drug
stringlengths
3
199
prompt
stringlengths
45
281
solution
stringclasses
2 values
problem_type
stringclasses
5 values
index
int64
1
1.8k
COc1ccc(-n2c(=O)c(C)nc3cnc(N4CCNCC4)nc32)cc1
Given the following SMILES string, predict whether the compound inhibits CYP2C19? COc1ccc(-n2c(=O)c(C)nc3cnc(N4CCNCC4)nc32)cc1
No
single_pred_adme_cyp2c19
101
CNC1C(O)C(NC)C2OC3(O)C(=O)CC(C)OC3OC2C1O
Does the following compound cause drug-induced liver injury (DILI)? CNC1C(O)C(NC)C2OC3(O)C(=O)CC(C)OC3OC2C1O
No
single_pred_tox_dili
102
C=CCSC1=Nc2sccc2C2=NC(=O)CN12
Given the following SMILES string, predict whether the compound inhibits CYP2C19? C=CCSC1=Nc2sccc2C2=NC(=O)CN12
Yes
single_pred_adme_cyp2c19
103
CCN(CC)c1ccc([N+]#N)cc1
Is the following compound AMES mutagenic? CCN(CC)c1ccc([N+]#N)cc1
Yes
single_pred_tox_ames
104
CC(C)(C)NC(=O)C1CC2CCCCC2CN1CC(O)C(Cc1ccccc1)NC(=O)C(CC(N)=O)NC(=O)c1ccc2ccccc2n1
Does the following compound cause drug-induced liver injury (DILI)? CC(C)(C)NC(=O)C1CC2CCCCC2CN1CC(O)C(Cc1ccccc1)NC(=O)C(CC(N)=O)NC(=O)c1ccc2ccccc2n1
Yes
single_pred_tox_dili
105
C[NH2+]CCC=C1c2ccccc2CCc2ccccc21
Does the following compound block the hERG channel? C[NH2+]CCC=C1c2ccccc2CCc2ccccc21
Yes
single_pred_tox_herg
106
COc1cc2c(cc1OC)-c1cc3ccc(OC)c(OC)c3c[n+]1CC2
Given the following SMILES string, predict whether the compound inhibits CYP2C19? COc1cc2c(cc1OC)-c1cc3ccc(OC)c(OC)c3c[n+]1CC2
No
single_pred_adme_cyp2c19
107
CN1C(=O)/C(=C\c2ccccc2)Sc2ccc(C(=O)N3CCN(c4ccccn4)CC3)cc21
Given the following SMILES string, predict whether the compound inhibits CYP2C19? CN1C(=O)/C(=C\c2ccccc2)Sc2ccc(C(=O)N3CCN(c4ccccn4)CC3)cc21
Yes
single_pred_adme_cyp2c19
108
CC(C)C(=O)NCCc1nc2ccccc2n1CCCOc1ccc(Cl)cc1
Given the following SMILES string, predict whether the compound inhibits CYP2C19? CC(C)C(=O)NCCc1nc2ccccc2n1CCCOc1ccc(Cl)cc1
Yes
single_pred_adme_cyp2c19
109
CC(C)(C)c1cc(Cc2cc(C(C)(C)C)c(O)c(C(C)(C)C)c2)cc(C(C)(C)C)c1O
Is the following compound AMES mutagenic? CC(C)(C)c1cc(Cc2cc(C(C)(C)C)c(O)c(C(C)(C)C)c2)cc(C(C)(C)C)c1O
No
single_pred_tox_ames
110
CN(CCc1ccccn1)Cc1ccc(Cl)cc1Cl
Given the following SMILES string, predict whether the compound inhibits CYP2C19? CN(CCc1ccccn1)Cc1ccc(Cl)cc1Cl
Yes
single_pred_adme_cyp2c19
111
CCOC(=O)c1ncn2c1CN(C)C(=O)c1cc(F)ccc1-2
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? CCOC(=O)c1ncn2c1CN(C)C(=O)c1cc(F)ccc1-2
No
single_pred_adme_pgp
112
NS(=O)(=O)Cc1noc2ccccc12
Does the following compound cause drug-induced liver injury (DILI)? NS(=O)(=O)Cc1noc2ccccc12
Yes
