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Q4.224
Q4
What drugs target the gene CD79B?
The drug that targets CD79B is Polatuzumab Vedotin.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CD79B %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_560', 'drugName': 'Polatuzumab Vedotin', 'newLinkedTargets_string': 'CD79B (ENSG00000007312), TUBB4B (ENSG00000188229), TUBB1 (ENSG00000101162), TUBA3C (ENSG00000198033), TUBA4A (ENSG00000127824), TUBB3 (ENSG00000258947), TUBA1A (ENSG00000167552), TUBB4A (ENSG00000104833), TUBB8 (ENSG00000...
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Q4.1258
Q4
What drugs target the gene RPL36?
The drug that targets RPL36 is Ataluren.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RPL36 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG00000083845), RPS7 (ENSG...
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Q4.939
Q4
What drugs target the gene NDUFA13?
The drugs that target NDUFA13 are Metformin and Metformin Hydrochloride.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NDUFA13 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (ENSG00000165264), NDUFA4 (...
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Q4.187
Q4
What drugs target the gene CCKAR?
The drugs that target CCKAR are Sincalide, Ceruletide Diethylamine, Ceruletide, and Proglumide.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CCKAR %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5575', 'drugName': 'Proglumide', 'newLinkedTargets_string': 'CCKBR (ENSG00000110148), CCKAR (ENSG00000163394)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2693', 'drugName': 'Sincalide', 'newLinkedTargets_string': 'CCKAR (ENSG00000163394)', 'drugIsApp...
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Q4.42
Q4
What drugs target the gene AFP?
There are no approved drugs targeting AFP, but the drug Yttrium Y 90 Tacatuzumab Tetraxetan, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%AFP %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_262', 'drugName': 'Yttrium Y 90 Tacatuzumab Tetraxetan', 'newLinkedTargets_string': 'AFP (ENSG00000081051)', 'drugIsApproved': False, 'maxClinicalTrialPhase': -1}]
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Q4.697
Q4
What drugs target the gene IL33?
There are no FDA approved drugs targeting the gene IL33. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Torudokimab, Etokimab, and Itepekimab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%IL33 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2908', 'drugName': 'Itepekimab', 'newLinkedTargets_string': 'IL33 (ENSG00000137033)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_2323', 'drugName': 'Etokimab', 'newLinkedTargets_string': 'IL33 (ENSG00000137033)', 'drugIsApproved': False, 'maxClinical...
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Q4.110
Q4
What drugs target the gene BDKRB2?
The drugs that target BDKRB2 are Icatibant Acetate and Icatibant.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%BDKRB2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3024', 'drugName': 'Icatibant', 'newLinkedTargets_string': 'BDKRB2 (ENSG00000168398)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_226', 'drugName': 'Icatibant Acetate', 'newLinkedTargets_string': 'BDKRB2 (ENSG00000168398)', 'drugIsApproved': True, 'ma...
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Q4.39
Q4
What drugs target the gene ADRB2?
The drugs that target ADRB2 are Oxprenolol Hydrochloride, Nebivolol, Nadolol, Arformoterol Tartrate, Rimiterol, Reproterol, Timolol Maleate, Vilanterol Trifenatate, Dipivefrin, Epinephrine, Carvedilol Phosphate, Penbutolol Sulfate, Sotalol, Levalbuterol Hydrochloride, Isoproterenol Hydrochloride, Clenbuterol, Dobutamin...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ADRB2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3721', 'drugName': 'Levosalbutamol', 'newLinkedTargets_string': 'ADRB2 (ENSG00000169252)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1445', 'drugName': 'Terbutaline Sulfate', 'newLinkedTargets_string': 'ADRB2 (ENSG00000169252)', 'drugIsApproved': Tru...
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Q4.571
Q4
What drugs target the gene HBA1?
The drug that targets HBA1 is Voxelotor.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%HBA1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2318', 'drugName': 'Voxelotor', 'newLinkedTargets_string': 'HBA1 (ENSG00000206172), HBA2 (ENSG00000188536), HBB (ENSG00000244734)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5816', 'drugName': 'Efaproxiral', 'newLinkedTargets_string': 'HBA1 (ENSG0000...
