drug
stringlengths
3
199
prompt
stringlengths
45
281
solution
stringclasses
2 values
problem_type
stringclasses
5 values
index
int64
1
1.8k
CC1(C)O[C@@H]2C[C@@H]3[C@H]4C[C@@H](F)C5=CC(=O)C=C[C@@]5(C)[C@@H]4[C@@H](O)C[C@]3(C)[C@@]2(C(=O)CO)O1
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? CC1(C)O[C@@H]2C[C@@H]3[C@H]4C[C@@H](F)C5=CC(=O)C=C[C@@]5(C)[C@@H]4[C@@H](O)C[C@]3(C)[C@@]2(C(=O)CO)O1
No
single_pred_adme_pgp
201
FC(F)(F)c1cc(NC(=S)N2c3ccccc3-n3cccc3[C@H]2c2cccnc2)cc(C(F)(F)F)c1
Given the following SMILES string, predict whether the compound inhibits CYP2C19? FC(F)(F)c1cc(NC(=S)N2c3ccccc3-n3cccc3[C@H]2c2cccnc2)cc(C(F)(F)F)c1
No
single_pred_adme_cyp2c19
202
Cc1ncc([N+](=O)[O-])n1C[C@H](O)CCl
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? Cc1ncc([N+](=O)[O-])n1C[C@H](O)CCl
No
single_pred_adme_pgp
203
Cc1nnc(C(C)C)n1C1C[C@@H]2CC[C@H](C1)N2CC[C@H](NC(=O)C1CCC(F)(F)CC1)c1ccccc1
Does the following compound block the hERG channel? Cc1nnc(C(C)C)n1C1C[C@@H]2CC[C@H](C1)N2CC[C@H](NC(=O)C1CCC(F)(F)CC1)c1ccccc1
No
single_pred_tox_herg
204
NC(=O)N1c2ccccc2C=Cc2ccccc21
Does the following compound cause drug-induced liver injury (DILI)? NC(=O)N1c2ccccc2C=Cc2ccccc21
Yes
single_pred_tox_dili
205
Clc1ccc(C2=CCC[C@H]3CC[C@@H]2N3)cn1
Given the following SMILES string, predict whether the compound inhibits CYP2C19? Clc1ccc(C2=CCC[C@H]3CC[C@@H]2N3)cn1
No
single_pred_adme_cyp2c19
206
OCc1ccc2cccc3c2c1-c1ccccc1-3
Is the following compound AMES mutagenic? OCc1ccc2cccc3c2c1-c1ccccc1-3
No
single_pred_tox_ames
207
ClC(Cl)=C(c1ccc(Cl)cc1)c1ccc(Cl)cc1
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? ClC(Cl)=C(c1ccc(Cl)cc1)c1ccc(Cl)cc1
No
single_pred_adme_pgp
208
O=C(COc1ccc2ccccc2c1Br)NNC(=O)Nc1ccccc1
Given the following SMILES string, predict whether the compound inhibits CYP2C19? O=C(COc1ccc2ccccc2c1Br)NNC(=O)Nc1ccccc1
Yes
single_pred_adme_cyp2c19
209
CC(C(=O)O)c1cccc(Oc2ccccc2)c1
Does the following compound cause drug-induced liver injury (DILI)? CC(C(=O)O)c1cccc(Oc2ccccc2)c1
Yes
single_pred_tox_dili
210
NC(=O)CI
Is the following compound AMES mutagenic? NC(=O)CI
No
single_pred_tox_ames
211
[N-]=[N+]=NCC(O)C(O)C(O)C(O)C=O
Is the following compound AMES mutagenic? [N-]=[N+]=NCC(O)C(O)C(O)C(O)C=O
Yes
single_pred_tox_ames
212
CC1CCC(NC(=O)N(CCCl)N=O)CC1
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? CC1CCC(NC(=O)N(CCCl)N=O)CC1
No
single_pred_adme_pgp
213
C[NH+](C)CCC1C=Nc2ccc(Cn3cncn3)cc21
Does the following compound block the hERG channel? C[NH+](C)CCC1C=Nc2ccc(Cn3cncn3)cc21
No
single_pred_tox_herg
214
O=[N+]([O-])c1cc(F)ccc1F
Is the following compound AMES mutagenic? O=[N+]([O-])c1cc(F)ccc1F
