assay_uid
stringlengths
9
15
positive_smiles
stringlengths
2
615
positive_smiles_hash
stringlengths
64
64
negative_smiles
listlengths
7
7
negative_smiles_hashes
listlengths
7
7
example_weight
float32
1
1.71
chembl:1785635
CCOC(=O)CNC(=O)NC1CCN(c2ccc(/C=C/c3cc(Cl)cc(Cn4ccnc4)c3)cc2)CC1
298a2b0a8229331facc7307205094abc78d32545d03c10337d99e1cc3a861493
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1.646333
chembl:1785635
CCOC(=O)CNC(=O)NC1CCN(c2ccc(/C=C/c3cc(Cl)cc(Cn4ccnc4)c3)cc2)CC1
298a2b0a8229331facc7307205094abc78d32545d03c10337d99e1cc3a861493
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1.646333
chembl:1785635
CC(C)S(=O)(=O)N1CCN(c2ccc(/C=C/c3cc(Cl)cc(Cn4ccnc4)c3)cc2)CC1
26704057248b31b23833d446e58811405c547dc97b6cc9316415f5808189e7f5
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1.644
chembl:1785635
CC(C)S(=O)(=O)N1CCN(c2ccc(/C=C/c3cc(Cl)cc(Cn4ccnc4)c3)cc2)CC1
26704057248b31b23833d446e58811405c547dc97b6cc9316415f5808189e7f5
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1.644
chembl:1785635
O=[N+]([O-])c1cccc(S(=O)(=O)N2CCN(c3ccc(/C=C/c4cc(Cl)cc(Cn5ccnc5)c4)cc3)CC2)c1
dd783485aa0bb85b93ea78563851fc698c3afe7bb6815d880874201fb9a5e6d2
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1.635
chembl:1785635
O=[N+]([O-])c1cccc(S(=O)(=O)N2CCN(c3ccc(/C=C/c4cc(Cl)cc(Cn5ccnc5)c4)cc3)CC2)c1
dd783485aa0bb85b93ea78563851fc698c3afe7bb6815d880874201fb9a5e6d2
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1.635
chembl:1785635
CC(C)S(=O)(=O)N1CCN(c2ccc(/C=C/c3cc(F)cc(-c4ccncc4)c3)cc2)CC1
e9ada42c6cd7cd39fb037e2a6d5702ca49ca3e5fb96a3643cbec8a53c91c6047
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1.632333
chembl:1785635
CC(C)S(=O)(=O)N1CCN(c2ccc(/C=C/c3cc(F)cc(-c4ccncc4)c3)cc2)CC1
e9ada42c6cd7cd39fb037e2a6d5702ca49ca3e5fb96a3643cbec8a53c91c6047
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1.632333
chembl:1785635
CCOC(=O)CNC(=O)N1CCN(c2ccc(/C=C/c3cc(Cl)cc(Cn4ccnc4)c3)cc2)CC1
c08d8d37ad9ffbacde09f7c3acef7326b0a374f30f0689b5fd4053b7462c6d2b
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1.628333
chembl:1785635
CCOC(=O)CNC(=O)N1CCN(c2ccc(/C=C/c3cc(Cl)cc(Cn4ccnc4)c3)cc2)CC1
c08d8d37ad9ffbacde09f7c3acef7326b0a374f30f0689b5fd4053b7462c6d2b
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1.628333
chembl:1785635
N#Cc1cccc(CN2CCN(c3ccc(/C=C/c4cc(Cl)cc(Cn5ccnc5)c4)cc3)CC2)c1
a5a3eb8fb36d3ead7a48e40eae3f5825294f0980a0f9a340700534f8b74c74d1
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1.626333
chembl:1785635
N#Cc1cccc(CN2CCN(c3ccc(/C=C/c4cc(Cl)cc(Cn5ccnc5)c4)cc3)CC2)c1
a5a3eb8fb36d3ead7a48e40eae3f5825294f0980a0f9a340700534f8b74c74d1
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1.626333
chembl:1785635
O=S(=O)(N1CCN(c2ccc(/C=C/c3cc(F)cc(-c4ccncc4)c3)cc2)CC1)C(F)(F)F
5417fcababc321ab5851b6ca7edd0b5be906ec2d454f029049b1fed7328df5dd
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1.625
chembl:1785635
O=S(=O)(N1CCN(c2ccc(/C=C/c3cc(F)cc(-c4ccncc4)c3)cc2)CC1)C(F)(F)F
5417fcababc321ab5851b6ca7edd0b5be906ec2d454f029049b1fed7328df5dd
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1.625
chembl:1785635
O=S(=O)(C1CC1)N1CCN(c2ccc(/C=C/c3cc(Cl)cc(Cn4ccnc4)c3)cc2)CC1
d292100e8daec205a57afc83bcf5512233600db8f19461542bf84ce1988502ce
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1.624
chembl:1785635
O=S(=O)(C1CC1)N1CCN(c2ccc(/C=C/c3cc(Cl)cc(Cn4ccnc4)c3)cc2)CC1
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chembl:1785635
O=S(=O)(C1CC1)N1CCN(c2ccc(/C=C/c3cc(F)cc(-c4ccncc4)c3)cc2)CC1
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chembl:1785635
O=S(=O)(C1CC1)N1CCN(c2ccc(/C=C/c3cc(F)cc(-c4ccncc4)c3)cc2)CC1
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1.622
chembl:1785635
O=S(=O)(C1CC1)N1CCN(c2ccc(/C=C/c3cc(Cl)cc(-c4ccncc4)c3)cc2)CC1
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1.621
chembl:1785635
O=S(=O)(C1CC1)N1CCN(c2ccc(/C=C/c3cc(Cl)cc(-c4ccncc4)c3)cc2)CC1
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chembl:1785635
CC(=O)N1CCN(c2ccc(/C=C/c3cc(F)cc(-c4ccncc4)c3)cc2)CC1
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chembl:1785635
CC(=O)N1CCN(c2ccc(/C=C/c3cc(F)cc(-c4ccncc4)c3)cc2)CC1
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1.620667
chembl:1785635
Fc1cc(CCc2ccc(-c3ccncc3)cc2)cc(-c2ccncc2)c1
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1.618667
chembl:1785635
Fc1cc(CCc2ccc(-c3ccncc3)cc2)cc(-c2ccncc2)c1
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chembl:1785635
O=S(=O)(c1cccc(OC(F)(F)F)c1)N1CCN(c2ccc(/C=C/c3cc(Cl)cc(Cn4ccnc4)c3)cc2)CC1
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1.617667
chembl:1785635
O=S(=O)(c1cccc(OC(F)(F)F)c1)N1CCN(c2ccc(/C=C/c3cc(Cl)cc(Cn4ccnc4)c3)cc2)CC1
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1.617667
chembl:1785635
CCS(=O)(=O)N1CCN(c2ccc(/C=C/c3cc(F)cc(-c4ccncc4)c3)cc2)CC1
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1.617667
chembl:1785635
CCS(=O)(=O)N1CCN(c2ccc(/C=C/c3cc(F)cc(-c4ccncc4)c3)cc2)CC1
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1.617667
chembl:1785635
CCS(=O)(=O)N1CCN(c2ccc(/C=C/c3cc(Cl)cc(Cn4ccnc4)c3)cc2)CC1
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1.617333
chembl:1785635
CCS(=O)(=O)N1CCN(c2ccc(/C=C/c3cc(Cl)cc(Cn4ccnc4)c3)cc2)CC1
14cfd420e021efe574d8def963dbf2e97406960c10fe5bb4e10720005ff1bef1
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1.617333
chembl:1785635
CC(C)S(=O)(=O)N1CCN(c2ccc(/C=C/c3cc(Cl)cc(-c4ccncc4)c3)cc2)CC1
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1.616667
chembl:1785635
CC(C)S(=O)(=O)N1CCN(c2ccc(/C=C/c3cc(Cl)cc(-c4ccncc4)c3)cc2)CC1
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1.616667
chembl:1785635
Clc1cc(/C=C/c2ccc(N3CCN(CC4CC4)CC3)cc2)cc(Cn2ccnc2)c1
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1.616
chembl:1785635
Clc1cc(/C=C/c2ccc(N3CCN(CC4CC4)CC3)cc2)cc(Cn2ccnc2)c1
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1.616
chembl:1785635
CC(C)S(=O)(=O)N1CCN(c2ccc(/C=C/c3cc(F)cc(Cn4ccnc4)c3)cc2)CC1
78f47d67143086b040d16018aa9e9217be42853099a349edde95f6044a85a9c1
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1.613667
chembl:1785635
CC(C)S(=O)(=O)N1CCN(c2ccc(/C=C/c3cc(F)cc(Cn4ccnc4)c3)cc2)CC1
78f47d67143086b040d16018aa9e9217be42853099a349edde95f6044a85a9c1
[ "O=C(c1cccc([N+](=O)[O-])c1)N1CCN(c2ccc(/C=C/c3cc(Cl)cc(Cn4ccnc4)c3)cc2)CC1", "CC(=O)N1CCN(c2ccc(/C=C/c3cc(F)cc(-c4cccnc4)c3)cc2)CC1", "CC(=O)N1CCN(c2ccc(/C=C/c3cc(Cl)cc(Cc4cccnc4)c3)cc2)CC1", "N=C(N)N1CCN(c2ccc(/C=C/c3cc(F)cc(Cn4ccnc4)c3)cc2)CC1", "Fc1cc(/C=C/c2ccc(N3CCN(C4=NCCO4)CC3)cc2)cc(Cn2ccnc2)c1", ...
