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Q4.915
Q4
What drugs target the gene MTNR1A?
The drugs that target MTNR1A are Agomelatine, Melatonin, Ramelteon, and Tasimelteon.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%MTNR1A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5938', 'drugName': 'Ramelteon', 'newLinkedTargets_string': 'MTNR1A (ENSG00000168412), MTNR1B (ENSG00000134640)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5737', 'drugName': 'Melatonin', 'newLinkedTargets_string': 'MTNR1A (ENSG00000168412), MTNR1B (E...
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Q4.1428
Q4
What drugs target the gene TH?
The drug that targets TH is Metyrosine.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TH %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2694', 'drugName': 'Metyrosine', 'newLinkedTargets_string': 'TH (ENSG00000180176)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}]
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Q4.929
Q4
What drugs target the gene NAE1?
There are no approved drugs targeting NAE1, but the drug Pevonedistat, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NAE1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3764', 'drugName': 'Pevonedistat', 'newLinkedTargets_string': 'UBA3 (ENSG00000144744), NAE1 (ENSG00000159593)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}]
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Q4.1055
Q4
What drugs target the gene PDE6C?
The drugs that target PDE6C are Pentoxifylline and Dipyridamole.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PDE6C %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6107', 'drugName': 'Dipyridamole', 'newLinkedTargets_string': 'PDE5A (ENSG00000138735), PDE4A (ENSG00000065989), PDE3A (ENSG00000172572), PDE6H (ENSG00000139053), PDE6G (ENSG00000185527), PDE2A (ENSG00000186642), PDE7A (ENSG00000205268), PDE1A (ENSG00000115252), PDE9A (ENSG00000160191), PD...
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Q4.79
Q4
What drugs target the gene ASGR1?
There are no FDA approved drugs targeting the gene ASGR1. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Vupanorsen Sodium and Vupanorsen.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ASGR1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2325', 'drugName': 'Vupanorsen', 'newLinkedTargets_string': 'ANGPTL3 (ENSG00000132855), ASGR1 (ENSG00000141505)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_2326', 'drugName': 'Vupanorsen', 'newLinkedTargets_string': 'ANGPTL3 (ENSG00000132855), ASGR1...
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Q4.86
Q4
What drugs target the gene ATP1B3?
The drugs that target ATP1B3 are Acetyldigitoxin, Deslanoside, Digoxin, Lanatoside C, and Digitoxin.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ATP1B3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2499', 'drugName': 'Digoxin', 'newLinkedTargets_string': 'ATP1A1 (ENSG00000163399), ATP1B2 (ENSG00000129244), ATP1B1 (ENSG00000143153), ATP1A2 (ENSG00000018625), ATP1B3 (ENSG00000069849), ATP1A3 (ENSG00000105409), ATP1A4 (ENSG00000132681), FXYD2 (ENSG00000137731)', 'drugIsApproved': True, ...
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Q4.946
Q4
What drugs target the gene NDUFA7?
The drugs that target NDUFA7 are Metformin and Metformin Hydrochloride.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NDUFA7 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (ENSG00000165264), NDUFA4 (...
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Q4.84
Q4
What drugs target the gene ATP1B1?
The drugs that target ATP1B1 are Acetyldigitoxin, Deslanoside, Digoxin, Lanatoside C, and Digitoxin.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ATP1B1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2499', 'drugName': 'Digoxin', 'newLinkedTargets_string': 'ATP1A1 (ENSG00000163399), ATP1B2 (ENSG00000129244), ATP1B1 (ENSG00000143153), ATP1A2 (ENSG00000018625), ATP1B3 (ENSG00000069849), ATP1A3 (ENSG00000105409), ATP1A4 (ENSG00000132681), FXYD2 (ENSG00000137731)', 'drugIsApproved': True, ...
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Q4.459
Q4
What drugs target the gene FGA?
The drug that targets FGA is Fibrinolysin and Human.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%FGA %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1199', 'drugName': 'Fibrinolysin, Human', 'newLinkedTargets_string': 'FGA (ENSG00000171560), FGB (ENSG00000171564), FGG (ENSG00000171557)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1397', 'drugName': 'Ancrod', 'newLinkedTargets_string': 'FGA (ENSG00...
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Q4.947
Q4
What drugs target the gene NDUFA8?
The drugs that target NDUFA8 are Metformin and Metformin Hydrochloride.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NDUFA8 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (ENSG00000165264), NDUFA4 (...
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Q4.681
Q4
What drugs target the gene IL18RAP?
There are no approved drugs targeting IL18RAP, but the drug Iboctadekin, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%IL18RAP %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2219', 'drugName': 'Iboctadekin', 'newLinkedTargets_string': 'IL18RAP (ENSG00000115607), IL18R1 (ENSG00000115604)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
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Q4.1532
Q4
What drugs target the gene WT1?
There are no FDA approved drugs targeting the gene WT1. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Galinpepimut-S and Ombipepimut-S.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%WT1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_240', 'drugName': 'Galinpepimut-S', 'newLinkedTargets_string': 'WT1 (ENSG00000184937)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_6067', 'drugName': 'Ombipepimut-S', 'newLinkedTargets_string': 'WT1 (ENSG00000184937)', 'drugIsApproved': False, 'maxCl...
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Q4.1114
Q4
What drugs target the gene PPARD?
The drug that targets PPARD is Bezafibrate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PPARD %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1564', 'drugName': 'Bezafibrate', 'newLinkedTargets_string': 'PPARG (ENSG00000132170), PPARA (ENSG00000186951), PPARD (ENSG00000112033)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1645', 'drugName': 'Lanifibranor', 'newLinkedTargets_string': 'PPARG (...
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Q4.438
Q4
What drugs target the gene F2?
The drugs that target F2 are Lepirudin, Dabigatran Etexilate, Ximelagatran, Argatroban, Desirudin, Antithrombin Alfa, Bivalirudin, and Dabigatran Etexilate Mesylate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%F2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1887', 'drugName': 'Metformin Hydrochloride', 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (ENSG00000165264), NDUFA4 (...
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Q4.775
Q4
What drugs target the gene KCNQ1?