Yes
single_pred_tox_ames
215
CCC[NH+](CCC)CCc1cccc2c1CC(=O)N2
Does the following compound block the hERG channel? CCC[NH+](CCC)CCc1cccc2c1CC(=O)N2
No
single_pred_tox_herg
216
CN(C)CCN(C)C
Is the following compound AMES mutagenic? CN(C)CCN(C)C
No
single_pred_tox_ames
217
COC(=O)C1=CO[C@H](C)[C@@H]2CN3CCc4c([nH]c5ccccc45)[C@@H]3C[C@@H]12
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? COC(=O)C1=CO[C@H](C)[C@@H]2CN3CCc4c([nH]c5ccccc45)[C@@H]3C[C@@H]12
No
single_pred_adme_pgp
218
Nc1c(CC(=O)O)cccc1C(=O)c1ccc(Br)cc1
Does the following compound cause drug-induced liver injury (DILI)? Nc1c(CC(=O)O)cccc1C(=O)c1ccc(Br)cc1
Yes
single_pred_tox_dili
219
COc1cc(Cc2cnc(N)nc2N)cc(OC)c1OC
Does the following compound block the hERG channel? COc1cc(Cc2cnc(N)nc2N)cc(OC)c1OC
No
single_pred_tox_herg
220
O=C1CN(CCc2ccc(F)cc2)CCN1[C@H]1CCc2cc(Cn3ccnc3)ccc2C1
Does the following compound block the hERG channel? O=C1CN(CCc2ccc(F)cc2)CCN1[C@H]1CCc2cc(Cn3ccnc3)ccc2C1
Yes
single_pred_tox_herg
221
CC(C)n1c(C=CC(O)CC(O)CC(=O)O)c(-c2ccc(F)cc2)c2ccccc21
Does the following compound cause drug-induced liver injury (DILI)? CC(C)n1c(C=CC(O)CC(O)CC(=O)O)c(-c2ccc(F)cc2)c2ccccc21
No
single_pred_tox_dili
222
COc1cccc2c1C(=O)c1c(O)c3c(c(O)c1C2=O)CC(O)(C(=O)CO)CC3OC1CC(N)C(O)C(C)O1
Does the following compound cause drug-induced liver injury (DILI)? COc1cccc2c1C(=O)c1c(O)c3c(c(O)c1C2=O)CC(O)(C(=O)CO)CC3OC1CC(N)C(O)C(C)O1
Yes
single_pred_tox_dili
223
O=C(NC1CCN(Cc2cc3c(cc2Cl)OCO3)CC1)c1cc(=O)c2ccc(F)cc2o1
Does the following compound block the hERG channel? O=C(NC1CCN(Cc2cc3c(cc2Cl)OCO3)CC1)c1cc(=O)c2ccc(F)cc2o1
Yes
single_pred_tox_herg
224
C1=CC2CCCCC2c2ccccc21
Is the following compound AMES mutagenic? C1=CC2CCCCC2c2ccccc21
Yes
single_pred_tox_ames
225
CC(=O)Nc1ccc(Nc2ccc([N+](=O)[O-])cc2)cc1
Is the following compound AMES mutagenic? CC(=O)Nc1ccc(Nc2ccc([N+](=O)[O-])cc2)cc1
Yes
single_pred_tox_ames
226
O=c1n(-c2ccccc2)c(=O)n2n1CC[C@H]1/C(=N\OCc3ccccc3)[C@H]3O[C@@H]3[C@@H](O)[C@@H]12
Given the following SMILES string, predict whether the compound inhibits CYP2C19? O=c1n(-c2ccccc2)c(=O)n2n1CC[C@H]1/C(=N\OCc3ccccc3)[C@H]3O[C@@H]3[C@@H](O)[C@@H]12
No
single_pred_adme_cyp2c19
227
Cc1oc(=O)oc1CN1CCN(c2cc3c(cc2F)c(=O)c(C(=O)O)c2n3[C@@H](C)S2)CC1
Does the following compound block the hERG channel? Cc1oc(=O)oc1CN1CCN(c2cc3c(cc2F)c(=O)c(C(=O)O)c2n3[C@@H](C)S2)CC1
No
single_pred_tox_herg
228
Cc1cccc(C)c1NC1=NCCCS1
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? Cc1cccc(C)c1NC1=NCCCS1
No
single_pred_adme_pgp
229
CC1=CC(=O)c2ccccc2C1=O
Is the following compound AMES mutagenic? CC1=CC(=O)c2ccccc2C1=O
