:7]-[C:8]-1>>[C:3]-[C:2]-[CH2;D2;+0:1]-[CH;D3;+0:4]1-[C:5]=[C:6]-[C:7]-[C:8]-1
null
[]
null
null
null
null
All reactions are carried out under an inert atmosphere. The starting material, (5-chloro-1-pentyloxy)(2,2-dimethylethyl) dimethylsilane {[(5-chloropentyl)oxy](1,1-dimethylethyl)dimethylsilane} (534 g, 2.26 moles), diluted in tetrahydrofuran (500 ml), is added portionwise to a refluxing solution of tetrahydrofuran and ...
10.6084/m9.figshare.5104873.v1
null
Secondary halide.Primary halide
null
C1=CCCC1
C1=CCCC1
C1=CCCC1
Other
O1CCCC1.O
null
null
CC(C)(C)[Si](C)(C)OCCCCCCl.ClC1C=CCC1>O1CCCC1.O>CC(C)(C)[Si](C)(C)OCCCCCC1C=CCC1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-7822be45e6a7487a81b1386880688f0e
CC(C)(C)[Si](C)(C)OCCCCCC1CCC2C1CC(=O)C2(Cl)Cl>>O=C1CC2CCC(CCCCCO)C2C1
ClC1(C2CCC(C2CC1=O)CCCCCO[Si](C)(C)C(C)(C)C)Cl.ClC1(C(CC2C(CCC12)CCCCCO[Si](C)(C)C(C)(C)C)=O)Cl.CCOCC>>OCCCCCC1C2CC(CC2CC1)=O
CC(C)(C)[Si](C)(C)[O:13][CH2:12][CH2:11][CH2:10][CH2:9][CH2:8][CH:7]1[CH2:6][CH2:5][CH:4]2[C:3](Cl)(Cl)[C:2](=[O:1])[CH2:15][CH:14]21>>[O:1]=[C:2]1[CH2:3][CH:4]2[CH2:5][CH2:6][CH:7]([CH2:8][CH2:9][CH2:10][CH2:11][CH2:12][OH:13])[CH:14]2[CH2:15]1
CC(C)(C)[Si](C)(C)OCCCCCC1CCC2C1CC(=O)C2(Cl)Cl
O=C1CC2CCC(CCCCCO)C2C1
null
[Zn]
C(C)(=O)O
Deprotection
OtherReaction
a6023071637a7a1fd55762c847d42bf9e4bf43a1deeb92c6f585037e3e1e93f6
134ea584ae06b324ee35fec219b8456a8da345492f4eb1044d490535f00a1b3e
O=C1CC2CCCC2C1
C-C(-C)(-C)-[Si](-C)(-C)-[O;H0;D2;+0:1]-[C:2]-[C:3].Cl-[C;H0;D4;+0:4]1(-Cl)-[C:5](=[O;D1;H0:6])-[C:7]-[C:8]-[C:9]-1-[C:10]>>[C:3]-[C:2]-[OH;D1;+0:1].[C:10]-[C:9]1-[C:8]-[C:7]-[C:5](=[O;D1;H0:6])-[CH2;D2;+0:4]-1
null
[]
70
CELSIUS
null
null
The starting material, 6,6-dichloro-2-(5-[(1,1-dimethylethyl)dimethylsiloxy]pent-1-yl)bicyclo[3.3.0]octan-7-one {1,1-dichloro-4-[5-[[(1,1-dimethylethyl)dimethylsilyl]oxy]pentyl]hexahydro-2(1H)-pentalenone}(12.1 g, 0.30 moles) is dissolved in glacial acetic acid (85 ml) and the solution is stirred while zinc (25 g) is s...