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Q4.1024
Q4
What drugs target the gene P2RX3?
There are no FDA approved drugs targeting the gene P2RX3. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Camlipixant and Gefapixant.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%P2RX3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_913', 'drugName': 'Gefapixant', 'newLinkedTargets_string': 'P2RX3 (ENSG00000109991)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_601', 'drugName': 'Camlipixant', 'newLinkedTargets_string': 'P2RX3 (ENSG00000109991)', 'drugIsApproved': False, 'maxClini...
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Q4.1299
Q4
What drugs target the gene RPS4Y1?
The drug that targets RPS4Y1 is Ataluren.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RPS4Y1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG00000083845), RPS7 (ENSG...
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Q4.1478
Q4
What drugs target the gene TRAV29DV5?
There are no FDA approved drugs targeting the gene TRAV29DV5. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Medi-500, Tol-101, and Maslimomab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TRAV29DV5 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1483', 'drugName': 'Medi-500', 'newLinkedTargets_string': 'TRAV29DV5 (ENSG00000211810), TRAC (ENSG00000277734), TRBV7-9 (ENSG00000278030), TRGV3 (ENSG00000211699)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_5971', 'drugName': 'Tol-101', 'newLinkedTa...
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Q4.486
Q4
What drugs target the gene FZD2?
There are no approved drugs targeting FZD2, but the drug Vantictumab, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%FZD2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5828', 'drugName': 'Vantictumab', 'newLinkedTargets_string': 'FZD2 (ENSG00000180340), FZD7 (ENSG00000155760), FZD1 (ENSG00000157240), FZD5 (ENSG00000163251), FZD8 (ENSG00000177283)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 1}, {'UUID': 'DrugGeneTargets_v2_5825', 'drugName': 'Vant...
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Q4.470
Q4
What drugs target the gene FKBP1A?
The drugs that target FKBP1A are Tacrolimus, Everolimus, Sirolimus, Pimecrolimus, and Temsirolimus.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%FKBP1A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5128', 'drugName': 'Tacrolimus', 'newLinkedTargets_string': 'FKBP1A (ENSG00000088832)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1925', 'drugName': 'Everolimus', 'newLinkedTargets_string': 'FKBP1A (ENSG00000088832)', 'drugIsApproved': True, 'maxClin...
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Q4.895
Q4
What drugs target the gene MMP13?
The drugs that target MMP13 are Doxycycline Anhydrous, Doxycycline Hyclate, Doxycycline, and Doxycycline Calcium.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%MMP13 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_289', 'drugName': 'Doxycycline Anhydrous', 'newLinkedTargets_string': 'MMP13 (ENSG00000137745), MMP8 (ENSG00000118113), MMP7 (ENSG00000137673), MMP1 (ENSG00000196611)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_287', 'drugName': 'Doxycycline Anhydrou...
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Q4.952
Q4
What drugs target the gene NDUFAF3?
The drugs that target NDUFAF3 are Metformin and Metformin Hydrochloride.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NDUFAF3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (ENSG00000165264), NDUFA4 (...
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Q4.25
Q4
What drugs target the gene ADH6?
The drug that targets ADH6 is Nitrefazole.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ADH6 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6344', 'drugName': 'Nitrefazole', 'newLinkedTargets_string': 'ADH1A (ENSG00000187758), ADH4 (ENSG00000198099), ADH1B (ENSG00000196616), ADH1C (ENSG00000248144), ADH7 (ENSG00000196344), ADH5 (ENSG00000197894), ADH6 (ENSG00000172955)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}]
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Q4.1036
Q4
What drugs target the gene PARP2?
The drugs that target PARP2 are Talazoparib, Olaparib, Talazoparib Tosylate, Rucaparib, Niraparib, Niraparib Tosylate, and Rucaparib Camsylate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PARP2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_100', 'drugName': 'Talazoparib', 'newLinkedTargets_string': 'PARP2 (ENSG00000129484), PARP1 (ENSG00000143799)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2224', 'drugName': 'Talazoparib Tosylate', 'newLinkedTargets_string': 'PARP2 (ENSG00000129484), ...