The drugs that target KCNQ1 are Dalfampridine, Guanidine, Amifampridine Phosphate, Ezogabine, Guanidine Hydrochloride, and Amifampridine.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%KCNQ1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2190', 'drugName': 'Guanidine', 'newLinkedTargets_string': 'KCNQ1 (ENSG00000053918), KCND3 (ENSG00000171385), KCNH2 (ENSG00000055118), KCNA2 (ENSG00000177301), KCNA1 (ENSG00000111262), KCNQ2 (ENSG00000075043), KCNQ3 (ENSG00000184156), KCNA7 (ENSG00000104848), KCNQ5 (ENSG00000185760), KCNQ4...
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Q4.648
Q4
What drugs target the gene IFNA4?
There are no FDA approved drugs targeting the gene IFNA4. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Rontalizumab and Sifalimumab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%IFNA4 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5087', 'drugName': 'Sifalimumab', 'newLinkedTargets_string': 'IFNA6 (ENSG00000120235), IFNA8 (ENSG00000120242), IFNA5 (ENSG00000147873), IFNA10 (ENSG00000186803), IFNA2 (ENSG00000188379), IFNA1 (ENSG00000197919), IFNA13 (ENSG00000233816), IFNA7 (ENSG00000214042), IFNA21 (ENSG00000137080), ...
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Q4.850
Q4
What drugs target the gene MAP3K10?
There are no approved drugs targeting MAP3K10, but the drug Cep-1347, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%MAP3K10 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6091', 'drugName': 'Cep-1347', 'newLinkedTargets_string': 'MAP3K13 (ENSG00000073803), MAP3K12 (ENSG00000139625), MAP3K10 (ENSG00000130758), MAP3K9 (ENSG00000006432), MAP3K11 (ENSG00000173327)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_6088', 'drugN...
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Q4.1414
Q4
What drugs target the gene TACSTD2?
The drug that targets TACSTD2 is Sacituzumab Govitecan.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TACSTD2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4818', 'drugName': 'Sacituzumab Govitecan', 'newLinkedTargets_string': 'TACSTD2 (ENSG00000184292), TOP1 (ENSG00000198900)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4819', 'drugName': 'Sacituzumab Govitecan', 'newLinkedTargets_string': 'TACSTD2 (ENS...
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Q4.1223
Q4
What drugs target the gene ROCK1?
The drugs that target ROCK1 are Belumosudil, Netarsudil Dimesylate, Netarsudil, and Belumosudil Mesylate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ROCK1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4693', 'drugName': 'Netarsudil Dimesylate', 'newLinkedTargets_string': 'ROCK2 (ENSG00000134318), ROCK1 (ENSG00000067900)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4213', 'drugName': 'Belumosudil', 'newLinkedTargets_string': 'ROCK2 (ENSG00000134318)...
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Q4.406
Q4
What drugs target the gene EPCAM?
The drug that targets EPCAM is Catumaxomab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%EPCAM %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2537', 'drugName': 'Catumaxomab', 'newLinkedTargets_string': 'CD3E (ENSG00000198851), CD3G (ENSG00000160654), CD3D (ENSG00000167286), EPCAM (ENSG00000119888)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2538', 'drugName': 'Catumaxomab', 'newLinkedTarg...
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Q4.1336
Q4
What drugs target the gene SCN5A?
The drugs that target SCN5A are Propoxycaine, Orphenadrine, Indecainide, Quinidine Polygalacturonate, Fosphenytoin Sodium, Prilocaine Hydrochloride, Zonisamide, Mexiletine, Flecainide Acetate, Hexylcaine Hydrochloride, Vernakalant, Fosphenytoin, Phenazopyridine Hydrochloride, Primidone, Phenytoin Sodium, Propafenone, T...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%SCN5A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_718', 'drugName': 'Vernakalant', 'newLinkedTargets_string': 'KCND3 (ENSG00000171385), KCNA5 (ENSG00000130037), KCNJ3 (ENSG00000162989), KCNJ5 (ENSG00000120457), KCNH2 (ENSG00000055118), SCN5A (ENSG00000183873)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets...
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Q4.1110
Q4
What drugs target the gene POLR2A?
There are no approved drugs targeting POLR2A, but the drug Tas-106, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%POLR2A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3830', 'drugName': 'Tas-106', 'newLinkedTargets_string': 'POLR1A (ENSG00000068654), POLR3A (ENSG00000148606), POLR2A (ENSG00000181222)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_3831', 'drugName': 'Tas-106', 'newLinkedTargets_string': 'POLR1A (ENSG...
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Q4.1429
Q4
What drugs target the gene THRA?
The drugs that target THRA are Liothyronine, Levothyroxine, Dextrothyroxine Sodium, Dextrothyroxine, Liothyronine Sodium, and Levothyroxine Sodium.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%THRA %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_637', 'drugName': 'Levothyroxine', 'newLinkedTargets_string': 'THRA (ENSG00000126351), THRB (ENSG00000151090)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4914', 'drugName': 'Liothyronine Sodium', 'newLinkedTargets_string': 'THRA (ENSG00000126351), TH...
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Q4.106
Q4
What drugs target the gene BCL2L2?
There are no FDA approved drugs targeting the gene BCL2L2. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Obatoclax, Obatoclax Mesylate, and Navitoclax.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%BCL2L2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2962', 'drugName': 'Obatoclax Mesylate', 'newLinkedTargets_string': 'BCL2 (ENSG00000171791), BCL2L1 (ENSG00000171552), MCL1 (ENSG00000143384), BCL2L2-PABPN1 (ENSG00000258643), BCL2L2 (ENSG00000129473), BCL2A1 (ENSG00000140379), BCL2L10 (ENSG00000137875)', 'drugIsApproved': False, 'maxClini...
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Q4.613
Q4
What drugs target the gene HSPA8?
There are no FDA approved drugs targeting the gene HSPA8. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Forigerimod and Forigerimod Acetate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%HSPA8 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1772', 'drugName': 'Forigerimod', 'newLinkedTargets_string': 'HSPA8 (ENSG00000109971)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_3527', 'drugName': 'Forigerimod Acetate', 'newLinkedTargets_string': 'HSPA8 (ENSG00000109971)', 'drugIsApproved': False...
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Q4.1338
Q4
What drugs target the gene SCN8A?