Yes
single_pred_tox_ames
230
CSc1ncnc2c1ncn2[C@@H]1O[C@@H](CO)[C@H](O)O[C@@H]1O
Given the following SMILES string, predict whether the compound inhibits CYP2C19? CSc1ncnc2c1ncn2[C@@H]1O[C@@H](CO)[C@H](O)O[C@@H]1O
No
single_pred_adme_cyp2c19
231
CC[C@@H](C)C(=O)O[C@@H]1C[C@H](C)C=C2C=C[C@H](C)[C@H](CC[C@H]3C[C@H](O)CC(=O)O3)[C@H]21
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? CC[C@@H](C)C(=O)O[C@@H]1C[C@H](C)C=C2C=C[C@H](C)[C@H](CC[C@H]3C[C@H](O)CC(=O)O3)[C@H]21
Yes
single_pred_adme_pgp
232
CC[N+](CC)=c1ccc2nc3c(cc(N)c4ccccc43)oc-2c1
Is the following compound AMES mutagenic? CC[N+](CC)=c1ccc2nc3c(cc(N)c4ccccc43)oc-2c1
Yes
single_pred_tox_ames
233
CC1(C)CC(C(=O)O)C(C)(C)N1O
Is the following compound AMES mutagenic? CC1(C)CC(C(=O)O)C(C)(C)N1O
No
single_pred_tox_ames
234
CCCC/C=C/C(NC(=O)c1ccc(-c2ccccc2)cc1)c1ccccc1
Given the following SMILES string, predict whether the compound inhibits CYP2C19? CCCC/C=C/C(NC(=O)c1ccc(-c2ccccc2)cc1)c1ccccc1
No
single_pred_adme_cyp2c19
235
CCCS(=O)CCC[NH+](CC)C[C@@H](O)COc1ccc(C#N)cc1
Does the following compound block the hERG channel? CCCS(=O)CCC[NH+](CC)C[C@@H](O)COc1ccc(C#N)cc1
Yes
single_pred_tox_herg
236
CC[C@H]1OC(=O)[C@@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H]([NH2+]C)[C@@H]2O)[C@](C)(O)C[C@@H](C)C(=O)[C@H](C)[C@@H](O)[C@]1(C)O
Does the following compound block the hERG channel? CC[C@H]1OC(=O)[C@@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H]([NH2+]C)[C@@H]2O)[C@](C)(O)C[C@@H](C)C(=O)[C@H](C)[C@@H](O)[C@]1(C)O
No
single_pred_tox_herg
237
COCO[C@@H]1CC(=O)O[C@H](C)[C@H](C)C(=O)O[C@@H](C(C)C)C(=O)N(C)[C@H]1Cc1ccccc1
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? COCO[C@@H]1CC(=O)O[C@H](C)[C@H](C)C(=O)O[C@@H](C(C)C)C(=O)N(C)[C@H]1Cc1ccccc1
Yes
single_pred_adme_pgp
238
COc1cc(O)c2c(=O)c(OC)c(-c3ccc4c(c3)O[C@H](c3ccc(O)c(OC)c3)[C@@H](CO)O4)oc2c1
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? COc1cc(O)c2c(=O)c(OC)c(-c3ccc4c(c3)O[C@H](c3ccc(O)c(OC)c3)[C@@H](CO)O4)oc2c1
Yes
single_pred_adme_pgp
239
COc1cc(NS(C)(=O)=O)ccc1Nc1c2ccccc2nc2ccccc12
Does the following compound cause drug-induced liver injury (DILI)? COc1cc(NS(C)(=O)=O)ccc1Nc1c2ccccc2nc2ccccc12
Yes
single_pred_tox_dili
240
CC(C)(C)c1ccc(OC[C@H]2CO2)cc1
Is the following compound AMES mutagenic? CC(C)(C)c1ccc(OC[C@H]2CO2)cc1
Yes
single_pred_tox_ames
241
CC(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)O
Given the following SMILES string, predict whether the compound inhibits CYP2C19? CC(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)O
No
single_pred_adme_cyp2c19
242