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Q4.1222
Q4
What drugs target the gene RNPEPL1?
There are no approved drugs targeting RNPEPL1, but the drug Tosedostat, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RNPEPL1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_582', 'drugName': 'Tosedostat', 'newLinkedTargets_string': 'ANPEP (ENSG00000166825), NPEPPS (ENSG00000141279), RNPEP (ENSG00000176393), METAP1 (ENSG00000164024), LNPEP (ENSG00000113441), DNPEP (ENSG00000123992), ENPEP (ENSG00000138792), XPNPEP1 (ENSG00000108039), LAP3 (ENSG00000002549), ME...
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Q4.69
Q4
What drugs target the gene APCS?
There are no FDA approved drugs targeting the gene APCS. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Miridesap and Dezamizumab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%APCS %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5164', 'drugName': 'Dezamizumab', 'newLinkedTargets_string': 'APCS (ENSG00000132703)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_1308', 'drugName': 'Miridesap', 'newLinkedTargets_string': 'APCS (ENSG00000132703)', 'drugIsApproved': False, 'maxClinic...
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Q4.889
Q4
What drugs target the gene MKNK2?
There are no approved drugs targeting MKNK2, but the drug Tomivosertib, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%MKNK2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1066', 'drugName': 'Tomivosertib', 'newLinkedTargets_string': 'MKNK2 (ENSG00000099875), MKNK1 (ENSG00000079277)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
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Q4.1297
Q4
What drugs target the gene RPS3A?
The drug that targets RPS3A is Ataluren.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RPS3A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG00000083845), RPS7 (ENSG...
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Q4.368
Q4
What drugs target the gene DNMT3A?
The drugs that target DNMT3A are Decitabine and Azacitidine.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%DNMT3A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4132', 'drugName': 'Azacitidine', 'newLinkedTargets_string': 'DNMT1 (ENSG00000130816), DNMT3A (ENSG00000119772)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4131', 'drugName': 'Azacitidine', 'newLinkedTargets_string': 'DNMT1 (ENSG00000130816), DNMT3A ...
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Q4.508
Q4
What drugs target the gene GABRQ?
The drugs that target GABRQ are Meprobamate, Acamprosate Calcium, Enflurane, Methohexital, Metharbital, Butabarbital, Flurazepam Hydrochloride, Pentobarbital Sodium, Acamprosate, Primidone, Temazepam, Flunitrazepam, Ganaxolone, Diazepam, Methyprylon, Thiopental, Clonazepam, Topiramate, Remimazolam Besylate, Brexanolone...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%GABRQ %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1494', 'drugName': 'Thiopental', 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089), GABRA3 (ENSG00000011677), GABRP (ENSG00000094755...
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Q4.855
Q4
What drugs target the gene MAP3K8?
There are no approved drugs targeting MAP3K8, but the drug Tilpisertib, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%MAP3K8 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6134', 'drugName': 'Tilpisertib', 'newLinkedTargets_string': 'MAP3K8 (ENSG00000107968)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
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Q4.1348
Q4
What drugs target the gene SELPLG?
There are no approved drugs targeting SELPLG, but the drug Neihulizumab, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%SELPLG %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3018', 'drugName': 'Neihulizumab', 'newLinkedTargets_string': 'SELPLG (ENSG00000110876)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
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Q4.385
Q4
What drugs target the gene E2F8?
There are no FDA approved drugs targeting the gene E2F8. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Edifoligide and Edifoligide Sodium.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%E2F8 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4614', 'drugName': 'Edifoligide Sodium', 'newLinkedTargets_string': 'E2F1 (ENSG00000101412), E2F2 (ENSG00000007968), E2F3 (ENSG00000112242), E2F4 (ENSG00000205250), E2F5 (ENSG00000133740), E2F6 (ENSG00000169016), E2F7 (ENSG00000165891), E2F8 (ENSG00000129173)', 'drugIsApproved': False, 'ma...
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Q4.739
Q4
What drugs target the gene KCNA6?