single_pred_tox_dili
113
CN1Cc2c(N)cccc2C(c2ccccc2)C1
Does the following compound cause drug-induced liver injury (DILI)? CN1Cc2c(N)cccc2C(c2ccccc2)C1
Yes
single_pred_tox_dili
114
C[C@H]1Sc2c(C(=O)O)c(=O)c3cc(F)c(N4CCNCC4)cc3n21
Does the following compound block the hERG channel? C[C@H]1Sc2c(C(=O)O)c(=O)c3cc(F)c(N4CCNCC4)cc3n21
No
single_pred_tox_herg
115
CC(O)C(=O)Nc1c(I)c(C(=O)NC(CO)CO)c(I)c(C(=O)NC(CO)CO)c1I
Does the following compound cause drug-induced liver injury (DILI)? CC(O)C(=O)Nc1c(I)c(C(=O)NC(CO)CO)c(I)c(C(=O)NC(CO)CO)c1I
No
single_pred_tox_dili
116
C1CCN2C[C@H]3C[C@@H](CN4CCCC[C@H]34)[C@H]2C1
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? C1CCN2C[C@H]3C[C@@H](CN4CCCC[C@H]34)[C@H]2C1
No
single_pred_adme_pgp
117
O=C(Cc1ccccc1)N/N=C/c1ccccc1OCc1ccc(Cl)cc1
Given the following SMILES string, predict whether the compound inhibits CYP2C19? O=C(Cc1ccccc1)N/N=C/c1ccccc1OCc1ccc(Cl)cc1
Yes
single_pred_adme_cyp2c19
118
c1ccc(OCC2CO2)cc1
Is the following compound AMES mutagenic? c1ccc(OCC2CO2)cc1
Yes
single_pred_tox_ames
119
CNC(=O)Oc1cc2ccccc2c2ccccc12
Is the following compound AMES mutagenic? CNC(=O)Oc1cc2ccccc2c2ccccc12
Yes
single_pred_tox_ames
120
CCN1C[C@]2(C)CC[C@H](OC)[C@]34[C@H]1[C@]1(OCO[C@@]15C[C@H](OC)[C@H]1C[C@]3(O)[C@]5(O)[C@@H]1OC)[C@H](C(C)=O)[C@@H]42
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? CCN1C[C@]2(C)CC[C@H](OC)[C@]34[C@H]1[C@]1(OCO[C@@]15C[C@H](OC)[C@H]1C[C@]3(O)[C@]5(O)[C@@H]1OC)[C@H](C(C)=O)[C@@H]42
No
single_pred_adme_pgp
121
CCN(CC(=O)O)CC(=O)O
Given the following SMILES string, predict whether the compound inhibits CYP2C19? CCN(CC(=O)O)CC(=O)O
No
single_pred_adme_cyp2c19
122
CC(C=CC1=C(C)CCCC1(C)C)=CC=CC(C)=CCO
Does the following compound cause drug-induced liver injury (DILI)? CC(C=CC1=C(C)CCCC1(C)C)=CC=CC(C)=CCO
No
single_pred_tox_dili
123
COc1cc2c(cc1O)C[C@H]1c3c(cc(O)c(OC)c3-2)CCN1C
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? COc1cc2c(cc1O)C[C@H]1c3c(cc(O)c(OC)c3-2)CCN1C
No
single_pred_adme_pgp
124
CNc1ccc2ccc3ccc(O)cc3c2c1
Is the following compound AMES mutagenic? CNc1ccc2ccc3ccc(O)cc3c2c1
Yes
single_pred_tox_ames
125
CN(C)NC(=O)CCC(=O)O
Is the following compound AMES mutagenic? CN(C)NC(=O)CCC(=O)O
No
single_pred_tox_ames
126
Nc1ncnc2c1ncn2[C@H]1O[C@H](CO)[C@H](O)[C@H]1O
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? Nc1ncnc2c1ncn2[C@H]1O[C@H](CO)[C@H](O)[C@H]1O
No
single_pred_adme_pgp
127
CC[C@H](CO)NC(=O)[C@@H]1C=C2c3cccc4[nH]cc(c34)C[C@H]2N(C)C1
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? CC[C@H](CO)NC(=O)[C@@H]1C=C2c3cccc4[nH]cc(c34)C[C@H]2N(C)C1