COc1ccc(-c2nc3cnc(Oc4cccc(Cl)c4)nc3n(CCC#N)c2=O)cc1
Given the following SMILES string, predict whether the compound inhibits CYP2C19? COc1ccc(-c2nc3cnc(Oc4cccc(Cl)c4)nc3n(CCC#N)c2=O)cc1
No
single_pred_adme_cyp2c19
243
CCOc1ccc(OCCOCCN2CCc3ccccc3C2)cc1
Given the following SMILES string, predict whether the compound inhibits CYP2C19? CCOc1ccc(OCCOCCN2CCc3ccccc3C2)cc1
Yes
single_pred_adme_cyp2c19
244
Cc1ccc(/C=C2\Sc3ccccc3C2=O)s1
Given the following SMILES string, predict whether the compound inhibits CYP2C19? Cc1ccc(/C=C2\Sc3ccccc3C2=O)s1
Yes
single_pred_adme_cyp2c19
245
C[N+](C)(C)CCNCCc1ccc(N=Nc2ccc([N+](=O)[O-])cc2Cl)cc1
Is the following compound AMES mutagenic? C[N+](C)(C)CCNCCc1ccc(N=Nc2ccc([N+](=O)[O-])cc2Cl)cc1
Yes
single_pred_tox_ames
246
COCCCCC(=NOCCN)c1ccc(C(F)(F)F)cc1
Does the following compound cause drug-induced liver injury (DILI)? COCCCCC(=NOCCN)c1ccc(C(F)(F)F)cc1
No
single_pred_tox_dili
247
CCl
Is the following compound AMES mutagenic? CCl
Yes
single_pred_tox_ames
248
Fc1ccc(C(OCCN2CCN(CCCc3ccccc3)CC2)c2ccc(F)cc2)cc1
Does the following compound block the hERG channel? Fc1ccc(C(OCCN2CCN(CCCc3ccccc3)CC2)c2ccc(F)cc2)cc1
Yes
single_pred_tox_herg
249
CC(C)C[C@H]1C(=O)N2CCCC2[C@]2(O)O[C@@](NC(=O)[C@H]3C=C4c5cccc6[nH]cc(c56)C[C@H]4N(C)C3)(C(C)C)C(=O)N12
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? CC(C)C[C@H]1C(=O)N2CCCC2[C@]2(O)O[C@@](NC(=O)[C@H]3C=C4c5cccc6[nH]cc(c56)C[C@H]4N(C)C3)(C(C)C)C(=O)N12
Yes
single_pred_adme_pgp
250
Cn1nnnc1SCC1=C(C(=O)O)N2C(=O)C(NC(=O)C(O)c3ccccc3)C2SC1
Does the following compound cause drug-induced liver injury (DILI)? Cn1nnnc1SCC1=C(C(=O)O)N2C(=O)C(NC(=O)C(O)c3ccccc3)C2SC1
Yes
single_pred_tox_dili
251
O=c1[nH]c2ccccc2n1C1CCN(CCCC(c2ccc(F)cc2)c2ccc(F)cc2)CC1
Does the following compound cause drug-induced liver injury (DILI)? O=c1[nH]c2ccccc2n1C1CCN(CCCC(c2ccc(F)cc2)c2ccc(F)cc2)CC1
No
single_pred_tox_dili
252
CC(C)(C)n1ncc2c(=O)n(Cc3ccc(Cl)cc3Cl)cnc21
Given the following SMILES string, predict whether the compound inhibits CYP2C19? CC(C)(C)n1ncc2c(=O)n(Cc3ccc(Cl)cc3Cl)cnc21
Yes
single_pred_adme_cyp2c19
253
O=C(N/N=C\c1ccc([N+](=O)[O-])o1)c1ccc(O)cc1
Given the following SMILES string, predict whether the compound inhibits CYP2C19? O=C(N/N=C\c1ccc([N+](=O)[O-])o1)c1ccc(O)cc1
No
single_pred_adme_cyp2c19
254
ClCCOCCCl
Is the following compound AMES mutagenic? ClCCOCCCl
Yes
single_pred_tox_ames
255
Cc1ccc(C)c(NC(=O)C2CC3c4ccccc4C2c2ccccc23)c1
Given the following SMILES string, predict whether the compound inhibits CYP2C19? Cc1ccc(C)c(NC(=O)C2CC3c4ccccc4C2c2ccccc23)c1
Yes
single_pred_adme_cyp2c19
256
CC(=O)OC1(C(C)=O)CCC2C3C=C(Cl)C4=CC(=O)OCC4(C)C3CCC21C
