assay_uid
stringlengths
9
15
positive_smiles
stringlengths
2
615
positive_smiles_hash
stringlengths
64
64
negative_smiles
listlengths
7
7
negative_smiles_hashes
listlengths
7
7
example_weight
float32
1
1.71
chembl:1665423
Fc1cccc2[nH]cc(Cc3c[nH]c4cccc(F)c34)c12
88f6fd062e971ae112b7dc7cf3cab9ddc33646ddf2106fa97fb644dd366975cf
[ "Cn1cc(Cc2cn(C)c3ccccc23)c2ccccc21", "CCCC(c1c[nH]c2ccccc12)c1c[nH]c2ccccc12", "COc1ccc2[nH]cc(Cc3c(O)[nH]c4ccccc34)c2c1", "Fc1cc2c(Cc3c[nH]c4cc(Cl)c(F)cc34)c[nH]c2cc1Cl", "COC(=O)c1ccc2[nH]cc(Cc3c[nH]c4ccccc34)c2c1", "O=C(O)c1ccc2[nH]cc(Cc3c[nH]c4ccc(C(=O)O)cc34)c2c1", "COc1ccc(C(c2c[nH]c3ccccc23)c2c[n...
[ "260106fc9b5eee5ee4a84d86b512b78a84a6b2e638cd379bb75a949f157ea33e", "64605f82c0fafe4f3e56aeb00c85e94b5537d4572607f530edd8e94a28ee486e", "d64c2b71f1500616c4cc44bf840c4a1f23a66cb799cf1d03764ee10649b723e7", "e69f8319837cf02fc558b29538dbcf7de8a59d4f5777e9372e65453cf91f8b14", "9cab3bbab19ff4661d6c77132d8c603f375...
1.624333
chembl:1665423
Fc1cccc2[nH]cc(Cc3c[nH]c4cccc(F)c34)c12
88f6fd062e971ae112b7dc7cf3cab9ddc33646ddf2106fa97fb644dd366975cf
[ "Clc1cc(Cl)c2c(Cc3c[nH]c4cc(Cl)cc(Cl)c34)c[nH]c2c1", "Oc1[nH]c2ccccc2c1Cc1ccc2[nH]ccc2c1", "COC(=O)c1ccc2[nH]cc(Cc3c[nH]c4ccc(C(=O)OC)cc34)c2c1", "COc1ccc2[nH]cc(C=C3C(=O)Nc4ccccc43)c2c1", "O=Cc1ccc2[nH]cc(Cc3c[nH]c4ccc(C=O)cc34)c2c1", "Oc1[nH]c2ccc(F)cc2c1Cc1c[nH]c2ccc(F)cc12", "O=C(O)c1ccc2[nH]cc(Cc3c...
[ "b191f902798da315087cf7b4516347a82b6246183ff9cbfc0959f570ff05561b", "c870cfec5d2e39fe776be5c6f842e867a6c97c6c8cde130d779a37a597100625", "f851c51bd47b4a91c20f1a7d9ae8e8794aa894f0d961f095f1a5294bf3c4460c", "e861dfd670d9976e28e41cbcc3267d1403221f0997569b0c2391bf3b44f2e6c3", "2881c6ced01d2c8d465b134d1f235e4a099...
1.624333
chembl:1665423
COc1ccc2[nH]cc(Cc3c[nH]c4ccc(OC)cc34)c2c1
de0274e5c852576fed8ba9e8614a7c335194fb0357c6ffb73619c9cca015018f
[ "Clc1cc(Cl)c2c(Cc3c[nH]c4cc(Cl)cc(Cl)c34)c[nH]c2c1", "Oc1[nH]c2ccccc2c1Cc1ccc2[nH]ccc2c1", "COC(=O)c1ccc2[nH]cc(Cc3c[nH]c4ccc(C(=O)OC)cc34)c2c1", "COc1ccc2[nH]cc(C=C3C(=O)Nc4ccccc43)c2c1", "O=Cc1ccc2[nH]cc(Cc3c[nH]c4ccc(C=O)cc34)c2c1", "Oc1[nH]c2ccc(F)cc2c1Cc1c[nH]c2ccc(F)cc12", "O=C(O)c1ccc2[nH]cc(Cc3c...
[ "b191f902798da315087cf7b4516347a82b6246183ff9cbfc0959f570ff05561b", "c870cfec5d2e39fe776be5c6f842e867a6c97c6c8cde130d779a37a597100625", "f851c51bd47b4a91c20f1a7d9ae8e8794aa894f0d961f095f1a5294bf3c4460c", "e861dfd670d9976e28e41cbcc3267d1403221f0997569b0c2391bf3b44f2e6c3", "2881c6ced01d2c8d465b134d1f235e4a099...
1.623
chembl:1665423
COc1ccc2[nH]cc(Cc3c[nH]c4ccc(OC)cc34)c2c1
de0274e5c852576fed8ba9e8614a7c335194fb0357c6ffb73619c9cca015018f
[ "Cc1ccc2c(Cc3c[nH]c4cc(C)ccc34)c[nH]c2c1", "Fc1cc2cc[nH]c2cc1F", "c1ccc2c(C(c3c[nH]c4ccccc34)c3c[nH]c4ccccc34)c[nH]c2c1", "O=C1Nc2ccccc2C1=Cc1c[nH]c2ccccc12", "O=[N+]([O-])c1ccc2[nH]cc(Cc3c[nH]c4ccc([N+](=O)[O-])cc34)c2c1", "Oc1ccc(C(c2c[nH]c3ccccc23)c2c[nH]c3ccccc23)cc1", "COc1ccc2[nH]cc(C=C3C(=O)Nc4cc...
[ "47d66df9731b2945b0a1a1cb00adb59cd38442fdabc4eb4f745b3cd32143ebda", "991dde3e76c426645057e85cae6baac8a28f1f0ccc2713dc1251c04f28fc09d9", "77f1bb36b2b599257d009e2d8fc9f8816218e45953bca080df9555aa98135107", "fca6d63fc3cec7f570fee6ad1d218dfa03001a3d41a8f414316fe16118083a4b", "cdb3d825db059fc5ea1dca5769682c79852...
1.623
chembl:1665423
Fc1ccc2[nH]cc(Cc3c[nH]c4ccc(F)c(F)c34)c2c1F
cb00cae90c04bc6096eb634d647f2e780d289477d78aef9fca8dadd5d6de32de
[ "Cc1ccc2c(Cc3c[nH]c4cc(C)ccc34)c[nH]c2c1", "Fc1cc2cc[nH]c2cc1F", "c1ccc2c(C(c3c[nH]c4ccccc34)c3c[nH]c4ccccc34)c[nH]c2c1", "O=C1Nc2ccccc2C1=Cc1c[nH]c2ccccc12", "O=[N+]([O-])c1ccc2[nH]cc(Cc3c[nH]c4ccc([N+](=O)[O-])cc34)c2c1", "Oc1ccc(C(c2c[nH]c3ccccc23)c2c[nH]c3ccccc23)cc1", "COc1ccc2[nH]cc(C=C3C(=O)Nc4cc...
[ "47d66df9731b2945b0a1a1cb00adb59cd38442fdabc4eb4f745b3cd32143ebda", "991dde3e76c426645057e85cae6baac8a28f1f0ccc2713dc1251c04f28fc09d9", "77f1bb36b2b599257d009e2d8fc9f8816218e45953bca080df9555aa98135107", "fca6d63fc3cec7f570fee6ad1d218dfa03001a3d41a8f414316fe16118083a4b", "cdb3d825db059fc5ea1dca5769682c79852...
1.622333
chembl:1665423
Fc1ccc2[nH]cc(Cc3c[nH]c4ccc(F)c(F)c34)c2c1F
cb00cae90c04bc6096eb634d647f2e780d289477d78aef9fca8dadd5d6de32de
[ "Cc1ccc(C(c2c[nH]c3ccccc23)c2c[nH]c3ccccc23)cc1", "CC(c1c[nH]c2cccc(F)c12)c1c[nH]c2cccc(F)c12", "CCC(c1c[nH]c2ccccc12)c1c[nH]c2ccccc12", "O=[N+]([O-])c1ccc(C(c2c[nH]c3ccccc23)c2c[nH]c3ccccc23)cc1", "COc1ccc2c(Cc3c[nH]c4cc(OC)ccc34)c[nH]c2c1", "c1ccc(COc2ccc3[nH]cc(Cc4c[nH]c5ccc(OCc6ccccc6)cc45)c3c2)cc1", ...
[ "e22afd95c4732f10f4f4737b993098bf4ea602948e8aa79eb576d9659c341e36", "87623e17e8ede5a82fffa6a26a049ff31ef8cf3afe4772b0c1d0b3a11de54a46", "b58c5ff9fc18abaff0038932c1aa5907c3b205367acf859e02cd123104583d0f", "513e609b47f300502886edd52fa5ca155e58966e72e6089bfddb905d1ad9ed2e", "cde7adb7ab42dbcdb669ec092d7d92de7b9...