No
single_pred_adme_pgp
128
CC(C)NC[C@H](O)c1cc(O)cc(O)c1
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? CC(C)NC[C@H](O)c1cc(O)cc(O)c1
No
single_pred_adme_pgp
129
CC(=O)CCl
Is the following compound AMES mutagenic? CC(=O)CCl
No
single_pred_tox_ames
130
CCn1nc(C(=O)O)c(=O)c2cc3c(cc21)OCO3
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? CCn1nc(C(=O)O)c(=O)c2cc3c(cc21)OCO3
No
single_pred_adme_pgp
131
CC(C)(C(=O)O)c1ccc([C@H](O)CCCN2CCC(C(O)(c3ccccc3)c3ccccc3)CC2)cc1
Does the following compound block the hERG channel? CC(C)(C(=O)O)c1ccc([C@H](O)CCCN2CCC(C(O)(c3ccccc3)c3ccccc3)CC2)cc1
Yes
single_pred_tox_herg
132
CN1CCC23c4c5ccc(O)c4OC2C(O)C=CC3C1C5
Does the following compound cause drug-induced liver injury (DILI)? CN1CCC23c4c5ccc(O)c4OC2C(O)C=CC3C1C5
No
single_pred_tox_dili
133
O=C1c2ccccc2C(=O)c2c(NC3CCCCC3)ccc(Nc3ccc(S(=O)(=O)O)cc3)c21
Given the following SMILES string, predict whether the compound inhibits CYP2C19? O=C1c2ccccc2C(=O)c2c(NC3CCCCC3)ccc(Nc3ccc(S(=O)(=O)O)cc3)c21
Yes
single_pred_adme_cyp2c19
134
CC(C)N=c1cc2n(-c3ccc(Cl)cc3)c3ccccc3nc-2cc1Nc1ccc(Cl)cc1
Given the following SMILES string, predict whether the compound inhibits CYP2C19? CC(C)N=c1cc2n(-c3ccc(Cl)cc3)c3ccccc3nc-2cc1Nc1ccc(Cl)cc1
No
single_pred_adme_cyp2c19
135
OCCN(CCO)c1nc(N2CCOCC2)c2nc(N(CCO)CCO)nc(N3CCOCC3)c2n1
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? OCCN(CCO)c1nc(N2CCOCC2)c2nc(N(CCO)CCO)nc(N3CCOCC3)c2n1
No
single_pred_adme_pgp
136
C[NH+](C)CCOC(c1ccccc1)c1ccccc1
Does the following compound block the hERG channel? C[NH+](C)CCOC(c1ccccc1)c1ccccc1
Yes
single_pred_tox_herg
137
COc1cc2c(c(OC)c1OC)-c1ccc(OC)c(=O)cc1C(NC(C)=O)CC2
Does the following compound cause drug-induced liver injury (DILI)? COc1cc2c(c(OC)c1OC)-c1ccc(OC)c(=O)cc1C(NC(C)=O)CC2
No
single_pred_tox_dili
138
C#CCSc1n[nH]c(-c2ccco2)n1
Does the following compound block the hERG channel? C#CCSc1n[nH]c(-c2ccco2)n1
No
single_pred_tox_herg
139
COc1cc2c(cc1OC)C(C(=O)Nc1ccc3c(c1)OCCO3)C(c1cccnc1)N(C)C2=O
Given the following SMILES string, predict whether the compound inhibits CYP2C19? COc1cc2c(cc1OC)C(C(=O)Nc1ccc3c(c1)OCCO3)C(c1cccnc1)N(C)C2=O
No
single_pred_adme_cyp2c19
140
Cc1noc(C)c1-c1ccc2ncnc(N(C)C)c2c1
Given the following SMILES string, predict whether the compound inhibits CYP2C19? Cc1noc(C)c1-c1ccc2ncnc(N(C)C)c2c1
Yes
single_pred_adme_cyp2c19
141
COc1ccc(CCN(C)CCCN(C(=O)c2ccc([N+](=O)[O-])cc2)c2ccc(OC)c(OC)c2)cc1OC