The drugs that target KCNA6 are Dalfampridine, Guanidine, Amifampridine Phosphate, Guanidine Hydrochloride, and Amifampridine.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%KCNA6 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5118', 'drugName': 'Guanidine Hydrochloride', 'newLinkedTargets_string': 'KCNQ1 (ENSG00000053918), KCND3 (ENSG00000171385), KCNH2 (ENSG00000055118), KCNA2 (ENSG00000177301), KCNA1 (ENSG00000111262), KCNQ2 (ENSG00000075043), KCNQ3 (ENSG00000184156), KCNA7 (ENSG00000104848), KCNQ5 (ENSG00000...
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Q4.722
Q4
What drugs target the gene ITGB1?
The drug that targets ITGB1 is Natalizumab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ITGB1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5016', 'drugName': 'Natalizumab', 'newLinkedTargets_string': 'ITGA4 (ENSG00000115232), ITGB7 (ENSG00000139626), ITGB1 (ENSG00000150093)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5015', 'drugName': 'Natalizumab', 'newLinkedTargets_string': 'ITGA4 (E...
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Genetic Target
Q4.456
Q4
What drugs target the gene FDPS?
The drugs that target FDPS are Risedronic Acid, Ibandronic Acid, Ibandronate Sodium, Pamidronate Disodium, Pamidronic Acid, Zoledronic Acid, Risedronate Sodium, Alendronate Sodium, and Alendronic Acid.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%FDPS %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4717', 'drugName': 'Risedronate Sodium', 'newLinkedTargets_string': 'FDPS (ENSG00000160752)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5882', 'drugName': 'Alendronic Acid', 'newLinkedTargets_string': 'FDPS (ENSG00000160752)', 'drugIsApproved': True,...
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Genetic Target
Q4.266
Q4
What drugs target the gene CHRNA3?
The drugs that target CHRNA3 are Mecamylamine, Mecamylamine Hydrochloride, Trimethaphan, Pentolinium Tartrate, Pentolinium, and Trimethaphan Camsylate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CHRNA3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5467', 'drugName': 'Trimethaphan Camsylate', 'newLinkedTargets_string': 'CHRNB4 (ENSG00000117971), CHRNA3 (ENSG00000080644)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4467', 'drugName': 'Trimethaphan', 'newLinkedTargets_string': 'CHRNB4 (ENSG0000011...
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Genetic Target
Q4.76
Q4
What drugs target the gene APP?
The drug that targets APP is Aducanumab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%APP %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4177', 'drugName': 'Aducanumab', 'newLinkedTargets_string': 'APP (ENSG00000142192)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3123', 'drugName': 'Tramiprosate', 'newLinkedTargets_string': 'APP (ENSG00000142192)', 'drugIsApproved': False, 'maxClinica...
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Genetic Target
Q4.446
Q4
What drugs target the gene FAAH?
The drug that targets FAAH is Acetaminophen.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%FAAH %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_147', 'drugName': 'Acetaminophen', 'newLinkedTargets_string': 'PTGS2 (ENSG00000073756), PTGS1 (ENSG00000095303), TRPV1 (ENSG00000196689), FAAH (ENSG00000117480)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_146', 'drugName': 'Acetaminophen', 'newLinked...
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Genetic Target
Q4.397
Q4
What drugs target the gene EGR1?
There are no approved drugs targeting EGR1, but the drug Brivoligide, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%EGR1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_862', 'drugName': 'Brivoligide', 'newLinkedTargets_string': 'EGR1 (ENSG00000120738)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
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Genetic Target
Q4.178
Q4
What drugs target the gene CASP3?
There are no approved drugs targeting CASP3, but the drug Emricasan, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CASP3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_45', 'drugName': 'Emricasan', 'newLinkedTargets_string': 'CASP4 (ENSG00000196954), CASP9 (ENSG00000132906), CASP3 (ENSG00000164305), CASP5 (ENSG00000137757), CASP6 (ENSG00000138794), CASP7 (ENSG00000165806), CASP8 (ENSG00000064012), CASP1 (ENSG00000137752), CASP2 (ENSG00000106144), CASP10 ...