The drugs that target SCN8A are Propoxycaine, Orphenadrine, Indecainide, Quinidine Polygalacturonate, Fosphenytoin Sodium, Prilocaine Hydrochloride, Zonisamide, Mexiletine, Hexylcaine Hydrochloride, Fosphenytoin, Phenazopyridine Hydrochloride, Primidone, Phenytoin Sodium, Propafenone, Topiramate, Chloroprocaine, Etidoc...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%SCN8A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1606', 'drugName': 'Chloroprocaine', 'newLinkedTargets_string': 'SCN1A (ENSG00000144285), SCN5A (ENSG00000183873), SCN4A (ENSG00000007314), SCN7A (ENSG00000136546), SCN2A (ENSG00000136531), SCN9A (ENSG00000169432), SCN3A (ENSG00000153253), SCN11A (ENSG00000168356), SCN8A (ENSG00000196876),...
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Q4.693
Q4
What drugs target the gene IL2RA?
The drugs that target IL2RA are Basiliximab, Aldesleukin, Denileukin Diftitox, and Daclizumab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%IL2RA %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5634', 'drugName': 'Denileukin Diftitox', 'newLinkedTargets_string': 'IL2RA (ENSG00000134460), IL2RG (ENSG00000147168), IL2RB (ENSG00000100385), EEF2 (ENSG00000167658)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5633', 'drugName': 'Denileukin Diftito...
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Q4.1360
Q4
What drugs target the gene SLC10A2?
The drugs that target SLC10A2 are Odevixibat, Maralixibat, and Maralixibat Chloride.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%SLC10A2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5835', 'drugName': 'Maralixibat', 'newLinkedTargets_string': 'SLC10A2 (ENSG00000125255)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5944', 'drugName': 'Maralixibat Chloride', 'newLinkedTargets_string': 'SLC10A2 (ENSG00000125255)', 'drugIsApproved': T...
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Q4.1473
Q4
What drugs target the gene TPH1?
The drugs that target TPH1 are Telotristat Etiprate, Telotristat Ethyl, and Telotristat.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TPH1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3468', 'drugName': 'Telotristat', 'newLinkedTargets_string': 'TPH2 (ENSG00000139287), TPH1 (ENSG00000129167)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1064', 'drugName': 'Telotristat Etiprate', 'newLinkedTargets_string': 'TPH2 (ENSG00000139287), TP...
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Q4.63
Q4
What drugs target the gene ANGPTL3?
The drug that targets ANGPTL3 is Evinacumab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ANGPTL3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5281', 'drugName': 'Evinacumab', 'newLinkedTargets_string': 'ANGPTL3 (ENSG00000132855)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2325', 'drugName': 'Vupanorsen', 'newLinkedTargets_string': 'ANGPTL3 (ENSG00000132855), ASGR1 (ENSG00000141505)', 'drug...
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Genetic Target
Q4.283
Q4
What drugs target the gene CNR1?
The drugs that target CNR1 are Nabilone, Dronabinol, Rimonabant, and Cannabidiol.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CNR1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4055', 'drugName': 'Cannabidiol', 'newLinkedTargets_string': 'CNR1 (ENSG00000118432)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3038', 'drugName': 'Dronabinol', 'newLinkedTargets_string': 'CNR1 (ENSG00000118432)', 'drugIsApproved': True, 'maxClinica...
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Genetic Target
Q4.783
Q4
What drugs target the gene KCNV1?
The drugs that target KCNV1 are Dalfampridine, Guanidine, Amifampridine Phosphate, Guanidine Hydrochloride, and Amifampridine.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%KCNV1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5118', 'drugName': 'Guanidine Hydrochloride', 'newLinkedTargets_string': 'KCNQ1 (ENSG00000053918), KCND3 (ENSG00000171385), KCNH2 (ENSG00000055118), KCNA2 (ENSG00000177301), KCNA1 (ENSG00000111262), KCNQ2 (ENSG00000075043), KCNQ3 (ENSG00000184156), KCNA7 (ENSG00000104848), KCNQ5 (ENSG00000...
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Q4.1037
Q4
What drugs target the gene PARP3?
The drugs that target PARP3 are Olaparib, Rucaparib, and Rucaparib Camsylate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PARP3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3166', 'drugName': 'Rucaparib', 'newLinkedTargets_string': 'PARP1 (ENSG00000143799), PARP3 (ENSG00000041880), PARP2 (ENSG00000129484)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_279', 'drugName': 'Olaparib', 'newLinkedTargets_string': 'PARP1 (ENSG000...
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Genetic Target
Q4.240
Q4
What drugs target the gene CDK19?
There are no FDA approved drugs targeting the gene CDK19. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Roniciclib, Pha-793887, Azd-5438, and At-7519.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CDK19 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1429', 'drugName': 'Roniciclib', 'newLinkedTargets_string': 'CDK1 (ENSG00000170312), CDK4 (ENSG00000135446), CDK2 (ENSG00000123374), CDK5 (ENSG00000164885), CDK6 (ENSG00000105810), CDK7 (ENSG00000134058), CDK3 (ENSG00000250506), CDK16 (ENSG00000102225), CDK18 (ENSG00000117266), CDK8 (ENSG0...
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Genetic Target
Q4.225
Q4
What drugs target the gene CD80?
The drugs that target CD80 are Abatacept and Belatacept.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CD80 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4093', 'drugName': 'Belatacept', 'newLinkedTargets_string': 'CD80 (ENSG00000121594), CD86 (ENSG00000114013)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4094', 'drugName': 'Belatacept', 'newLinkedTargets_string': 'CD80 (ENSG00000121594), CD86 (ENSG000...
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Q4.147
Q4
What drugs target the gene CACNA1F?
The drugs that target CACNA1F are Gabapentin, Nicardipine, Clevidipine, Terodiline Hydrochloride, Nicardipine Hydrochloride, Amlodipine Maleate, Lacidipine, Lercanidipine, Diltiazem Hydrochloride, Nimodipine, Amlodipine, Phloroglucinol, Nitrendipine, Suloctidil, Amlodipine Besylate, Pregabalin, Diltiazem Malate, Nifedi...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CACNA1F %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6292', 'drugName': 'Terodiline', 'newLinkedTargets_string': 'CHRM3 (ENSG00000133019), CHRM4 (ENSG00000180720), CHRM1 (ENSG00000168539), CHRM2 (ENSG00000181072), CHRM5 (ENSG00000184984), CACNA1H (ENSG00000196557), CACNA2D1 (ENSG00000153956), CACNA1C (ENSG00000151067), CACNA2D3 (ENSG00000157...