1.622333
chembl:1665423
O=C(c1c[nH]c2ccccc12)c1c[nH]c2ccccc12
e207b154b9e5d0d470070be55e5c59fcf5e23bbc51eda8310b1ea4a90394ddc7
[ "Cc1ccc(C(c2c[nH]c3ccccc23)c2c[nH]c3ccccc23)cc1", "CC(c1c[nH]c2cccc(F)c12)c1c[nH]c2cccc(F)c12", "CCC(c1c[nH]c2ccccc12)c1c[nH]c2ccccc12", "O=[N+]([O-])c1ccc(C(c2c[nH]c3ccccc23)c2c[nH]c3ccccc23)cc1", "COc1ccc2c(Cc3c[nH]c4cc(OC)ccc34)c[nH]c2c1", "c1ccc(COc2ccc3[nH]cc(Cc4c[nH]c5ccc(OCc6ccccc6)cc45)c3c2)cc1", ...
[ "e22afd95c4732f10f4f4737b993098bf4ea602948e8aa79eb576d9659c341e36", "87623e17e8ede5a82fffa6a26a049ff31ef8cf3afe4772b0c1d0b3a11de54a46", "b58c5ff9fc18abaff0038932c1aa5907c3b205367acf859e02cd123104583d0f", "513e609b47f300502886edd52fa5ca155e58966e72e6089bfddb905d1ad9ed2e", "cde7adb7ab42dbcdb669ec092d7d92de7b9...
1.617
chembl:1665423
O=C(c1c[nH]c2ccccc12)c1c[nH]c2ccccc12
e207b154b9e5d0d470070be55e5c59fcf5e23bbc51eda8310b1ea4a90394ddc7
[ "c1cc2c(c(C(c3c[nH]c4ccccc34)c3c[nH]c4ccccc34)c1)OCO2", "c1cnc2[nH]cc(Cc3c[nH]c4ncccc34)c2c1", "CCCCC(c1c[nH]c2ccccc12)c1c[nH]c2ccccc12", "Cc1ccc2[nH]cc(Cc3c[nH]c4ccc(C)cc34)c2c1", "Clc1ccc(C(c2c[nH]c3ccccc23)c2c[nH]c3ccccc23)cc1", "O=C1Nc2ccc(F)cc2C1=Cc1c[nH]c2ccc(F)cc12", "Fc1ccc(C(c2c[nH]c3ccccc23)c2...
[ "b26d5a2f077abacc5a8c83a4bd1490481378ae46f24c0e08887d8d7668ad6972", "166656477a3c97c1065998f7622ea709d572d81e4ca32bf263b54693fa8e71dd", "cb257c1cf140ecf8eb1a3d34938dc46c96c48c44ce2d7206c6aa5d2eec91d063", "d893ca0b615a065f1acbe8145d695bf9312a9caf594305f40a3d6ffeef2df406", "fb71c3c12129d44c7d5899e15e17196317f...
1.617
chembl:1665423
Fc1ccc2c(Cc3c[nH]c4cc(F)ccc34)c[nH]c2c1
956dbaffbd47b32e7b1c6b71d22c97f08c9a4fdfced19157120178726e70bb00
[ "c1cc2c(c(C(c3c[nH]c4ccccc34)c3c[nH]c4ccccc34)c1)OCO2", "c1cnc2[nH]cc(Cc3c[nH]c4ncccc34)c2c1", "CCCCC(c1c[nH]c2ccccc12)c1c[nH]c2ccccc12", "Cc1ccc2[nH]cc(Cc3c[nH]c4ccc(C)cc34)c2c1", "Clc1ccc(C(c2c[nH]c3ccccc23)c2c[nH]c3ccccc23)cc1", "O=C1Nc2ccc(F)cc2C1=Cc1c[nH]c2ccc(F)cc12", "Fc1ccc(C(c2c[nH]c3ccccc23)c2...
[ "b26d5a2f077abacc5a8c83a4bd1490481378ae46f24c0e08887d8d7668ad6972", "166656477a3c97c1065998f7622ea709d572d81e4ca32bf263b54693fa8e71dd", "cb257c1cf140ecf8eb1a3d34938dc46c96c48c44ce2d7206c6aa5d2eec91d063", "d893ca0b615a065f1acbe8145d695bf9312a9caf594305f40a3d6ffeef2df406", "fb71c3c12129d44c7d5899e15e17196317f...
1.615
chembl:1665423
Fc1ccc2c(Cc3c[nH]c4cc(F)ccc34)c[nH]c2c1
956dbaffbd47b32e7b1c6b71d22c97f08c9a4fdfced19157120178726e70bb00
[ "N#Cc1ccc2[nH]cc(Cc3c[nH]c4ccc(C#N)cc34)c2c1", "O=C1Nc2ccccc2C1=Cc1c[nH]c2ccc(F)cc12", "Cn1cc(Cc2c[nH]c3ccccc23)c2ccccc21", "CC(c1c[nH]c2ccccc12)c1c[nH]c2ccccc12", "CC(C)C(c1c[nH]c2ccccc12)c1c[nH]c2ccccc12", "COc1cccc2c(Cc3c[nH]c4c(OC)cccc34)c[nH]c12", "COc1cccc2[nH]cc(Cc3c[nH]c4cccc(OC)c34)c12" ]
[ "93175a9c07eaf886ab612a9edbf53cace2924ca1e57750021d763e4d21f5bb4f", "2411eb192ce38d8bf29e0afe5fe0e1fb480d60e1302c0e1588d115e890f02aa3", "4929bf3dbfc71d95a3e54a5834fc7a9ad874c51582fb9b56d02550b7baddf23d", "8289bdc5883b81055c3858bf5b547403dc9d3cb1afc423b08e2892b9070fdd3b", "92c88b8a35d975a6e0b8e7793a9d172a203...
1.615
chembl:1665423
CCCCCCCC=CCCc1c(O)c(O)cc(O)c1O
6cfb8932f596c340cf8ba1c2efecbdb5ad3ba5d727d1fa87e9b8583437e3a8b8
[ "N#Cc1ccc2[nH]cc(Cc3c[nH]c4ccc(C#N)cc34)c2c1", "O=C1Nc2ccccc2C1=Cc1c[nH]c2ccc(F)cc12", "Cn1cc(Cc2c[nH]c3ccccc23)c2ccccc21", "CC(c1c[nH]c2ccccc12)c1c[nH]c2ccccc12", "CC(C)C(c1c[nH]c2ccccc12)c1c[nH]c2ccccc12", "COc1cccc2c(Cc3c[nH]c4c(OC)cccc34)c[nH]c12", "COc1cccc2[nH]cc(Cc3c[nH]c4cccc(OC)c34)c12" ]
[ "93175a9c07eaf886ab612a9edbf53cace2924ca1e57750021d763e4d21f5bb4f", "2411eb192ce38d8bf29e0afe5fe0e1fb480d60e1302c0e1588d115e890f02aa3", "4929bf3dbfc71d95a3e54a5834fc7a9ad874c51582fb9b56d02550b7baddf23d", "8289bdc5883b81055c3858bf5b547403dc9d3cb1afc423b08e2892b9070fdd3b", "92c88b8a35d975a6e0b8e7793a9d172a203...
1.611667
chembl:1665423
CCCCCCCC=CCCc1c(O)c(O)cc(O)c1O
6cfb8932f596c340cf8ba1c2efecbdb5ad3ba5d727d1fa87e9b8583437e3a8b8
[ "Clc1ccc2c(Cc3c[nH]c4cc(Cl)ccc34)c[nH]c2c1", "Cc1[nH]c2ccccc2c1Cc1c(C)[nH]c2ccccc12", "O=C1Nc2ccccc2C1=Cc1ccc2[nH]ccc2c1", "Cn1cc(Cc2cn(C)c3ccccc23)c2ccccc21", "CCCC(c1c[nH]c2ccccc12)c1c[nH]c2ccccc12", "COc1ccc2[nH]cc(Cc3c(O)[nH]c4ccccc34)c2c1", "Fc1cc2c(Cc3c[nH]c4cc(Cl)c(F)cc34)c[nH]c2cc1Cl" ]
[ "96a54c548d04255af54db5a726b048ef7a86f82096269cbe3b74cf47b51c565c", "a67428239496e9d3292d08e003d14463d3bcfe83de88fb0487d975dece69b0fe", "ce4f7fbccb7e8f9caef5835f409f76bc79442ea7acb717fd35c4c120375ea044", "260106fc9b5eee5ee4a84d86b512b78a84a6b2e638cd379bb75a949f157ea33e", "64605f82c0fafe4f3e56aeb00c85e94b553...
1.611667
chembl:1665423
Cc1cccc2[nH]cc(Cc3c[nH]c4cccc(C)c34)c12
66b4d0e74ad31cc6d4030fce6c4f0b3b8000919d5af69fe7658e123f36fd0d26
[ "Clc1ccc2c(Cc3c[nH]c4cc(Cl)ccc34)c[nH]c2c1", "Cc1[nH]c2ccccc2c1Cc1c(C)[nH]c2ccccc12", "O=C1Nc2ccccc2C1=Cc1ccc2[nH]ccc2c1", "Cn1cc(Cc2cn(C)c3ccccc23)c2ccccc21", "CCCC(c1c[nH]c2ccccc12)c1c[nH]c2ccccc12", "COc1ccc2[nH]cc(Cc3c(O)[nH]c4ccccc34)c2c1", "Fc1cc2c(Cc3c[nH]c4cc(Cl)c(F)cc34)c[nH]c2cc1Cl" ]
[ "96a54c548d04255af54db5a726b048ef7a86f82096269cbe3b74cf47b51c565c", "a67428239496e9d3292d08e003d14463d3bcfe83de88fb0487d975dece69b0fe", "ce4f7fbccb7e8f9caef5835f409f76bc79442ea7acb717fd35c4c120375ea044", "260106fc9b5eee5ee4a84d86b512b78a84a6b2e638cd379bb75a949f157ea33e", "64605f82c0fafe4f3e56aeb00c85e94b553...