Is the following compound AMES mutagenic? CC(=O)OC1(C(C)=O)CCC2C3C=C(Cl)C4=CC(=O)OCC4(C)C3CCC21C
No
single_pred_tox_ames
257
COc1ccc(C=NC(CO)C(O)c2ccc([N+](=O)[O-])cc2)cc1
Given the following SMILES string, predict whether the compound inhibits CYP2C19? COc1ccc(C=NC(CO)C(O)c2ccc([N+](=O)[O-])cc2)cc1
No
single_pred_adme_cyp2c19
258
CC12c3ccccc3C(c3ccccc31)C1C(=O)N(Cc3cccnc3)C(=O)C12
Given the following SMILES string, predict whether the compound inhibits CYP2C19? CC12c3ccccc3C(c3ccccc31)C1C(=O)N(Cc3cccnc3)C(=O)C12
Yes
single_pred_adme_cyp2c19
259
NC1=NC(=O)C(c2ccccc2)O1
Does the following compound cause drug-induced liver injury (DILI)? NC1=NC(=O)C(c2ccccc2)O1
Yes
single_pred_tox_dili
260
COc1cccc(CCc2ccccc2OCCN2CCN(c3ccc(F)cc3)CC2)c1
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? COc1cccc(CCc2ccccc2OCCN2CCN(c3ccc(F)cc3)CC2)c1
Yes
single_pred_adme_pgp
261
CCCCCCC[C@H]1OC(=O)CC[C@H](Cc2ccccc2)N(C)C(=O)[C@H](C(C)C)OC(=O)[C@H]1C
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? CCCCCCC[C@H]1OC(=O)CC[C@H](Cc2ccccc2)N(C)C(=O)[C@H](C(C)C)OC(=O)[C@H]1C
Yes
single_pred_adme_pgp
262
COc1cc2c(c(O)c1O)C(=O)c1c(O)cc(C)cc1C2=O
Is the following compound AMES mutagenic? COc1cc2c(c(O)c1O)C(=O)c1c(O)cc(C)cc1C2=O
Yes
single_pred_tox_ames
263
CCCn1nnc(NC(=O)Cc2ccccc2)n1
Given the following SMILES string, predict whether the compound inhibits CYP2C19? CCCn1nnc(NC(=O)Cc2ccccc2)n1
Yes
single_pred_adme_cyp2c19
264
O=C(O)c1cc(Cl)cc(Cl)c1
Is the following compound AMES mutagenic? O=C(O)c1cc(Cl)cc(Cl)c1
No
single_pred_tox_ames
265
COC(=O)C1=C(C)NC(C)=C(C(=O)OCCCN2CCC(c3ccccc3)(c3ccccc3)CC2)[C@H]1c1cccc([N+](=O)[O-])c1
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? COC(=O)C1=C(C)NC(C)=C(C(=O)OCCCN2CCC(c3ccccc3)(c3ccccc3)CC2)[C@H]1c1cccc([N+](=O)[O-])c1
Yes
single_pred_adme_pgp
266
O=c1c(-c2cccs2)nc2cnc(Nc3ccccc3)nc2n1C[C@H]1CCCO1
Given the following SMILES string, predict whether the compound inhibits CYP2C19? O=c1c(-c2cccs2)nc2cnc(Nc3ccccc3)nc2n1C[C@H]1CCCO1
No
single_pred_adme_cyp2c19
267
Cc1cnc(NC(=O)C2=C(O)c3ccccc3S(=O)(=O)N2C)s1
Does the following compound block the hERG channel? Cc1cnc(NC(=O)C2=C(O)c3ccccc3S(=O)(=O)N2C)s1
No
single_pred_tox_herg
268
CN(C)CCCC1(c2ccc(F)cc2)OCc2cc(C#N)ccc21
Does the following compound cause drug-induced liver injury (DILI)? CN(C)CCCC1(c2ccc(F)cc2)OCc2cc(C#N)ccc21
No
single_pred_tox_dili
269
OCc1cccc2c1-c1cccc3cccc-2c13
Is the following compound AMES mutagenic? OCc1cccc2c1-c1cccc3cccc-2c13
No
single_pred_tox_ames
270
CN[C@@H](C)Cc1ccccc1
Is the following compound AMES mutagenic? CN[C@@H](C)Cc1ccccc1
No
single_pred_tox_ames