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Genetic Target
Q4.1434
Q4
What drugs target the gene TLR3?
There are no FDA approved drugs targeting the gene TLR3. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Bevasiranib, Bevasiranib Sodium, and Rintatolimod.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TLR3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4726', 'drugName': 'Bevasiranib', 'newLinkedTargets_string': 'TLR3 (ENSG00000164342)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_4727', 'drugName': 'Bevasiranib', 'newLinkedTargets_string': 'TLR3 (ENSG00000164342)', 'drugIsApproved': False, 'maxClin...
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Q4.375
Q4
What drugs target the gene DRD3?
The drugs that target DRD3 are Promazine Hydrochloride, Haloperidol Decanoate, Loxapine Succinate, Bromocriptine, Levomepromazine, Pramipexole, Droperidol, Cariprazine, Amisulpride, Ropinirole, Olanzapine Pamoate, Ropinirole Hydrochloride, Rotigotine, Amoxapine, Olanzapine, Chlorpromazine Hydrochloride, Chlorpromazine,...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%DRD3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4041', 'drugName': 'Loxapine', 'newLinkedTargets_string': 'HTR2A (ENSG00000102468), HTR2C (ENSG00000147246), DRD2 (ENSG00000149295), DRD3 (ENSG00000151577), DRD4 (ENSG00000069696)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1241', 'drugName': 'Caripr...
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Q4.1271
Q4
What drugs target the gene RPL9?
The drug that targets RPL9 is Ataluren.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RPL9 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG00000083845), RPS7 (ENSG...
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Q4.120
Q4
What drugs target the gene BRD2?
There are no FDA approved drugs targeting the gene BRD2. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Bms-986158, Apabetalone, Pelabresib, Ro-6870810, Birabresib, and Molibresib.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%BRD2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_866', 'drugName': 'Pelabresib', 'newLinkedTargets_string': 'BRD2 (ENSG00000204256), BRD4 (ENSG00000141867), BRDT (ENSG00000137948), BRD3 (ENSG00000169925)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_746', 'drugName': 'Apabetalone', 'newLinkedTargets...
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Q4.1153
Q4
What drugs target the gene PSMA3?
The drugs that target PSMA3 are Bortezomib, Carfilzomib, Ixazomib, and Ixazomib Citrate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PSMA3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3334', 'drugName': 'Ixazomib', 'newLinkedTargets_string': 'PSMD1 (ENSG00000173692), PSMB2 (ENSG00000126067), PSMB1 (ENSG00000008018), PSMB5 (ENSG00000100804), PSMB8 (ENSG00000204264), PSMB9 (ENSG00000240065), PSMB6 (ENSG00000142507), PSMD14 (ENSG00000115233), PSMA1 (ENSG00000129084), PSMA2...
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Q4.252
Q4
What drugs target the gene CETP?
There are no FDA approved drugs targeting the gene CETP. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Torcetrapib, Obicetrapib, Anacetrapib, Dalcetrapib, Rocacetrapib, and Evacetrapib.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CETP %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5790', 'drugName': 'Evacetrapib', 'newLinkedTargets_string': 'CETP (ENSG00000087237)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_2315', 'drugName': 'Obicetrapib', 'newLinkedTargets_string': 'CETP (ENSG00000087237)', 'drugIsApproved': False, 'maxClin...
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Q4.1481
Q4
What drugs target the gene TRGV3?
There are no FDA approved drugs targeting the gene TRGV3. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Medi-500, Tol-101, and Maslimomab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TRGV3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1483', 'drugName': 'Medi-500', 'newLinkedTargets_string': 'TRAV29DV5 (ENSG00000211810), TRAC (ENSG00000277734), TRBV7-9 (ENSG00000278030), TRGV3 (ENSG00000211699)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_5971', 'drugName': 'Tol-101', 'newLinkedTa...
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Q4.1239
Q4
What drugs target the gene RPL18A?
The drug that targets RPL18A is Ataluren.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RPL18A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG00000083845), RPS7 (ENSG...
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Q4.920
Q4
What drugs target the gene MUC16?
The drug that targets MUC16 is Igovomab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%MUC16 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_640', 'drugName': 'Igovomab', 'newLinkedTargets_string': 'MUC16 (ENSG00000181143)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3687', 'drugName': 'Oregovomab', 'newLinkedTargets_string': 'MUC16 (ENSG00000181143)', 'drugIsApproved': False, 'maxClinical...
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Q4.10
Q4
What drugs target the gene ACACB?
There are no FDA approved drugs targeting the gene ACACB. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Olumacostat Glasaretil, Clesacostat, Pf-05175157, and Firsocostat.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ACACB %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1425', 'drugName': 'Olumacostat Glasaretil', 'newLinkedTargets_string': 'ACACA (ENSG00000278540), ACACB (ENSG00000076555)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_2233', 'drugName': 'Clesacostat', 'newLinkedTargets_string': 'ACACA (ENSG0000027854...
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Q4.451
Q4
What drugs target the gene FCGR1A?
There are no FDA approved drugs targeting the gene FCGR1A. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Mdx-210 and Mdx-447.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%FCGR1A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4872', 'drugName': 'Mdx-447', 'newLinkedTargets_string': 'EGFR (ENSG00000146648), FCGR1A (ENSG00000150337)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_4871', 'drugName': 'Mdx-447', 'newLinkedTargets_string': 'EGFR (ENSG00000146648), FCGR1A (ENSG0000...
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Q4.911
Q4
What drugs target the gene MT-ND4?
The drugs that target MT-ND4 are Metformin and Metformin Hydrochloride.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%MT-ND4 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (ENSG00000165264), NDUFA4 (...
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Q4.713
Q4
What drugs target the gene IRAK4?
There are no approved drugs targeting IRAK4, but the drug Zimlovisertib, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%IRAK4 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4254', 'drugName': 'Zimlovisertib', 'newLinkedTargets_string': 'IRAK4 (ENSG00000198001)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
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Q4.257
Q4
What drugs target the gene CHEK2?
There are no FDA approved drugs targeting the gene CHEK2. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Prexasertib and Xl-844.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CHEK2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_562', 'drugName': 'Prexasertib', 'newLinkedTargets_string': 'CHEK1 (ENSG00000149554), CHEK2 (ENSG00000183765)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_563', 'drugName': 'Prexasertib', 'newLinkedTargets_string': 'CHEK1 (ENSG00000149554), CHEK2 (EN...