1.608667
chembl:1665423
Cc1cccc2[nH]cc(Cc3c[nH]c4cccc(C)c34)c12
66b4d0e74ad31cc6d4030fce6c4f0b3b8000919d5af69fe7658e123f36fd0d26
[ "COC(=O)c1ccc2[nH]cc(Cc3c[nH]c4ccccc34)c2c1", "O=C(O)c1ccc2[nH]cc(Cc3c[nH]c4ccc(C(=O)O)cc34)c2c1", "COc1ccc(C(c2c[nH]c3ccccc23)c2c[nH]c3ccccc23)cc1", "Clc1cc(Cl)c2c(Cc3c[nH]c4cc(Cl)cc(Cl)c34)c[nH]c2c1", "Oc1[nH]c2ccccc2c1Cc1ccc2[nH]ccc2c1", "COC(=O)c1ccc2[nH]cc(Cc3c[nH]c4ccc(C(=O)OC)cc34)c2c1", "COc1ccc...
[ "9cab3bbab19ff4661d6c77132d8c603f375aed88cc2f6db7f01bdfa4c31d490b", "a619001c11ff01a4a2dcc5199345c289ce71e18d7d43e18e303f1512ff631266", "9ffacca1d077b94eb8db64f5a568bcf1f927e6f849f2e86e61bea70b31cf1827", "b191f902798da315087cf7b4516347a82b6246183ff9cbfc0959f570ff05561b", "c870cfec5d2e39fe776be5c6f842e867a6c...
1.608667
chembl:1670780
O=C(O)/C=C/C(O)c1ccc(OCc2ccc(Br)cc2)cc1
e07923f5bb0b0dde48a4dad084bd04e7db31d3a2ed800a5b7b0e89398ea76c32
[ "O=C(O)C1=C(c2ccccc2)C(O)CC1", "Cc1ccc(C2=C(C(=O)O)CCC2O)cc1", "O=C(O)C1CCC[C@@H](O)C1", "O=C(O)C1CC[C@@](O)(c2ccccc2)C1", "O=C(O)C1=CCCC1", "O=C(O)C1CC(O)C1", "O=C(O)C1=C(c2ccc(Cl)cc2)C(O)CC1" ]
[ "41c0d704df614fea31279a188d786cd27abdeaa000ebf9f007904f4614b5ee03", "65d9061fe520936afbdf6796f37a92b2380a01a1b3f6529e39517b52716fcad2", "576d3a9c89912e9d49de43ac9bb16d5f4383a299851cbd31dd64211dda1cdc65", "731c8fd5ccdc3d54894458e0fe671dc923beecabe8ca3e5fd634d2f580905de9", "f837711c63c0292945378748d63969f5440...
1.588
chembl:1670780
O=C(O)/C=C/C(O)c1ccc(OCc2ccc(Br)cc2)cc1
e07923f5bb0b0dde48a4dad084bd04e7db31d3a2ed800a5b7b0e89398ea76c32
[ "COc1cccc(CC2=C(C(=O)O)CCC2O)c1", "O=C(O)C1=C(c2ccc(Cl)c(Cl)c2)C(O)CC1", "O=C(O)C1=C(Cc2ccccc2)C(O)CC1", "O=C(O)C1CCC(O)C1", "CC1=C(C(=O)O)CCC1O", "O=C(O)C1=CC(c2ccccc2)CC1", "COc1ccc(C2=C(C(=O)O)CCC2O)cc1" ]
[ "3c7a15d8001f18157916259df4f9ec99eaaff32155090c1e57c57caae3f3aa73", "b1dcadaf5a757b36fb04a5962f26e4e3a3da850b4d5fe6fc86ac7f343e54e4e6", "4649c6f532a7b4b36e0da22fe28f9d67514f4ee625f7b9bee2f714b5c6d32aaa", "241d12649f1ca02abe843e489ba8e76d65229807aceb98ba015596dcf8040a79", "ac8ce23be75716c5948ace075ac2c3deb08...
1.588
chembl:1670780
O=C(O)/C=C/C(O)c1ccc(Cc2ccccc2)cc1
e436cc765b35229577539d2d0fd3feb9c47275ecdf0e5e1cb48ffc7ecac8780e
[ "COc1cccc(CC2=C(C(=O)O)CCC2O)c1", "O=C(O)C1=C(c2ccc(Cl)c(Cl)c2)C(O)CC1", "O=C(O)C1=C(Cc2ccccc2)C(O)CC1", "O=C(O)C1CCC(O)C1", "CC1=C(C(=O)O)CCC1O", "O=C(O)C1=CC(c2ccccc2)CC1", "COc1ccc(C2=C(C(=O)O)CCC2O)cc1" ]
[ "3c7a15d8001f18157916259df4f9ec99eaaff32155090c1e57c57caae3f3aa73", "b1dcadaf5a757b36fb04a5962f26e4e3a3da850b4d5fe6fc86ac7f343e54e4e6", "4649c6f532a7b4b36e0da22fe28f9d67514f4ee625f7b9bee2f714b5c6d32aaa", "241d12649f1ca02abe843e489ba8e76d65229807aceb98ba015596dcf8040a79", "ac8ce23be75716c5948ace075ac2c3deb08...
1.584
chembl:1670780
O=C(O)/C=C/C(O)c1ccc(Cc2ccccc2)cc1
e436cc765b35229577539d2d0fd3feb9c47275ecdf0e5e1cb48ffc7ecac8780e
[ "CCC1=C(C(=O)O)CCC1O", "O=C(O)[C@]12CC[C@@H](O)[C@H]1C2", "C=CCC1=C(C(=O)O)CCC1O", "O=C(O)C1=C(c2ccccc2)C(O)CC1", "Cc1ccc(C2=C(C(=O)O)CCC2O)cc1", "O=C(O)C1CCC[C@@H](O)C1", "O=C(O)C1CC[C@@](O)(c2ccccc2)C1" ]
[ "270acd38334855ce112d9ee3f864c4916d456ce817c8b436af34c3c8008f1648", "96f02734e7a4d6285bf0c83f7bf25f8eb811b9da241768b166b1f5fe5e84f4a2", "51ae9170034ddac9092031776335a24594ebd66f592860e6f80c24e0a9d06d35", "41c0d704df614fea31279a188d786cd27abdeaa000ebf9f007904f4614b5ee03", "65d9061fe520936afbdf6796f37a92b2380...
1.584
chembl:1670780
O=C(O)/C=C/C(O)c1ccc(OCc2ccccc2)cc1
b87ac57bd84bf7d6dd6149b34897d6b587652745cf10c830dde8b0836576578f
[ "CCC1=C(C(=O)O)CCC1O", "O=C(O)[C@]12CC[C@@H](O)[C@H]1C2", "C=CCC1=C(C(=O)O)CCC1O", "O=C(O)C1=C(c2ccccc2)C(O)CC1", "Cc1ccc(C2=C(C(=O)O)CCC2O)cc1", "O=C(O)C1CCC[C@@H](O)C1", "O=C(O)C1CC[C@@](O)(c2ccccc2)C1" ]
[ "270acd38334855ce112d9ee3f864c4916d456ce817c8b436af34c3c8008f1648", "96f02734e7a4d6285bf0c83f7bf25f8eb811b9da241768b166b1f5fe5e84f4a2", "51ae9170034ddac9092031776335a24594ebd66f592860e6f80c24e0a9d06d35", "41c0d704df614fea31279a188d786cd27abdeaa000ebf9f007904f4614b5ee03", "65d9061fe520936afbdf6796f37a92b2380...
1.581
chembl:1670780
O=C(O)/C=C/C(O)c1ccc(OCc2ccccc2)cc1
b87ac57bd84bf7d6dd6149b34897d6b587652745cf10c830dde8b0836576578f
[ "O=C(O)C1=CCCC1", "O=C(O)C1CC(O)C1", "O=C(O)C1=C(c2ccc(Cl)cc2)C(O)CC1", "COc1cccc(CC2=C(C(=O)O)CCC2O)c1", "O=C(O)C1=C(c2ccc(Cl)c(Cl)c2)C(O)CC1", "O=C(O)C1=C(Cc2ccccc2)C(O)CC1", "O=C(O)C1CCC(O)C1" ]
[ "f837711c63c0292945378748d63969f5440f3f3ac2e3c8605c4e593b354c5e79", "dbe79c2fcccd4cb0ca5e930789c795c139fd496cc163eeabbc411c5ee2e9b50c", "64d2921bc629f9ce44dd861b41db3f9bff04503a4acbaa4797ec92863784341c", "3c7a15d8001f18157916259df4f9ec99eaaff32155090c1e57c57caae3f3aa73", "b1dcadaf5a757b36fb04a5962f26e4e3a3d...