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1.613667
chembl:1785635
CS(=O)(=O)N1CCN(c2ccc(/C=C/c3cc(F)cc(-c4ccncc4)c3)cc2)CC1
935c5a89ba93fd5f6c720b91028f32574fa9e41c891ec7212fd8fa073689db4c
[ "O=C(c1cccc([N+](=O)[O-])c1)N1CCN(c2ccc(/C=C/c3cc(Cl)cc(Cn4ccnc4)c3)cc2)CC1", "CC(=O)N1CCN(c2ccc(/C=C/c3cc(F)cc(-c4cccnc4)c3)cc2)CC1", "CC(=O)N1CCN(c2ccc(/C=C/c3cc(Cl)cc(Cc4cccnc4)c3)cc2)CC1", "N=C(N)N1CCN(c2ccc(/C=C/c3cc(F)cc(Cn4ccnc4)c3)cc2)CC1", "Fc1cc(/C=C/c2ccc(N3CCN(C4=NCCO4)CC3)cc2)cc(Cn2ccnc2)c1", ...
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1.612667
chembl:1785635
CS(=O)(=O)N1CCN(c2ccc(/C=C/c3cc(F)cc(-c4ccncc4)c3)cc2)CC1
935c5a89ba93fd5f6c720b91028f32574fa9e41c891ec7212fd8fa073689db4c
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1.612667
chembl:1785635
Fc1cc(/C=C/c2ccc(N3CCN(CC4CC4)CC3)cc2)cc(-c2ccncc2)c1
97391629f52159f691cdbf1f5f22f12bec0e918e44177fc60540f77502cf539c
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1.612
chembl:1785635
Fc1cc(/C=C/c2ccc(N3CCN(CC4CC4)CC3)cc2)cc(-c2ccncc2)c1
97391629f52159f691cdbf1f5f22f12bec0e918e44177fc60540f77502cf539c
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1.612
chembl:1785635
CS(=O)(=O)N1CCN(c2ccc(/C=C/c3cc(Cl)cc(-c4ccncc4)c3)cc2)CC1
7a56746df454f27a29ed7909342e5bef8b424db08b0c25784abf93237e8b5f17
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1.611
chembl:1785635
CS(=O)(=O)N1CCN(c2ccc(/C=C/c3cc(Cl)cc(-c4ccncc4)c3)cc2)CC1
7a56746df454f27a29ed7909342e5bef8b424db08b0c25784abf93237e8b5f17
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1.611
chembl:1785635
Fc1cc(/C=C/c2ccc(-c3ccncc3)cc2)cc(-c2ccncc2)c1
4803f0feab7500b52a4c9cea2068a7b26073f967ccc611d1cba519df5ed9c6fd
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1.610667
chembl:1785635
Fc1cc(/C=C/c2ccc(-c3ccncc3)cc2)cc(-c2ccncc2)c1
4803f0feab7500b52a4c9cea2068a7b26073f967ccc611d1cba519df5ed9c6fd
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1.610667
chembl:1801488
COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(OC)cc4)ccc32)cc1
9382cf5f0c95127019f4e5ef51ba1708b1b45bfcc7f62038ddaf8a897487d726
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1.585
chembl:1801488
COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(OC)cc4)ccc32)cc1
9382cf5f0c95127019f4e5ef51ba1708b1b45bfcc7f62038ddaf8a897487d726
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[ "97a744cb5940b79956a6910f17b61b88615d0ed985e34754bdcfb5f08343f85c", "f6b1d48c1cdc5d50696ad6d7d21f1c2645fe394000ec5c71ea7f962184ee5f60", "7ebdb017871fdbee29b177bb780126f50c1e46df285b7c8f156a1be1e33b36fe", "e6101de344a3cac7c0cc98ffe2e9eac89cf6b3e5ca8a2b34ebb949da80c4e8ec", "fa87c5cd9059dc443914cb124a0732e4d6c...
1.585
chembl:1801488
COc1ccc(-c2ccc3c(c2)C(=O)C(=O)N3Cc2ccccc2OC)cc1
9109f8a48d01104b4508563590222fa0f9245114846614f2b8e5e0beb6713e49
[ "Cc1ccc2c(c1)C(=O)C(=O)N2", "O=C1Nc2ccc(F)cc2C1=O", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(C)cc4)ccc32)cc1", "O=C1Nc2ccc(Cl)cc2C1=O", "COc1ccc(CN2C(=O)/C(=C\\c3ccc(C(F)(F)F)cc3)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3c(-c4ccc(OC)cc4)cccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3ccc(-c4ccc(OC)cc4)cc32)c...
[ "97a744cb5940b79956a6910f17b61b88615d0ed985e34754bdcfb5f08343f85c", "f6b1d48c1cdc5d50696ad6d7d21f1c2645fe394000ec5c71ea7f962184ee5f60", "7ebdb017871fdbee29b177bb780126f50c1e46df285b7c8f156a1be1e33b36fe", "e6101de344a3cac7c0cc98ffe2e9eac89cf6b3e5ca8a2b34ebb949da80c4e8ec", "fa87c5cd9059dc443914cb124a0732e4d6c...
1.571333
chembl:1801488
COc1ccc(-c2ccc3c(c2)C(=O)C(=O)N3Cc2ccccc2OC)cc1
9109f8a48d01104b4508563590222fa0f9245114846614f2b8e5e0beb6713e49
[ "O=C1Nc2ccccc2C1=O", "COc1ccc(Cn2c(O)c(N=O)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(OC)c(OC)c4)ccc32)cc1", "O=C1Nc2ccc(Br)cc2C1=O", "COc1ccc(Cn2c(O)cc3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(OC(C)C)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(F)(F)c3cc(-c4ccc(OC)cc4)...
[ "5518611e3076e1a5209c531d063d23cd36df581395ed72bcc8bf515b3f873196", "c048a48684f447b7c7cdbf38eae6f30daa409c67f8fc19d29d202e29de024985", "cb731fcf6345af364441c9254f47cd5950257cfbd0a1cc3a8437de573d943164", "2338bccb34ceebc4708f442271a99b0f3d6eca56b3aef0f43d17be4705da81c4", "404f1da9ee430e576f53cb872eaa3910eb1...
1.571333
chembl:1801488
COc1ccc(-c2ccc3c(c2)C(=O)C(=O)N3Cc2ccc(Cl)cc2)cc1
ae25dbd474b35cbedceebb5497389ae190185778d63349f679654f95d051dd2c
[ "O=C1Nc2ccccc2C1=O", "COc1ccc(Cn2c(O)c(N=O)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(OC)c(OC)c4)ccc32)cc1", "O=C1Nc2ccc(Br)cc2C1=O", "COc1ccc(Cn2c(O)cc3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(OC(C)C)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(F)(F)c3cc(-c4ccc(OC)cc4)...
[ "5518611e3076e1a5209c531d063d23cd36df581395ed72bcc8bf515b3f873196", "c048a48684f447b7c7cdbf38eae6f30daa409c67f8fc19d29d202e29de024985", "cb731fcf6345af364441c9254f47cd5950257cfbd0a1cc3a8437de573d943164", "2338bccb34ceebc4708f442271a99b0f3d6eca56b3aef0f43d17be4705da81c4", "404f1da9ee430e576f53cb872eaa3910eb1...
1.561667
chembl:1801488
COc1ccc(-c2ccc3c(c2)C(=O)C(=O)N3Cc2ccc(Cl)cc2)cc1
ae25dbd474b35cbedceebb5497389ae190185778d63349f679654f95d051dd2c
[ "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccncc4)ccc32)cc1", "COc1ccc(CN2C(=O)C3(OCCO3)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccccc4OC)ccc32)cc1", "COc1ccc(-c2ccc3c(c2)C(=O)C(=O)N3c2ccc(OC)cc2)cc1", "COc1ccc(CN2C(=O)/C(=C\\c3ccccc3)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc2c(c1)C(=O)C(=O)N2", "C...
[ "9962fd6f7c70ea95458960df7d9e3f60e54ac931b9d8598965b9379cdf1701cb", "20ad785f524a001eb45b3ace687e3601c878131a62e1f27fb7dbf284990240fa", "aabe0eb965b5e933f141ef01bc7fee378fef1d39eee6e431df7cb24b5376bcf4", "c285b904f8d4adad8afc74c354125bc2f04baf66f6e20f5206886dfa5539a159", "886216776a89cadcf0fcd4242f034b8cb7f...
1.561667
chembl:1801488
COc1ccc(-c2ccc3c(c2)C(=O)C(=O)N3Cc2cccc(Cl)c2)cc1
ff22e989e26db1d112960f7edca5bcffae570eeb8246386b2b759fc2aa21d8a2
[ "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccncc4)ccc32)cc1", "COc1ccc(CN2C(=O)C3(OCCO3)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccccc4OC)ccc32)cc1", "COc1ccc(-c2ccc3c(c2)C(=O)C(=O)N3c2ccc(OC)cc2)cc1", "COc1ccc(CN2C(=O)/C(=C\\c3ccccc3)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc2c(c1)C(=O)C(=O)N2", "C...
[ "9962fd6f7c70ea95458960df7d9e3f60e54ac931b9d8598965b9379cdf1701cb", "20ad785f524a001eb45b3ace687e3601c878131a62e1f27fb7dbf284990240fa", "aabe0eb965b5e933f141ef01bc7fee378fef1d39eee6e431df7cb24b5376bcf4", "c285b904f8d4adad8afc74c354125bc2f04baf66f6e20f5206886dfa5539a159", "886216776a89cadcf0fcd4242f034b8cb7f...