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Q4.597
Q4
What drugs target the gene HMGCR?
The drugs that target HMGCR are Pitavastatin Calcium, Cerivastatin, Fluvastatin Sodium, Fluvastatin, Pitavastatin Sodium, Pravastatin Sodium, Pitavastatin Magnesium, Cerivastatin Sodium, Simvastatin, Atorvastatin Calcium, Lovastatin, Atorvastatin, Rosuvastatin Calcium, Pravastatin, Pitavastatin, and Rosuvastatin.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%HMGCR %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1184', 'drugName': 'Fluvastatin Sodium', 'newLinkedTargets_string': 'HMGCR (ENSG00000113161)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5208', 'drugName': 'Rosuvastatin Calcium', 'newLinkedTargets_string': 'HMGCR (ENSG00000113161)', 'drugIsApproved'...
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Q4.391
Q4
What drugs target the gene EFNB2?
There are no approved drugs targeting EFNB2, but the drug Sephb4-Hsa, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%EFNB2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6169', 'drugName': 'Sephb4-Hsa', 'newLinkedTargets_string': 'EFNB2 (ENSG00000125266)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
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Q4.1321
Q4
What drugs target the gene RXRB?
The drugs that target RXRB are Etretinate, Alitretinoin, Bexarotene, and Acitretin.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RXRB %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5080', 'drugName': 'Acitretin', 'newLinkedTargets_string': 'RXRB (ENSG00000204231), RARG (ENSG00000172819), RXRG (ENSG00000143171), RARB (ENSG00000077092), RARA (ENSG00000131759), RXRA (ENSG00000186350)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_701...
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Q4.1231
Q4
What drugs target the gene RPL11?
The drug that targets RPL11 is Ataluren.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RPL11 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG00000083845), RPS7 (ENSG...
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Q4.560
Q4
What drugs target the gene GSK3B?
The drugs that target GSK3B are Lithium Citrate and Lithium Carbonate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%GSK3B %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3119', 'drugName': 'Lithium Carbonate', 'newLinkedTargets_string': 'IMPA1 (ENSG00000133731), GSK3A (ENSG00000105723), GSK3B (ENSG00000082701)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5478', 'drugName': 'Lithium Citrate', 'newLinkedTargets_string':...
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Q4.1320
Q4
What drugs target the gene RXRA?
The drugs that target RXRA are Etretinate, Alitretinoin, Danthron, Bexarotene, and Acitretin.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RXRA %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_701', 'drugName': 'Alitretinoin', 'newLinkedTargets_string': 'RXRB (ENSG00000204231), RARG (ENSG00000172819), RXRG (ENSG00000143171), RARB (ENSG00000077092), RARA (ENSG00000131759), RXRA (ENSG00000186350)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3...
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Q4.867
Q4
What drugs target the gene MARCKS?
There are no approved drugs targeting MARCKS, but the drug Bio-11006, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%MARCKS %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5771', 'drugName': 'Bio-11006', 'newLinkedTargets_string': 'MARCKS (ENSG00000277443)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
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Genetic Target
Q4.462
Q4
What drugs target the gene FGF2?
There are no approved drugs targeting FGF2, but the drug Muparfostat, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%FGF2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5103', 'drugName': 'Muparfostat', 'newLinkedTargets_string': 'HPSE (ENSG00000173083), FGF1 (ENSG00000113578), FGF2 (ENSG00000138685), VEGFA (ENSG00000112715)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_5102', 'drugName': 'Muparfostat', 'newLinkedTar...
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Genetic Target
Q4.728
Q4
What drugs target the gene ITGB8?
There are no approved drugs targeting ITGB8, but the drug Abituzumab, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ITGB8 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1968', 'drugName': 'Abituzumab', 'newLinkedTargets_string': 'ITGAV (ENSG00000138448), ITGB6 (ENSG00000115221), ITGB5 (ENSG00000082781), ITGB3 (ENSG00000259207), ITGB1 (ENSG00000150093), ITGB8 (ENSG00000105855)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTarget...
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Genetic Target
Q4.1417
Q4
What drugs target the gene TEC?
There are no approved drugs targeting TEC, but the drug Pf-06651600, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TEC %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4380', 'drugName': 'Pf-06651600', 'newLinkedTargets_string': 'ITK (ENSG00000113263), BMX (ENSG00000102010), TEC (ENSG00000135605), TXK (ENSG00000074966), BTK (ENSG00000010671), JAK3 (ENSG00000105639)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_4381'...
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Genetic Target
Q4.146
Q4
What drugs target the gene CACNA1E?
The drugs that target CACNA1E are Gabapentin, Terodiline Hydrochloride, Phloroglucinol, Suloctidil, Pregabalin, Gabapentin Enacarbil, Bepridil Hydrochloride, Bepridil, and Terodiline.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CACNA1E %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_142', 'drugName': 'Gabapentin', 'newLinkedTargets_string': 'CACNA1H (ENSG00000196557), CACNA2D1 (ENSG00000153956), CACNA1C (ENSG00000151067), CACNA2D3 (ENSG00000157445), CACNA1S (ENSG00000081248), CACNA2D2 (ENSG00000007402), CACNA1D (ENSG00000157388), CACNA1A (ENSG00000141837), CACNA1B (EN...
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Genetic Target
Q4.504
Q4
What drugs target the gene GABRG1?
The drugs that target GABRG1 are Meprobamate, Acamprosate Calcium, Enflurane, Methohexital, Metharbital, Butabarbital, Flurazepam Hydrochloride, Pentobarbital Sodium, Acamprosate, Primidone, Temazepam, Flunitrazepam, Ganaxolone, Diazepam, Methyprylon, Thiopental, Clonazepam, Topiramate, Remimazolam Besylate, Brexanolon...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%GABRG1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1494', 'drugName': 'Thiopental', 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089), GABRA3 (ENSG00000011677), GABRP (ENSG00000094755...
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Genetic Target
Q4.1175
Q4
What drugs target the gene PSMC6?