1.581
chembl:1670780
O=C(O)/C=C/C(O)c1ccc(CCc2ccccc2)cc1
dc3a125a51aa50bd0bee5ea27c1e2c93f47620993dd32546108464b6fb908f79
[ "O=C(O)C1=CCCC1", "O=C(O)C1CC(O)C1", "O=C(O)C1=C(c2ccc(Cl)cc2)C(O)CC1", "COc1cccc(CC2=C(C(=O)O)CCC2O)c1", "O=C(O)C1=C(c2ccc(Cl)c(Cl)c2)C(O)CC1", "O=C(O)C1=C(Cc2ccccc2)C(O)CC1", "O=C(O)C1CCC(O)C1" ]
[ "f837711c63c0292945378748d63969f5440f3f3ac2e3c8605c4e593b354c5e79", "dbe79c2fcccd4cb0ca5e930789c795c139fd496cc163eeabbc411c5ee2e9b50c", "64d2921bc629f9ce44dd861b41db3f9bff04503a4acbaa4797ec92863784341c", "3c7a15d8001f18157916259df4f9ec99eaaff32155090c1e57c57caae3f3aa73", "b1dcadaf5a757b36fb04a5962f26e4e3a3d...
1.579667
chembl:1670780
O=C(O)/C=C/C(O)c1ccc(CCc2ccccc2)cc1
dc3a125a51aa50bd0bee5ea27c1e2c93f47620993dd32546108464b6fb908f79
[ "CC1=C(C(=O)O)CCC1O", "O=C(O)C1=CC(c2ccccc2)CC1", "COc1ccc(C2=C(C(=O)O)CCC2O)cc1", "CCC1=C(C(=O)O)CCC1O", "O=C(O)[C@]12CC[C@@H](O)[C@H]1C2", "C=CCC1=C(C(=O)O)CCC1O", "O=C(O)C1=C(c2ccccc2)C(O)CC1" ]
[ "ac8ce23be75716c5948ace075ac2c3deb088d4e1b564c7675292450d5a03b29c", "e81f02bb1287c7eabe246e1df71cffa23c788fea808e1250f3d73b22ba0215ac", "3618ce5b3a2f60f276c2c549fd96601049097b1837b769d3a006870dcfc42a01", "270acd38334855ce112d9ee3f864c4916d456ce817c8b436af34c3c8008f1648", "96f02734e7a4d6285bf0c83f7bf25f8eb81...
1.579667
chembl:1670780
O=C(O)/C=C/C(O)c1ccc(-c2ccccc2)cc1
e6302ba0e029adfe74cfda761fc9e186aaeec35e90e6b4986b381b1b92764f5a
[ "CC1=C(C(=O)O)CCC1O", "O=C(O)C1=CC(c2ccccc2)CC1", "COc1ccc(C2=C(C(=O)O)CCC2O)cc1", "CCC1=C(C(=O)O)CCC1O", "O=C(O)[C@]12CC[C@@H](O)[C@H]1C2", "C=CCC1=C(C(=O)O)CCC1O", "O=C(O)C1=C(c2ccccc2)C(O)CC1" ]
[ "ac8ce23be75716c5948ace075ac2c3deb088d4e1b564c7675292450d5a03b29c", "e81f02bb1287c7eabe246e1df71cffa23c788fea808e1250f3d73b22ba0215ac", "3618ce5b3a2f60f276c2c549fd96601049097b1837b769d3a006870dcfc42a01", "270acd38334855ce112d9ee3f864c4916d456ce817c8b436af34c3c8008f1648", "96f02734e7a4d6285bf0c83f7bf25f8eb81...
1.571333
chembl:1670780
O=C(O)/C=C/C(O)c1ccc(-c2ccccc2)cc1
e6302ba0e029adfe74cfda761fc9e186aaeec35e90e6b4986b381b1b92764f5a
[ "Cc1ccc(C2=C(C(=O)O)CCC2O)cc1", "O=C(O)C1CCC[C@@H](O)C1", "O=C(O)C1CC[C@@](O)(c2ccccc2)C1", "O=C(O)C1=CCCC1", "O=C(O)C1CC(O)C1", "O=C(O)C1=C(c2ccc(Cl)cc2)C(O)CC1", "COc1cccc(CC2=C(C(=O)O)CCC2O)c1" ]
[ "65d9061fe520936afbdf6796f37a92b2380a01a1b3f6529e39517b52716fcad2", "576d3a9c89912e9d49de43ac9bb16d5f4383a299851cbd31dd64211dda1cdc65", "731c8fd5ccdc3d54894458e0fe671dc923beecabe8ca3e5fd634d2f580905de9", "f837711c63c0292945378748d63969f5440f3f3ac2e3c8605c4e593b354c5e79", "dbe79c2fcccd4cb0ca5e930789c795c139f...
1.571333
chembl:1670780
O=C(O)C1=C[C@H](O)CC1
4f3e70b3a50cec1bbfb5ef6b70558e6cad21f19fbe50d170baf10b0434054d67
[ "Cc1ccc(C2=C(C(=O)O)CCC2O)cc1", "O=C(O)C1CCC[C@@H](O)C1", "O=C(O)C1CC[C@@](O)(c2ccccc2)C1", "O=C(O)C1=CCCC1", "O=C(O)C1CC(O)C1", "O=C(O)C1=C(c2ccc(Cl)cc2)C(O)CC1", "COc1cccc(CC2=C(C(=O)O)CCC2O)c1" ]
[ "65d9061fe520936afbdf6796f37a92b2380a01a1b3f6529e39517b52716fcad2", "576d3a9c89912e9d49de43ac9bb16d5f4383a299851cbd31dd64211dda1cdc65", "731c8fd5ccdc3d54894458e0fe671dc923beecabe8ca3e5fd634d2f580905de9", "f837711c63c0292945378748d63969f5440f3f3ac2e3c8605c4e593b354c5e79", "dbe79c2fcccd4cb0ca5e930789c795c139f...
1.565333
chembl:1670780
O=C(O)C1=C[C@H](O)CC1
4f3e70b3a50cec1bbfb5ef6b70558e6cad21f19fbe50d170baf10b0434054d67
[ "O=C(O)C1=C(c2ccc(Cl)c(Cl)c2)C(O)CC1", "O=C(O)C1=C(Cc2ccccc2)C(O)CC1", "O=C(O)C1CCC(O)C1", "CC1=C(C(=O)O)CCC1O", "O=C(O)C1=CC(c2ccccc2)CC1", "COc1ccc(C2=C(C(=O)O)CCC2O)cc1", "CCC1=C(C(=O)O)CCC1O" ]
[ "b1dcadaf5a757b36fb04a5962f26e4e3a3da850b4d5fe6fc86ac7f343e54e4e6", "4649c6f532a7b4b36e0da22fe28f9d67514f4ee625f7b9bee2f714b5c6d32aaa", "241d12649f1ca02abe843e489ba8e76d65229807aceb98ba015596dcf8040a79", "ac8ce23be75716c5948ace075ac2c3deb088d4e1b564c7675292450d5a03b29c", "e81f02bb1287c7eabe246e1df71cffa23c7...
1.565333
chembl:1670780
O=C(O)C1=CC(O)CC1
d965e58d5315a6271e5cac4666f45ee6b76fe8acf982cf4dc930d12b242b55b5
[ "O=C(O)C1=C(c2ccc(Cl)c(Cl)c2)C(O)CC1", "O=C(O)C1=C(Cc2ccccc2)C(O)CC1", "O=C(O)C1CCC(O)C1", "CC1=C(C(=O)O)CCC1O", "O=C(O)C1=CC(c2ccccc2)CC1", "COc1ccc(C2=C(C(=O)O)CCC2O)cc1", "CCC1=C(C(=O)O)CCC1O" ]
[ "b1dcadaf5a757b36fb04a5962f26e4e3a3da850b4d5fe6fc86ac7f343e54e4e6", "4649c6f532a7b4b36e0da22fe28f9d67514f4ee625f7b9bee2f714b5c6d32aaa", "241d12649f1ca02abe843e489ba8e76d65229807aceb98ba015596dcf8040a79", "ac8ce23be75716c5948ace075ac2c3deb088d4e1b564c7675292450d5a03b29c", "e81f02bb1287c7eabe246e1df71cffa23c7...
1.563
chembl:1670780
O=C(O)C1=CC(O)CC1
d965e58d5315a6271e5cac4666f45ee6b76fe8acf982cf4dc930d12b242b55b5
[ "O=C(O)[C@]12CC[C@@H](O)[C@H]1C2", "C=CCC1=C(C(=O)O)CCC1O", "O=C(O)C1=C(c2ccccc2)C(O)CC1", "Cc1ccc(C2=C(C(=O)O)CCC2O)cc1", "O=C(O)C1CCC[C@@H](O)C1", "O=C(O)C1CC[C@@](O)(c2ccccc2)C1", "O=C(O)C1=CCCC1" ]
[ "96f02734e7a4d6285bf0c83f7bf25f8eb811b9da241768b166b1f5fe5e84f4a2", "51ae9170034ddac9092031776335a24594ebd66f592860e6f80c24e0a9d06d35", "41c0d704df614fea31279a188d786cd27abdeaa000ebf9f007904f4614b5ee03", "65d9061fe520936afbdf6796f37a92b2380a01a1b3f6529e39517b52716fcad2", "576d3a9c89912e9d49de43ac9bb16d5f438...