1.558333
chembl:1801488
COc1ccc(-c2ccc3c(c2)C(=O)C(=O)N3Cc2cccc(Cl)c2)cc1
ff22e989e26db1d112960f7edca5bcffae570eeb8246386b2b759fc2aa21d8a2
[ "COc1ccc(CN2C(=O)/C(=C\\c3ccc(C(C)C)cc3)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(F)c(Cl)c4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(O)cc4)ccc32)cc1", "CCC=Cc1ccc2[nH]c(O)c(O)c2c1", "COc1ccc(CN2C(=O)C(C)(O)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "Cc1ccc2c(c1)C(=O)C(=O)N2", "O=C1Nc2ccc...
[ "1d58312e01e6f598a39ea92b894982aef4a0265cb88e02aaaf4850a8fb6505d3", "b93ae4854fa6a37bddc5d1ade66bf449bf0604f59f312c43a0e50aa833e55593", "274bad82abd467b1c7ac433d739606ae037c7fdd90342fa7742e233eff8fa5e3", "d62311babd26106395c51df3a7116b5c5085d0ee43a289a10c773c8f011c01f7", "90388bcdeadc46688b50621eceaef1ac7eb...
1.558333
chembl:1801488
COc1ccc(-c2ccc3c(c2)C(=O)C(=O)N3Cc2ccc(C)cc2)cc1
4029969be580d9467735581e198b1905c8c3a5448d0caed5ee12d05d975634b8
[ "COc1ccc(CN2C(=O)/C(=C\\c3ccc(C(C)C)cc3)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(F)c(Cl)c4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(O)cc4)ccc32)cc1", "CCC=Cc1ccc2[nH]c(O)c(O)c2c1", "COc1ccc(CN2C(=O)C(C)(O)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "Cc1ccc2c(c1)C(=O)C(=O)N2", "O=C1Nc2ccc...
[ "1d58312e01e6f598a39ea92b894982aef4a0265cb88e02aaaf4850a8fb6505d3", "b93ae4854fa6a37bddc5d1ade66bf449bf0604f59f312c43a0e50aa833e55593", "274bad82abd467b1c7ac433d739606ae037c7fdd90342fa7742e233eff8fa5e3", "d62311babd26106395c51df3a7116b5c5085d0ee43a289a10c773c8f011c01f7", "90388bcdeadc46688b50621eceaef1ac7eb...
1.557667
chembl:1801488
COc1ccc(-c2ccc3c(c2)C(=O)C(=O)N3Cc2ccc(C)cc2)cc1
4029969be580d9467735581e198b1905c8c3a5448d0caed5ee12d05d975634b8
[ "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(C)cc4)ccc32)cc1", "O=C1Nc2ccc(Cl)cc2C1=O", "COc1ccc(CN2C(=O)/C(=C\\c3ccc(C(F)(F)F)cc3)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3c(-c4ccc(OC)cc4)cccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3ccc(-c4ccc(OC)cc4)cc32)cc1", "O=C1Nc2ccccc2C1=O", "COc1ccc(Cn2c(O)c(N=O)c3cc...
[ "7ebdb017871fdbee29b177bb780126f50c1e46df285b7c8f156a1be1e33b36fe", "e6101de344a3cac7c0cc98ffe2e9eac89cf6b3e5ca8a2b34ebb949da80c4e8ec", "fa87c5cd9059dc443914cb124a0732e4d6cd889e2af559934d0df92c91d543ba", "1486d5ee417d89c8005180d7e9a366e473858b9845c47a35aecc20684809711c", "c1aed19ed4670b9363ea4f89904570e91ae...
1.557667
chembl:1801488
CC[C@@]1(O)C(=O)OCc2c1cc1n(c2=O)Cc2cc3ccccc3nc2-1
e52bf76887e001a7500c71cc7243bda87e9313846267a9700753c970e4425e4d
[ "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(C)cc4)ccc32)cc1", "O=C1Nc2ccc(Cl)cc2C1=O", "COc1ccc(CN2C(=O)/C(=C\\c3ccc(C(F)(F)F)cc3)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3c(-c4ccc(OC)cc4)cccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3ccc(-c4ccc(OC)cc4)cc32)cc1", "O=C1Nc2ccccc2C1=O", "COc1ccc(Cn2c(O)c(N=O)c3cc...
[ "7ebdb017871fdbee29b177bb780126f50c1e46df285b7c8f156a1be1e33b36fe", "e6101de344a3cac7c0cc98ffe2e9eac89cf6b3e5ca8a2b34ebb949da80c4e8ec", "fa87c5cd9059dc443914cb124a0732e4d6cd889e2af559934d0df92c91d543ba", "1486d5ee417d89c8005180d7e9a366e473858b9845c47a35aecc20684809711c", "c1aed19ed4670b9363ea4f89904570e91ae...
1.556
chembl:1801488
CC[C@@]1(O)C(=O)OCc2c1cc1n(c2=O)Cc2cc3ccccc3nc2-1
e52bf76887e001a7500c71cc7243bda87e9313846267a9700753c970e4425e4d
[ "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(OC)c(OC)c4)ccc32)cc1", "O=C1Nc2ccc(Br)cc2C1=O", "COc1ccc(Cn2c(O)cc3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(OC(C)C)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(F)(F)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccncc4)ccc32)cc1", "COc1ccc(CN2C...
[ "cb731fcf6345af364441c9254f47cd5950257cfbd0a1cc3a8437de573d943164", "2338bccb34ceebc4708f442271a99b0f3d6eca56b3aef0f43d17be4705da81c4", "404f1da9ee430e576f53cb872eaa3910eb16a5d65055e950ca34f5e0c991d266", "c4990598cc291b556fff63f69ade724ce17fa523a39c2b6b813e49927f6d1a26", "16076c7e9c9579ef55f00066ad292b022ba...
1.556
chembl:1801488
COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(Cl)cc4)ccc32)cc1
33ad19b1ca515fdf2a07ad33a446e8eefc06b90cc462bb477bc4577797df4f7d
[ "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(OC)c(OC)c4)ccc32)cc1", "O=C1Nc2ccc(Br)cc2C1=O", "COc1ccc(Cn2c(O)cc3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(OC(C)C)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(F)(F)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccncc4)ccc32)cc1", "COc1ccc(CN2C...
[ "cb731fcf6345af364441c9254f47cd5950257cfbd0a1cc3a8437de573d943164", "2338bccb34ceebc4708f442271a99b0f3d6eca56b3aef0f43d17be4705da81c4", "404f1da9ee430e576f53cb872eaa3910eb16a5d65055e950ca34f5e0c991d266", "c4990598cc291b556fff63f69ade724ce17fa523a39c2b6b813e49927f6d1a26", "16076c7e9c9579ef55f00066ad292b022ba...
1.555667
chembl:1801488
COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(Cl)cc4)ccc32)cc1
33ad19b1ca515fdf2a07ad33a446e8eefc06b90cc462bb477bc4577797df4f7d
[ "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccccc4OC)ccc32)cc1", "COc1ccc(-c2ccc3c(c2)C(=O)C(=O)N3c2ccc(OC)cc2)cc1", "COc1ccc(CN2C(=O)/C(=C\\c3ccccc3)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc2c(c1)C(=O)C(=O)N2", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc5ccccc5c4)ccc32)cc1", "COc1ccc(CN2C(=O)/C(=C\\c3ccc(C(C)C)cc3)c3cc(-c4ccc(OC)...
[ "aabe0eb965b5e933f141ef01bc7fee378fef1d39eee6e431df7cb24b5376bcf4", "c285b904f8d4adad8afc74c354125bc2f04baf66f6e20f5206886dfa5539a159", "886216776a89cadcf0fcd4242f034b8cb7f1d6af9d2b0a74859f2df16f7baa4c", "7e307bb8d9b03f359cd4cb452d85fc01b5b2667270538bba83ee5cb9c72088df", "17bc81a97c03faef2ac10d6094abd0ad369...
1.555667
chembl:1801488
COc1ccc(-c2ccc3c(c2)C(=O)C(=O)N3Cc2ccc3ccccc3c2)cc1
2c4256ce9b7c0482e5ab5b6200f77697c6c388231ace64a09751736231da18b1
[ "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccccc4OC)ccc32)cc1", "COc1ccc(-c2ccc3c(c2)C(=O)C(=O)N3c2ccc(OC)cc2)cc1", "COc1ccc(CN2C(=O)/C(=C\\c3ccccc3)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc2c(c1)C(=O)C(=O)N2", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc5ccccc5c4)ccc32)cc1", "COc1ccc(CN2C(=O)/C(=C\\c3ccc(C(C)C)cc3)c3cc(-c4ccc(OC)...
[ "aabe0eb965b5e933f141ef01bc7fee378fef1d39eee6e431df7cb24b5376bcf4", "c285b904f8d4adad8afc74c354125bc2f04baf66f6e20f5206886dfa5539a159", "886216776a89cadcf0fcd4242f034b8cb7f1d6af9d2b0a74859f2df16f7baa4c", "7e307bb8d9b03f359cd4cb452d85fc01b5b2667270538bba83ee5cb9c72088df", "17bc81a97c03faef2ac10d6094abd0ad369...