The drugs that target PSMC6 are Bortezomib, Carfilzomib, Ixazomib, and Ixazomib Citrate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PSMC6 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_559', 'drugName': 'Bortezomib', 'newLinkedTargets_string': 'PSMD1 (ENSG00000173692), PSMB2 (ENSG00000126067), PSMB1 (ENSG00000008018), PSMB5 (ENSG00000100804), PSMB8 (ENSG00000204264), PSMB9 (ENSG00000240065), PSMB6 (ENSG00000142507), PSMD14 (ENSG00000115233), PSMA1 (ENSG00000129084), PSMA...
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Genetic Target
Q4.744
Q4
What drugs target the gene KCNC2?
The drugs that target KCNC2 are Dalfampridine, Guanidine, Amifampridine Phosphate, Guanidine Hydrochloride, and Amifampridine.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%KCNC2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5118', 'drugName': 'Guanidine Hydrochloride', 'newLinkedTargets_string': 'KCNQ1 (ENSG00000053918), KCND3 (ENSG00000171385), KCNH2 (ENSG00000055118), KCNA2 (ENSG00000177301), KCNA1 (ENSG00000111262), KCNQ2 (ENSG00000075043), KCNQ3 (ENSG00000184156), KCNA7 (ENSG00000104848), KCNQ5 (ENSG00000...
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Genetic Target
Q4.1420
Q4
What drugs target the gene TFPI?
There are no FDA approved drugs targeting the gene TFPI. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Concizumab, Andexanet Alfa, Marstacimab, and Bay-1093884.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TFPI %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6201', 'drugName': 'Marstacimab', 'newLinkedTargets_string': 'TFPI (ENSG00000003436)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_5154', 'drugName': 'Andexanet Alfa', 'newLinkedTargets_string': 'TFPI (ENSG00000003436)', 'drugIsApproved': False, 'maxC...
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Genetic Target
Q4.736
Q4
What drugs target the gene KCNA3?
The drugs that target KCNA3 are Dalfampridine, Guanidine, Amifampridine Phosphate, Guanidine Hydrochloride, and Amifampridine.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%KCNA3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5118', 'drugName': 'Guanidine Hydrochloride', 'newLinkedTargets_string': 'KCNQ1 (ENSG00000053918), KCND3 (ENSG00000171385), KCNH2 (ENSG00000055118), KCNA2 (ENSG00000177301), KCNA1 (ENSG00000111262), KCNQ2 (ENSG00000075043), KCNQ3 (ENSG00000184156), KCNA7 (ENSG00000104848), KCNQ5 (ENSG00000...
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Genetic Target
Q4.542
Q4
What drugs target the gene GRIA4?
The drugs that target GRIA4 are Topiramate and Perampanel.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%GRIA4 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2165', 'drugName': 'Perampanel', 'newLinkedTargets_string': 'GRIA4 (ENSG00000152578), GRIA3 (ENSG00000125675), GRIA2 (ENSG00000120251), GRIA1 (ENSG00000155511)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1593', 'drugName': 'Topiramate', 'newLinkedTar...
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Genetic Target
Q4.179
Q4
What drugs target the gene CASP4?
There are no approved drugs targeting CASP4, but the drug Emricasan, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CASP4 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_45', 'drugName': 'Emricasan', 'newLinkedTargets_string': 'CASP4 (ENSG00000196954), CASP9 (ENSG00000132906), CASP3 (ENSG00000164305), CASP5 (ENSG00000137757), CASP6 (ENSG00000138794), CASP7 (ENSG00000165806), CASP8 (ENSG00000064012), CASP1 (ENSG00000137752), CASP2 (ENSG00000106144), CASP10 ...
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Genetic Target
Q4.1483
Q4
What drugs target the gene TRPA1?
The drugs that target TRPA1 are Butamben Picrate, Butamben, and Menthol.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TRPA1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5721', 'drugName': 'Menthol', 'newLinkedTargets_string': 'TRPA1 (ENSG00000104321), TRPM8 (ENSG00000144481)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5054', 'drugName': 'Butamben', 'newLinkedTargets_string': 'TRPA1 (ENSG00000104321), TRPV4 (ENSG0000...
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Q4.702
Q4
What drugs target the gene IL5RA?
The drug that targets IL5RA is Benralizumab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%IL5RA %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5224', 'drugName': 'Benralizumab', 'newLinkedTargets_string': 'IL5RA (ENSG00000091181)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}]
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Genetic Target
Q4.969
Q4
What drugs target the gene NDUFS3?
The drugs that target NDUFS3 are Metformin and Metformin Hydrochloride.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NDUFS3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (ENSG00000165264), NDUFA4 (...
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Genetic Target
Q4.1069
Q4
What drugs target the gene PDK3?
The drug that targets PDK3 is Sodium Dichloroacetate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PDK3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2764', 'drugName': 'Sodium Dichloroacetate', 'newLinkedTargets_string': 'PDK2 (ENSG00000005882), PDK3 (ENSG00000067992), PDK4 (ENSG00000004799), PDK1 (ENSG00000152256)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}]
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Genetic Target
Q4.903
Q4
What drugs target the gene MPO?
There are no approved drugs targeting MPO, but the drug Verdiperstat, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%MPO %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1006', 'drugName': 'Verdiperstat', 'newLinkedTargets_string': 'MPO (ENSG00000005381)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}]
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Genetic Target
Q4.927
Q4
What drugs target the gene MYL4?
The drug that targets MYL4 is Mavacamten.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%MYL4 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1036', 'drugName': 'Mavacamten', 'newLinkedTargets_string': 'MYH7 (ENSG00000092054), MYH6 (ENSG00000197616), MYH7B (ENSG00000078814), MYL3 (ENSG00000160808), MYL2 (ENSG00000111245), MYL7 (ENSG00000106631), MYL4 (ENSG00000198336)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID...
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Genetic Target
Q4.1531
Q4
What drugs target the gene WEE1?
There are no FDA approved drugs targeting the gene WEE1. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Adavosertib and Azenosertib.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%WEE1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5552', 'drugName': 'Azenosertib', 'newLinkedTargets_string': 'WEE1 (ENSG00000166483)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_224', 'drugName': 'Adavosertib', 'newLinkedTargets_string': 'WEE1 (ENSG00000166483)', 'drugIsApproved': False, 'maxClini...
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Genetic Target
Q4.8
Q4
What drugs target the gene ABL1?