1.563
chembl:1670780
O=C(O)C1CC[C@@](O)(c2ccc(-c3ccccc3)cc2)C1
a6e41ed24722dbb824aaa3974fb9b7e9c0d0e25516a97134beb86f6e770fe1ee
[ "O=C(O)[C@]12CC[C@@H](O)[C@H]1C2", "C=CCC1=C(C(=O)O)CCC1O", "O=C(O)C1=C(c2ccccc2)C(O)CC1", "Cc1ccc(C2=C(C(=O)O)CCC2O)cc1", "O=C(O)C1CCC[C@@H](O)C1", "O=C(O)C1CC[C@@](O)(c2ccccc2)C1", "O=C(O)C1=CCCC1" ]
[ "96f02734e7a4d6285bf0c83f7bf25f8eb811b9da241768b166b1f5fe5e84f4a2", "51ae9170034ddac9092031776335a24594ebd66f592860e6f80c24e0a9d06d35", "41c0d704df614fea31279a188d786cd27abdeaa000ebf9f007904f4614b5ee03", "65d9061fe520936afbdf6796f37a92b2380a01a1b3f6529e39517b52716fcad2", "576d3a9c89912e9d49de43ac9bb16d5f438...
1.543
chembl:1670780
O=C(O)C1CC[C@@](O)(c2ccc(-c3ccccc3)cc2)C1
a6e41ed24722dbb824aaa3974fb9b7e9c0d0e25516a97134beb86f6e770fe1ee
[ "O=C(O)C1CC(O)C1", "O=C(O)C1=C(c2ccc(Cl)cc2)C(O)CC1", "COc1cccc(CC2=C(C(=O)O)CCC2O)c1", "O=C(O)C1=C(c2ccc(Cl)c(Cl)c2)C(O)CC1", "O=C(O)C1=C(Cc2ccccc2)C(O)CC1", "O=C(O)C1CCC(O)C1", "CC1=C(C(=O)O)CCC1O" ]
[ "dbe79c2fcccd4cb0ca5e930789c795c139fd496cc163eeabbc411c5ee2e9b50c", "64d2921bc629f9ce44dd861b41db3f9bff04503a4acbaa4797ec92863784341c", "3c7a15d8001f18157916259df4f9ec99eaaff32155090c1e57c57caae3f3aa73", "b1dcadaf5a757b36fb04a5962f26e4e3a3da850b4d5fe6fc86ac7f343e54e4e6", "4649c6f532a7b4b36e0da22fe28f9d67514...
1.543
chembl:1673771
O=[N+]([O-])c1cn2c(n1)OC[C@H](Oc1ccc(-c3ccc(OC(F)(F)F)cc3)nc1)C2
977f6d95c09269c36ec44c702a56857a1dedb74c68bec2de5b3e36e2f61475fd
[ "O=C(N[C@H]1COc2nc([N+](=O)[O-])cn2C1)c1cccc(OC(F)(F)F)c1", "O=[N+]([O-])c1nc2n(n1)CC(OCc1ccc(-c3ccc(OC(F)(F)F)cc3)cn1)CO2", "O=[N+]([O-])c1cn2c(n1)OC[C@H](NCc1ccc(OC(F)(F)F)cc1)C2", "O=[N+]([O-])c1cn2c(n1)OCCC(OCc1ccc(OCc3ccccc3)cc1)C2", "O=C(Nc1ccccc1OC(F)(F)F)N[C@H]1COc2nc([N+](=O)[O-])cn2C1", "O=C(N[C...
[ "f30bd8cddbe2d2b07e0aa23eff25fc97e517fb91b8217731cc0ac244e5b710ae", "3e83c4d74f02e18154d29cd119703829434223c4946ead9c392e69ed2b31c7d4", "96ed32e7e7bd7a9dc648b1547ff36445b964662665a713c5afa2504e4674cdda", "433929c24f676b0b439cd24a8042efcf16fa9ab4a403ef680a5991d76662ff12", "99ed03530c51027dd84f96bbcac49ed7eab...
1.571333
chembl:1673771
O=[N+]([O-])c1cn2c(n1)OC[C@H](Oc1ccc(-c3ccc(OC(F)(F)F)cc3)nc1)C2
977f6d95c09269c36ec44c702a56857a1dedb74c68bec2de5b3e36e2f61475fd
[ "O=[N+]([O-])c1cn2c(n1)OC[C@H](OCc1ccc(-c3ccc(OC(F)(F)F)c(F)c3)nc1)C2", "O=C(O[C@H]1COc2nc([N+](=O)[O-])cn2C1)N1CCN(c2ccc(OC(F)(F)F)cc2)CC1", "O=[N+]([O-])c1cn2c(n1)OC[C@H](Oc1cc(-c3ccc(F)cc3)ncn1)C2", "O=C(N[C@H]1COc2nc([N+](=O)[O-])cn2C1)c1ccccc1OC(F)(F)F", "O=C(Nc1ccc(OC(F)(F)F)cc1)N[C@@H]1COc2nc([N+](=O...
[ "d594f6f183b274dfc6285cdb49924abe20c94e2f2c176e5b1c7b908f43bd9303", "241dd74760d4a400d4a346f2efaaf5fbd60a25c75743ca372914b22818f8abdd", "7fcfc5d2d10089447832caaf6788dc64a166beb6d10b85fd6e03e406d83caf0e", "1507848e07ee35bef2a043ad5e0adabd3f0f0f43bb0ec61511d182b802543332", "06c1e6d198976664162b82474839edc5bb3...
1.571333
chembl:1673771
O=[N+]([O-])c1cn2c(n1)OC[C@H](Oc1ccc(-c3ccc(F)cc3)nc1)C2
4728ce5c7a2677420481b5bfb34f9b7cd124d684a2ed5230cf3baeeebd125373
[ "O=[N+]([O-])c1cn2c(n1)OC[C@H](OCc1ccc(-c3ccc(OC(F)(F)F)c(F)c3)nc1)C2", "O=C(O[C@H]1COc2nc([N+](=O)[O-])cn2C1)N1CCN(c2ccc(OC(F)(F)F)cc2)CC1", "O=[N+]([O-])c1cn2c(n1)OC[C@H](Oc1cc(-c3ccc(F)cc3)ncn1)C2", "O=C(N[C@H]1COc2nc([N+](=O)[O-])cn2C1)c1ccccc1OC(F)(F)F", "O=C(Nc1ccc(OC(F)(F)F)cc1)N[C@@H]1COc2nc([N+](=O...
[ "d594f6f183b274dfc6285cdb49924abe20c94e2f2c176e5b1c7b908f43bd9303", "241dd74760d4a400d4a346f2efaaf5fbd60a25c75743ca372914b22818f8abdd", "7fcfc5d2d10089447832caaf6788dc64a166beb6d10b85fd6e03e406d83caf0e", "1507848e07ee35bef2a043ad5e0adabd3f0f0f43bb0ec61511d182b802543332", "06c1e6d198976664162b82474839edc5bb3...
1.565
chembl:1673771
O=[N+]([O-])c1cn2c(n1)OC[C@H](Oc1ccc(-c3ccc(F)cc3)nc1)C2
4728ce5c7a2677420481b5bfb34f9b7cd124d684a2ed5230cf3baeeebd125373
[ "O=[N+]([O-])c1cn2c(n1)OC[C@@H](OCc1cccnc1-c1ccc(OC(F)(F)F)cc1)C2", "O=C(Nc1ccc(OC(F)(F)F)cc1)N[C@H]1COc2nc([N+](=O)[O-])cn2C1", "CC1(OCc2ccc(OC(F)(F)F)cc2)COc2nc([N+](=O)[O-])cn2C1", "O=[N+]([O-])c1nc2n(n1)CC(Oc1ccc(OC(F)(F)F)cc1)CO2", "O=[N+]([O-])c1cn2c(n1)OCC(OCc1ccc(OCc3ccccc3)cc1)CC2", "O=[N+]([O-])...
[ "7f543ddbbd80a94f25eda2a9b0a53f441dbb3f977697ec7d5ffc446d3d88fd0a", "669b667e3bdb40c5749ff3fb90b0909efc89558a59bdc108e2bdf18ccbfdae88", "47366f28f7a5e6fd6d6b48c3f8c331f1d8757aab795c0d022d138bd4dca4145b", "c967da40ce707d020cbf7357874e69ac2ac4a2fc20e9e95d7408d71162996b38", "28857e3a537d1ec06557afc3bdac20a795a...