Does the following compound block the hERG channel? COc1ccc(CCN(C)CCCN(C(=O)c2ccc([N+](=O)[O-])cc2)c2ccc(OC)c(OC)c2)cc1OC
Yes
single_pred_tox_herg
142
CNCCC(Oc1cccc2ccccc12)c1cccs1
Does the following compound cause drug-induced liver injury (DILI)? CNCCC(Oc1cccc2ccccc12)c1cccs1
Yes
single_pred_tox_dili
143
CC(=O)c1c(C)cc(C)c(CSc2nc3ccc(NC(=O)c4cccc5ccccc45)cc3s2)c1C
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? CC(=O)c1c(C)cc(C)c(CSc2nc3ccc(NC(=O)c4cccc5ccccc45)cc3s2)c1C
Yes
single_pred_adme_pgp
144
C=Cc1ccc(C)cc1
Is the following compound AMES mutagenic? C=Cc1ccc(C)cc1
No
single_pred_tox_ames
145
COc1cc(C[C@@H]2NCCc3cc(O)c(O)cc32)cc(OC)c1OC
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? COc1cc(C[C@@H]2NCCc3cc(O)c(O)cc32)cc(OC)c1OC
No
single_pred_adme_pgp
146
NC(=O)c1cnccn1
Is the following compound AMES mutagenic? NC(=O)c1cnccn1
No
single_pred_tox_ames
147
c1ccc2c(c1)cc([C@@H]1CO1)c1ccccc12
Is the following compound AMES mutagenic? c1ccc2c(c1)cc([C@@H]1CO1)c1ccccc12
Yes
single_pred_tox_ames
148
O=C1NCCN1CC[NH+]1CCC(c2cn(-c3ccccc3)c3ccc(Cl)cc23)CC1
Does the following compound block the hERG channel? O=C1NCCN1CC[NH+]1CCC(c2cn(-c3ccccc3)c3ccc(Cl)cc23)CC1
No
single_pred_tox_herg
149
CO/N=C(/C(=O)N[C@H]1C(=O)N2C(C(=O)O)=C(COC(C)=O)CS[C@@H]12)c1csc(N)n1
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? CO/N=C(/C(=O)N[C@H]1C(=O)N2C(C(=O)O)=C(COC(C)=O)CS[C@@H]12)c1csc(N)n1
Yes
single_pred_adme_pgp
150
CC1=CC(=O)CC(C)(C)C1
Is the following compound AMES mutagenic? CC1=CC(=O)CC(C)(C)C1
No
single_pred_tox_ames
151
OCC(S)CS
Does the following compound cause drug-induced liver injury (DILI)? OCC(S)CS
Yes
single_pred_tox_dili
152
NCCNC[C@@H](O)CO
Does the following compound block the hERG channel? NCCNC[C@@H](O)CO
No
single_pred_tox_herg
153
O[C@H](CNC[C@@H](O)[C@H]1CCc2cc(F)ccc2O1)[C@H]1CCc2cc(F)ccc2O1
Does the following compound block the hERG channel? O[C@H](CNC[C@@H](O)[C@H]1CCc2cc(F)ccc2O1)[C@H]1CCc2cc(F)ccc2O1
Yes
single_pred_tox_herg
154
CCN=[N+](C)[O-]
Is the following compound AMES mutagenic? CCN=[N+](C)[O-]
No
single_pred_tox_ames
155
N/C(=N\O)c1cn([C@@H]2O[C@@H](CO)[C@H](O)[C@@H]2O)c2ncnc(NO)c12
Given the following SMILES string, predict whether the compound inhibits CYP2C19? N/C(=N\O)c1cn([C@@H]2O[C@@H](CO)[C@H](O)[C@@H]2O)c2ncnc(NO)c12
No
single_pred_adme_cyp2c19
156
COc1ccc(C2Sc3ccccc3N(CCN(C)C)C(=O)C2OC(C)=O)cc1
Does the following compound cause drug-induced liver injury (DILI)? COc1ccc(C2Sc3ccccc3N(CCN(C)C)C(=O)C2OC(C)=O)cc1
Yes
single_pred_tox_dili
157
O=c1[nH]c2ccccc2n1C1CCN(CCCC(c2ccc(F)cc2)c2ccc(F)cc2)CC1