10.6084/m9.figshare.5104873.v1
null
Tertiary halide.Tertiary halide.Ketone.TMS ether protective group
Ketone.Primary alcohol
C1CC2CCCC2C1
C1CC2CCCC2C1
C1CC2CCCC2C1
HCl
[Zn].C(C)(=O)O
70
null
CC(C)(C)[Si](C)(C)OCCCCCC1CCC2C1CC(=O)C2(Cl)Cl>[Zn].C(C)(=O)O>O=C1CC2CCC(CCCCCO)C2C1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-44bfa0d5f31a44aa9684818b80bf5a65
CC(C)(C)[Si](C)(C)OCCCCCC1C=CCC1>>OCCCCCC1C=CCC1
CC(C)(C)[Si](OCCCCCC1C=CCC1)(C)C.F.C([O-])(O)=O.[Na+]>>OCCCCCC1C=CCC1
CC(C)(C)[Si](C)(C)[O:1][CH2:2][CH2:3][CH2:4][CH2:5][CH2:6][CH:7]1[CH:8]=[CH:9][CH2:10][CH2:11]1>>[OH:1][CH2:2][CH2:3][CH2:4][CH2:5][CH2:6][CH:7]1[CH:8]=[CH:9][CH2:10][CH2:11]1
CC(C)(C)[Si](C)(C)OCCCCCC1C=CCC1
OCCCCCC1C=CCC1
null
null
C(C)#N
Deprotection
Alcohol deprotection from silyl ethers
6ff8c9c41093ab5237b871dd4689ba6431022d615e227d3774901a983c846e4b
84d9f5b4e7757c58e584c26c7d52c9a3f594fbcb0c0d22f34765a93a932fcd5b
C1=CCCC1
C-C(-C)(-C)-[Si](-C)(-C)-[O;H0;D2;+0:1]-[C:2]-[C:3]>>[C:3]-[C:2]-[OH;D1;+0:1]
null
[]
null
null
10
MINUTE
3-(5-[(1,1-Dimethylethyl)dimethylsiloxy]pent-1-yl)cyclopentene (300 g, 1.170 moles) is diluted with acetonitrile (3000 ml) and a 40% stock solution of hydrofluoric acid (166 ml) is added. The reaction is stirred at room temperature for 10 minutes and then slowly neutralized with a saturated solution of sodium bicarbona...
10.6084/m9.figshare.5104873.v1
null
TMS ether protective group
Primary alcohol
null
null
C1=CCCC1
Other
C(C)#N
null
0.166667
CC(C)(C)[Si](C)(C)OCCCCCC1C=CCC1>C(C)#N>OCCCCCC1C=CCC1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-a798ca8805c3407eb1901260aed8dce8
CCC(CC=O)C1C=CCC1.CCC(CC=O)C1CC=CC1>>CCC(O)CCCCC1C=CCC1
C=1CC(CC1)C(CC=O)CC.C(C)[Mg]Br.S(O)(O)(=O)=O.C1=CC(CC1)C(CC=O)CC>>OC(CCCCC1C=CCC1)CC
CC[CH:8]([CH2:7]C=[O:4])[CH:9]1[CH:10]=[CH:11][CH2:12][CH2:13]1.O=[CH:6][CH2:5][CH:3](C1CC=CC1)[CH2:2][CH3:1]>>[CH3:1][CH2:2][CH:3]([OH:4])[CH2:5][CH2:6][CH2:7][CH2:8][CH:9]1[CH:10]=[CH:11][CH2:12][CH2:13]1
CCC(CC=O)C1C=CCC1.CCC(CC=O)C1CC=CC1
CCC(O)CCCCC1C=CCC1
null
null
O1CCCC1.O
Heteroatom Alkylation and Arylation
OtherReaction
e36ded412ea1d7c6f9df5824d7ce6c857249051a6957dd698d740bd96921a6a1
8bfc6d7c0e522e7b1f11bf2b693fafd682d1ff34472ac7c26c6e3f71ef89dcf0
C1=CCCC1
C-C-[CH;D3;+0:1](-[CH2;D2;+0:2]-C=[O;H0;D1;+0:3])-[C:4]1-[C:5]=[C:6]-[C:7]-[C:8]-1.O=[CH;D2;+0:9]-[C:10]-[CH;D3;+0:11](-[C:12]-[C;D1;H3:13])-C1-C-C=C-C-1>>[C;D1;H3:13]-[C:12]-[CH;D3;+0:11](-[OH;D1;+0:3])-[C:10]-[CH2;D2;+0:9]-[CH2;D2;+0:2]-[CH2;D2;+0:1]-[C:4]1-[C:5]=[C:6]-[C:7]-[C:8]-1
null
[]
-30
CELSIUS
null
null
All work is performed in an inert atmosphere using anhydrous tetrahydrofuran. The starting material, 3-(5-cyclopenten-3-yl) valeraldehyde {2-cyclopentene-1-pentanal} (75 g, 0.493 moles) is dissolved in tetrahydrofuran (750 ml) and cooled in a -30° C. ethanol/dry ice bath. Ethyl magnesium bromide (0.493 moles) is added ...