1.555667
chembl:1801488
COc1ccc(-c2ccc3c(c2)C(=O)C(=O)N3Cc2ccc3ccccc3c2)cc1
2c4256ce9b7c0482e5ab5b6200f77697c6c388231ace64a09751736231da18b1
[ "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(O)cc4)ccc32)cc1", "CCC=Cc1ccc2[nH]c(O)c(O)c2c1", "COc1ccc(CN2C(=O)C(C)(O)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "Cc1ccc2c(c1)C(=O)C(=O)N2", "O=C1Nc2ccc(F)cc2C1=O", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(C)cc4)ccc32)cc1", "O=C1Nc2ccc(Cl)cc2C1=O" ]
[ "274bad82abd467b1c7ac433d739606ae037c7fdd90342fa7742e233eff8fa5e3", "d62311babd26106395c51df3a7116b5c5085d0ee43a289a10c773c8f011c01f7", "90388bcdeadc46688b50621eceaef1ac7ebf817067142975d956629fa4c1195c", "97a744cb5940b79956a6910f17b61b88615d0ed985e34754bdcfb5f08343f85c", "f6b1d48c1cdc5d50696ad6d7d21f1c2645f...
1.555667
chembl:1801488
COc1ccc(-c2ccc3c(c2)C(=O)C(=O)N3Cc2ccc(C(F)(F)F)cc2)cc1
78c7cb20b36e910a180c2cf2dbf72a406a219e0bc55e14e426a6beaca65ed691
[ "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(O)cc4)ccc32)cc1", "CCC=Cc1ccc2[nH]c(O)c(O)c2c1", "COc1ccc(CN2C(=O)C(C)(O)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "Cc1ccc2c(c1)C(=O)C(=O)N2", "O=C1Nc2ccc(F)cc2C1=O", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(C)cc4)ccc32)cc1", "O=C1Nc2ccc(Cl)cc2C1=O" ]
[ "274bad82abd467b1c7ac433d739606ae037c7fdd90342fa7742e233eff8fa5e3", "d62311babd26106395c51df3a7116b5c5085d0ee43a289a10c773c8f011c01f7", "90388bcdeadc46688b50621eceaef1ac7ebf817067142975d956629fa4c1195c", "97a744cb5940b79956a6910f17b61b88615d0ed985e34754bdcfb5f08343f85c", "f6b1d48c1cdc5d50696ad6d7d21f1c2645f...
1.555667
chembl:1801488
COc1ccc(-c2ccc3c(c2)C(=O)C(=O)N3Cc2ccc(C(F)(F)F)cc2)cc1
78c7cb20b36e910a180c2cf2dbf72a406a219e0bc55e14e426a6beaca65ed691
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[ "fa87c5cd9059dc443914cb124a0732e4d6cd889e2af559934d0df92c91d543ba", "1486d5ee417d89c8005180d7e9a366e473858b9845c47a35aecc20684809711c", "c1aed19ed4670b9363ea4f89904570e91ae2a6abea98f7d9fc410893573e62a4", "5518611e3076e1a5209c531d063d23cd36df581395ed72bcc8bf515b3f873196", "c048a48684f447b7c7cdbf38eae6f30daa4...
1.555667
chembl:1801488
COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(OC(F)(F)F)cc4)ccc32)cc1
90149208dea098bf80e3100ec697d18e49670e67555a5528e423b6ac3754845f
[ "COc1ccc(CN2C(=O)/C(=C\\c3ccc(C(F)(F)F)cc3)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3c(-c4ccc(OC)cc4)cccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3ccc(-c4ccc(OC)cc4)cc32)cc1", "O=C1Nc2ccccc2C1=O", "COc1ccc(Cn2c(O)c(N=O)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(OC)c(OC)c4)ccc32)c...
[ "fa87c5cd9059dc443914cb124a0732e4d6cd889e2af559934d0df92c91d543ba", "1486d5ee417d89c8005180d7e9a366e473858b9845c47a35aecc20684809711c", "c1aed19ed4670b9363ea4f89904570e91ae2a6abea98f7d9fc410893573e62a4", "5518611e3076e1a5209c531d063d23cd36df581395ed72bcc8bf515b3f873196", "c048a48684f447b7c7cdbf38eae6f30daa4...
1.554667
chembl:1801488
COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(OC(F)(F)F)cc4)ccc32)cc1
90149208dea098bf80e3100ec697d18e49670e67555a5528e423b6ac3754845f
[ "COc1ccc(Cn2c(O)cc3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(OC(C)C)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(F)(F)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccncc4)ccc32)cc1", "COc1ccc(CN2C(=O)C3(OCCO3)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccccc4OC)c...
[ "404f1da9ee430e576f53cb872eaa3910eb16a5d65055e950ca34f5e0c991d266", "c4990598cc291b556fff63f69ade724ce17fa523a39c2b6b813e49927f6d1a26", "16076c7e9c9579ef55f00066ad292b022ba0be00eefcdb5d0f3a773a26df37a3", "9962fd6f7c70ea95458960df7d9e3f60e54ac931b9d8598965b9379cdf1701cb", "20ad785f524a001eb45b3ace687e3601c87...
1.554667
chembl:1801488
COc1ccc(-c2ccc3c(c2)C(=O)C(=O)N3Cc2cc(C)cc(C)c2)cc1
145f11d20ea9cd807aca3d62f98204ed1b1a56f2cead892fa82dcaa2f756c744
[ "COc1ccc(Cn2c(O)cc3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(OC(C)C)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(F)(F)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccncc4)ccc32)cc1", "COc1ccc(CN2C(=O)C3(OCCO3)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccccc4OC)c...
[ "404f1da9ee430e576f53cb872eaa3910eb16a5d65055e950ca34f5e0c991d266", "c4990598cc291b556fff63f69ade724ce17fa523a39c2b6b813e49927f6d1a26", "16076c7e9c9579ef55f00066ad292b022ba0be00eefcdb5d0f3a773a26df37a3", "9962fd6f7c70ea95458960df7d9e3f60e54ac931b9d8598965b9379cdf1701cb", "20ad785f524a001eb45b3ace687e3601c87...
1.554667
chembl:1801488
COc1ccc(-c2ccc3c(c2)C(=O)C(=O)N3Cc2cc(C)cc(C)c2)cc1
145f11d20ea9cd807aca3d62f98204ed1b1a56f2cead892fa82dcaa2f756c744
[ "COc1ccc(CN2C(=O)/C(=C\\c3ccccc3)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc2c(c1)C(=O)C(=O)N2", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc5ccccc5c4)ccc32)cc1", "COc1ccc(CN2C(=O)/C(=C\\c3ccc(C(C)C)cc3)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(F)c(Cl)c4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4c...
[ "886216776a89cadcf0fcd4242f034b8cb7f1d6af9d2b0a74859f2df16f7baa4c", "7e307bb8d9b03f359cd4cb452d85fc01b5b2667270538bba83ee5cb9c72088df", "17bc81a97c03faef2ac10d6094abd0ad3690030e112c016692f830438668fc7a", "1d58312e01e6f598a39ea92b894982aef4a0265cb88e02aaaf4850a8fb6505d3", "b93ae4854fa6a37bddc5d1ade66bf449bf0...
1.554667
chembl:1801488
COc1ccc(-c2ccc3c(c2)C(=O)C(=O)N3Cc2ccc3c(c2)OCO3)cc1
9de7059cc64bc3015fd0c4be0eebe56b636a628efcfd834b2731dc79a4933f68
[ "COc1ccc(CN2C(=O)/C(=C\\c3ccccc3)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc2c(c1)C(=O)C(=O)N2", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc5ccccc5c4)ccc32)cc1", "COc1ccc(CN2C(=O)/C(=C\\c3ccc(C(C)C)cc3)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(F)c(Cl)c4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4c...
[ "886216776a89cadcf0fcd4242f034b8cb7f1d6af9d2b0a74859f2df16f7baa4c", "7e307bb8d9b03f359cd4cb452d85fc01b5b2667270538bba83ee5cb9c72088df", "17bc81a97c03faef2ac10d6094abd0ad3690030e112c016692f830438668fc7a", "1d58312e01e6f598a39ea92b894982aef4a0265cb88e02aaaf4850a8fb6505d3", "b93ae4854fa6a37bddc5d1ade66bf449bf0...
1.553667
chembl:1801488
COc1ccc(-c2ccc3c(c2)C(=O)C(=O)N3Cc2ccc3c(c2)OCO3)cc1
9de7059cc64bc3015fd0c4be0eebe56b636a628efcfd834b2731dc79a4933f68
[ "COc1ccc(CN2C(=O)C(C)(O)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "Cc1ccc2c(c1)C(=O)C(=O)N2", "O=C1Nc2ccc(F)cc2C1=O", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(C)cc4)ccc32)cc1", "O=C1Nc2ccc(Cl)cc2C1=O", "COc1ccc(CN2C(=O)/C(=C\\c3ccc(C(F)(F)F)cc3)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3c(-c4ccc(OC)cc4)cccc32...
[ "90388bcdeadc46688b50621eceaef1ac7ebf817067142975d956629fa4c1195c", "97a744cb5940b79956a6910f17b61b88615d0ed985e34754bdcfb5f08343f85c", "f6b1d48c1cdc5d50696ad6d7d21f1c2645fe394000ec5c71ea7f962184ee5f60", "7ebdb017871fdbee29b177bb780126f50c1e46df285b7c8f156a1be1e33b36fe", "e6101de344a3cac7c0cc98ffe2e9eac89cf...