1.565
chembl:1673771
O=[N+]([O-])c1cn2c(n1)OC[C@H](Oc1cccc(-c3ccc(OC(F)(F)F)cc3)n1)C2
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chembl:1673771
O=[N+]([O-])c1cn2c(n1)OC[C@H](Oc1cccc(-c3ccc(OC(F)(F)F)cc3)n1)C2
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chembl:1673771
O=[N+]([O-])c1cn2c(n1)OC[C@H](OCC#Cc1ccc(OC(F)(F)F)cc1)C2
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chembl:1673771
O=[N+]([O-])c1cn2c(n1)OC[C@H](OCC#Cc1ccc(OC(F)(F)F)cc1)C2
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chembl:1673771
O=[N+]([O-])c1cn2c(n1)OC[C@H](Oc1cccc(-c3ccc(F)cc3)n1)C2
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chembl:1673771
O=[N+]([O-])c1cn2c(n1)OC[C@H](Oc1cccc(-c3ccc(F)cc3)n1)C2
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chembl:1673771
O=[N+]([O-])c1cn2c(n1)OC[C@H](Oc1ccc(-c3ccc(F)cc3)cn1)C2
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chembl:1673771
O=[N+]([O-])c1cn2c(n1)OC[C@H](Oc1ccc(-c3ccc(F)cc3)cn1)C2
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chembl:1673771
O=[N+]([O-])c1cn2c(n1)OC[C@H](OCC#Cc1ccc(C(F)(F)F)cn1)C2
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chembl:1673771
O=[N+]([O-])c1cn2c(n1)OC[C@H](OCC#Cc1ccc(C(F)(F)F)cn1)C2
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chembl:1673771
O=[N+]([O-])c1cn2c(n1)OC[C@H](OCc1cccc(-c3ccc(OC(F)(F)F)cc3F)n1)C2
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chembl:1673771
O=[N+]([O-])c1cn2c(n1)OC[C@H](OCc1cccc(-c3ccc(OC(F)(F)F)cc3F)n1)C2
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chembl:1673771
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chembl:1673771
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chembl:1673771
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chembl:1673771
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chembl:1673771
O=[N+]([O-])c1cn2c(n1)OC[C@H](Oc1ccc(OC(F)(F)F)cc1)C2
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chembl:1673771
O=[N+]([O-])c1cn2c(n1)OC[C@H](Oc1ccc(OC(F)(F)F)cc1)C2
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chembl:1673771
O=[N+]([O-])c1cn2c(n1)OC[C@H](OCc1ccc(-c3ccc(OC(F)(F)F)cc3Cl)cn1)C2
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chembl:1673771
O=[N+]([O-])c1cn2c(n1)OC[C@H](OCc1ccc(-c3ccc(OC(F)(F)F)cc3Cl)cn1)C2
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chembl:1673771
O=[N+]([O-])c1cn2c(n1)OC[C@H](OCc1ccc(-c3ccc(OC(F)(F)F)cc3Cl)nc1)C2
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chembl:1673771
O=[N+]([O-])c1cn2c(n1)OC[C@H](OCc1ccc(-c3ccc(OC(F)(F)F)cc3Cl)nc1)C2
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chembl:1673771
O=[N+]([O-])c1cn2c(n1)OC[C@H](OCc1ccc(-c3ccc(OC(F)(F)F)cc3F)cn1)C2
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chembl:1673771
O=[N+]([O-])c1cn2c(n1)OC[C@H](OCc1ccc(-c3ccc(OC(F)(F)F)cc3F)cn1)C2
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1.548667
chembl:1673771
O=[N+]([O-])c1cn2c(n1)OC[C@H](OCc1cccc(-c3ccc(OC(F)(F)F)cc3)n1)C2
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chembl:1673771
O=[N+]([O-])c1cn2c(n1)OC[C@H](OCc1cccc(-c3ccc(OC(F)(F)F)cc3)n1)C2
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1.548333
chembl:1673771
O=[N+]([O-])c1cn2c(n1)OC[C@H](OCc1ccc(-c3ccc(OC(F)F)cc3)cn1)C2
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chembl:1673771
O=[N+]([O-])c1cn2c(n1)OC[C@H](OCc1ccc(-c3ccc(OC(F)F)cc3)cn1)C2
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chembl:1673771
O=[N+]([O-])c1cn2c(n1)OC[C@H](Oc1ccc(-c3ccc(OC(F)(F)F)cc3)cn1)C2
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chembl:1673771
O=[N+]([O-])c1cn2c(n1)OC[C@H](Oc1ccc(-c3ccc(OC(F)(F)F)cc3)cn1)C2
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chembl:1673771
O=[N+]([O-])c1cn2c(n1)OC[C@H](Oc1ncc(-c3ccc(OC(F)(F)F)cc3)cn1)C2
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chembl:1673771
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chembl:1673771
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chembl:1673771
O=[N+]([O-])c1cn2c(n1)OC[C@H](OCc1cccc(-c3ccc(F)cc3)n1)C2
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1.546333
chembl:1673771
O=[N+]([O-])c1cn2c(n1)OC[C@H](OCc1cccc(-c3ccc(F)cc3)n1)C2
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chembl:1673771
O=[N+]([O-])c1cn2c(n1)OC[C@H](Oc1ncc(-c3ccc(F)cc3)cn1)C2
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chembl:1673771
O=[N+]([O-])c1cn2c(n1)OC[C@H](Oc1ncc(-c3ccc(F)cc3)cn1)C2
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chembl:1673771
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chembl:1673771
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chembl:1673771
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chembl:1673771
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chembl:1673771
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chembl:1673771
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chembl:1673771
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312a2303c80b8b64ee24a70868fb2064d0b1c53bbfff59a22d39f125570cf90f
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[ "166e814a728e1969f1ee57775d8ede995e4d27c4bba529b8a9abdc17494d274e", "7f543ddbbd80a94f25eda2a9b0a53f441dbb3f977697ec7d5ffc446d3d88fd0a", "669b667e3bdb40c5749ff3fb90b0909efc89558a59bdc108e2bdf18ccbfdae88", "47366f28f7a5e6fd6d6b48c3f8c331f1d8757aab795c0d022d138bd4dca4145b", "c967da40ce707d020cbf7357874e69ac2ac...
1.543667
chembl:1673771
O=[N+]([O-])c1cn2c(n1)OCC(Oc1ccc(OC(F)(F)F)cc1)C2
edb849188af19ae6bdfb9ece99841076ffe44f1c315bfd5c9fdd9809a8428992
[ "O=[N+]([O-])c1cn2c(n1)OC[C@@H](OCc1ccc(OC(F)(F)F)cc1)C2", "O=[N+]([O-])c1cn2c(n1)OC[C@@H](OCc1cccnc1-c1ccc(OC(F)(F)F)cc1)C2", "O=C(Nc1ccc(OC(F)(F)F)cc1)N[C@H]1COc2nc([N+](=O)[O-])cn2C1", "CC1(OCc2ccc(OC(F)(F)F)cc2)COc2nc([N+](=O)[O-])cn2C1", "O=[N+]([O-])c1nc2n(n1)CC(Oc1ccc(OC(F)(F)F)cc1)CO2", "O=[N+]([O...
[ "166e814a728e1969f1ee57775d8ede995e4d27c4bba529b8a9abdc17494d274e", "7f543ddbbd80a94f25eda2a9b0a53f441dbb3f977697ec7d5ffc446d3d88fd0a", "669b667e3bdb40c5749ff3fb90b0909efc89558a59bdc108e2bdf18ccbfdae88", "47366f28f7a5e6fd6d6b48c3f8c331f1d8757aab795c0d022d138bd4dca4145b", "c967da40ce707d020cbf7357874e69ac2ac...
1.542333
chembl:1673771
O=[N+]([O-])c1cn2c(n1)OCC(Oc1ccc(OC(F)(F)F)cc1)C2
edb849188af19ae6bdfb9ece99841076ffe44f1c315bfd5c9fdd9809a8428992
[ "O=[N+]([O-])c1cn2c(n1)OC[C@H](OCc1ccc(-c3ccc(OC(F)(F)F)cc3)cc1)C2", "O=[N+]([O-])c1nc2n(n1)CC(OCc1ccc(OC(F)(F)F)cc1)CO2", "O=[N+]([O-])c1cc2n(n1)CC(OCc1ccc(OC(F)(F)F)cc1)CO2", "O=[N+]([O-])c1cn2c(n1)OC[C@@H](OCc1ccc(OCc3ccccc3)cc1)C2", "O=[N+]([O-])c1nc2n(n1)CC(Oc1ccc(C(F)(F)F)cn1)CO2", "O=[N+]([O-])c1cn...
[ "672c6e2a2f40061bb9ede144c184dde4da55ab1337c670cdcf8ad24094fb2db8", "7688deadc142defadfcd19a625337342d528f4a6657aaa2b2aa487101bdd13f8", "a2a820be8500b999a55a9fb07e202f1811794ff54e4cedaf176e57a9ba74250a", "96d5829cbe568f9daf472f0cfdb7398a8f5b354be1e95345546fe13f20e6cb27", "0450ae0fcf2498497d1a610055a12ce2f64...
1.542333
chembl:1676735
C[N+](C)(C)CCc1ccc2ccoc2c1
2bb800f52793ed5b275c2bb3aae5ed2d914367a9c649a87c028189d1f143626b
[ "COc1cccc2c1C[N+](C)(C)CC2", "c1cncc(COC2CCCNC2)c1", "COc1cccc(/C=C/C[N+](C)(C)C)c1", "COc1ccccc1C[N+](C)(C)C", "COc1cccc2c1CC[N+](C)(C)C2", "CN1CCC(COCc2cccnc2)C1", "CCOc1cccc(CC[N+](C)(C)C)c1" ]
[ "2eb1d51473dd0fa7439db66d7a8edac2a923ecea4e7f7f7864bba692624b9fe2", "f0e92f3ec29cc8080b45bb2b6f936ebae32c52b7faed9f1252ac903322dbdbaa", "4e462fd7df0a794aeb303d003e578e36dab8e285dc803c4438365166f9bfa2ff", "869f862a5847ea5ea3db5b62bf14b5f8e4250296c85c4df708a9ab057910b64d", "ccabb494fe32fa98281c7a2f23127006798...