The drugs that target ABL1 are Nilotinib Hydrochloride Monohydrate, Regorafenib, Ponatinib, Imatinib, Umbralisib Tosylate, Imatinib Mesylate, Asciminib, Bosutinib, Asciminib Hydrochloride, Dasatinib, Umbralisib, Nilotinib, and Ponatinib Hydrochloride.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ABL1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_802', 'drugName': 'Regorafenib', 'newLinkedTargets_string': 'EPHA2 (ENSG00000142627), TEK (ENSG00000120156), MAPK11 (ENSG00000185386), RAF1 (ENSG00000132155), FRK (ENSG00000111816), PDGFRB (ENSG00000113721), PDGFRA (ENSG00000134853), KIT (ENSG00000157404), FGFR1 (ENSG00000077782), DDR2 (EN...
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Genetic Target
Q4.908
Q4
What drugs target the gene MT-ND1?
The drugs that target MT-ND1 are Metformin and Metformin Hydrochloride.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%MT-ND1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (ENSG00000165264), NDUFA4 (...
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Genetic Target
Q4.672
Q4
What drugs target the gene IL13RA1?
There are no approved drugs targeting IL13RA1, but the drug Cintredekin Besudotox, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%IL13RA1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2466', 'drugName': 'Cintredekin Besudotox', 'newLinkedTargets_string': 'IL4R (ENSG00000077238), IL13RA1 (ENSG00000131724), IL13RA2 (ENSG00000123496)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_2467', 'drugName': 'Cintredekin Besudotox', 'newLinkedTa...
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Genetic Target
Q4.1436
Q4
What drugs target the gene TLR5?
There are no approved drugs targeting TLR5, but the drug Entolimod, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TLR5 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3738', 'drugName': 'Entolimod', 'newLinkedTargets_string': 'TLR5 (ENSG00000187554)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
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Genetic Target
Q4.359
Q4
What drugs target the gene DHCR24?
The drug that targets DHCR24 is Triparanol.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%DHCR24 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3812', 'drugName': 'Triparanol', 'newLinkedTargets_string': 'DHCR24 (ENSG00000116133)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}]
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Genetic Target
Q4.788
Q4
What drugs target the gene KIF11?
There are no FDA approved drugs targeting the gene KIF11. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Azd-4877, Ispinesib, Litronesib, and Filanesib.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%KIF11 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5386', 'drugName': 'Litronesib', 'newLinkedTargets_string': 'KIF11 (ENSG00000138160)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_3893', 'drugName': 'Ispinesib', 'newLinkedTargets_string': 'KIF11 (ENSG00000138160)', 'drugIsApproved': False, 'maxClini...
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Genetic Target
Q4.740
Q4
What drugs target the gene KCNA7?
The drugs that target KCNA7 are Dalfampridine, Guanidine, Amifampridine Phosphate, Guanidine Hydrochloride, and Amifampridine.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%KCNA7 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5118', 'drugName': 'Guanidine Hydrochloride', 'newLinkedTargets_string': 'KCNQ1 (ENSG00000053918), KCND3 (ENSG00000171385), KCNH2 (ENSG00000055118), KCNA2 (ENSG00000177301), KCNA1 (ENSG00000111262), KCNQ2 (ENSG00000075043), KCNQ3 (ENSG00000184156), KCNA7 (ENSG00000104848), KCNQ5 (ENSG00000...
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Genetic Target
Q4.331
Q4
What drugs target the gene CTSC?
There are no approved drugs targeting CTSC, but the drug Brensocatib, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CTSC %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1902', 'drugName': 'Brensocatib', 'newLinkedTargets_string': 'CTSC (ENSG00000109861)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}]
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Genetic Target
Q4.1230
Q4
What drugs target the gene RPL10A?
The drug that targets RPL10A is Ataluren.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RPL10A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG00000083845), RPS7 (ENSG...
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Genetic Target
Q4.1176
Q4
What drugs target the gene PSMD1?
The drugs that target PSMD1 are Bortezomib, Carfilzomib, Ixazomib, and Ixazomib Citrate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PSMD1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_559', 'drugName': 'Bortezomib', 'newLinkedTargets_string': 'PSMD1 (ENSG00000173692), PSMB2 (ENSG00000126067), PSMB1 (ENSG00000008018), PSMB5 (ENSG00000100804), PSMB8 (ENSG00000204264), PSMB9 (ENSG00000240065), PSMB6 (ENSG00000142507), PSMD14 (ENSG00000115233), PSMA1 (ENSG00000129084), PSMA...
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Genetic Target
Q4.1270
Q4
What drugs target the gene RPL8?
The drug that targets RPL8 is Ataluren.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RPL8 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG00000083845), RPS7 (ENSG...
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Genetic Target
Q4.260
Q4
What drugs target the gene CHRM2?
The drugs that target CHRM2 are Oxybutynin, Terodiline Hydrochloride, Oxybutynin Chloride, Tolterodine, Fesoterodine, Solifenacin Succinate, Atropine Sulfate, Bethanechol, Darifenacin Hydrobromide, Propantheline, Tolterodine Tartrate, Solifenacin, Fesoterodine Fumarate, Atropine, Darifenacin, Alcuronium, Propantheline ...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CHRM2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3301', 'drugName': 'Tolterodine Tartrate', 'newLinkedTargets_string': 'CHRM3 (ENSG00000133019), CHRM2 (ENSG00000181072)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_871', 'drugName': 'Oxybutynin Chloride', 'newLinkedTargets_string': 'CHRM3 (ENSG000001...
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Q4.1255
Q4
What drugs target the gene RPL34?
The drug that targets RPL34 is Ataluren.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RPL34 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG00000083845), RPS7 (ENSG...
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Q4.374
Q4
What drugs target the gene DRD2?
The drugs that target DRD2 are Promazine Hydrochloride, Thiethylperazine Maleate, Perphenazine, Triflupromazine, Benzquinamide, Prochlorperazine, Fluphenazine Decanoate, Haloperidol Decanoate, Loxapine Succinate, Trimipramine Maleate, Bromocriptine, Levomepromazine, Veralipride, Molindone, Fluspirilene, Fluphenazine En...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%DRD2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5204', 'drugName': 'Metoclopramide Hydrochloride', 'newLinkedTargets_string': 'HTR4 (ENSG00000164270), HTR3A (ENSG00000166736), DRD2 (ENSG00000149295)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_426', 'drugName': 'Prochlorperazine', 'newLinkedTargets...
