uuid stringlengths 4 8 | template_uuid stringclasses 40
values | question stringlengths 13 193 | answer stringlengths 29 2.2k | benchmark_query stringlengths 133 622 | execution_results stringlengths 2 1.14M | query_type stringclasses 2
values | sql_category stringclasses 26
values | bio_category stringclasses 14
values |
|---|---|---|---|---|---|---|---|---|
Q4.228 | Q4 | What drugs target the gene CDC7? | There are no FDA approved drugs targeting the gene CDC7. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Bms-863233, Rxdx-103, Nms-1116354, and Simurosertib. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%CDC7 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_1097', 'drugName': 'Bms-863233', 'newLinkedTargets_string': 'CDC7 (ENSG00000097046)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_5195', 'drugName': 'Simurosertib', 'newLinkedTargets_string': 'CDC7 (ENSG00000097046)', 'drugIsApproved': False, 'maxClin... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.1056 | Q4 | What drugs target the gene PDE6D? | The drugs that target PDE6D are Pentoxifylline and Dipyridamole. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%PDE6D %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_6107', 'drugName': 'Dipyridamole', 'newLinkedTargets_string': 'PDE5A (ENSG00000138735), PDE4A (ENSG00000065989), PDE3A (ENSG00000172572), PDE6H (ENSG00000139053), PDE6G (ENSG00000185527), PDE2A (ENSG00000186642), PDE7A (ENSG00000205268), PDE1A (ENSG00000115252), PDE9A (ENSG00000160191), PD... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.230 | Q4 | What drugs target the gene CDK1? | There are no FDA approved drugs targeting the gene CDK1. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Dinaciclib, Zotiraciclib, Roniciclib, Ag-24322, Pha-793887, Azd-5438, At-7519, Riviciclib, Rg-547, Rgb-286638, Alvocidib, Milciclib, and Seliciclib. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%CDK1 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_5622', 'drugName': 'Alvocidib', 'newLinkedTargets_string': 'CDK1 (ENSG00000170312), CDK7 (ENSG00000134058), CDK9 (ENSG00000136807), CDK6 (ENSG00000105810), CDK2 (ENSG00000123374), CDK4 (ENSG00000135446)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_49... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.1312 | Q4 | What drugs target the gene RPTOR? | There are no approved drugs targeting RPTOR, but the drug Indoximod, which potentially targets this gene, is currently undergoing clinical trials. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%RPTOR %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_2816', 'drugName': 'Indoximod', 'newLinkedTargets_string': 'MTOR (ENSG00000198793), RPTOR (ENSG00000141564), MLST8 (ENSG00000167965)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}] | general | Select, Similarity Search, Order By | Genetic Target |
Q4.1330 | Q4 | What drugs target the gene SCN10A? | The drugs that target SCN10A are Propoxycaine, Orphenadrine, Indecainide, Quinidine Polygalacturonate, Fosphenytoin Sodium, Prilocaine Hydrochloride, Zonisamide, Mexiletine, Hexylcaine Hydrochloride, Fosphenytoin, Phenazopyridine Hydrochloride, Primidone, Phenytoin Sodium, Propafenone, Topiramate, Chloroprocaine, Dibuc... | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%SCN10A %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_3875', 'drugName': 'Dronedarone Hydrochloride', 'newLinkedTargets_string': 'CACNA1C (ENSG00000151067), CACNA1S (ENSG00000081248), CACNA1D (ENSG00000157388), CACNA1F (ENSG00000102001), HCN4 (ENSG00000138622), SCN1A (ENSG00000144285), SCN5A (ENSG00000183873), SCN4A (ENSG00000007314), SCN7A (... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.214 | Q4 | What drugs target the gene CD4? | The drug that targets CD4 is Ibalizumab. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%CD4 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_1583', 'drugName': 'Ibalizumab', 'newLinkedTargets_string': 'CD4 (ENSG00000010610)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4573', 'drugName': 'Zanolimumab', 'newLinkedTargets_string': 'CD4 (ENSG00000010610)', 'drugIsApproved': False, 'maxClinical... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.890 | Q4 | What drugs target the gene MLNR? | There are no FDA approved drugs targeting the gene MLNR. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Mitemcinal, Atilmotin, Mitemcinal Fumarate, and Camicinal. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%MLNR %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_4697', 'drugName': 'Camicinal', 'newLinkedTargets_string': 'MLNR (ENSG00000102539)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_232', 'drugName': 'Mitemcinal', 'newLinkedTargets_string': 'MLNR (ENSG00000102539)', 'drugIsApproved': False, 'maxClinical... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.81 | Q4 | What drugs target the gene ATP1A2? | The drugs that target ATP1A2 are Acetyldigitoxin, Deslanoside, Digoxin, Lanatoside C, and Digitoxin. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%ATP1A2 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_2499', 'drugName': 'Digoxin', 'newLinkedTargets_string': 'ATP1A1 (ENSG00000163399), ATP1B2 (ENSG00000129244), ATP1B1 (ENSG00000143153), ATP1A2 (ENSG00000018625), ATP1B3 (ENSG00000069849), ATP1A3 (ENSG00000105409), ATP1A4 (ENSG00000132681), FXYD2 (ENSG00000137731)', 'drugIsApproved': True, ... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.150 | Q4 | What drugs target the gene CACNA1I? | The drugs that target CACNA1I are Gabapentin, Mibefradil Dihydrochloride, Terodiline Hydrochloride, Mibefradil, Phloroglucinol, Phensuximide, Suloctidil, Pregabalin, Methsuximide, Gabapentin Enacarbil, Trimethadione, Paramethadione, Bepridil Hydrochloride, Ethosuximide, Bepridil, and Terodiline. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%CACNA1I %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_4418', 'drugName': 'Trimethadione', 'newLinkedTargets_string': 'CACNA1H (ENSG00000196557), CACNA1G (ENSG00000006283), CACNA1I (ENSG00000100346)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4085', 'drugName': 'Methsuximide', 'newLinkedTargets_string': ... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.819 | Q4 | What drugs target the gene LGALS3? | There are no FDA approved drugs targeting the gene LGALS3. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Olitigaltin, Davanat, and Belapectin. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%LGALS3 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_6390', 'drugName': 'Belapectin', 'newLinkedTargets_string': 'LGALS3 (ENSG00000131981)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_3707', 'drugName': 'Olitigaltin', 'newLinkedTargets_string': 'LGALS3 (ENSG00000131981)', 'drugIsApproved': False, 'maxC... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.1208 | Q4 | What drugs target the gene RAMP1? | The drugs that target RAMP1 are Pramlintide and Pramlintide Acetate. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%RAMP1 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_2396', 'drugName': 'Pramlintide Acetate', 'newLinkedTargets_string': 'CALCR (ENSG00000004948), RAMP1 (ENSG00000132329), RAMP2 (ENSG00000131477), RAMP3 (ENSG00000122679)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_358', 'drugName': 'Pramlintide', 'new... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.941 | Q4 | What drugs target the gene NDUFA3? | The drugs that target NDUFA3 are Metformin and Metformin Hydrochloride. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%NDUFA3 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (ENSG00000165264), NDUFA4 (... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.676 | Q4 | What drugs target the gene IL17A? | The drugs that target IL17A are Bimekizumab, Secukinumab, and Ixekizumab. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%IL17A %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_306', 'drugName': 'Bimekizumab', 'newLinkedTargets_string': 'IL17F (ENSG00000112116), IL17A (ENSG00000112115)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3578', 'drugName': 'Ixekizumab', 'newLinkedTargets_string': 'IL17A (ENSG00000112115)', 'drugIsAp... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.1183 | Q4 | What drugs target the gene PSMD4? | The drugs that target PSMD4 are Bortezomib, Carfilzomib, Ixazomib, and Ixazomib Citrate. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%PSMD4 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_559', 'drugName': 'Bortezomib', 'newLinkedTargets_string': 'PSMD1 (ENSG00000173692), PSMB2 (ENSG00000126067), PSMB1 (ENSG00000008018), PSMB5 (ENSG00000100804), PSMB8 (ENSG00000204264), PSMB9 (ENSG00000240065), PSMB6 (ENSG00000142507), PSMD14 (ENSG00000115233), PSMA1 (ENSG00000129084), PSMA... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.558 | Q4 | What drugs target the gene GRM5? | There are no FDA approved drugs targeting the gene GRM5. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Dipraglurant, Basimglurant, Azd2516, Raseglurant, Rg7342, Ly545694, Azd2066, Stx107, and Mavoglurant. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%GRM5 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_2800', 'drugName': 'Azd2066', 'newLinkedTargets_string': 'GRM5 (ENSG00000168959)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_3225', 'drugName': 'Stx107', 'newLinkedTargets_string': 'GRM5 (ENSG00000168959)', 'drugIsApproved': False, 'maxClinicalTrial... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.936 | Q4 | What drugs target the gene NDUFA10? | The drugs that target NDUFA10 are Metformin and Metformin Hydrochloride. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%NDUFA10 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (ENSG00000165264), NDUFA4 (... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.135 | Q4 | What drugs target the gene CA3? | The drugs that target CA3 are Ethoxzolamide and Sulthiame. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%CA3 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_6095', 'drugName': 'Sulthiame', 'newLinkedTargets_string': 'CA2 (ENSG00000104267), CA7 (ENSG00000168748), CA1 (ENSG00000133742), CA3 (ENSG00000164879), CA6 (ENSG00000131686), CA12 (ENSG00000074410), CA14 (ENSG00000118298), CA9 (ENSG00000107159), CA4 (ENSG00000167434), CA13 (ENSG00000185015... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.1133 | Q4 | What drugs target the gene PRKAG3? | There are no approved drugs targeting PRKAG3, but the drug Acadesine, which potentially targets this gene, is currently undergoing clinical trials. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%PRKAG3 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_5888', 'drugName': 'Acadesine', 'newLinkedTargets_string': 'PRKAA2 (ENSG00000162409), PRKAB2 (ENSG00000131791), PRKAG1 (ENSG00000181929), PRKAG2 (ENSG00000106617), PRKAB1 (ENSG00000111725), PRKAA1 (ENSG00000132356), PRKAG3 (ENSG00000115592)', 'drugIsApproved': False, 'maxClinicalTrialPhase... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.828 | Q4 | What drugs target the gene LPAR1? | There are no approved drugs targeting LPAR1, but the drug Bms-986020, which potentially targets this gene, is currently undergoing clinical trials. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%LPAR1 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_1832', 'drugName': 'Bms-986020', 'newLinkedTargets_string': 'LPAR1 (ENSG00000198121)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}] | general | Select, Similarity Search, Order By | Genetic Target |
Q4.410 | Q4 | What drugs target the gene EPHA3? | The drug that targets EPHA3 is Vandetanib. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%EPHA3 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_1935', 'drugName': 'Vandetanib', 'newLinkedTargets_string': 'TEK (ENSG00000120156), ERBB2 (ENSG00000141736), EGFR (ENSG00000146648), ERBB4 (ENSG00000178568), ERBB3 (ENSG00000065361), EPHA2 (ENSG00000142627), EPHB2 (ENSG00000133216), EPHA5 (ENSG00000145242), EPHA4 (ENSG00000116106), EPHA8 (... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.370 | Q4 | What drugs target the gene DPEP1? | The drugs that target DPEP1 are Cilastatin Sodium and Cilastatin. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%DPEP1 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_1365', 'drugName': 'Cilastatin', 'newLinkedTargets_string': 'DPEP1 (ENSG00000015413)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_185', 'drugName': 'Cilastatin Sodium', 'newLinkedTargets_string': 'DPEP1 (ENSG00000015413)', 'drugIsApproved': True, 'max... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.510 | Q4 | What drugs target the gene GAS6? | There are no approved drugs targeting GAS6, but the drug Batiraxcept, which potentially targets this gene, is currently undergoing clinical trials. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%GAS6 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_5288', 'drugName': 'Batiraxcept', 'newLinkedTargets_string': 'GAS6 (ENSG00000183087)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}] | general | Select, Similarity Search, Order By | Genetic Target |
Q4.1211 | Q4 | What drugs target the gene RARA? | The drugs that target RARA are Etretinate, Alitretinoin, Adapalene, Isotretinoin, Acitretin, Tazarotene, and Tretinoin. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%RARA %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_343', 'drugName': 'Etretinate', 'newLinkedTargets_string': 'RXRB (ENSG00000204231), RARG (ENSG00000172819), RXRG (ENSG00000143171), RARB (ENSG00000077092), RARA (ENSG00000131759), RXRA (ENSG00000186350)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_508... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.507 | Q4 | What drugs target the gene GABRP? | The drugs that target GABRP are Meprobamate, Acamprosate Calcium, Enflurane, Methohexital, Metharbital, Butabarbital, Flurazepam Hydrochloride, Pentobarbital Sodium, Acamprosate, Primidone, Temazepam, Flunitrazepam, Ganaxolone, Diazepam, Methyprylon, Thiopental, Clonazepam, Topiramate, Remimazolam Besylate, Brexanolone... | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%GABRP %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_1494', 'drugName': 'Thiopental', 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089), GABRA3 (ENSG00000011677), GABRP (ENSG00000094755... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.1365 | Q4 | What drugs target the gene SLC22A12? | The drugs that target SLC22A12 are Sulfinpyrazone, Lesinurad, and Benzbromarone. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%SLC22A12 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_1001', 'drugName': 'Lesinurad', 'newLinkedTargets_string': 'SLC22A12 (ENSG00000197891)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3284', 'drugName': 'Benzbromarone', 'newLinkedTargets_string': 'SLC22A12 (ENSG00000197891)', 'drugIsApproved': True, 'm... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.349 | Q4 | What drugs target the gene CYP3A43? | The drugs that target CYP3A43 are Ritonavir and Cobicistat. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%CYP3A43 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_2751', 'drugName': 'Ritonavir', 'newLinkedTargets_string': 'CYP3A4 (ENSG00000160868), CYP3A5 (ENSG00000106258), CYP3A43 (ENSG00000021461), CYP3A7 (ENSG00000160870)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2752', 'drugName': 'Ritonavir', 'newLinked... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.388 | Q4 | What drugs target the gene EDNRB? | The drugs that target EDNRB are Bosentan, Sitaxentan, Ambrisentan, Macitentan, and Sitaxentan Sodium. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%EDNRB %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_1670', 'drugName': 'Sitaxentan', 'newLinkedTargets_string': 'EDNRB (ENSG00000136160), EDNRA (ENSG00000151617)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3910', 'drugName': 'Ambrisentan', 'newLinkedTargets_string': 'EDNRB (ENSG00000136160), EDNRA (EN... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.1 | Q4 | What drugs target the gene A2M? | The drugs that target A2M are Technetium Tc 99M Succimer and Technetium Succimer. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%A2M %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_2885', 'drugName': 'Technetium Tc 99M Succimer', 'newLinkedTargets_string': 'A2M (ENSG00000175899)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4248', 'drugName': 'Technetium Succimer', 'newLinkedTargets_string': 'A2M (ENSG00000175899)', 'drugIsApprov... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.362 | Q4 | What drugs target the gene DIO1? | The drug that targets DIO1 is Propylthiouracil. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%DIO1 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_394', 'drugName': 'Propylthiouracil', 'newLinkedTargets_string': 'TPO (ENSG00000115705), DIO1 (ENSG00000211452)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_395', 'drugName': 'Propylthiouracil', 'newLinkedTargets_string': 'TPO (ENSG00000115705), DIO1 ... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.899 | Q4 | What drugs target the gene MMP7? | The drugs that target MMP7 are Doxycycline Anhydrous, Doxycycline Hyclate, Doxycycline, and Doxycycline Calcium. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%MMP7 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_285', 'drugName': 'Doxycycline Anhydrous', 'newLinkedTargets_string': 'MMP13 (ENSG00000137745), MMP8 (ENSG00000118113), MMP7 (ENSG00000137673), MMP1 (ENSG00000196611)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3046', 'drugName': 'Doxycycline', 'newL... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.833 | Q4 | What drugs target the gene LTB4R? | There are no FDA approved drugs targeting the gene LTB4R. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Cp-195543, Amelubant, Nomacopan, and Etalocib. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%LTB4R %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_1191', 'drugName': 'Nomacopan', 'newLinkedTargets_string': 'LTB4R2 (ENSG00000213906), LTB4R (ENSG00000213903), C5 (ENSG00000106804)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_1192', 'drugName': 'Nomacopan', 'newLinkedTargets_string': 'LTB4R2 (ENSG0... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.1451 | Q4 | What drugs target the gene TNFRSF8? | The drug that targets TNFRSF8 is Brentuximab Vedotin. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%TNFRSF8 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_1085', 'drugName': 'Brentuximab Vedotin', 'newLinkedTargets_string': 'TNFRSF8 (ENSG00000120949), TUBB4B (ENSG00000188229), TUBB1 (ENSG00000101162), TUBA3C (ENSG00000198033), TUBA4A (ENSG00000127824), TUBB3 (ENSG00000258947), TUBA1A (ENSG00000167552), TUBB4A (ENSG00000104833), TUBB8 (ENSG00... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.477 | Q4 | What drugs target the gene FNTB? | The drug that targets FNTB is Lonafarnib. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%FNTB %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_5762', 'drugName': 'Lonafarnib', 'newLinkedTargets_string': 'FNTA (ENSG00000168522), FNTB (ENSG00000257365)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3546', 'drugName': 'Tipifarnib', 'newLinkedTargets_string': 'FNTA (ENSG00000168522), FNTB (ENSG000... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.1313 | Q4 | What drugs target the gene RRM1? | The drugs that target RRM1 are Gemcitabine Hydrochloride, Gemcitabine, Clofarabine, Fludarabine Phosphate, Gallium Nitrate, and Hydroxyurea. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%RRM1 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_4', 'drugName': 'Gemcitabine Hydrochloride', 'newLinkedTargets_string': 'POLA1 (ENSG00000101868), POLD4 (ENSG00000175482), POLD3 (ENSG00000077514), POLD1 (ENSG00000062822), POLD2 (ENSG00000106628), POLE (ENSG00000177084), POLA2 (ENSG00000014138), PRIM1 (ENSG00000198056), PRIM2 (ENSG0000014... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.58 | Q4 | What drugs target the gene ALOX5? | The drugs that target ALOX5 are Zileuton, Balsalazide, Balsalazide Disodium, Sulfasalazine, Meclofenamate Sodium, Olsalazine Sodium, Olsalazine, Meclofenamic Acid, and Mesalamine. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%ALOX5 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_3724', 'drugName': 'Meclofenamate Sodium', 'newLinkedTargets_string': 'ALOX5 (ENSG00000012779), PTGS2 (ENSG00000073756), PTGS1 (ENSG00000095303)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3016', 'drugName': 'Sulfasalazine', 'newLinkedTargets_string'... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.641 | Q4 | What drugs target the gene IFNA10? | There are no FDA approved drugs targeting the gene IFNA10. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Rontalizumab and Sifalimumab. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%IFNA10 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_5087', 'drugName': 'Sifalimumab', 'newLinkedTargets_string': 'IFNA6 (ENSG00000120235), IFNA8 (ENSG00000120242), IFNA5 (ENSG00000147873), IFNA10 (ENSG00000186803), IFNA2 (ENSG00000188379), IFNA1 (ENSG00000197919), IFNA13 (ENSG00000233816), IFNA7 (ENSG00000214042), IFNA21 (ENSG00000137080), ... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.1339 | Q4 | What drugs target the gene SCN9A? | The drugs that target SCN9A are Propoxycaine, Orphenadrine, Indecainide, Quinidine Polygalacturonate, Fosphenytoin Sodium, Prilocaine Hydrochloride, Zonisamide, Mexiletine, Hexylcaine Hydrochloride, Fosphenytoin, Phenazopyridine Hydrochloride, Primidone, Phenytoin Sodium, Propafenone, Topiramate, Chloroprocaine, Etidoc... | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%SCN9A %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_2948', 'drugName': 'Proparacaine Hydrochloride', 'newLinkedTargets_string': 'SCN1A (ENSG00000144285), SCN5A (ENSG00000183873), SCN4A (ENSG00000007314), SCN7A (ENSG00000136546), SCN2A (ENSG00000136531), SCN9A (ENSG00000169432), SCN3A (ENSG00000153253), SCN11A (ENSG00000168356), SCN8A (ENSG0... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.1073 | Q4 | What drugs target the gene PGF? | The drug that targets PGF is Aflibercept. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%PGF %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_998', 'drugName': 'Aflibercept', 'newLinkedTargets_string': 'VEGFA (ENSG00000112715), PGF (ENSG00000119630)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_997', 'drugName': 'Aflibercept', 'newLinkedTargets_string': 'VEGFA (ENSG00000112715), PGF (ENSG000... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.1529 | Q4 | What drugs target the gene VKORC1? | The drugs that target VKORC1 are Warfarin Sodium, Phenprocoumon, Dicumarol, Acenocoumarol, Warfarin, Phenindione, and Warfarin Potassium. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%VKORC1 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_5347', 'drugName': 'Warfarin Potassium', 'newLinkedTargets_string': 'VKORC1 (ENSG00000167397)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1631', 'drugName': 'Dicumarol', 'newLinkedTargets_string': 'VKORC1 (ENSG00000167397)', 'drugIsApproved': True, '... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.174 | Q4 | What drugs target the gene CASP10? | There are no approved drugs targeting CASP10, but the drug Emricasan, which potentially targets this gene, is currently undergoing clinical trials. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%CASP10 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_45', 'drugName': 'Emricasan', 'newLinkedTargets_string': 'CASP4 (ENSG00000196954), CASP9 (ENSG00000132906), CASP3 (ENSG00000164305), CASP5 (ENSG00000137757), CASP6 (ENSG00000138794), CASP7 (ENSG00000165806), CASP8 (ENSG00000064012), CASP1 (ENSG00000137752), CASP2 (ENSG00000106144), CASP10 ... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.452 | Q4 | What drugs target the gene FCGR2B? | There are no approved drugs targeting FCGR2B, but the drug Obexelimab, which potentially targets this gene, is currently undergoing clinical trials. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%FCGR2B %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_2610', 'drugName': 'Obexelimab', 'newLinkedTargets_string': 'CD19 (ENSG00000177455), FCGR2B (ENSG00000072694)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_2611', 'drugName': 'Obexelimab', 'newLinkedTargets_string': 'CD19 (ENSG00000177455), FCGR2B (EN... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.127 | Q4 | What drugs target the gene C3? | The drug that targets C3 is Pegcetacoplan. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%C3 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_5818', 'drugName': 'Ocriplasmin', 'newLinkedTargets_string': 'FN1 (ENSG00000115414), COL1A2 (ENSG00000164692), COL1A1 (ENSG00000108821), COL2A1 (ENSG00000139219), COL3A1 (ENSG00000168542), COL4A1 (ENSG00000187498), COL5A1 (ENSG00000130635), COL6A1 (ENSG00000142156), COL11A1 (ENSG0000006071... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.1010 | Q4 | What drugs target the gene NRAS? | There are no approved drugs targeting NRAS, but the drug Salirasib, which potentially targets this gene, is currently undergoing clinical trials. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%NRAS %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_3775', 'drugName': 'Salirasib', 'newLinkedTargets_string': 'HRAS (ENSG00000174775), NRAS (ENSG00000213281), KRAS (ENSG00000133703)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}] | general | Select, Similarity Search, Order By | Genetic Target |
Q4.533 | Q4 | What drugs target the gene GPD2? | The drugs that target GPD2 are Metformin and Metformin Hydrochloride. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%GPD2 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_1886', 'drugName': 'Metformin', 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (ENSG00000165264), NDUFA4 (ENSG0000018904... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.862 | Q4 | What drugs target the gene MAPK8? | There are no FDA approved drugs targeting the gene MAPK8. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Tanzisertib, Cc-401, and Bentamapimod. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%MAPK8 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_2634', 'drugName': 'Cc-401', 'newLinkedTargets_string': 'MAPK9 (ENSG00000050748), MAPK8 (ENSG00000107643), MAPK10 (ENSG00000109339)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_2632', 'drugName': 'Cc-401', 'newLinkedTargets_string': 'MAPK9 (ENSG00000... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.718 | Q4 | What drugs target the gene ITGA5? | There are no FDA approved drugs targeting the gene ITGA5. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Atn-161, Volociximab, and Pf-04605412. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%ITGA5 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_1021', 'drugName': 'Volociximab', 'newLinkedTargets_string': 'ITGB1 (ENSG00000150093), ITGA5 (ENSG00000161638)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_174', 'drugName': 'Atn-161', 'newLinkedTargets_string': 'ITGB1 (ENSG00000150093), ITGA5 (ENSG0... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.92 | Q4 | What drugs target the gene ATR? | There are no FDA approved drugs targeting the gene ATR. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: M4344, Berzosertib, Ceralasertib, and Elimusertib. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%ATR %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_4153', 'drugName': 'Ceralasertib', 'newLinkedTargets_string': 'ATR (ENSG00000175054)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_3704', 'drugName': 'Berzosertib', 'newLinkedTargets_string': 'ATR (ENSG00000175054)', 'drugIsApproved': False, 'maxClini... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.1487 | Q4 | What drugs target the gene TRPV4? | The drugs that target TRPV4 are Butamben Picrate and Butamben. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%TRPV4 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_5053', 'drugName': 'Butamben', 'newLinkedTargets_string': 'TRPA1 (ENSG00000104321), TRPV4 (ENSG00000111199)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5054', 'drugName': 'Butamben', 'newLinkedTargets_string': 'TRPA1 (ENSG00000104321), TRPV4 (ENSG000... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.183 | Q4 | What drugs target the gene CASP8? | There are no FDA approved drugs targeting the gene CASP8. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Emricasan and Nivocasan. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%CASP8 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_1848', 'drugName': 'Nivocasan', 'newLinkedTargets_string': 'CASP8 (ENSG00000064012), CASP1 (ENSG00000137752), CASP9 (ENSG00000132906)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_1847', 'drugName': 'Nivocasan', 'newLinkedTargets_string': 'CASP8 (ENSG... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.880 | Q4 | What drugs target the gene METAP1? | There are no approved drugs targeting METAP1, but the drug Tosedostat, which potentially targets this gene, is currently undergoing clinical trials. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%METAP1 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_582', 'drugName': 'Tosedostat', 'newLinkedTargets_string': 'ANPEP (ENSG00000166825), NPEPPS (ENSG00000141279), RNPEP (ENSG00000176393), METAP1 (ENSG00000164024), LNPEP (ENSG00000113441), DNPEP (ENSG00000123992), ENPEP (ENSG00000138792), XPNPEP1 (ENSG00000108039), LAP3 (ENSG00000002549), ME... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.1035 | Q4 | What drugs target the gene PARP1? | The drugs that target PARP1 are Talazoparib, Olaparib, Talazoparib Tosylate, Rucaparib, Niraparib, Niraparib Tosylate, and Rucaparib Camsylate. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%PARP1 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_4882', 'drugName': 'Niraparib Tosylate', 'newLinkedTargets_string': 'PARP2 (ENSG00000129484), PARP1 (ENSG00000143799)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3166', 'drugName': 'Rucaparib', 'newLinkedTargets_string': 'PARP1 (ENSG00000143799), PAR... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.791 | Q4 | What drugs target the gene KIR2DL2? | There are no FDA approved drugs targeting the gene KIR2DL2. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Iph-2101 and Lirilumab. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%KIR2DL2 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_4725', 'drugName': 'Iph-2101', 'newLinkedTargets_string': 'KIR2DL2 (ENSG00000275546), KIR2DL1 (ENSG00000125498), KIR2DL3 (ENSG00000243772)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_5180', 'drugName': 'Lirilumab', 'newLinkedTargets_string': 'KIR2DL... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.416 | Q4 | What drugs target the gene EPHB1? | The drug that targets EPHB1 is Vandetanib. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%EPHB1 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_1936', 'drugName': 'Vandetanib', 'newLinkedTargets_string': 'TEK (ENSG00000120156), ERBB2 (ENSG00000141736), EGFR (ENSG00000146648), ERBB4 (ENSG00000178568), ERBB3 (ENSG00000065361), EPHA2 (ENSG00000142627), EPHB2 (ENSG00000133216), EPHA5 (ENSG00000145242), EPHA4 (ENSG00000116106), EPHA8 (... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.253 | Q4 | What drugs target the gene CFB? | There are no approved drugs targeting CFB, but the drug Iptacopan, which potentially targets this gene, is currently undergoing clinical trials. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%CFB %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_3164', 'drugName': 'Iptacopan', 'newLinkedTargets_string': 'CFB (ENSG00000243649)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}] | general | Select, Similarity Search, Order By | Genetic Target |
Q4.70 | Q4 | What drugs target the gene APEX1? | There are no approved drugs targeting APEX1, but the drug Apx-3330, which potentially targets this gene, is currently undergoing clinical trials. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%APEX1 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_3210', 'drugName': 'Apx-3330', 'newLinkedTargets_string': 'APEX1 (ENSG00000100823)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}] | general | Select, Similarity Search, Order By | Genetic Target |
Q4.808 | Q4 | What drugs target the gene LAMB2? | The drug that targets LAMB2 is Ocriplasmin. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%LAMB2 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_5818', 'drugName': 'Ocriplasmin', 'newLinkedTargets_string': 'FN1 (ENSG00000115414), COL1A2 (ENSG00000164692), COL1A1 (ENSG00000108821), COL2A1 (ENSG00000139219), COL3A1 (ENSG00000168542), COL4A1 (ENSG00000187498), COL5A1 (ENSG00000130635), COL6A1 (ENSG00000142156), COL11A1 (ENSG0000006071... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.133 | Q4 | What drugs target the gene CA14? | The drugs that target CA14 are Ethoxzolamide and Sulthiame. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%CA14 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_6095', 'drugName': 'Sulthiame', 'newLinkedTargets_string': 'CA2 (ENSG00000104267), CA7 (ENSG00000168748), CA1 (ENSG00000133742), CA3 (ENSG00000164879), CA6 (ENSG00000131686), CA12 (ENSG00000074410), CA14 (ENSG00000118298), CA9 (ENSG00000107159), CA4 (ENSG00000167434), CA13 (ENSG00000185015... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.302 | Q4 | What drugs target the gene COL5A1? | The drugs that target COL5A1 are Collagenase Clostridium Histolyticum and Ocriplasmin. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%COL5A1 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_5818', 'drugName': 'Ocriplasmin', 'newLinkedTargets_string': 'FN1 (ENSG00000115414), COL1A2 (ENSG00000164692), COL1A1 (ENSG00000108821), COL2A1 (ENSG00000139219), COL3A1 (ENSG00000168542), COL4A1 (ENSG00000187498), COL5A1 (ENSG00000130635), COL6A1 (ENSG00000142156), COL11A1 (ENSG0000006071... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.1092 | Q4 | What drugs target the gene PLA2G7? | There are no FDA approved drugs targeting the gene PLA2G7. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Rilapladib and Darapladib. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%PLA2G7 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_5024', 'drugName': 'Darapladib', 'newLinkedTargets_string': 'PLA2G7 (ENSG00000146070)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_3181', 'drugName': 'Rilapladib', 'newLinkedTargets_string': 'PLA2G7 (ENSG00000146070)', 'drugIsApproved': False, 'maxCl... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.328 | Q4 | What drugs target the gene CTAG1B? | There are no approved drugs targeting CTAG1B, but the drug Rasdegafusp Alfa, which potentially targets this gene, is currently undergoing clinical trials. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%CTAG1B %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_5339', 'drugName': 'Rasdegafusp Alfa', 'newLinkedTargets_string': 'LY75 (ENSG00000054219), CTAG1B (ENSG00000184033), CTAG1A (ENSG00000268651)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_5340', 'drugName': 'Rasdegafusp Alfa', 'newLinkedTargets_string... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.1501 | Q4 | What drugs target the gene TUBB1? | The drugs that target TUBB1 are Polatuzumab Vedotin, Cabazitaxel, Vinflunine, Brentuximab Vedotin, Docetaxel, Belantamab Mafodotin, Paclitaxel, Vinorelbine, Ixabepilone, Enfortumab Vedotin, Eribulin Mesylate, Vincristine Sulfate, Tisotumab Vedotin, Vinblastine, Colchicine, Vincristine, Eribulin, Trastuzumab Emtansine, ... | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%TUBB1 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_1084', 'drugName': 'Brentuximab Vedotin', 'newLinkedTargets_string': 'TNFRSF8 (ENSG00000120949), TUBB4B (ENSG00000188229), TUBB1 (ENSG00000101162), TUBA3C (ENSG00000198033), TUBA4A (ENSG00000127824), TUBB3 (ENSG00000258947), TUBA1A (ENSG00000167552), TUBB4A (ENSG00000104833), TUBB8 (ENSG00... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.1534 | Q4 | What drugs target the gene XPNPEP1? | There are no approved drugs targeting XPNPEP1, but the drug Tosedostat, which potentially targets this gene, is currently undergoing clinical trials. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%XPNPEP1 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_582', 'drugName': 'Tosedostat', 'newLinkedTargets_string': 'ANPEP (ENSG00000166825), NPEPPS (ENSG00000141279), RNPEP (ENSG00000176393), METAP1 (ENSG00000164024), LNPEP (ENSG00000113441), DNPEP (ENSG00000123992), ENPEP (ENSG00000138792), XPNPEP1 (ENSG00000108039), LAP3 (ENSG00000002549), ME... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.502 | Q4 | What drugs target the gene GABRD? | The drugs that target GABRD are Meprobamate, Acamprosate Calcium, Enflurane, Methohexital, Metharbital, Butabarbital, Flurazepam Hydrochloride, Pentobarbital Sodium, Acamprosate, Primidone, Temazepam, Flunitrazepam, Ganaxolone, Diazepam, Methyprylon, Thiopental, Clonazepam, Topiramate, Remimazolam Besylate, Brexanolone... | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%GABRD %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_1494', 'drugName': 'Thiopental', 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089), GABRA3 (ENSG00000011677), GABRP (ENSG00000094755... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.343 | Q4 | What drugs target the gene CYP11B1? | The drugs that target CYP11B1 are Levoketoconazole, Osilodrostat Phosphate, Osilodrostat, and Mitotane. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%CYP11B1 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_3930', 'drugName': 'Levoketoconazole', 'newLinkedTargets_string': 'CYP11B1 (ENSG00000160882), CYP11B2 (ENSG00000179142), CYP17A1 (ENSG00000148795), CYP11A1 (ENSG00000140459)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3932', 'drugName': 'Levoketocona... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.837 | Q4 | What drugs target the gene LY6E? | There are no approved drugs targeting LY6E, but the drug Rg-7841, which potentially targets this gene, is currently undergoing clinical trials. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%LY6E %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_831', 'drugName': 'Rg-7841', 'newLinkedTargets_string': 'LY6E (ENSG00000160932), TUBB4B (ENSG00000188229), TUBB1 (ENSG00000101162), TUBA3C (ENSG00000198033), TUBA4A (ENSG00000127824), TUBB3 (ENSG00000258947), TUBA1A (ENSG00000167552), TUBB4A (ENSG00000104833), TUBB8 (ENSG00000261456), TUBB... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.366 | Q4 | What drugs target the gene DMD? | The drugs that target DMD are Viltolarsen, Eteplirsen, Golodirsen, and Casimersen. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%DMD %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_3184', 'drugName': 'Eteplirsen', 'newLinkedTargets_string': 'DMD (ENSG00000198947)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2014', 'drugName': 'Viltolarsen', 'newLinkedTargets_string': 'DMD (ENSG00000198947)', 'drugIsApproved': True, 'maxClinicalT... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.498 | Q4 | What drugs target the gene GABRA6? | The drugs that target GABRA6 are Meprobamate, Acamprosate Calcium, Enflurane, Methohexital, Metharbital, Butabarbital, Flurazepam Hydrochloride, Pentobarbital Sodium, Acamprosate, Primidone, Temazepam, Flunitrazepam, Ganaxolone, Diazepam, Methyprylon, Thiopental, Clonazepam, Topiramate, Remimazolam Besylate, Brexanolon... | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%GABRA6 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_1108', 'drugName': 'Temazepam', 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089), GABRA3 (ENSG00000011677), GABRP (ENSG00000094755)... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.1430 | Q4 | What drugs target the gene THRB? | The drugs that target THRB are Liothyronine, Levothyroxine, Dextrothyroxine Sodium, Dextrothyroxine, Liothyronine Sodium, and Levothyroxine Sodium. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%THRB %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_4368', 'drugName': 'Dextrothyroxine Sodium', 'newLinkedTargets_string': 'THRA (ENSG00000126351), THRB (ENSG00000151090)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5964', 'drugName': 'Levothyroxine Sodium', 'newLinkedTargets_string': 'THRA (ENSG00000... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.340 | Q4 | What drugs target the gene CXCR2? | There are no FDA approved drugs targeting the gene CXCR2. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Ladarixin, Elubrixin, Navarixin, Reparixin, Sx-682, and Danirixin. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%CXCR2 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_2754', 'drugName': 'Reparixin', 'newLinkedTargets_string': 'CXCR1 (ENSG00000163464), CXCR2 (ENSG00000180871)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_400', 'drugName': 'Ladarixin', 'newLinkedTargets_string': 'CXCR2 (ENSG00000180871), CXCR1 (ENSG0... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.423 | Q4 | What drugs target the gene ERAP1? | There are no approved drugs targeting ERAP1, but the drug Tosedostat, which potentially targets this gene, is currently undergoing clinical trials. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%ERAP1 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_582', 'drugName': 'Tosedostat', 'newLinkedTargets_string': 'ANPEP (ENSG00000166825), NPEPPS (ENSG00000141279), RNPEP (ENSG00000176393), METAP1 (ENSG00000164024), LNPEP (ENSG00000113441), DNPEP (ENSG00000123992), ENPEP (ENSG00000138792), XPNPEP1 (ENSG00000108039), LAP3 (ENSG00000002549), ME... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.166 | Q4 | What drugs target the gene CACNG7? | The drugs that target CACNG7 are Gabapentin, Terodiline Hydrochloride, Phloroglucinol, Suloctidil, Pregabalin, Gabapentin Enacarbil, Bepridil Hydrochloride, Bepridil, and Terodiline. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%CACNG7 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_142', 'drugName': 'Gabapentin', 'newLinkedTargets_string': 'CACNA1H (ENSG00000196557), CACNA2D1 (ENSG00000153956), CACNA1C (ENSG00000151067), CACNA2D3 (ENSG00000157445), CACNA1S (ENSG00000081248), CACNA2D2 (ENSG00000007402), CACNA1D (ENSG00000157388), CACNA1A (ENSG00000141837), CACNA1B (EN... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.29 | Q4 | What drugs target the gene ADORA2A? | The drugs that target ADORA2A are Theophylline Sodium Glycinate, Adenosine, Theophylline Glycinate, Istradefylline, Regadenoson, Oxtriphylline, Pentoxifylline, Theophylline, Caffeine, Aminophylline, Caffeine, and Citrated. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%ADORA2A %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_5472', 'drugName': 'Aminophylline', 'newLinkedTargets_string': 'PDE4A (ENSG00000065989), PDE4D (ENSG00000113448), PDE4B (ENSG00000184588), PDE4C (ENSG00000105650), PDE3A (ENSG00000172572), PDE3B (ENSG00000152270), ADORA1 (ENSG00000163485), ADORA2B (ENSG00000170425), ADORA3 (ENSG00000282608... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.519 | Q4 | What drugs target the gene GHSR? | The drugs that target GHSR are Macimorelin Acetate and Macimorelin. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%GHSR %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_5129', 'drugName': 'Macimorelin', 'newLinkedTargets_string': 'GHSR (ENSG00000121853)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_942', 'drugName': 'Macimorelin Acetate', 'newLinkedTargets_string': 'GHSR (ENSG00000121853)', 'drugIsApproved': True, 'ma... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.195 | Q4 | What drugs target the gene CCR4? | The drug that targets CCR4 is Mogamulizumab. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%CCR4 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_879', 'drugName': 'Mogamulizumab', 'newLinkedTargets_string': 'CCR4 (ENSG00000183813)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}] | general | Select, Similarity Search, Order By | Genetic Target |