1.553667
chembl:1801488
COc1ccc(-c2ccc3c(c2)C(=O)C(=O)N3Cc2ccccc2Cl)cc1
5d1f950055f3faa74be0b3dc3f7c08035befb91628556b6bdc5c68a9fdc277fb
[ "COc1ccc(CN2C(=O)C(C)(O)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "Cc1ccc2c(c1)C(=O)C(=O)N2", "O=C1Nc2ccc(F)cc2C1=O", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(C)cc4)ccc32)cc1", "O=C1Nc2ccc(Cl)cc2C1=O", "COc1ccc(CN2C(=O)/C(=C\\c3ccc(C(F)(F)F)cc3)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3c(-c4ccc(OC)cc4)cccc32...
[ "90388bcdeadc46688b50621eceaef1ac7ebf817067142975d956629fa4c1195c", "97a744cb5940b79956a6910f17b61b88615d0ed985e34754bdcfb5f08343f85c", "f6b1d48c1cdc5d50696ad6d7d21f1c2645fe394000ec5c71ea7f962184ee5f60", "7ebdb017871fdbee29b177bb780126f50c1e46df285b7c8f156a1be1e33b36fe", "e6101de344a3cac7c0cc98ffe2e9eac89cf...
1.549
chembl:1801488
COc1ccc(-c2ccc3c(c2)C(=O)C(=O)N3Cc2ccccc2Cl)cc1
5d1f950055f3faa74be0b3dc3f7c08035befb91628556b6bdc5c68a9fdc277fb
[ "COc1ccc(CN2C(=O)C(=O)c3ccc(-c4ccc(OC)cc4)cc32)cc1", "O=C1Nc2ccccc2C1=O", "COc1ccc(Cn2c(O)c(N=O)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(OC)c(OC)c4)ccc32)cc1", "O=C1Nc2ccc(Br)cc2C1=O", "COc1ccc(Cn2c(O)cc3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(OC(C)C)cc4)cc...
[ "c1aed19ed4670b9363ea4f89904570e91ae2a6abea98f7d9fc410893573e62a4", "5518611e3076e1a5209c531d063d23cd36df581395ed72bcc8bf515b3f873196", "c048a48684f447b7c7cdbf38eae6f30daa409c67f8fc19d29d202e29de024985", "cb731fcf6345af364441c9254f47cd5950257cfbd0a1cc3a8437de573d943164", "2338bccb34ceebc4708f442271a99b0f3d6...
1.549
chembl:1801488
COc1ccc(-c2ccc3c(c2)C(=O)C(=O)N3Cc2cccc(OC)c2)cc1
75a9d76a4220cb92a000fd6519aefebbdf7d1939ba84f6525da34fdbc9654d91
[ "COc1ccc(CN2C(=O)C(=O)c3ccc(-c4ccc(OC)cc4)cc32)cc1", "O=C1Nc2ccccc2C1=O", "COc1ccc(Cn2c(O)c(N=O)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(OC)c(OC)c4)ccc32)cc1", "O=C1Nc2ccc(Br)cc2C1=O", "COc1ccc(Cn2c(O)cc3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(OC(C)C)cc4)cc...
[ "c1aed19ed4670b9363ea4f89904570e91ae2a6abea98f7d9fc410893573e62a4", "5518611e3076e1a5209c531d063d23cd36df581395ed72bcc8bf515b3f873196", "c048a48684f447b7c7cdbf38eae6f30daa409c67f8fc19d29d202e29de024985", "cb731fcf6345af364441c9254f47cd5950257cfbd0a1cc3a8437de573d943164", "2338bccb34ceebc4708f442271a99b0f3d6...
1.547
chembl:1801488
COc1ccc(-c2ccc3c(c2)C(=O)C(=O)N3Cc2cccc(OC)c2)cc1
75a9d76a4220cb92a000fd6519aefebbdf7d1939ba84f6525da34fdbc9654d91
[ "COc1ccc(CN2C(=O)C(F)(F)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccncc4)ccc32)cc1", "COc1ccc(CN2C(=O)C3(OCCO3)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccccc4OC)ccc32)cc1", "COc1ccc(-c2ccc3c(c2)C(=O)C(=O)N3c2ccc(OC)cc2)cc1", "COc1ccc(CN2C(=O)/C(=C\\c3ccccc3)c3cc(-c4c...
[ "16076c7e9c9579ef55f00066ad292b022ba0be00eefcdb5d0f3a773a26df37a3", "9962fd6f7c70ea95458960df7d9e3f60e54ac931b9d8598965b9379cdf1701cb", "20ad785f524a001eb45b3ace687e3601c878131a62e1f27fb7dbf284990240fa", "aabe0eb965b5e933f141ef01bc7fee378fef1d39eee6e431df7cb24b5376bcf4", "c285b904f8d4adad8afc74c354125bc2f04...
1.547
chembl:1801488
COc1ccc(-c2ccc3c(c2)C(=O)C(=O)N3CCOc2ccccc2)cc1
4720bb5f81f36517cd9fc7eeaa636bd1d5b4a8f04a4a8992073648cb5bfd26c6
[ "COc1ccc(CN2C(=O)C(F)(F)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccncc4)ccc32)cc1", "COc1ccc(CN2C(=O)C3(OCCO3)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccccc4OC)ccc32)cc1", "COc1ccc(-c2ccc3c(c2)C(=O)C(=O)N3c2ccc(OC)cc2)cc1", "COc1ccc(CN2C(=O)/C(=C\\c3ccccc3)c3cc(-c4c...
[ "16076c7e9c9579ef55f00066ad292b022ba0be00eefcdb5d0f3a773a26df37a3", "9962fd6f7c70ea95458960df7d9e3f60e54ac931b9d8598965b9379cdf1701cb", "20ad785f524a001eb45b3ace687e3601c878131a62e1f27fb7dbf284990240fa", "aabe0eb965b5e933f141ef01bc7fee378fef1d39eee6e431df7cb24b5376bcf4", "c285b904f8d4adad8afc74c354125bc2f04...
1.547
chembl:1801488
COc1ccc(-c2ccc3c(c2)C(=O)C(=O)N3CCOc2ccccc2)cc1
4720bb5f81f36517cd9fc7eeaa636bd1d5b4a8f04a4a8992073648cb5bfd26c6
[ "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc5ccccc5c4)ccc32)cc1", "COc1ccc(CN2C(=O)/C(=C\\c3ccc(C(C)C)cc3)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(F)c(Cl)c4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(O)cc4)ccc32)cc1", "CCC=Cc1ccc2[nH]c(O)c(O)c2c1", "COc1ccc(CN2C(=O)C(C)(O)c3cc(-c4ccc(OC)cc...
[ "17bc81a97c03faef2ac10d6094abd0ad3690030e112c016692f830438668fc7a", "1d58312e01e6f598a39ea92b894982aef4a0265cb88e02aaaf4850a8fb6505d3", "b93ae4854fa6a37bddc5d1ade66bf449bf0604f59f312c43a0e50aa833e55593", "274bad82abd467b1c7ac433d739606ae037c7fdd90342fa7742e233eff8fa5e3", "d62311babd26106395c51df3a7116b5c508...
1.547
chembl:1801488
COc1ccc(Cn2c(O)c(O)c3cc(-c4ccc(OC)cc4)ccc32)cc1
22be12a07e70dfc844f923f93ecc60235a06514fc3c7c7700cb06b309ab55667
[ "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc5ccccc5c4)ccc32)cc1", "COc1ccc(CN2C(=O)/C(=C\\c3ccc(C(C)C)cc3)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(F)c(Cl)c4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(O)cc4)ccc32)cc1", "CCC=Cc1ccc2[nH]c(O)c(O)c2c1", "COc1ccc(CN2C(=O)C(C)(O)c3cc(-c4ccc(OC)cc...
[ "17bc81a97c03faef2ac10d6094abd0ad3690030e112c016692f830438668fc7a", "1d58312e01e6f598a39ea92b894982aef4a0265cb88e02aaaf4850a8fb6505d3", "b93ae4854fa6a37bddc5d1ade66bf449bf0604f59f312c43a0e50aa833e55593", "274bad82abd467b1c7ac433d739606ae037c7fdd90342fa7742e233eff8fa5e3", "d62311babd26106395c51df3a7116b5c508...
1.547
chembl:1801488
COc1ccc(Cn2c(O)c(O)c3cc(-c4ccc(OC)cc4)ccc32)cc1
22be12a07e70dfc844f923f93ecc60235a06514fc3c7c7700cb06b309ab55667
[ "O=C1Nc2ccc(F)cc2C1=O", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(C)cc4)ccc32)cc1", "O=C1Nc2ccc(Cl)cc2C1=O", "COc1ccc(CN2C(=O)/C(=C\\c3ccc(C(F)(F)F)cc3)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3c(-c4ccc(OC)cc4)cccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3ccc(-c4ccc(OC)cc4)cc32)cc1", "O=C1Nc2ccccc2C1=O" ]
[ "f6b1d48c1cdc5d50696ad6d7d21f1c2645fe394000ec5c71ea7f962184ee5f60", "7ebdb017871fdbee29b177bb780126f50c1e46df285b7c8f156a1be1e33b36fe", "e6101de344a3cac7c0cc98ffe2e9eac89cf6b3e5ca8a2b34ebb949da80c4e8ec", "fa87c5cd9059dc443914cb124a0732e4d6cd889e2af559934d0df92c91d543ba", "1486d5ee417d89c8005180d7e9a366e4738...