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Q4.1128
Q4
What drugs target the gene PRKACA?
There are no approved drugs targeting PRKACA, but the drug Gsk-690693, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PRKACA %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1835', 'drugName': 'Gsk-690693', 'newLinkedTargets_string': 'PRKACB (ENSG00000142875), PRKACA (ENSG00000072062), PRKACG (ENSG00000165059), AKT2 (ENSG00000105221), AKT3 (ENSG00000117020), AKT1 (ENSG00000142208), PRKD3 (ENSG00000115825), PRKCI (ENSG00000163558), PRKCA (ENSG00000154229), PRKC...
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Q4.954
Q4
What drugs target the gene NDUFB1?
The drugs that target NDUFB1 are Metformin and Metformin Hydrochloride.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NDUFB1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (ENSG00000165264), NDUFA4 (...
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Q4.144
Q4
What drugs target the gene CACNA1C?
The drugs that target CACNA1C are Gabapentin, Nicardipine, Clevidipine, Terodiline Hydrochloride, Nicardipine Hydrochloride, Amlodipine Maleate, Lacidipine, Lercanidipine, Diltiazem Hydrochloride, Nimodipine, Amlodipine, Phloroglucinol, Nitrendipine, Suloctidil, Amlodipine Besylate, Pregabalin, Diltiazem Malate, Nifedi...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CACNA1C %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6292', 'drugName': 'Terodiline', 'newLinkedTargets_string': 'CHRM3 (ENSG00000133019), CHRM4 (ENSG00000180720), CHRM1 (ENSG00000168539), CHRM2 (ENSG00000181072), CHRM5 (ENSG00000184984), CACNA1H (ENSG00000196557), CACNA2D1 (ENSG00000153956), CACNA1C (ENSG00000151067), CACNA2D3 (ENSG00000157...
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Q4.528
Q4
What drugs target the gene GNRHR?
The drugs that target GNRHR are Ganirelix Acetate, Goserelin Acetate, Leuprolide Mesylate, Gonadorelin, Linzagolix, Nafarelin Acetate, Nafarelin, Degarelix, Relugolix, Goserelin, Leuprolide, Cetrorelix, Gonadorelin Acetate, Histrelin Acetate, Cetrorelix Acetate, Triptorelin, Histrelin, Triptorelin Pamoate, Leuprolide A...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%GNRHR %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4802', 'drugName': 'Leuprolide Acetate', 'newLinkedTargets_string': 'GNRHR (ENSG00000109163)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2259', 'drugName': 'Goserelin', 'newLinkedTargets_string': 'GNRHR (ENSG00000109163)', 'drugIsApproved': True, 'ma...
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Q4.1164
Q4
What drugs target the gene PSMB4?
The drugs that target PSMB4 are Bortezomib, Carfilzomib, Ixazomib, and Ixazomib Citrate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PSMB4 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3334', 'drugName': 'Ixazomib', 'newLinkedTargets_string': 'PSMD1 (ENSG00000173692), PSMB2 (ENSG00000126067), PSMB1 (ENSG00000008018), PSMB5 (ENSG00000100804), PSMB8 (ENSG00000204264), PSMB9 (ENSG00000240065), PSMB6 (ENSG00000142507), PSMD14 (ENSG00000115233), PSMA1 (ENSG00000129084), PSMA2...
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Q4.234
Q4
What drugs target the gene CDK13?
There are no FDA approved drugs targeting the gene CDK13. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Roniciclib, Pha-793887, Azd-5438, and At-7519.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CDK13 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1429', 'drugName': 'Roniciclib', 'newLinkedTargets_string': 'CDK1 (ENSG00000170312), CDK4 (ENSG00000135446), CDK2 (ENSG00000123374), CDK5 (ENSG00000164885), CDK6 (ENSG00000105810), CDK7 (ENSG00000134058), CDK3 (ENSG00000250506), CDK16 (ENSG00000102225), CDK18 (ENSG00000117266), CDK8 (ENSG0...
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Q4.1212
Q4
What drugs target the gene RARB?
The drugs that target RARB are Etretinate, Alitretinoin, Adapalene, Isotretinoin, Acitretin, Tazarotene, and Tretinoin.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RARB %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5080', 'drugName': 'Acitretin', 'newLinkedTargets_string': 'RXRB (ENSG00000204231), RARG (ENSG00000172819), RXRG (ENSG00000143171), RARB (ENSG00000077092), RARA (ENSG00000131759), RXRA (ENSG00000186350)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_701...
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Q4.1459
Q4
What drugs target the gene TNKS?
There are no approved drugs targeting TNKS, but the drug 2X-121, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TNKS %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1419', 'drugName': '2X-121', 'newLinkedTargets_string': 'TNKS2 (ENSG00000107854), TNKS (ENSG00000173273), PARP1 (ENSG00000143799), PARP2 (ENSG00000129484)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_1420', 'drugName': '2X-121', 'newLinkedTargets_str...
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Q4.442
Q4
What drugs target the gene F5?
The drug that targets F5 is Drotrecogin Alfa (Activated).
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%F5 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2502', 'drugName': 'Drotrecogin Alfa (Activated)', 'newLinkedTargets_string': 'F8 (ENSG00000185010), F5 (ENSG00000198734)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2503', 'drugName': 'Drotrecogin Alfa (Activated)', 'newLinkedTargets_string': 'F8 (E...
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Q4.534
Q4
What drugs target the gene GPNMB?
There are no FDA approved drugs targeting the gene GPNMB. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Glembatumumab and Glembatumumab Vedotin.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%GPNMB %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6315', 'drugName': 'Glembatumumab Vedotin', 'newLinkedTargets_string': 'GPNMB (ENSG00000136235), TUBB4B (ENSG00000188229), TUBB1 (ENSG00000101162), TUBA3C (ENSG00000198033), TUBA4A (ENSG00000127824), TUBB3 (ENSG00000258947), TUBA1A (ENSG00000167552), TUBB4A (ENSG00000104833), TUBB8 (ENSG00...
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Q4.1232
Q4
What drugs target the gene RPL12?
The drug that targets RPL12 is Ataluren.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RPL12 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG00000083845), RPS7 (ENSG...
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