271
CC1OC(OC2C(CO)OC(OC3C(CO)OC(O)C(O)C3O)C(O)C2O)C(O)C(O)C1NC1C=C(CO)C(O)C(O)C1O
Does the following compound cause drug-induced liver injury (DILI)? CC1OC(OC2C(CO)OC(OC3C(CO)OC(O)C(O)C3O)C(O)C2O)C(O)C(O)C1NC1C=C(CO)C(O)C(O)C1O
Yes
single_pred_tox_dili
272
Nc1ccc(Oc2c(Cl)cc(Cl)cc2Cl)cc1
Is the following compound AMES mutagenic? Nc1ccc(Oc2c(Cl)cc(Cl)cc2Cl)cc1
Yes
single_pred_tox_ames
273
O=S(=O)(Cc1ccccc1)N1C2c3ccccc3-c3ccccc3C21
Is the following compound AMES mutagenic? O=S(=O)(Cc1ccccc1)N1C2c3ccccc3-c3ccccc3C21
Yes
single_pred_tox_ames
274
CCc1ccc(OCC(=O)NC(=S)Nc2ccc(F)cc2)c(Br)c1
Given the following SMILES string, predict whether the compound inhibits CYP2C19? CCc1ccc(OCC(=O)NC(=S)Nc2ccc(F)cc2)c(Br)c1
Yes
single_pred_adme_cyp2c19
275
CC1COc2c(N3CCN(C)CC3)c(F)cc3c(=O)c(C(=O)O)cn1c23
Does the following compound cause drug-induced liver injury (DILI)? CC1COc2c(N3CCN(C)CC3)c(F)cc3c(=O)c(C(=O)O)cn1c23
Yes
single_pred_tox_dili
276
O=C(CSC1=NCCN1)Nc1ccccc1
Given the following SMILES string, predict whether the compound inhibits CYP2C19? O=C(CSC1=NCCN1)Nc1ccccc1
No
single_pred_adme_cyp2c19
277
CCNc1nc(Cl)nc(NC(C)C)n1
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? CCNc1nc(Cl)nc(NC(C)C)n1
No
single_pred_adme_pgp
278
CC[NH+](CC)CC#CCOC(=O)C(O)(c1ccccc1)C1CCCCC1
Does the following compound block the hERG channel? CC[NH+](CC)CC#CCOC(=O)C(O)(c1ccccc1)C1CCCCC1
Yes
single_pred_tox_herg
279
Cc1ccc([N+](=O)[O-])cc1S(=O)(=O)O
Is the following compound AMES mutagenic? Cc1ccc([N+](=O)[O-])cc1S(=O)(=O)O
No
single_pred_tox_ames
280
COc1ccc2[nH]cc(CCN)c2c1
Given the following SMILES string, predict whether the compound inhibits CYP2C19? COc1ccc2[nH]cc(CCN)c2c1
No
single_pred_adme_cyp2c19
281
COc1cccc(-c2cc(C(F)(F)F)nc(N3CCN(c4ccccc4)CC3)n2)c1
Given the following SMILES string, predict whether the compound inhibits CYP2C19? COc1cccc(-c2cc(C(F)(F)F)nc(N3CCN(c4ccccc4)CC3)n2)c1
Yes
single_pred_adme_cyp2c19
282
O=C([O-])CCc1nc(-c2ccccc2)c(-c2ccccc2)o1
Does the following compound block the hERG channel? O=C([O-])CCc1nc(-c2ccccc2)c(-c2ccccc2)o1
No
single_pred_tox_herg
283
c1ccc(Nc2ccc3ccccc3c2)cc1
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? c1ccc(Nc2ccc3ccccc3c2)cc1
No
single_pred_adme_pgp
284
CN(CCC#N)c1ccc(N=Nc2ccc3ncsc3c2)cc1
Is the following compound AMES mutagenic? CN(CCC#N)c1ccc(N=Nc2ccc3ncsc3c2)cc1
Yes
single_pred_tox_ames
285
CN(C)C1C(O)=C(C(N)=O)C(=O)C2(O)C(O)=C3C(=O)c4c(O)cccc4C(C)(O)C3C(O)C12
Is the following compound AMES mutagenic? CN(C)C1C(O)=C(C(N)=O)C(=O)C2(O)C(O)=C3C(=O)c4c(O)cccc4C(C)(O)C3C(O)C12
No
single_pred_tox_ames
286
O=[N+]([O-])c1ccc(/C=C/c2cccc(Cl)c2)cc1