Q4.1116 | Q4 | What drugs target the gene PPAT? | The drugs that target PPAT are Azathioprine, Mercaptopurine, and Azathioprine Sodium. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%PPAT %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_5406', 'drugName': 'Mercaptopurine', 'newLinkedTargets_string': 'PPAT (ENSG00000128059)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2137', 'drugName': 'Mercaptopurine', 'newLinkedTargets_string': 'PPAT (ENSG00000128059)', 'drugIsApproved': True, 'max... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.1395 | Q4 | What drugs target the gene SRD5A3? | The drugs that target SRD5A3 are Dutasteride and Abiraterone. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%SRD5A3 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_6320', 'drugName': 'Abiraterone', 'newLinkedTargets_string': 'AR (ENSG00000169083), CYP17A1 (ENSG00000148795), SRD5A1 (ENSG00000145545), SRD5A2 (ENSG00000277893), SRD5A3 (ENSG00000128039)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_433', 'drugName': ... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.950 | Q4 | What drugs target the gene NDUFAF1? | The drugs that target NDUFAF1 are Metformin and Metformin Hydrochloride. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%NDUFAF1 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (ENSG00000165264), NDUFA4 (... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.1394 | Q4 | What drugs target the gene SRD5A2? | The drugs that target SRD5A2 are Dutasteride, Finasteride, and Abiraterone. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%SRD5A2 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_6321', 'drugName': 'Abiraterone', 'newLinkedTargets_string': 'AR (ENSG00000169083), CYP17A1 (ENSG00000148795), SRD5A1 (ENSG00000145545), SRD5A2 (ENSG00000277893), SRD5A3 (ENSG00000128039)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5461', 'drugName':... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.171 | Q4 | What drugs target the gene CALCRL? | The drugs that target CALCRL are Ubrogepant, Rimegepant, Atogepant, Rimegepant Sulfate, and Erenumab. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%CALCRL %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_3190', 'drugName': 'Rimegepant Sulfate', 'newLinkedTargets_string': 'CALCRL (ENSG00000064989)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5361', 'drugName': 'Erenumab', 'newLinkedTargets_string': 'CALCRL (ENSG00000064989)', 'drugIsApproved': True, 'm... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.169 | Q4 | What drugs target the gene CALCB? | The drugs that target CALCB are Galcanezumab, Eptinezumab, and Fremanezumab. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%CALCB %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_1901', 'drugName': 'Galcanezumab', 'newLinkedTargets_string': 'CALCA (ENSG00000110680), CALCB (ENSG00000175868)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5545', 'drugName': 'Fremanezumab', 'newLinkedTargets_string': 'CALCA (ENSG00000110680), CALCB ... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.656 | Q4 | What drugs target the gene IFNG? | The drug that targets IFNG is Emapalumab. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%IFNG %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_3856', 'drugName': 'Emapalumab', 'newLinkedTargets_string': 'IFNG (ENSG00000111537)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4201', 'drugName': 'Fontolizumab', 'newLinkedTargets_string': 'IFNG (ENSG00000111537)', 'drugIsApproved': False, 'maxClini... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.175 | Q4 | What drugs target the gene CASP12? | There are no approved drugs targeting CASP12, but the drug Emricasan, which potentially targets this gene, is currently undergoing clinical trials. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%CASP12 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_45', 'drugName': 'Emricasan', 'newLinkedTargets_string': 'CASP4 (ENSG00000196954), CASP9 (ENSG00000132906), CASP3 (ENSG00000164305), CASP5 (ENSG00000137757), CASP6 (ENSG00000138794), CASP7 (ENSG00000165806), CASP8 (ENSG00000064012), CASP1 (ENSG00000137752), CASP2 (ENSG00000106144), CASP10 ... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.521 | Q4 | What drugs target the gene GLA? | The drugs that target GLA are Migalastat Hydrochloride and Migalastat. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%GLA %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_3147', 'drugName': 'Migalastat', 'newLinkedTargets_string': 'GLA (ENSG00000102393)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_549', 'drugName': 'Migalastat Hydrochloride', 'newLinkedTargets_string': 'GLA (ENSG00000102393)', 'drugIsApproved': True, '... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.1244 | Q4 | What drugs target the gene RPL23A? | The drug that targets RPL23A is Ataluren. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%RPL23A %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG00000083845), RPS7 (ENSG... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.1210 | Q4 | What drugs target the gene RAMP3? | The drugs that target RAMP3 are Pramlintide and Pramlintide Acetate. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%RAMP3 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_359', 'drugName': 'Pramlintide', 'newLinkedTargets_string': 'CALCR (ENSG00000004948), RAMP1 (ENSG00000132329), RAMP2 (ENSG00000131477), RAMP3 (ENSG00000122679)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2395', 'drugName': 'Pramlintide Acetate', 'new... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.917 | Q4 | What drugs target the gene MTOR? | The drugs that target MTOR are Perhexiline and Perhexiline Maleate. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%MTOR %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_1725', 'drugName': 'Perhexiline Maleate', 'newLinkedTargets_string': 'MTOR (ENSG00000198793), CPT2 (ENSG00000157184), CPT1B (ENSG00000205560)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_919', 'drugName': 'Perhexiline', 'newLinkedTargets_string': 'MTO... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.494 | Q4 | What drugs target the gene GABRA2? | The drugs that target GABRA2 are Meprobamate, Acamprosate Calcium, Enflurane, Methohexital, Metharbital, Butabarbital, Flurazepam Hydrochloride, Pentobarbital Sodium, Acamprosate, Primidone, Temazepam, Flunitrazepam, Ganaxolone, Diazepam, Methyprylon, Thiopental, Clonazepam, Topiramate, Remimazolam Besylate, Brexanolon... | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%GABRA2 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_2854', 'drugName': 'Chlordiazepoxide Hydrochloride', 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089), GABRA3 (ENSG00000011677), GA... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.958 | Q4 | What drugs target the gene NDUFB3? | The drugs that target NDUFB3 are Metformin and Metformin Hydrochloride. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%NDUFB3 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (ENSG00000165264), NDUFA4 (... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.74 | Q4 | What drugs target the gene APOB? | The drugs that target APOB are Mipomersen Sodium and Mipomersen. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%APOB %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_3718', 'drugName': 'Mipomersen Sodium', 'newLinkedTargets_string': 'APOB (ENSG00000084674)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5688', 'drugName': 'Mipomersen', 'newLinkedTargets_string': 'APOB (ENSG00000084674)', 'drugIsApproved': True, 'maxC... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.1285 | Q4 | What drugs target the gene RPS2? | The drug that targets RPS2 is Ataluren. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%RPS2 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG00000083845), RPS7 (ENSG... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.591 | Q4 | What drugs target the gene HGF? | There are no FDA approved drugs targeting the gene HGF. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Rilotumumab and Ficlatuzumab. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%HGF %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_1237', 'drugName': 'Rilotumumab', 'newLinkedTargets_string': 'HGF (ENSG00000019991)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_5496', 'drugName': 'Ficlatuzumab', 'newLinkedTargets_string': 'HGF (ENSG00000019991)', 'drugIsApproved': False, 'maxClini... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.755 | Q4 | What drugs target the gene KCNH1? | The drugs that target KCNH1 are Dalfampridine, Guanidine, Amifampridine Phosphate, Guanidine Hydrochloride, and Amifampridine. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%KCNH1 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_5118', 'drugName': 'Guanidine Hydrochloride', 'newLinkedTargets_string': 'KCNQ1 (ENSG00000053918), KCND3 (ENSG00000171385), KCNH2 (ENSG00000055118), KCNA2 (ENSG00000177301), KCNA1 (ENSG00000111262), KCNQ2 (ENSG00000075043), KCNQ3 (ENSG00000184156), KCNA7 (ENSG00000104848), KCNQ5 (ENSG00000... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.661 | Q4 | What drugs target the gene IGF1R? | The drugs that target IGF1R are Mecasermin Rinfabate, Teprotumumab, and Mecasermin. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%IGF1R %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_672', 'drugName': 'Mecasermin Rinfabate', 'newLinkedTargets_string': 'IGF1R (ENSG00000140443)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1336', 'drugName': 'Teprotumumab', 'newLinkedTargets_string': 'IGF1R (ENSG00000140443)', 'drugIsApproved': True,... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.847 | Q4 | What drugs target the gene MAP2K1? | The drugs that target MAP2K1 are Trametinib Dimethyl Sulfoxide, Binimetinib, Selumetinib, Cobimetinib, Selumetinib Sulfate, Trametinib, and Cobimetinib Fumarate. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%MAP2K1 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_6005', 'drugName': 'Cobimetinib Fumarate', 'newLinkedTargets_string': 'MAP2K1 (ENSG00000169032), MAP2K2 (ENSG00000126934)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3657', 'drugName': 'Cobimetinib', 'newLinkedTargets_string': 'MAP2K1 (ENSG0000016903... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.236 | Q4 | What drugs target the gene CDK15? | There are no FDA approved drugs targeting the gene CDK15. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Roniciclib, Pha-793887, Azd-5438, and At-7519. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%CDK15 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_1429', 'drugName': 'Roniciclib', 'newLinkedTargets_string': 'CDK1 (ENSG00000170312), CDK4 (ENSG00000135446), CDK2 (ENSG00000123374), CDK5 (ENSG00000164885), CDK6 (ENSG00000105810), CDK7 (ENSG00000134058), CDK3 (ENSG00000250506), CDK16 (ENSG00000102225), CDK18 (ENSG00000117266), CDK8 (ENSG0... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.737 | Q4 | What drugs target the gene KCNA4? | The drugs that target KCNA4 are Dalfampridine, Guanidine, Amifampridine Phosphate, Guanidine Hydrochloride, and Amifampridine. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%KCNA4 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_5118', 'drugName': 'Guanidine Hydrochloride', 'newLinkedTargets_string': 'KCNQ1 (ENSG00000053918), KCND3 (ENSG00000171385), KCNH2 (ENSG00000055118), KCNA2 (ENSG00000177301), KCNA1 (ENSG00000111262), KCNQ2 (ENSG00000075043), KCNQ3 (ENSG00000184156), KCNA7 (ENSG00000104848), KCNQ5 (ENSG00000... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.216 | Q4 | What drugs target the gene CD40LG? | There are no FDA approved drugs targeting the gene CD40LG. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Ruplizumab, At-1501, Dazodalibep, Dapirolizumab Pegol, Ravagalimab, and Toralizumab. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%CD40LG %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_230', 'drugName': 'Ruplizumab', 'newLinkedTargets_string': 'CD40LG (ENSG00000102245)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_4952', 'drugName': 'Dapirolizumab Pegol', 'newLinkedTargets_string': 'CD40LG (ENSG00000102245)', 'drugIsApproved': False... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.164 | Q4 | What drugs target the gene CACNG5? | The drugs that target CACNG5 are Gabapentin, Terodiline Hydrochloride, Phloroglucinol, Suloctidil, Pregabalin, Gabapentin Enacarbil, Bepridil Hydrochloride, Bepridil, and Terodiline. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%CACNG5 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_142', 'drugName': 'Gabapentin', 'newLinkedTargets_string': 'CACNA1H (ENSG00000196557), CACNA2D1 (ENSG00000153956), CACNA1C (ENSG00000151067), CACNA2D3 (ENSG00000157445), CACNA1S (ENSG00000081248), CACNA2D2 (ENSG00000007402), CACNA1D (ENSG00000157388), CACNA1A (ENSG00000141837), CACNA1B (EN... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.134 | Q4 | What drugs target the gene CA2? | The drugs that target CA2 are Dichlorphenamide, Dorzolamide, Acetazolamide, Topiramate, Dorzolamide Hydrochloride, Ethoxzolamide, Brinzolamide, Methazolamide, Sulthiame, and Acetazolamide Sodium. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%CA2 %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_469', 'drugName': 'Acetazolamide', 'newLinkedTargets_string': 'CA12 (ENSG00000074410), CA2 (ENSG00000104267), CA4 (ENSG00000167434), CA1 (ENSG00000133742)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_468', 'drugName': 'Acetazolamide', 'newLinkedTarget... | general | Select, Similarity Search, Order By | Genetic Target |
Q4.1129 | Q4 | What drugs target the gene PRKACB? | There are no approved drugs targeting PRKACB, but the drug Gsk-690693, which potentially targets this gene, is currently undergoing clinical trials. | SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase
FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated`
WHERE newLinkedTargets_string LIKE '%PRKACB %'
ORDER BY maxClinicalTrialPhase DESC
LIMIT 100 | [{'UUID': 'DrugGeneTargets_v2_1835', 'drugName': 'Gsk-690693', 'newLinkedTargets_string': 'PRKACB (ENSG00000142875), PRKACA (ENSG00000072062), PRKACG (ENSG00000165059), AKT2 (ENSG00000105221), AKT3 (ENSG00000117020), AKT1 (ENSG00000142208), PRKD3 (ENSG00000115825), PRKCI (ENSG00000163558), PRKCA (ENSG00000154229), PRKC... | general | Select, Similarity Search, Order By | Genetic Target |
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