1.547
chembl:1801488
COc1ccc(-c2ccc3c(c2)C(=O)C(=O)N3Cc2ccc(Br)cc2)cc1
04acf9c13a224c54c0d3490656725bf20eda06490389631dc2e758e6c7fff575
[ "O=C1Nc2ccc(F)cc2C1=O", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(C)cc4)ccc32)cc1", "O=C1Nc2ccc(Cl)cc2C1=O", "COc1ccc(CN2C(=O)/C(=C\\c3ccc(C(F)(F)F)cc3)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3c(-c4ccc(OC)cc4)cccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3ccc(-c4ccc(OC)cc4)cc32)cc1", "O=C1Nc2ccccc2C1=O" ]
[ "f6b1d48c1cdc5d50696ad6d7d21f1c2645fe394000ec5c71ea7f962184ee5f60", "7ebdb017871fdbee29b177bb780126f50c1e46df285b7c8f156a1be1e33b36fe", "e6101de344a3cac7c0cc98ffe2e9eac89cf6b3e5ca8a2b34ebb949da80c4e8ec", "fa87c5cd9059dc443914cb124a0732e4d6cd889e2af559934d0df92c91d543ba", "1486d5ee417d89c8005180d7e9a366e4738...
1.547
chembl:1801488
COc1ccc(-c2ccc3c(c2)C(=O)C(=O)N3Cc2ccc(Br)cc2)cc1
04acf9c13a224c54c0d3490656725bf20eda06490389631dc2e758e6c7fff575
[ "COc1ccc(Cn2c(O)c(N=O)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(OC)c(OC)c4)ccc32)cc1", "O=C1Nc2ccc(Br)cc2C1=O", "COc1ccc(Cn2c(O)cc3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(OC(C)C)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(F)(F)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(...
[ "c048a48684f447b7c7cdbf38eae6f30daa409c67f8fc19d29d202e29de024985", "cb731fcf6345af364441c9254f47cd5950257cfbd0a1cc3a8437de573d943164", "2338bccb34ceebc4708f442271a99b0f3d6eca56b3aef0f43d17be4705da81c4", "404f1da9ee430e576f53cb872eaa3910eb16a5d65055e950ca34f5e0c991d266", "c4990598cc291b556fff63f69ade724ce17...
1.547
chembl:1801488
COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(C(F)(F)F)cc4)ccc32)cc1
11e4933bdb45a79a17e4ae6559ef5901b7686fcd92f1bd63670aea88850394f2
[ "COc1ccc(Cn2c(O)c(N=O)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(OC)c(OC)c4)ccc32)cc1", "O=C1Nc2ccc(Br)cc2C1=O", "COc1ccc(Cn2c(O)cc3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(OC(C)C)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(F)(F)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(...
[ "c048a48684f447b7c7cdbf38eae6f30daa409c67f8fc19d29d202e29de024985", "cb731fcf6345af364441c9254f47cd5950257cfbd0a1cc3a8437de573d943164", "2338bccb34ceebc4708f442271a99b0f3d6eca56b3aef0f43d17be4705da81c4", "404f1da9ee430e576f53cb872eaa3910eb16a5d65055e950ca34f5e0c991d266", "c4990598cc291b556fff63f69ade724ce17...
1.544667
chembl:1801488
COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(C(F)(F)F)cc4)ccc32)cc1
11e4933bdb45a79a17e4ae6559ef5901b7686fcd92f1bd63670aea88850394f2
[ "COc1ccc(CN2C(=O)C3(OCCO3)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccccc4OC)ccc32)cc1", "COc1ccc(-c2ccc3c(c2)C(=O)C(=O)N3c2ccc(OC)cc2)cc1", "COc1ccc(CN2C(=O)/C(=C\\c3ccccc3)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc2c(c1)C(=O)C(=O)N2", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc5ccccc5c4)ccc32)cc1"...
[ "20ad785f524a001eb45b3ace687e3601c878131a62e1f27fb7dbf284990240fa", "aabe0eb965b5e933f141ef01bc7fee378fef1d39eee6e431df7cb24b5376bcf4", "c285b904f8d4adad8afc74c354125bc2f04baf66f6e20f5206886dfa5539a159", "886216776a89cadcf0fcd4242f034b8cb7f1d6af9d2b0a74859f2df16f7baa4c", "7e307bb8d9b03f359cd4cb452d85fc01b5b...
1.544667
chembl:1801488
COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(C#N)cc4)ccc32)cc1
2565d3565fbef39c6ec3e7060c216666ec959f60ef9053c84e7cc53405f23064
[ "COc1ccc(CN2C(=O)C3(OCCO3)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccccc4OC)ccc32)cc1", "COc1ccc(-c2ccc3c(c2)C(=O)C(=O)N3c2ccc(OC)cc2)cc1", "COc1ccc(CN2C(=O)/C(=C\\c3ccccc3)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc2c(c1)C(=O)C(=O)N2", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc5ccccc5c4)ccc32)cc1"...
[ "20ad785f524a001eb45b3ace687e3601c878131a62e1f27fb7dbf284990240fa", "aabe0eb965b5e933f141ef01bc7fee378fef1d39eee6e431df7cb24b5376bcf4", "c285b904f8d4adad8afc74c354125bc2f04baf66f6e20f5206886dfa5539a159", "886216776a89cadcf0fcd4242f034b8cb7f1d6af9d2b0a74859f2df16f7baa4c", "7e307bb8d9b03f359cd4cb452d85fc01b5b...
1.543333
chembl:1801488
COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(C#N)cc4)ccc32)cc1
2565d3565fbef39c6ec3e7060c216666ec959f60ef9053c84e7cc53405f23064
[ "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(F)c(Cl)c4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(O)cc4)ccc32)cc1", "CCC=Cc1ccc2[nH]c(O)c(O)c2c1", "COc1ccc(CN2C(=O)C(C)(O)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "Cc1ccc2c(c1)C(=O)C(=O)N2", "O=C1Nc2ccc(F)cc2C1=O", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(C)cc4)ccc32)cc1" ]
[ "b93ae4854fa6a37bddc5d1ade66bf449bf0604f59f312c43a0e50aa833e55593", "274bad82abd467b1c7ac433d739606ae037c7fdd90342fa7742e233eff8fa5e3", "d62311babd26106395c51df3a7116b5c5085d0ee43a289a10c773c8f011c01f7", "90388bcdeadc46688b50621eceaef1ac7ebf817067142975d956629fa4c1195c", "97a744cb5940b79956a6910f17b61b88615...
1.543333
chembl:1801488
COc1ccc(-c2ccc3c(c2)C(=O)C(=O)N3)cc1
91a62b6a98a191c12e5f991b65b457abda18cff2d6e537164ac99f805461c03e
[ "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(F)c(Cl)c4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(O)cc4)ccc32)cc1", "CCC=Cc1ccc2[nH]c(O)c(O)c2c1", "COc1ccc(CN2C(=O)C(C)(O)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "Cc1ccc2c(c1)C(=O)C(=O)N2", "O=C1Nc2ccc(F)cc2C1=O", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(C)cc4)ccc32)cc1" ]
[ "b93ae4854fa6a37bddc5d1ade66bf449bf0604f59f312c43a0e50aa833e55593", "274bad82abd467b1c7ac433d739606ae037c7fdd90342fa7742e233eff8fa5e3", "d62311babd26106395c51df3a7116b5c5085d0ee43a289a10c773c8f011c01f7", "90388bcdeadc46688b50621eceaef1ac7ebf817067142975d956629fa4c1195c", "97a744cb5940b79956a6910f17b61b88615...
1.542333
chembl:1801488
COc1ccc(-c2ccc3c(c2)C(=O)C(=O)N3)cc1
91a62b6a98a191c12e5f991b65b457abda18cff2d6e537164ac99f805461c03e
[ "O=C1Nc2ccc(Cl)cc2C1=O", "COc1ccc(CN2C(=O)/C(=C\\c3ccc(C(F)(F)F)cc3)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3c(-c4ccc(OC)cc4)cccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3ccc(-c4ccc(OC)cc4)cc32)cc1", "O=C1Nc2ccccc2C1=O", "COc1ccc(Cn2c(O)c(N=O)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3c...
[ "e6101de344a3cac7c0cc98ffe2e9eac89cf6b3e5ca8a2b34ebb949da80c4e8ec", "fa87c5cd9059dc443914cb124a0732e4d6cd889e2af559934d0df92c91d543ba", "1486d5ee417d89c8005180d7e9a366e473858b9845c47a35aecc20684809711c", "c1aed19ed4670b9363ea4f89904570e91ae2a6abea98f7d9fc410893573e62a4", "5518611e3076e1a5209c531d063d23cd36d...
1.542333
chembl:1801488
COc1ccc(-c2ccc3c(c2)C(=O)C(=O)N3Cc2ccc(Cl)c(Cl)c2)cc1
3bb522508ddac1a2d91e33d58d79f253deff985ae39a455d3dce630758915eee
[ "O=C1Nc2ccc(Cl)cc2C1=O", "COc1ccc(CN2C(=O)/C(=C\\c3ccc(C(F)(F)F)cc3)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3c(-c4ccc(OC)cc4)cccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3ccc(-c4ccc(OC)cc4)cc32)cc1", "O=C1Nc2ccccc2C1=O", "COc1ccc(Cn2c(O)c(N=O)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3c...
[ "e6101de344a3cac7c0cc98ffe2e9eac89cf6b3e5ca8a2b34ebb949da80c4e8ec", "fa87c5cd9059dc443914cb124a0732e4d6cd889e2af559934d0df92c91d543ba", "1486d5ee417d89c8005180d7e9a366e473858b9845c47a35aecc20684809711c", "c1aed19ed4670b9363ea4f89904570e91ae2a6abea98f7d9fc410893573e62a4", "5518611e3076e1a5209c531d063d23cd36d...