1.663
chembl:1676735
C[N+](C)(C)CCc1ccc2ccoc2c1
2bb800f52793ed5b275c2bb3aae5ed2d914367a9c649a87c028189d1f143626b
[ "COc1cccc(C#CC[N+](C)(C)C)c1", "COc1cccc(CC[N+](C)(C)C)c1", "COc1cccc(C(O)C[N+](C)(C)C)c1", "C[N+](C)(C)CCOC(N)=O", "C[N+](C)(C)CCc1cccc(O)c1", "CN1CCCC(OCc2cccnc2)C1", "COc1cccc2c1CCC(C[N+](C)(C)C)C2" ]
[ "cfadbb477844fd832232b67c485838efe38bd66e513ee082dc91f1a7de62b36b", "d6f4660200eb0a863a88926c44f628c11bfcc779c57a600be4464e911ba10eb6", "1a8be913d9d8258258660c21545ef4bfd9d1e66d141cc7c138dd6a7d91ace92b", "953419ff59925c74dc5f7b1b06d1eb8f05e545b706e0e7e57f2c2d11ddb43e5f", "ea067a63dc46809b837f2fee561c7b2616d...
1.663
chembl:1676735
C[N+](C)(C)CCCc1ccc2ccoc2c1
401322a0b852a165cb4cb4064754f0cddbc84be205d281250af0b003da8abf51
[ "COc1cccc(C#CC[N+](C)(C)C)c1", "COc1cccc(CC[N+](C)(C)C)c1", "COc1cccc(C(O)C[N+](C)(C)C)c1", "C[N+](C)(C)CCOC(N)=O", "C[N+](C)(C)CCc1cccc(O)c1", "CN1CCCC(OCc2cccnc2)C1", "COc1cccc2c1CCC(C[N+](C)(C)C)C2" ]
[ "cfadbb477844fd832232b67c485838efe38bd66e513ee082dc91f1a7de62b36b", "d6f4660200eb0a863a88926c44f628c11bfcc779c57a600be4464e911ba10eb6", "1a8be913d9d8258258660c21545ef4bfd9d1e66d141cc7c138dd6a7d91ace92b", "953419ff59925c74dc5f7b1b06d1eb8f05e545b706e0e7e57f2c2d11ddb43e5f", "ea067a63dc46809b837f2fee561c7b2616d...
1.648333
chembl:1676735
C[N+](C)(C)CCCc1ccc2ccoc2c1
401322a0b852a165cb4cb4064754f0cddbc84be205d281250af0b003da8abf51
[ "c1cncc(COCC2CCNC2)c1", "CN(C)C1CCc2cccc(O)c2C1", "COc1cccc2c1C[N+](C)(C)CC2", "c1cncc(COC2CCCNC2)c1", "COc1cccc(/C=C/C[N+](C)(C)C)c1", "COc1ccccc1C[N+](C)(C)C", "COc1cccc2c1CC[N+](C)(C)C2" ]
[ "6a7b5de6cf039f6232848de05de9d67a47193eb9077fa5e44de6bd379129525c", "7c91a1a538cabf19f880fabef41e56525d2c16250d06a0ccbe586e7b449e347d", "2eb1d51473dd0fa7439db66d7a8edac2a923ecea4e7f7f7864bba692624b9fe2", "f0e92f3ec29cc8080b45bb2b6f936ebae32c52b7faed9f1252ac903322dbdbaa", "4e462fd7df0a794aeb303d003e578e36dab...
1.648333
chembl:1676735
COc1cccc(C(=O)C[N+](C)(C)C)c1
aa8b4832bfcceeaec70fbfb65c1df25befd42d54b8402509c59c58f7c15cd44c
[ "c1cncc(COCC2CCNC2)c1", "CN(C)C1CCc2cccc(O)c2C1", "COc1cccc2c1C[N+](C)(C)CC2", "c1cncc(COC2CCCNC2)c1", "COc1cccc(/C=C/C[N+](C)(C)C)c1", "COc1ccccc1C[N+](C)(C)C", "COc1cccc2c1CC[N+](C)(C)C2" ]
[ "6a7b5de6cf039f6232848de05de9d67a47193eb9077fa5e44de6bd379129525c", "7c91a1a538cabf19f880fabef41e56525d2c16250d06a0ccbe586e7b449e347d", "2eb1d51473dd0fa7439db66d7a8edac2a923ecea4e7f7f7864bba692624b9fe2", "f0e92f3ec29cc8080b45bb2b6f936ebae32c52b7faed9f1252ac903322dbdbaa", "4e462fd7df0a794aeb303d003e578e36dab...
1.634
chembl:1676735
COc1cccc(C(=O)C[N+](C)(C)C)c1
aa8b4832bfcceeaec70fbfb65c1df25befd42d54b8402509c59c58f7c15cd44c
[ "CN1CCC(COCc2cccnc2)C1", "CCOc1cccc(CC[N+](C)(C)C)c1", "COc1cccc(C#CC[N+](C)(C)C)c1", "COc1cccc(CC[N+](C)(C)C)c1", "COc1cccc(C(O)C[N+](C)(C)C)c1", "C[N+](C)(C)CCOC(N)=O", "C[N+](C)(C)CCc1cccc(O)c1" ]
[ "fdb935065556007b7a76ee14c6f766be368234cd194d430644227eef282e7e6c", "2eba37ec39cec457f592c51f20606c50646d9c78d749302b66363070696c376f", "cfadbb477844fd832232b67c485838efe38bd66e513ee082dc91f1a7de62b36b", "d6f4660200eb0a863a88926c44f628c11bfcc779c57a600be4464e911ba10eb6", "1a8be913d9d8258258660c21545ef4bfd9d...
1.634
chembl:1676735
COc1cccc(CCC[N+](C)(C)C)c1
9029f56bf55e0fe8f63252ecb37e838064b77b22c46ef7e6c01dd63e99f6a77e
[ "CN1CCC(COCc2cccnc2)C1", "CCOc1cccc(CC[N+](C)(C)C)c1", "COc1cccc(C#CC[N+](C)(C)C)c1", "COc1cccc(CC[N+](C)(C)C)c1", "COc1cccc(C(O)C[N+](C)(C)C)c1", "C[N+](C)(C)CCOC(N)=O", "C[N+](C)(C)CCc1cccc(O)c1" ]
[ "fdb935065556007b7a76ee14c6f766be368234cd194d430644227eef282e7e6c", "2eba37ec39cec457f592c51f20606c50646d9c78d749302b66363070696c376f", "cfadbb477844fd832232b67c485838efe38bd66e513ee082dc91f1a7de62b36b", "d6f4660200eb0a863a88926c44f628c11bfcc779c57a600be4464e911ba10eb6", "1a8be913d9d8258258660c21545ef4bfd9d...
1.624333
chembl:1676735
COc1cccc(CCC[N+](C)(C)C)c1
9029f56bf55e0fe8f63252ecb37e838064b77b22c46ef7e6c01dd63e99f6a77e
[ "CN1CCCC(OCc2cccnc2)C1", "COc1cccc2c1CCC(C[N+](C)(C)C)C2", "c1cncc(COCC2CCNC2)c1", "CN(C)C1CCc2cccc(O)c2C1", "COc1cccc2c1C[N+](C)(C)CC2", "c1cncc(COC2CCCNC2)c1", "COc1cccc(/C=C/C[N+](C)(C)C)c1" ]
[ "ab08f3d8218288a0dc8f56c5231b26fe645ca36a8407f05eebe7ca9d53300cba", "dddc7767c62dbde05ca7d0eb00f3163d8fbf51138a48f025e8975ec010ce7a57", "6a7b5de6cf039f6232848de05de9d67a47193eb9077fa5e44de6bd379129525c", "7c91a1a538cabf19f880fabef41e56525d2c16250d06a0ccbe586e7b449e347d", "2eb1d51473dd0fa7439db66d7a8edac2a92...
1.624333
chembl:1676735
C[N+](C)(C)CC#CCOC1=NOCC1
6b31f2fc5b69bf3a54afcc8cf9e3aff32b3edafc32aaaa87814d0bb7b5e4ced9
[ "CN1CCCC(OCc2cccnc2)C1", "COc1cccc2c1CCC(C[N+](C)(C)C)C2", "c1cncc(COCC2CCNC2)c1", "CN(C)C1CCc2cccc(O)c2C1", "COc1cccc2c1C[N+](C)(C)CC2", "c1cncc(COC2CCCNC2)c1", "COc1cccc(/C=C/C[N+](C)(C)C)c1" ]
[ "ab08f3d8218288a0dc8f56c5231b26fe645ca36a8407f05eebe7ca9d53300cba", "dddc7767c62dbde05ca7d0eb00f3163d8fbf51138a48f025e8975ec010ce7a57", "6a7b5de6cf039f6232848de05de9d67a47193eb9077fa5e44de6bd379129525c", "7c91a1a538cabf19f880fabef41e56525d2c16250d06a0ccbe586e7b449e347d", "2eb1d51473dd0fa7439db66d7a8edac2a92...
1.623667
chembl:1676735
C[N+](C)(C)CC#CCOC1=NOCC1
6b31f2fc5b69bf3a54afcc8cf9e3aff32b3edafc32aaaa87814d0bb7b5e4ced9
[ "COc1ccccc1C[N+](C)(C)C", "COc1cccc2c1CC[N+](C)(C)C2", "CN1CCC(COCc2cccnc2)C1", "CCOc1cccc(CC[N+](C)(C)C)c1", "COc1cccc(C#CC[N+](C)(C)C)c1", "COc1cccc(CC[N+](C)(C)C)c1", "COc1cccc(C(O)C[N+](C)(C)C)c1" ]
[ "869f862a5847ea5ea3db5b62bf14b5f8e4250296c85c4df708a9ab057910b64d", "ccabb494fe32fa98281c7a2f2312700679899dcc91e4cb2b7f0e4dd41a81f02e", "fdb935065556007b7a76ee14c6f766be368234cd194d430644227eef282e7e6c", "2eba37ec39cec457f592c51f20606c50646d9c78d749302b66363070696c376f", "cfadbb477844fd832232b67c485838efe38...