10.6084/m9.figshare.5104873.v1
null
Aldehyde.Aldehyde
Secondary alcohol
C1=CCCC1
null
C1=CCCC1
HO-
O1CCCC1.O
-30
null
CCC(CC=O)C1C=CCC1.CCC(CC=O)C1CC=CC1>O1CCCC1.O>CCC(O)CCCCC1C=CCC1
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-34afba9a9704414cbb10f1ebd75ae625
CC(C)(C)[Si](C)(C)Cl.CCC(O)CCCCC1C=CCC1.CCC(O)CCCCC1C=CCC1.c1c[nH]cn1>>CCC(CCCCC1C=CCC1)OCC(C)(C)[SiH](C)C.CCC(CCCCC1C=CCC1)O[Si](C)(C)C(C)(C)C
N1C=NC=C1.OC(CCCCC1C=CCC1)CC.C(C)C(CCCCC1C=CCC1)O.[Si](C)(C)(C(C)(C)C)Cl>>C1(C=CCC1)CCCCC(CC)OCC(C)(C)[SiH](C)C.CC(C)(C)[Si](OC(CCCCC1C=CCC1)CC)(C)C
Cl[Si:18]([C:15]([CH3:16])([CH3:17])[CH3:37])([CH3:19])[CH3:40].[CH3:1][CH2:2][CH:3]([CH2:4][CH2:5][CH2:6][CH2:7][CH:8]1[CH:9]=[CH:10][CH2:11][CH2:12]1)[OH:13].[CH3:21][CH2:22][CH:23]([CH2:24][CH2:25][CH2:26][CH2:27][CH:28]1[CH:29]=[CH:30][CH2:31][CH2:32]1)[OH:33].n1[cH:14][nH][cH:20][cH:36]1>>[CH3:1][CH2:2][CH:3]([CH2...
CC(C)(C)[Si](C)(C)Cl.CCC(O)CCCCC1C=CCC1.CCC(O)CCCCC1C=CCC1.c1c[nH]cn1
CCC(CCCCC1C=CCC1)OCC(C)(C)[SiH](C)C.CCC(CCCCC1C=CCC1)O[Si](C)(C)C(C)(C)C
null
null
CN(C=O)C
Heteroatom Alkylation and Arylation
OtherReaction
94bbf83bb4e309c242af61604eb8d59215d1fad5e5a6fa3369286f414da72c62
12e47ce768a9e0b4fc42c8b8462594651faaf7fa9858d4c8019f2073451198b4
C1=CCCC1.C1=CCCC1
Cl-[Si;H0;D4;+0:1](-[C;D1;H3:2])(-[CH3;D1;+0:3])-[C;H0;D4;+0:4](-[C;D1;H3:5])(-[C;D1;H3:6])-[CH3;D1;+0:7].[C:8]-[C:9](-[C:10])-[OH;D1;+0:11].[C:12]-[C:13](-[C:14])-[OH;D1;+0:15].[cH;D2;+0:16]1:[nH]:[cH;D2;+0:17]:[cH;D2;+0:18]:n:1>>[C:12]-[C:13](-[C:14])-[O;H0;D2;+0:15]-[#14:19](-[C;D1;H3:20])(-[CH3;D1;+0:18])-[C;H0;D4;...
null
[]
null
null
null
null
The procedure followed is the same as that described in Example 7 and 8 using 3-(5-hydroxyhept-1-yl)cyclopentene {alpha-ethyl-2-cyclopenten-1-pentanol} (32.5 g, 0.177 moles), t-butyldimethylsilylchloride (29.3 g, 0.194 moles), imidazole (13.3 g, 0.194 moles), and dimethylformamide (163 ml). The crude product is fractio...