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Genetic Target
Q4.1343
Q4
What drugs target the gene SCTR?
The drugs that target SCTR are Secretin Synthetic Porcine, Secretin, and Secretin Synthetic Human.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%SCTR %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4400', 'drugName': 'Secretin', 'newLinkedTargets_string': 'SCTR (ENSG00000080293)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4712', 'drugName': 'Secretin Synthetic Human', 'newLinkedTargets_string': 'SCTR (ENSG00000080293)', 'drugIsApproved': True, ...
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Genetic Target
Q4.1113
Q4
What drugs target the gene PPARA?
The drugs that target PPARA are Fenofibric Acid, Fenofibrate, Bezafibrate, Clofibrate, Choline Fenofibrate, Ciprofibrate, and Gemfibrozil.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PPARA %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_347', 'drugName': 'Fenofibric Acid', 'newLinkedTargets_string': 'PPARA (ENSG00000186951)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4561', 'drugName': 'Ciprofibrate', 'newLinkedTargets_string': 'PPARA (ENSG00000186951)', 'drugIsApproved': True, 'max...
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Genetic Target
Q4.1059
Q4
What drugs target the gene PDE7A?
The drugs that target PDE7A are Flavoxate, Flavoxate Hydrochloride, Pentoxifylline, and Dipyridamole.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PDE7A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_766', 'drugName': 'Flavoxate', 'newLinkedTargets_string': 'PDE8B (ENSG00000113231), PDE8A (ENSG00000073417), PDE7A (ENSG00000205268), PDE7B (ENSG00000171408), PDE4A (ENSG00000065989), PDE4D (ENSG00000113448), PDE4B (ENSG00000184588), PDE4C (ENSG00000105650)', 'drugIsApproved': True, 'maxCl...
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Genetic Target
Q4.599
Q4
What drugs target the gene HPD?
The drug that targets HPD is Nitisinone.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%HPD %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4714', 'drugName': 'Nitisinone', 'newLinkedTargets_string': 'HPD (ENSG00000158104)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}]
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Genetic Target
Q4.62
Q4
What drugs target the gene ANGPT2?
The drug that targets ANGPT2 is Faricimab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ANGPT2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_864', 'drugName': 'Faricimab', 'newLinkedTargets_string': 'ANGPT2 (ENSG00000091879), VEGFA (ENSG00000112715)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_865', 'drugName': 'Faricimab', 'newLinkedTargets_string': 'ANGPT2 (ENSG00000091879), VEGFA (ENSG0...
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Genetic Target
Q4.877
Q4
What drugs target the gene MEN1?
There are no FDA approved drugs targeting the gene MEN1. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Revumenib and Sndx-5613.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%MEN1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1716', 'drugName': 'Revumenib', 'newLinkedTargets_string': 'MEN1 (ENSG00000133895), KMT2A (ENSG00000118058)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 1}, {'UUID': 'DrugGeneTargets_v2_3382', 'drugName': 'Sndx-5613', 'newLinkedTargets_string': 'MEN1 (ENSG00000133895), KMT2A (ENSG00...
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Genetic Target
Q4.1146
Q4
What drugs target the gene PRMT5?
There are no approved drugs targeting PRMT5, but the drug Pemrametostat, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PRMT5 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1649', 'drugName': 'Pemrametostat', 'newLinkedTargets_string': 'PRMT5 (ENSG00000100462)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
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Genetic Target
Q4.1442
Q4
What drugs target the gene TNF?
The drugs that target TNF are Golimumab, Etanercept, Adalimumab, Certolizumab Pegol, and Infliximab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TNF %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6275', 'drugName': 'Infliximab', 'newLinkedTargets_string': 'TNF (ENSG00000232810)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_393', 'drugName': 'Golimumab', 'newLinkedTargets_string': 'TNF (ENSG00000232810)', 'drugIsApproved': True, 'maxClinicalTria...
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Genetic Target
Q4.280
Q4
What drugs target the gene CLEC4C?
There are no approved drugs targeting CLEC4C, but the drug Litifilimab, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CLEC4C %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4112', 'drugName': 'Litifilimab', 'newLinkedTargets_string': 'CLEC4C (ENSG00000198178)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}]
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Q4.37
Q4
What drugs target the gene ADRA2C?