1.541667
chembl:1801488
COc1ccc(-c2ccc3c(c2)C(=O)C(=O)N3Cc2ccc(Cl)c(Cl)c2)cc1
3bb522508ddac1a2d91e33d58d79f253deff985ae39a455d3dce630758915eee
[ "O=C1Nc2ccc(Br)cc2C1=O", "COc1ccc(Cn2c(O)cc3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccc(OC(C)C)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(F)(F)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C(=O)C(=O)c3cc(-c4ccncc4)ccc32)cc1", "COc1ccc(CN2C(=O)C3(OCCO3)c3cc(-c4ccc(OC)cc4)ccc32)cc1", "COc1ccc(CN2C...
[ "2338bccb34ceebc4708f442271a99b0f3d6eca56b3aef0f43d17be4705da81c4", "404f1da9ee430e576f53cb872eaa3910eb16a5d65055e950ca34f5e0c991d266", "c4990598cc291b556fff63f69ade724ce17fa523a39c2b6b813e49927f6d1a26", "16076c7e9c9579ef55f00066ad292b022ba0be00eefcdb5d0f3a773a26df37a3", "9962fd6f7c70ea95458960df7d9e3f60e54...
1.541667
chembl:1802954
COc1nn(-c2ccc(NC(=O)OCc3ccccc3)c(C)c2)c(=O)o1
a5f6313df88bce9540bfaeb0c7094d6bc2a105ca7b677567c7ac0eaea6617552
[ "CCCCCCCCCCCCCC(=NO)c1cc(-c2cccc(F)c2)ccc1O", "CCC(=NO)c1cc(-c2ccc(O)c(F)c2)ccc1O", "CCCCCCCCCC(=NO)c1cc(-c2ccc(OC)c(F)c2)ccc1O", "COc1ccc(-c2ccc(O)c(C(=NO)c3ccccc3)c2)cc1F", "CC(=NO)c1cc(-c2ccc(O)c(F)c2)ccc1O", "COc1ccc(-c2ccc(O)c(C(Cc3ccccc3)=NO)c2)cc1F", "CCCCCCCC(=NO)c1cc(-c2ccc(OC)cc2)ccc1O" ]
[ "ecf9f9eb3438eb0290dc445ab00ac036ff4e78a6c7595eab40c61d7af5681145", "f89e134890bb931afa03ddfc1e29fa3aebc1733e2b746dec865777860b70ef47", "6512137d7f7297ee6b6b7c5d6d5c3c7f349eeaf62ae02939c6d83b2f6e814315", "52522b5b582a16d24174ef30af2cfac3b1da7ba8f7acb6355c8d79e9daf3e2f9", "df7713f4be1301a3ec7022acfc3637caaba...
1.636667
chembl:1802954
COc1nn(-c2ccc(NC(=O)OCc3ccccc3)c(C)c2)c(=O)o1
a5f6313df88bce9540bfaeb0c7094d6bc2a105ca7b677567c7ac0eaea6617552
[ "CCCCCCCCCCCCCC(=NO)c1cc(-c2ccc(OC)cc2)ccc1O", "COc1ccc(-c2ccc(O)c(C(=NO)c3ccccc3)c2)cc1", "COc1ccc(-c2ccc(O)c(C(Cc3ccccc3)=NO)c2)cc1", "CCCCCCCCCCCCCCCC(=NO)c1cc(-c2ccc(OC)cc2)ccc1O", "CCCCCCCCCCCC(=NO)c1cc(-c2ccc(OC)cc2)ccc1O", "CCCCCCCC(=NO)c1cc(-c2ccc(OC)c(F)c2)ccc1O", "CCCCC(=NO)c1cc(-c2ccc(OC)c(F)...
[ "21f82473b56aab1afcfda9a287bc4740e98882930d808aac06be699d05db7f68", "ef0125502e3906e7f136151813d343c8865e0c49e0c28ae7fa89d6e3e8e03b42", "aad6776a9620361fd27ea3b608a38592811a68917c31690d7197c2a0b02c3e75", "bf3d77d271e6a0187404a97ce30a4b592747f57cf22fccd00597a3b331a8d00b", "4cdf811b2e685d3bbf5a0d254cd6ed3d20a...
1.636667
chembl:1802954
CCCCCCCCCCCCCC(=NO)c1cc(-c2ccc(O)c(F)c2)ccc1O
0e7c7c20c99ec72598fdf9d9e2fc3c5ba595923f6e35741c127699a0cdcd643a
[ "CCCCCCCCCCCCCC(=NO)c1cc(-c2ccc(OC)cc2)ccc1O", "COc1ccc(-c2ccc(O)c(C(=NO)c3ccccc3)c2)cc1", "COc1ccc(-c2ccc(O)c(C(Cc3ccccc3)=NO)c2)cc1", "CCCCCCCCCCCCCCCC(=NO)c1cc(-c2ccc(OC)cc2)ccc1O", "CCCCCCCCCCCC(=NO)c1cc(-c2ccc(OC)cc2)ccc1O", "CCCCCCCC(=NO)c1cc(-c2ccc(OC)c(F)c2)ccc1O", "CCCCC(=NO)c1cc(-c2ccc(OC)c(F)...
[ "21f82473b56aab1afcfda9a287bc4740e98882930d808aac06be699d05db7f68", "ef0125502e3906e7f136151813d343c8865e0c49e0c28ae7fa89d6e3e8e03b42", "aad6776a9620361fd27ea3b608a38592811a68917c31690d7197c2a0b02c3e75", "bf3d77d271e6a0187404a97ce30a4b592747f57cf22fccd00597a3b331a8d00b", "4cdf811b2e685d3bbf5a0d254cd6ed3d20a...
1.614
chembl:1802954
CCCCCCCCCCCCCC(=NO)c1cc(-c2ccc(O)c(F)c2)ccc1O
0e7c7c20c99ec72598fdf9d9e2fc3c5ba595923f6e35741c127699a0cdcd643a
[ "CCCCCCCCCCCCCC(=NO)c1cc(-c2ccccc2)ccc1O", "CCCCCCCCCCCC(=NO)c1cc(-c2ccc(OC)c(F)c2)ccc1O", "CCCCCCCCCC(=NO)c1cc(-c2ccc(OC)cc2)ccc1O", "CCCCC(=NO)c1cc(-c2ccc(OC)cc2)ccc1O", "CCCCCCCCCCCCCCCC(=NO)c1cc(-c2ccc(OC)c(F)c2)ccc1O", "CCCCCCCCCCCCCC(=NO)c1cc(-c2ccc(OC)c(F)c2)ccc1O", "CCCCCCCCCCCCCC(=NO)c1cc(-c2cc...
[ "18a402b43babd6c462aa6e0087470083f6aaa0ad7fdc611221a0f1a3a848fbb3", "8c56e1a7782f18562950a015e029181ab35fdc59f0309909c14dee7d98f01442", "2a5c9f48ffb8b38ab024e459a4f71a26e1b2ccabcaaf7f2de09469a3855c5523", "72cd08eb5f35b287a30c5e8aa3526725bebb750386a92b9c1634e576074c91c8", "9fab67258758aefd41f6444beffce3fac53...
1.614
chembl:1802954
CCCCCCCCCCCC(=NO)c1cc(-c2ccc(O)c(F)c2)ccc1O
d94225258bab8d92e9f4213abdcc1966e7c84b7e6a63fc8da169ef598a7a1735
[ "CCCCCCCCCCCCCC(=NO)c1cc(-c2ccccc2)ccc1O", "CCCCCCCCCCCC(=NO)c1cc(-c2ccc(OC)c(F)c2)ccc1O", "CCCCCCCCCC(=NO)c1cc(-c2ccc(OC)cc2)ccc1O", "CCCCC(=NO)c1cc(-c2ccc(OC)cc2)ccc1O", "CCCCCCCCCCCCCCCC(=NO)c1cc(-c2ccc(OC)c(F)c2)ccc1O", "CCCCCCCCCCCCCC(=NO)c1cc(-c2ccc(OC)c(F)c2)ccc1O", "CCCCCCCCCCCCCC(=NO)c1cc(-c2cc...
[ "18a402b43babd6c462aa6e0087470083f6aaa0ad7fdc611221a0f1a3a848fbb3", "8c56e1a7782f18562950a015e029181ab35fdc59f0309909c14dee7d98f01442", "2a5c9f48ffb8b38ab024e459a4f71a26e1b2ccabcaaf7f2de09469a3855c5523", "72cd08eb5f35b287a30c5e8aa3526725bebb750386a92b9c1634e576074c91c8", "9fab67258758aefd41f6444beffce3fac53...