10.6084/m9.figshare.5104873.v1
null
Secondary alcohol.Secondary alcohol.Silyl protective group
Ether.TMS ether protective group
c1c[nH]cn1
null
C1=CCCC1.C1=CCCC1
null
CN(C=O)C
null
null
CC(C)(C)[Si](C)(C)Cl.CCC(O)CCCCC1C=CCC1.CCC(O)CCCCC1C=CCC1.c1c[nH]cn1>CN(C=O)C>CCC(CCCCC1C=CCC1)OCC(C)(C)[SiH](C)C.CCC(CCCCC1C=CCC1)O[Si](C)(C)C(C)(C)C
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-5263750bf1284597acc5550363a196ee
CCC(O)CCCCC1CCC2CC(=O)CC12>>CCC(=O)CCCCC1CCC2CC(=O)CC12
[Cr](=O)(=O)([O-])O[Cr](=O)(=O)[O-].[NH+]1=CC=CC=C1.[NH+]1=CC=CC=C1.OC(CCCCC1C2CC(CC2CC1)=O)CC.OC(CCCCC1C2CC(CC2CC1)=O)CC.OC(CCCCC1C2CC(CC2CC1)=O)CC>>O=C(CCCCC1C2CC(CC2CC1)=O)CC
[CH3:1][CH2:2][CH:3]([OH:4])[CH2:5][CH2:6][CH2:7][CH2:8][CH:9]1[CH2:10][CH2:11][CH:12]2[CH2:13][C:14](=[O:15])[CH2:16][CH:17]12>>[CH3:1][CH2:2][C:3](=[O:4])[CH2:5][CH2:6][CH2:7][CH2:8][CH:9]1[CH2:10][CH2:11][CH:12]2[CH2:13][C:14](=[O:15])[CH2:16][CH:17]12
CCC(O)CCCCC1CCC2CC(=O)CC12
CCC(=O)CCCCC1CCC2CC(=O)CC12
null
null
C(Cl)Cl
Oxidation
Oxidation or Dehydrogenation of Alcohols to Aldehydes and Ketones
c7c20d2959ac48847b03cc1265962cf99a8ec8a85900c087dabb30077298c66c
767cfd93f5821ebb9e1e72addd9cb404b20b0c821d246ae6b87a5776b74a455b
O=C1CC2CCCC2C1
[C:1]-[C:2]-[CH;D3;+0:3](-[OH;D1;+0:4])-[C:5]-[C;D1;H3:6]>>[C:1]-[C:2]-[C;H0;D3;+0:3](=[O;H0;D1;+0:4])-[C:5]-[C;D1;H3:6]
null
[]
null
null
null
null
The procedure followed is the same as that described in Example 13 substituting the starting material from Example 3, 2-(5-hydroxyhept-1-yl)bicyclo[3.3.0]octan-7-one {hexahydro-4-(5-hydroxyheptyl)-2(1H)-pentalenone} (2.0 g, 8.4 mmoles) and pyridinium dichromate (4.7 g, 12.6 mmoles) in methylene chloride (10 ml). The cr...