The drugs that target ADRA2C are Oxymetazoline, Naphazoline Hydrochloride, Oxymetazoline Hydrochloride, Tetrahydrozoline, Clonidine, Moxisylyte, Dipivefrin, Epinephrine, Tetrahydrozoline Hydrochloride, Alseroxylon, Guanabenz Acetate, Dipivefrin Hydrochloride, Labetalol, Dexmedetomidine, Norepinephrine Bitartrate, Pheno...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ADRA2C %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4923', 'drugName': 'Brimonidine Tartrate', 'newLinkedTargets_string': 'ADRA2A (ENSG00000150594), ADRA2C (ENSG00000184160), ADRA2B (ENSG00000274286)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5012', 'drugName': 'Tizanidine Hydrochloride', 'newLinkedT...
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Q4.666
Q4
What drugs target the gene IL10RA?
There are no approved drugs targeting IL10RA, but the drug Pegilodecakin, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%IL10RA %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4152', 'drugName': 'Pegilodecakin', 'newLinkedTargets_string': 'IL10RB (ENSG00000243646), IL10RA (ENSG00000110324)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}]
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Genetic Target
Q4.1385
Q4
What drugs target the gene SNCA?
There are no FDA approved drugs targeting the gene SNCA. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Prasinezumab and Cinpanemab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%SNCA %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1283', 'drugName': 'Prasinezumab', 'newLinkedTargets_string': 'SNCA (ENSG00000145335)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_5903', 'drugName': 'Cinpanemab', 'newLinkedTargets_string': 'SNCA (ENSG00000145335)', 'drugIsApproved': False, 'maxClin...
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Genetic Target
Q4.1344
Q4
What drugs target the gene SDC1?
There are no approved drugs targeting SDC1, but the drug Indatuximab Ravtansine, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%SDC1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_294', 'drugName': 'Indatuximab Ravtansine', 'newLinkedTargets_string': 'SDC1 (ENSG00000115884)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 1}]
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Genetic Target
Q4.983
Q4
What drugs target the gene NISCH?
The drug that targets NISCH is Moxonidine.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NISCH %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2347', 'drugName': 'Moxonidine', 'newLinkedTargets_string': 'NISCH (ENSG00000010322)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3253', 'drugName': 'Rilmenidine', 'newLinkedTargets_string': 'NISCH (ENSG00000010322)', 'drugIsApproved': False, 'maxClin...
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Genetic Target
Q4.743
Q4
What drugs target the gene KCNC1?
The drugs that target KCNC1 are Dalfampridine, Guanidine, Amifampridine Phosphate, Guanidine Hydrochloride, and Amifampridine.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%KCNC1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5118', 'drugName': 'Guanidine Hydrochloride', 'newLinkedTargets_string': 'KCNQ1 (ENSG00000053918), KCND3 (ENSG00000171385), KCNH2 (ENSG00000055118), KCNA2 (ENSG00000177301), KCNA1 (ENSG00000111262), KCNQ2 (ENSG00000075043), KCNQ3 (ENSG00000184156), KCNA7 (ENSG00000104848), KCNQ5 (ENSG00000...
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Genetic Target
Q4.193
Q4
What drugs target the gene CCR1?
There are no FDA approved drugs targeting the gene CCR1. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Bms-817399, Ccx354, and Azd4818.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CCR1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_194', 'drugName': 'Bms-817399', 'newLinkedTargets_string': 'CCR1 (ENSG00000163823)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_200', 'drugName': 'Ccx354', 'newLinkedTargets_string': 'CCR1 (ENSG00000163823)', 'drugIsApproved': False, 'maxClinicalTria...
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Genetic Target
Q4.924
Q4
What drugs target the gene MYH7B?
The drug that targets MYH7B is Mavacamten.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%MYH7B %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1036', 'drugName': 'Mavacamten', 'newLinkedTargets_string': 'MYH7 (ENSG00000092054), MYH6 (ENSG00000197616), MYH7B (ENSG00000078814), MYL3 (ENSG00000160808), MYL2 (ENSG00000111245), MYL7 (ENSG00000106631), MYL4 (ENSG00000198336)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID...