1.613333
chembl:1802954
CCCCCCCCCCCC(=NO)c1cc(-c2ccc(O)c(F)c2)ccc1O
d94225258bab8d92e9f4213abdcc1966e7c84b7e6a63fc8da169ef598a7a1735
[ "CCC(=NO)c1cc(-c2ccc(O)c(F)c2)ccc1O", "CCCCCCCCCC(=NO)c1cc(-c2ccc(OC)c(F)c2)ccc1O", "COc1ccc(-c2ccc(O)c(C(=NO)c3ccccc3)c2)cc1F", "CC(=NO)c1cc(-c2ccc(O)c(F)c2)ccc1O", "COc1ccc(-c2ccc(O)c(C(Cc3ccccc3)=NO)c2)cc1F", "CCCCCCCC(=NO)c1cc(-c2ccc(OC)cc2)ccc1O", "CCCCCCCCCCCCCC(=NO)c1cc(-c2ccc(OC)cc2)ccc1O" ]
[ "f89e134890bb931afa03ddfc1e29fa3aebc1733e2b746dec865777860b70ef47", "6512137d7f7297ee6b6b7c5d6d5c3c7f349eeaf62ae02939c6d83b2f6e814315", "52522b5b582a16d24174ef30af2cfac3b1da7ba8f7acb6355c8d79e9daf3e2f9", "df7713f4be1301a3ec7022acfc3637caaba682cdd3f619622ee62fa167d641b3", "cdcb2852b97648f1f40882ec10b6141b8af...
1.613333
chembl:1802954
CCCCCCCCCCCCCC(=NO)c1cc(-c2ccc(O)cc2)ccc1O
7809aaed7595dfd2d08b1ffc1094680112b33928375a6456856be9c993e44778
[ "CCC(=NO)c1cc(-c2ccc(O)c(F)c2)ccc1O", "CCCCCCCCCC(=NO)c1cc(-c2ccc(OC)c(F)c2)ccc1O", "COc1ccc(-c2ccc(O)c(C(=NO)c3ccccc3)c2)cc1F", "CC(=NO)c1cc(-c2ccc(O)c(F)c2)ccc1O", "COc1ccc(-c2ccc(O)c(C(Cc3ccccc3)=NO)c2)cc1F", "CCCCCCCC(=NO)c1cc(-c2ccc(OC)cc2)ccc1O", "CCCCCCCCCCCCCC(=NO)c1cc(-c2ccc(OC)cc2)ccc1O" ]
[ "f89e134890bb931afa03ddfc1e29fa3aebc1733e2b746dec865777860b70ef47", "6512137d7f7297ee6b6b7c5d6d5c3c7f349eeaf62ae02939c6d83b2f6e814315", "52522b5b582a16d24174ef30af2cfac3b1da7ba8f7acb6355c8d79e9daf3e2f9", "df7713f4be1301a3ec7022acfc3637caaba682cdd3f619622ee62fa167d641b3", "cdcb2852b97648f1f40882ec10b6141b8af...
1.612
chembl:1802954
CCCCCCCCCCCCCC(=NO)c1cc(-c2ccc(O)cc2)ccc1O
7809aaed7595dfd2d08b1ffc1094680112b33928375a6456856be9c993e44778
[ "COc1ccc(-c2ccc(O)c(C(=NO)c3ccccc3)c2)cc1", "COc1ccc(-c2ccc(O)c(C(Cc3ccccc3)=NO)c2)cc1", "CCCCCCCCCCCCCCCC(=NO)c1cc(-c2ccc(OC)cc2)ccc1O", "CCCCCCCCCCCC(=NO)c1cc(-c2ccc(OC)cc2)ccc1O", "CCCCCCCC(=NO)c1cc(-c2ccc(OC)c(F)c2)ccc1O", "CCCCC(=NO)c1cc(-c2ccc(OC)c(F)c2)ccc1O", "CCCCCCCCCCCCCC(=NO)c1cc(-c2ccccc2)c...
[ "ef0125502e3906e7f136151813d343c8865e0c49e0c28ae7fa89d6e3e8e03b42", "aad6776a9620361fd27ea3b608a38592811a68917c31690d7197c2a0b02c3e75", "bf3d77d271e6a0187404a97ce30a4b592747f57cf22fccd00597a3b331a8d00b", "4cdf811b2e685d3bbf5a0d254cd6ed3d20aab0644f836481ebfafb190e2786da", "1063f495f5abb9bc26c435f6fb1bc72e471...
1.612
chembl:1802954
O=C(c1ccc(Cl)cc1)C1CCN(C(=O)c2cccc(O)c2)CC1
cc4ad13b89dff54c91cf7ab9138e3b4edbd8126a2ef3e6a96043d6aeebee15b1
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[ "ef0125502e3906e7f136151813d343c8865e0c49e0c28ae7fa89d6e3e8e03b42", "aad6776a9620361fd27ea3b608a38592811a68917c31690d7197c2a0b02c3e75", "bf3d77d271e6a0187404a97ce30a4b592747f57cf22fccd00597a3b331a8d00b", "4cdf811b2e685d3bbf5a0d254cd6ed3d20aab0644f836481ebfafb190e2786da", "1063f495f5abb9bc26c435f6fb1bc72e471...
1.611
chembl:1802954
O=C(c1ccc(Cl)cc1)C1CCN(C(=O)c2cccc(O)c2)CC1
cc4ad13b89dff54c91cf7ab9138e3b4edbd8126a2ef3e6a96043d6aeebee15b1
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[ "8c56e1a7782f18562950a015e029181ab35fdc59f0309909c14dee7d98f01442", "2a5c9f48ffb8b38ab024e459a4f71a26e1b2ccabcaaf7f2de09469a3855c5523", "72cd08eb5f35b287a30c5e8aa3526725bebb750386a92b9c1634e576074c91c8", "9fab67258758aefd41f6444beffce3fac53644a1e6c872bc2f069232ab4b2ebf", "803a7c2ebdaeafcafde336bb17a968b5783...
1.611
chembl:1802954
CCCCCCCCCCCCCCCC(=NO)c1cc(-c2ccc(O)c(F)c2)ccc1O
b142a38f8491522f81d12c501cfe7a92b999902a4feb1545dc11cf9e7635339f
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[ "8c56e1a7782f18562950a015e029181ab35fdc59f0309909c14dee7d98f01442", "2a5c9f48ffb8b38ab024e459a4f71a26e1b2ccabcaaf7f2de09469a3855c5523", "72cd08eb5f35b287a30c5e8aa3526725bebb750386a92b9c1634e576074c91c8", "9fab67258758aefd41f6444beffce3fac53644a1e6c872bc2f069232ab4b2ebf", "803a7c2ebdaeafcafde336bb17a968b5783...
1.609667
chembl:1802954
CCCCCCCCCCCCCCCC(=NO)c1cc(-c2ccc(O)c(F)c2)ccc1O
b142a38f8491522f81d12c501cfe7a92b999902a4feb1545dc11cf9e7635339f
[ "CCCCCCCCCC(=NO)c1cc(-c2ccc(OC)c(F)c2)ccc1O", "COc1ccc(-c2ccc(O)c(C(=NO)c3ccccc3)c2)cc1F", "CC(=NO)c1cc(-c2ccc(O)c(F)c2)ccc1O", "COc1ccc(-c2ccc(O)c(C(Cc3ccccc3)=NO)c2)cc1F", "CCCCCCCC(=NO)c1cc(-c2ccc(OC)cc2)ccc1O", "CCCCCCCCCCCCCC(=NO)c1cc(-c2ccc(OC)cc2)ccc1O", "COc1ccc(-c2ccc(O)c(C(=NO)c3ccccc3)c2)cc1"...
[ "6512137d7f7297ee6b6b7c5d6d5c3c7f349eeaf62ae02939c6d83b2f6e814315", "52522b5b582a16d24174ef30af2cfac3b1da7ba8f7acb6355c8d79e9daf3e2f9", "df7713f4be1301a3ec7022acfc3637caaba682cdd3f619622ee62fa167d641b3", "cdcb2852b97648f1f40882ec10b6141b8af087d43f77a47e32a8cf963f2b5c76", "4c247cb16eee4e2d448a34687b481e76cb5...
1.609667
chembl:1802954
CCCCCCCCCCCCCCCC(=NO)c1cc(-c2ccc(O)cc2)ccc1O
c012508769e95ce7a3e071bf8bd705243e99a25da1b3c40a8f523bbfd4d4435a
[ "CCCCCCCCCC(=NO)c1cc(-c2ccc(OC)c(F)c2)ccc1O", "COc1ccc(-c2ccc(O)c(C(=NO)c3ccccc3)c2)cc1F", "CC(=NO)c1cc(-c2ccc(O)c(F)c2)ccc1O", "COc1ccc(-c2ccc(O)c(C(Cc3ccccc3)=NO)c2)cc1F", "CCCCCCCC(=NO)c1cc(-c2ccc(OC)cc2)ccc1O", "CCCCCCCCCCCCCC(=NO)c1cc(-c2ccc(OC)cc2)ccc1O", "COc1ccc(-c2ccc(O)c(C(=NO)c3ccccc3)c2)cc1"...
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1.609
chembl:1802954
CCCCCCCCCCCCCCCC(=NO)c1cc(-c2ccc(O)cc2)ccc1O
c012508769e95ce7a3e071bf8bd705243e99a25da1b3c40a8f523bbfd4d4435a
[ "COc1ccc(-c2ccc(O)c(C(Cc3ccccc3)=NO)c2)cc1", "CCCCCCCCCCCCCCCC(=NO)c1cc(-c2ccc(OC)cc2)ccc1O", "CCCCCCCCCCCC(=NO)c1cc(-c2ccc(OC)cc2)ccc1O", "CCCCCCCC(=NO)c1cc(-c2ccc(OC)c(F)c2)ccc1O", "CCCCC(=NO)c1cc(-c2ccc(OC)c(F)c2)ccc1O", "CCCCCCCCCCCCCC(=NO)c1cc(-c2ccccc2)ccc1O", "CCCCCCCCCCCC(=NO)c1cc(-c2ccc(OC)c(F)...
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1.609