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? O=c1[nH]c2ccccc2n1C1CCN(CCCC(c2ccc(F)cc2)c2ccc(F)cc2)CC1
Yes
single_pred_adme_pgp
158
CN1c2ccccc2C(NCCCCCCC(=O)O)c2ccc(Cl)cc2S1(=O)=O
Does the following compound cause drug-induced liver injury (DILI)? CN1c2ccccc2C(NCCCCCCC(=O)O)c2ccc(Cl)cc2S1(=O)=O
Yes
single_pred_tox_dili
159
CC1CCC(=C(C#N)C(=O)Nc2cccc(Cl)c2)CC1
Given the following SMILES string, predict whether the compound inhibits CYP2C19? CC1CCC(=C(C#N)C(=O)Nc2cccc(Cl)c2)CC1
Yes
single_pred_adme_cyp2c19
160
COc1ccc(NC(=O)CCNS(=O)(=O)c2ccc3c(c2)c(=O)n(C)c(=O)n3C)cc1
Given the following SMILES string, predict whether the compound inhibits CYP2C19? COc1ccc(NC(=O)CCNS(=O)(=O)c2ccc3c(c2)c(=O)n(C)c(=O)n3C)cc1
No
single_pred_adme_cyp2c19
161
N#CC(=N)C(N)C#N
Is the following compound AMES mutagenic? N#CC(=N)C(N)C#N
No
single_pred_tox_ames
162
CC(C)=CCCC(C)CC=O
Is the following compound AMES mutagenic? CC(C)=CCCC(C)CC=O
No
single_pred_tox_ames
163
CN1CCN(CCCNC(=O)c2ccc(CSCc3cccc(Cl)c3)o2)CC1
Given the following SMILES string, predict whether the compound inhibits CYP2C19? CN1CCN(CCCNC(=O)c2ccc(CSCc3cccc(Cl)c3)o2)CC1
No
single_pred_adme_cyp2c19
164
CCCCCCCCCCCC(CC1OC(=O)C1CCCCCC)OC(=O)C(CC(C)C)NC=O
Does the following compound cause drug-induced liver injury (DILI)? CCCCCCCCCCCC(CC1OC(=O)C1CCCCCC)OC(=O)C(CC(C)C)NC=O
Yes
single_pred_tox_dili
165
CC(C)(C)c1cccc(Oc2nn[nH]n2)c1
Given the following SMILES string, predict whether the compound inhibits CYP2C19? CC(C)(C)c1cccc(Oc2nn[nH]n2)c1
Yes
single_pred_adme_cyp2c19
166
CC(C)CC1NC(=O)C(Cc2ccccc2)NC(=O)C(CCN)NC(=O)C(NC(=O)C(CCN)NC(=O)C(NC(=O)C(CCN)NC(=O)O)C(C)O)CCNC(=O)C(C(C)O)NC(=O)C(CCN)NC(=O)C(CCN)NC1=O
Does the following compound cause drug-induced liver injury (DILI)? CC(C)CC1NC(=O)C(Cc2ccccc2)NC(=O)C(CCN)NC(=O)C(NC(=O)C(CCN)NC(=O)C(NC(=O)C(CCN)NC(=O)O)C(C)O)CCNC(=O)C(C(C)O)NC(=O)C(CCN)NC(=O)C(CCN)NC1=O
No
single_pred_tox_dili
167
CNc1ccc2ncc(C)nc2c1N
Is the following compound AMES mutagenic? CNc1ccc2ncc(C)nc2c1N
No
single_pred_tox_ames
168
Cc1ccc(/C(=C\CN2CCCC2)c2cccc(/C=C/C(=O)O)n2)cc1
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? Cc1ccc(/C(=C\CN2CCCC2)c2cccc(/C=C/C(=O)O)n2)cc1
No
single_pred_adme_pgp
169
COc1ccc(C[NH2+]CC(O)COc2ccc3[nH]c(=O)ccc3c2)cc1OC
Does the following compound block the hERG channel? COc1ccc(C[NH2+]CC(O)COc2ccc3[nH]c(=O)ccc3c2)cc1OC
Yes
single_pred_tox_herg
170
N[C@H](CNO)C(=O)O
Does the following compound block the hERG channel? N[C@H](CNO)C(=O)O
No
single_pred_tox_herg
171
CC(C)(C#N)N=NC(C)(C)C#N