1.623667
chembl:1676735
C[N+](C)(C)C1CCc2ccc3ccoc3c2C1
773740ab7ac87ddbef416a83ca48e9dabef4eba45d9c641e96a28950feda6817
[ "COc1ccccc1C[N+](C)(C)C", "COc1cccc2c1CC[N+](C)(C)C2", "CN1CCC(COCc2cccnc2)C1", "CCOc1cccc(CC[N+](C)(C)C)c1", "COc1cccc(C#CC[N+](C)(C)C)c1", "COc1cccc(CC[N+](C)(C)C)c1", "COc1cccc(C(O)C[N+](C)(C)C)c1" ]
[ "869f862a5847ea5ea3db5b62bf14b5f8e4250296c85c4df708a9ab057910b64d", "ccabb494fe32fa98281c7a2f2312700679899dcc91e4cb2b7f0e4dd41a81f02e", "fdb935065556007b7a76ee14c6f766be368234cd194d430644227eef282e7e6c", "2eba37ec39cec457f592c51f20606c50646d9c78d749302b66363070696c376f", "cfadbb477844fd832232b67c485838efe38...
1.622333
chembl:1676735
C[N+](C)(C)C1CCc2ccc3ccoc3c2C1
773740ab7ac87ddbef416a83ca48e9dabef4eba45d9c641e96a28950feda6817
[ "C[N+](C)(C)CCOC(N)=O", "C[N+](C)(C)CCc1cccc(O)c1", "CN1CCCC(OCc2cccnc2)C1", "COc1cccc2c1CCC(C[N+](C)(C)C)C2", "c1cncc(COCC2CCNC2)c1", "CN(C)C1CCc2cccc(O)c2C1", "COc1cccc2c1C[N+](C)(C)CC2" ]
[ "953419ff59925c74dc5f7b1b06d1eb8f05e545b706e0e7e57f2c2d11ddb43e5f", "ea067a63dc46809b837f2fee561c7b2616d680b4c35cae5c8b1c819fa1729d8b", "ab08f3d8218288a0dc8f56c5231b26fe645ca36a8407f05eebe7ca9d53300cba", "dddc7767c62dbde05ca7d0eb00f3163d8fbf51138a48f025e8975ec010ce7a57", "6a7b5de6cf039f6232848de05de9d67a471...
1.622333
chembl:1676735
CNCCc1cccc(OC)c1
e344804a065b2f1806d25295b3ef5b49b74163d25e7a45a44a9061fd190ac367
[ "C[N+](C)(C)CCOC(N)=O", "C[N+](C)(C)CCc1cccc(O)c1", "CN1CCCC(OCc2cccnc2)C1", "COc1cccc2c1CCC(C[N+](C)(C)C)C2", "c1cncc(COCC2CCNC2)c1", "CN(C)C1CCc2cccc(O)c2C1", "COc1cccc2c1C[N+](C)(C)CC2" ]
[ "953419ff59925c74dc5f7b1b06d1eb8f05e545b706e0e7e57f2c2d11ddb43e5f", "ea067a63dc46809b837f2fee561c7b2616d680b4c35cae5c8b1c819fa1729d8b", "ab08f3d8218288a0dc8f56c5231b26fe645ca36a8407f05eebe7ca9d53300cba", "dddc7767c62dbde05ca7d0eb00f3163d8fbf51138a48f025e8975ec010ce7a57", "6a7b5de6cf039f6232848de05de9d67a471...
1.612667
chembl:1676735
CNCCc1cccc(OC)c1
e344804a065b2f1806d25295b3ef5b49b74163d25e7a45a44a9061fd190ac367
[ "c1cncc(COC2CCCNC2)c1", "COc1cccc(/C=C/C[N+](C)(C)C)c1", "COc1ccccc1C[N+](C)(C)C", "COc1cccc2c1CC[N+](C)(C)C2", "CN1CCC(COCc2cccnc2)C1", "CCOc1cccc(CC[N+](C)(C)C)c1", "COc1cccc(C#CC[N+](C)(C)C)c1" ]
[ "f0e92f3ec29cc8080b45bb2b6f936ebae32c52b7faed9f1252ac903322dbdbaa", "4e462fd7df0a794aeb303d003e578e36dab8e285dc803c4438365166f9bfa2ff", "869f862a5847ea5ea3db5b62bf14b5f8e4250296c85c4df708a9ab057910b64d", "ccabb494fe32fa98281c7a2f2312700679899dcc91e4cb2b7f0e4dd41a81f02e", "fdb935065556007b7a76ee14c6f766be368...
1.612667
chembl:1676736
C[N+](C)(C)CC#CCOC1=NOCC1
6b31f2fc5b69bf3a54afcc8cf9e3aff32b3edafc32aaaa87814d0bb7b5e4ced9
[ "C[N+]1(C)CCC(OCc2nccs2)C1", "COc1cccc(C#CC[N+](C)(C)C)c1", "c1cncc(COC2CCCNC2)c1", "CN1CCCC(OCc2cccnc2)C1", "CCOc1cccc(CC[N+](C)(C)C)c1", "COc1cccc(CC[N+](C)(C)C)c1", "C[N+](C)(C)CCc1ccc2c(c1)OCC2" ]
[ "504a3c1b2ae0fadf8db24342e47ae2229c283ad15a4834407334de890d58a413", "cfadbb477844fd832232b67c485838efe38bd66e513ee082dc91f1a7de62b36b", "f0e92f3ec29cc8080b45bb2b6f936ebae32c52b7faed9f1252ac903322dbdbaa", "ab08f3d8218288a0dc8f56c5231b26fe645ca36a8407f05eebe7ca9d53300cba", "2eba37ec39cec457f592c51f20606c50646...
1.685333
chembl:1676736
C[N+](C)(C)CC#CCOC1=NOCC1
6b31f2fc5b69bf3a54afcc8cf9e3aff32b3edafc32aaaa87814d0bb7b5e4ced9
[ "CN1CCC(COCc2cccnc2)C1", "C[N+](C)(C)CCc1cccc(O)c1", "COc1cccc2c1CCC(C[N+](C)(C)C)C2", "COc1cccc(C2CC2C[N+](C)(C)C)c1", "COc1cccc(/C=C/C[N+](C)(C)C)c1", "c1cncc(COCC2CCNC2)c1", "COc1cccc2c1CC[N+](C)(C)C2" ]
[ "fdb935065556007b7a76ee14c6f766be368234cd194d430644227eef282e7e6c", "ea067a63dc46809b837f2fee561c7b2616d680b4c35cae5c8b1c819fa1729d8b", "dddc7767c62dbde05ca7d0eb00f3163d8fbf51138a48f025e8975ec010ce7a57", "2f5889006e6c88f35545a30598f33802142fbaae7eadd8b0065835099aa0adee", "4e462fd7df0a794aeb303d003e578e36dab...
1.685333
chembl:1676736
C[N+](C)(C)CCc1ccc2ccoc2c1
2bb800f52793ed5b275c2bb3aae5ed2d914367a9c649a87c028189d1f143626b
[ "CN1CCC(COCc2cccnc2)C1", "C[N+](C)(C)CCc1cccc(O)c1", "COc1cccc2c1CCC(C[N+](C)(C)C)C2", "COc1cccc(C2CC2C[N+](C)(C)C)c1", "COc1cccc(/C=C/C[N+](C)(C)C)c1", "c1cncc(COCC2CCNC2)c1", "COc1cccc2c1CC[N+](C)(C)C2" ]
[ "fdb935065556007b7a76ee14c6f766be368234cd194d430644227eef282e7e6c", "ea067a63dc46809b837f2fee561c7b2616d680b4c35cae5c8b1c819fa1729d8b", "dddc7767c62dbde05ca7d0eb00f3163d8fbf51138a48f025e8975ec010ce7a57", "2f5889006e6c88f35545a30598f33802142fbaae7eadd8b0065835099aa0adee", "4e462fd7df0a794aeb303d003e578e36dab...
1.636667
chembl:1676736
C[N+](C)(C)CCc1ccc2ccoc2c1
2bb800f52793ed5b275c2bb3aae5ed2d914367a9c649a87c028189d1f143626b
[ "COc1cccc(C(O)C[N+](C)(C)C)c1", "CN(C)C1CCc2cccc(O)c2C1", "COc1ccccc1C[N+](C)(C)C", "C[N+]1(C)CCC(OCc2nccs2)C1", "COc1cccc(C#CC[N+](C)(C)C)c1", "c1cncc(COC2CCCNC2)c1", "CN1CCCC(OCc2cccnc2)C1" ]
[ "1a8be913d9d8258258660c21545ef4bfd9d1e66d141cc7c138dd6a7d91ace92b", "7c91a1a538cabf19f880fabef41e56525d2c16250d06a0ccbe586e7b449e347d", "869f862a5847ea5ea3db5b62bf14b5f8e4250296c85c4df708a9ab057910b64d", "504a3c1b2ae0fadf8db24342e47ae2229c283ad15a4834407334de890d58a413", "cfadbb477844fd832232b67c485838efe38...
1.636667