Is the following compound AMES mutagenic? O=[N+]([O-])c1ccc(/C=C/c2cccc(Cl)c2)cc1
Yes
single_pred_tox_ames
287
C[NH+]1[C@H]2CC[C@@H]1[C@@H](C(=O)[O-])[C@H](OC(=O)c1ccccc1)C2
Does the following compound block the hERG channel? C[NH+]1[C@H]2CC[C@@H]1[C@@H](C(=O)[O-])[C@H](OC(=O)c1ccccc1)C2
No
single_pred_tox_herg
288
C[N+](C)(C)CC(O)CC(=O)[O-]
Does the following compound cause drug-induced liver injury (DILI)? C[N+](C)(C)CC(O)CC(=O)[O-]
No
single_pred_tox_dili
289
COCc1ccc(-n2cc(C3CC[NH+](CCN4CCNC4=O)CC3)c3cc(Cl)ccc32)cc1
Does the following compound block the hERG channel? COCc1ccc(-n2cc(C3CC[NH+](CCN4CCNC4=O)CC3)c3cc(Cl)ccc32)cc1
Yes
single_pred_tox_herg
290
CN1CCN(Cc2ccc3c(c2)Cc2c(-c4csc(C#CCOc5ccccc5)c4)n[nH]c2-3)C(=O)C1
Does the following compound block the hERG channel? CN1CCN(Cc2ccc3c(c2)Cc2c(-c4csc(C#CCOc5ccccc5)c4)n[nH]c2-3)C(=O)C1
No
single_pred_tox_herg
291
CCN(CC)C(=O)Nc1ccc(OCC(O)CNC(C)(C)C)c(C(C)=O)c1
Is the following compound AMES mutagenic? CCN(CC)C(=O)Nc1ccc(OCC(O)CNC(C)(C)C)c(C(C)=O)c1
No
single_pred_tox_ames
292
C=C1C/C(=C\C)C(=O)O[C@H]2CCN3CC=C(COC(=O)[C@]1(C)O)C23
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? C=C1C/C(=C\C)C(=O)O[C@H]2CCN3CC=C(COC(=O)[C@]1(C)O)C23
No
single_pred_adme_pgp
293
COc1cc([C@H]2c3cc4c(cc3[C@H](O[C@@H]3O[C@@H]5CO[C@@H](C)O[C@H]5[C@@H](O)[C@@H]3O)[C@H]3COC(=O)[C@H]23)OCO4)cc(OC)c1O
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? COc1cc([C@H]2c3cc4c(cc3[C@H](O[C@@H]3O[C@@H]5CO[C@@H](C)O[C@H]5[C@@H](O)[C@@H]3O)[C@H]3COC(=O)[C@H]23)OCO4)cc(OC)c1O
No
single_pred_adme_pgp
294
COc1ccc2c(c1)N(C[C@@H](C)CN(C)C)c1ccccc1S2
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? COc1ccc2c(c1)N(C[C@@H](C)CN(C)C)c1ccccc1S2
Yes
single_pred_adme_pgp
295
N#CCCC#N
Is the following compound AMES mutagenic? N#CCCC#N
No
single_pred_tox_ames
296
CCCCCCC[C@H]1OC(=O)C[C@@H](OCOC)[C@H](Cc2ccccc2)N(C)C(=O)C(C)(C)OC(=O)[C@H]1C
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? CCCCCCC[C@H]1OC(=O)C[C@@H](OCOC)[C@H](Cc2ccccc2)N(C)C(=O)C(C)(C)OC(=O)[C@H]1C
Yes
single_pred_adme_pgp
297
Cc1ccc2c(c1)N(CCC(=O)NCC1CCCO1)C(=O)CO2
Given the following SMILES string, predict whether the compound inhibits CYP2C19? Cc1ccc2c(c1)N(CCC(=O)NCC1CCCO1)C(=O)CO2
No
single_pred_adme_cyp2c19
298
COC(=O)c1ccc(-c2nc(-c3ccc(N(C)C)cc3)c(-c3ccc(N(C)C)cc3)[nH]2)cc1
Given the SMILES of a compound, does it inhibit P-glycoprotein (P-gp)? COC(=O)c1ccc(-c2nc(-c3ccc(N(C)C)cc3)c(-c3ccc(N(C)C)cc3)[nH]2)cc1
Yes
single_pred_adme_pgp
299
O=Cc1ccc2ccc3cccc4ccc1c2c34
Is the following compound AMES mutagenic? O=Cc1ccc2ccc3cccc4ccc1c2c34
Yes
single_pred_tox_ames
300