Is the following compound AMES mutagenic? CC(C)(C#N)N=NC(C)(C)C#N
No
single_pred_tox_ames
172
Nc1nc2ccc(OC(F)(F)F)cc2s1
Does the following compound cause drug-induced liver injury (DILI)? Nc1nc2ccc(OC(F)(F)F)cc2s1
Yes
single_pred_tox_dili
173
Cc1ccc(NCC2(O)OCC(O)C(O)C2O)cc1
Is the following compound AMES mutagenic? Cc1ccc(NCC2(O)OCC(O)C(O)C2O)cc1
No
single_pred_tox_ames
174
CCC(=O)c1ccc(OCc2ccc(C(=O)OC)cc2)c(OC)c1
Given the following SMILES string, predict whether the compound inhibits CYP2C19? CCC(=O)c1ccc(OCc2ccc(C(=O)OC)cc2)c(OC)c1
Yes
single_pred_adme_cyp2c19
175
CC(C)N=C=NC(C)C
Is the following compound AMES mutagenic? CC(C)N=C=NC(C)C
No
single_pred_tox_ames
176
O=c1cnc2cnc(Oc3ccccc3)nc2n1CCc1ccccc1
Given the following SMILES string, predict whether the compound inhibits CYP2C19? O=c1cnc2cnc(Oc3ccccc3)nc2n1CCc1ccccc1
Yes
single_pred_adme_cyp2c19
177
CCNc1ncc2nc(CCc3ccccc3)c(=O)n(Cc3cccc(OC)c3)c2n1
Given the following SMILES string, predict whether the compound inhibits CYP2C19? CCNc1ncc2nc(CCc3ccccc3)c(=O)n(Cc3cccc(OC)c3)c2n1
Yes
single_pred_adme_cyp2c19
178
CCc1c(C)[nH]c2c1/C(=N/NC(=O)Nc1ccccc1)CCC2
Does the following compound block the hERG channel? CCc1c(C)[nH]c2c1/C(=N/NC(=O)Nc1ccccc1)CCC2
Yes
single_pred_tox_herg
179
O[C@@H](COc1cccc2ncccc12)CN1CCN(C2c3ccccc3C3C(c4ccccc42)C3(F)F)CC1
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? O[C@@H](COc1cccc2ncccc12)CN1CCN(C2c3ccccc3C3C(c4ccccc42)C3(F)F)CC1
Yes
single_pred_adme_pgp
180
CC(=O)Oc1ccc(C(=C2CCCCC2)c2ccc(OC(C)=O)cc2)cc1
Does the following compound cause drug-induced liver injury (DILI)? CC(=O)Oc1ccc(C(=C2CCCCC2)c2ccc(OC(C)=O)cc2)cc1
Yes
single_pred_tox_dili
181
C[C@@H](N)CN
Is the following compound AMES mutagenic? C[C@@H](N)CN
No
single_pred_tox_ames
182
COc1ccc(CN(CCN(C)C)c2ccccn2)cc1
Does the following compound cause drug-induced liver injury (DILI)? COc1ccc(CN(CCN(C)C)c2ccccn2)cc1
No
single_pred_tox_dili
183
COc1ccc2c3c1OC1C(=O)CCC4C(C2)N(C)CCC314
Does the following compound cause drug-induced liver injury (DILI)? COc1ccc2c3c1OC1C(=O)CCC4C(C2)N(C)CCC314
No
single_pred_tox_dili
184
NS(=O)(=O)c1cc(C(=O)O)c(NCc2ccco2)cc1Cl
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? NS(=O)(=O)c1cc(C(=O)O)c(NCc2ccco2)cc1Cl
No
single_pred_adme_pgp
185
CC(C)C(=O)Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1
Does the following compound cause drug-induced liver injury (DILI)? CC(C)C(=O)Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1
Yes
single_pred_tox_dili
186
NC(=O)c1cnccn1
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? NC(=O)c1cnccn1