10.6084/m9.figshare.5104873.v1
null
Secondary alcohol
Ketone
null
null
C1CC2CCCC2C1
null
C(Cl)Cl
null
null
CCC(O)CCCCC1CCC2CC(=O)CC12>C(Cl)Cl>CCC(=O)CCCCC1CCC2CC(=O)CC12
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-3dd62530494549a98c1c58849b00b4ae
CC(=O)O.CCC(O)CCCCC1CCC2CC(=O)CC12>>CCC(CCCCC1CCC2CC(=O)CC12)OC(C)=O
C(C)(=O)O.OC(CCCCC1C2CC(CC2CC1)=O)CC.OC(CCCCC1C2CC(CC2CC1)=O)CC.OC(CCCCC1C2CC(CC2CC1)=O)CC>>C(C)(=O)OC(CCCCC1C2CC(CC2CC1)=O)CC
[OH:17][C:18]([CH3:19])=[O:20].O[CH:3]([CH2:2][CH3:1])[CH2:4][CH2:5][CH2:6][CH2:7][CH:8]1[CH2:9][CH2:10][CH:11]2[CH2:12][C:13](=[O:14])[CH2:15][CH:16]12>>[CH3:1][CH2:2][CH:3]([CH2:4][CH2:5][CH2:6][CH2:7][CH:8]1[CH2:9][CH2:10][CH:11]2[CH2:12][C:13](=[O:14])[CH2:15][CH:16]12)[O:17][C:18]([CH3:19])=[O:20]
CC(=O)O.CCC(O)CCCCC1CCC2CC(=O)CC12
CCC(CCCCC1CCC2CC(=O)CC12)OC(C)=O
null
null
null
Heteroatom Alkylation and Arylation
Esterification of Carboxylic Acids
55fde8dca0a408407bb776c4e1e9a22d6eeb5c734b0d7975d23baba4292968d2
505f7b4da8def84a80ac616845cb7b0566b14f3232b5b9d3480d84d3e0d284a0
O=C1CC2CCCC2C1
O-[CH;D3;+0:1](-[C:2]-[C;D1;H3:3])-[C:4]-[C:5].[C;D1;H3:6]-[C:7](=[O;D1;H0:8])-[OH;D1;+0:9]>>[C:5]-[C:4]-[CH;D3;+0:1](-[C:2]-[C;D1;H3:3])-[O;H0;D2;+0:9]-[C:7](-[C;D1;H3:6])=[O;D1;H0:8]
null
[]
70
CELSIUS
4
HOUR
The starting material from Example 3, 2-(5-hydroxyhept-1-yl)bicyclo[3.3.0]octan-7-one {hexahydro-4-(5-hydroxyheptyl)-2(1H)-pentalenone} (2.5 g, 10.5 mmoles) is diluted with glacial acetic acid (10 ml) and stirred in a 70° C. water bath for 4 hours. The reaction is cooled to room temperature and partitioned between ethe...
10.6084/m9.figshare.5104873.v1
null
Carboxylic acid.Secondary alcohol
Ester
null
null
C1CC2CCCC2C1
HO-
null
70
4
CC(=O)O.CCC(O)CCCCC1CCC2CC(=O)CC12>>CCC(CCCCC1CCC2CC(=O)CC12)OC(C)=O
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-a562188c5ed14659b721a63cea1485be
CC(=O)O.O=C1CC2CCC(CCCCCO)C2C1>>CC(=O)OCCCCCC1CCC2CC(=O)CC12
C(C)(=O)O.OCCCCCC1C2CC(CC2CC1)=O.OCCCCCC1C2CC(CC2CC1)=O.O>>C(C)(=O)OCCCCCC1C2CC(CC2CC1)=O
[CH3:1][C:2](=[O:3])[OH:4].O[CH2:5][CH2:6][CH2:7][CH2:8][CH2:9][CH:10]1[CH2:11][CH2:12][CH:13]2[CH2:14][C:15](=[O:16])[CH2:17][CH:18]12>>[CH3:1][C:2](=[O:3])[O:4][CH2:5][CH2:6][CH2:7][CH2:8][CH2:9][CH:10]1[CH2:11][CH2:12][CH:13]2[CH2:14][C:15](=[O:16])[CH2:17][CH:18]12
CC(=O)O.O=C1CC2CCC(CCCCCO)C2C1
CC(=O)OCCCCCC1CCC2CC(=O)CC12
null
null
null
Heteroatom Alkylation and Arylation
Esterification of Carboxylic Acids
3f9a9ace480b666da05fcfe5450d12b5c1ea5b0d435c195e1dd4bd20281604bb
dcbf04ec563ed0e9dfc79070490a028958024079a671c385858bb18cc8ec995a
O=C1CC2CCCC2C1
O-[CH2;D2;+0:1]-[C:2]-[C:3].[C;D1;H3:4]-[C:5](=[O;D1;H0:6])-[OH;D1;+0:7]>>[C:3]-[C:2]-[CH2;D2;+0:1]-[O;H0;D2;+0:7]-[C:5](-[C;D1;H3:4])=[O;D1;H0:6]
null
[]
75
CELSIUS
null
null
The starting material 2-(5-hydroxypent-1-yl)bicyclo[3.3.0]octan-7-one {hexahydro-4-(5-hydroxypentyl)-2(1H)-pentalenone} (0.8 g, 3.8 mmoles) is diluted with glacial acetic acid (7 ml). The reaction is stirred and heated in a 75° C. oil bath for 24 hours, after which time water (20 ml) is added and the reaction partition...