No
single_pred_adme_pgp
187
N/C(=N\O)c1ccccc1
Is the following compound AMES mutagenic? N/C(=N\O)c1ccccc1
Yes
single_pred_tox_ames
188
COc1cccc2c1C(=O)c1c(O)c3c(c(O)c1C2=O)C[C@](O)(C(=O)CO)C[C@@H]3O[C@H]1C[C@@H](N)[C@H](O)[C@@H](C)O1
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? COc1cccc2c1C(=O)c1c(O)c3c(c(O)c1C2=O)C[C@](O)(C(=O)CO)C[C@@H]3O[C@H]1C[C@@H](N)[C@H](O)[C@@H](C)O1
No
single_pred_adme_pgp
189
CCC(CCC(C)=O)COC(=O)CCCCC(=O)O
Is the following compound AMES mutagenic? CCC(CCC(C)=O)COC(=O)CCCCC(=O)O
No
single_pred_tox_ames
190
Nc1c2c(nc3ccccc13)CCCC2
Does the following compound block the hERG channel? Nc1c2c(nc3ccccc13)CCCC2
No
single_pred_tox_herg
191
N#Cc1c2n(c3c(NS(=O)(=O)Cc4ccccc4)ncnc13)CCCC2
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? N#Cc1c2n(c3c(NS(=O)(=O)Cc4ccccc4)ncnc13)CCCC2
Yes
single_pred_adme_pgp
192
CN1CCN(CCCN(C(=O)Nc2ccc(F)c(C(F)(F)F)c2)[C@@H]2C[C@@H](c3ccc4c(c3)[C@H](N)NO4)[C@@H]3C[C@H]32)CC1
Does the following compound block the hERG channel? CN1CCN(CCCN(C(=O)Nc2ccc(F)c(C(F)(F)F)c2)[C@@H]2C[C@@H](c3ccc4c(c3)[C@H](N)NO4)[C@@H]3C[C@H]32)CC1
Yes
single_pred_tox_herg
193
CC1C=CC=CCCC=CC=CC=CC=CC(OC2OC(C)C(O)C(N)C2O)CC(O)C(C(=O)O)C(O)CC(=O)CC(O)C(O)CCC(O)CC(O)CC(O)CC(=O)OC(C)C(C)C1O
Does the following compound cause drug-induced liver injury (DILI)? CC1C=CC=CCCC=CC=CC=CC=CC(OC2OC(C)C(O)C(N)C2O)CC(O)C(C(=O)O)C(O)CC(=O)CC(O)C(O)CCC(O)CC(O)CC(O)CC(=O)OC(C)C(C)C1O
No
single_pred_tox_dili
194
N#Cc1ccc(C(c2ccc(C#N)cc2)n2cncn2)cc1
Does the following compound block the hERG channel? N#Cc1ccc(C(c2ccc(C#N)cc2)n2cncn2)cc1
No
single_pred_tox_herg
195
COc1cccc(/C(O)=C2/C(=O)C(=O)N(c3cc(C)on3)C2c2cccs2)c1
Given the following SMILES string, predict whether the compound inhibits CYP2C19? COc1cccc(/C(O)=C2/C(=O)C(=O)N(c3cc(C)on3)C2c2cccs2)c1
No
single_pred_adme_cyp2c19
196
Cc1cccc(N(NC(=O)C(C)(C)O)C(=O)c2ccccc2)c1
Given the following SMILES string, predict whether the compound inhibits CYP2C19? Cc1cccc(N(NC(=O)C(C)(C)O)C(=O)c2ccccc2)c1
Yes
single_pred_adme_cyp2c19
197
Cc1ccc(N)c(O)c1
Is the following compound AMES mutagenic? Cc1ccc(N)c(O)c1
Yes
single_pred_tox_ames
198
CC(C)COC[C@@H](CN(Cc1ccccc1)c1ccccc1)[NH+]1CCCC1
Does the following compound block the hERG channel? CC(C)COC[C@@H](CN(Cc1ccccc1)c1ccccc1)[NH+]1CCCC1
Yes
single_pred_tox_herg
199
COc1cccc(CCN2CCN(c3ncnc4c(C#N)c5n(c34)CCCC5)CC2)c1
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? COc1cccc(CCN2CCN(c3ncnc4c(C#N)c5n(c34)CCCC5)CC2)c1
Yes
single_pred_adme_pgp
200