10.6084/m9.figshare.5104873.v1
null
Carboxylic acid.Primary alcohol
Ester
null
null
C1CC2CCCC2C1
HO-
null
75
null
CC(=O)O.O=C1CC2CCC(CCCCCO)C2C1>>CC(=O)OCCCCCC1CCC2CC(=O)CC12
ord_dataset-c34472859da14a81bfe0f74e60f15c43
ord-6a2b05eb167f4a6fbf7b18ece3ffb063
CC(C)(C)[Si](C)(C)Cl.CCC(O)CCCl.CCC(O)CCCl.CN(C)C=O.c1c[nH]cn1>>CCC(CCCl)O[Si](C)(C)C(C)(C)C.CCC(CCCl)O[Si](C)(C)CC(C)C
N1C=NC=C1.ClCCC(CC)O.ClCCC(CC)O.CN(C=O)C.[Si](C)(C)(C(C)(C)C)Cl>>ClCCC(O[Si](C)(C)C(C)(C)C)CC.ClCCC(CC)O[Si](C)(C)CC(C)C
Cl[Si:8]([CH3:9])([CH3:10])[C:11]([CH3:12])([CH3:14])[CH3:28].[CH3:1][CH2:2][CH:3]([CH2:4][CH2:5][Cl:6])[OH:7].[CH3:15][CH2:16][CH:17]([CH2:18][CH2:19][Cl:20])[OH:21].O=[CH:25]N([CH3:13])[CH3:24].n1[cH:23][nH][cH:26][cH:27]1>>[CH3:1][CH2:2][CH:3]([CH2:4][CH2:5][Cl:6])[O:7][Si:8]([CH3:9])([CH3:10])[C:11]([CH3:12])([CH3:...
CC(C)(C)[Si](C)(C)Cl.CCC(O)CCCl.CCC(O)CCCl.CN(C)C=O.c1c[nH]cn1
CCC(CCCl)O[Si](C)(C)C(C)(C)C.CCC(CCCl)O[Si](C)(C)CC(C)C
null
null
null
C-C Coupling
OtherReaction
1b5c9e6d22618862c0cf92ff421ed927a52f1a47e9c948a659dea2c61724f3a1
e458a5c983718128b844b37d14f7422d92bf47d4d49e64ffe85804e9f4a928f4
null
Cl-[Si;H0;D4;+0:1](-[C;D1;H3:2])(-[C;D1;H3:3])-[C;H0;D4;+0:4](-[C;D1;H3:5])(-[C;D1;H3:6])-[CH3;D1;+0:7].O=[CH;D2;+0:8]-N(-[CH3;D1;+0:9])-[CH3;D1;+0:10].[C:11]-[C:12](-[C:13])-[OH;D1;+0:14].[C:15]-[C:16](-[C:17])-[OH;D1;+0:18].[cH;D2;+0:19]1:[nH]:[cH;D2;+0:20]:[cH;D2;+0:21]:n:1>>[C:15]-[C:16](-[C:17])-[O;H0;D2;+0:18]-[#...
null
[]
null
null
null
null
The procedure followed is the same as that described in Example 7 substituting 5-chloropentan-3-ol {1-chloro-3-pentanol} (50 g, 0.41 moles), tert-butyldimethylsilyl chloride (71g, 0.47 moles), imidazole (32.6 g, 0.48 moles), and dimethylformamide (150 ml). The crude product is fractionally distilled under vacuum leavin...
10.6084/m9.figshare.5104873.v1
null
Tertiary amide.Secondary alcohol.Secondary alcohol.Silyl protective group
TMS ether protective group.Silyl protective group
c1c[nH]cn1
null
null
Other
null
null
null
CC(C)(C)[Si](C)(C)Cl.CCC(O)CCCl.CCC(O)CCCl.CN(C)C=O.c1c[nH]cn1>>CCC(CCCl)O[Si](C)(C)C(C)(C)C.CCC(CCCl)O[Si](C)(C)CC(C)C