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Q4.458
Q4
What drugs target the gene FFAR2?
There are no approved drugs targeting FFAR2, but the drug Glpg-0974, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%FFAR2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5482', 'drugName': 'Glpg-0974', 'newLinkedTargets_string': 'FFAR2 (ENSG00000126262)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
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Genetic Target
Q4.680
Q4
What drugs target the gene IL18R1?
There are no approved drugs targeting IL18R1, but the drug Iboctadekin, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%IL18R1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2219', 'drugName': 'Iboctadekin', 'newLinkedTargets_string': 'IL18RAP (ENSG00000115607), IL18R1 (ENSG00000115604)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
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Q4.765
Q4
What drugs target the gene KCNJ3?
The drug that targets KCNJ3 is Vernakalant.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%KCNJ3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_716', 'drugName': 'Vernakalant', 'newLinkedTargets_string': 'KCND3 (ENSG00000171385), KCNA5 (ENSG00000130037), KCNJ3 (ENSG00000162989), KCNJ5 (ENSG00000120457), KCNH2 (ENSG00000055118), SCN5A (ENSG00000183873)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets...
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Genetic Target
Q4.1386
Q4
What drugs target the gene SOAT1?
The drug that targets SOAT1 is Benfluorex.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%SOAT1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5285', 'drugName': 'Benfluorex', 'newLinkedTargets_string': 'SOAT1 (ENSG00000057252)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_6272', 'drugName': 'Pactimibe', 'newLinkedTargets_string': 'SOAT2 (ENSG00000167780), SOAT1 (ENSG00000057252)', 'drugIsApp...
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Genetic Target
Q4.733
Q4
What drugs target the gene KCNA1?
The drugs that target KCNA1 are Dalfampridine, Guanidine, Amifampridine Phosphate, Guanidine Hydrochloride, and Amifampridine.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%KCNA1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5118', 'drugName': 'Guanidine Hydrochloride', 'newLinkedTargets_string': 'KCNQ1 (ENSG00000053918), KCND3 (ENSG00000171385), KCNH2 (ENSG00000055118), KCNA2 (ENSG00000177301), KCNA1 (ENSG00000111262), KCNQ2 (ENSG00000075043), KCNQ3 (ENSG00000184156), KCNA7 (ENSG00000104848), KCNQ5 (ENSG00000...
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Genetic Target
Q4.414
Q4
What drugs target the gene EPHA7?
The drug that targets EPHA7 is Vandetanib.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%EPHA7 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1936', 'drugName': 'Vandetanib', 'newLinkedTargets_string': 'TEK (ENSG00000120156), ERBB2 (ENSG00000141736), EGFR (ENSG00000146648), ERBB4 (ENSG00000178568), ERBB3 (ENSG00000065361), EPHA2 (ENSG00000142627), EPHB2 (ENSG00000133216), EPHA5 (ENSG00000145242), EPHA4 (ENSG00000116106), EPHA8 (...
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Genetic Target
Q4.830
Q4
What drugs target the gene LTA?
There are no FDA approved drugs targeting the gene LTA. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Pateclizumab and Baminercept.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%LTA %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_937', 'drugName': 'Pateclizumab', 'newLinkedTargets_string': 'LTA (ENSG00000226979)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_5474', 'drugName': 'Baminercept', 'newLinkedTargets_string': 'LTA (ENSG00000226979), LTB (ENSG00000227507), TNFSF14 (ENSG...
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Q4.620
Q4
What drugs target the gene HTR2A?
The drugs that target HTR2A are Promazine Hydrochloride, Haloperidol Decanoate, Loxapine Succinate, Pimavanserin, Trimipramine Maleate, Molindone, Zimeldine, Asenapine, Droperidol, Trazodone, Cyclobenzaprine, Amisulpride, Olanzapine Pamoate, Ziprasidone, Thiothixene Hydrochloride, Clothiapine, Olanzapine, Aripiprazole,...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%HTR2A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4892', 'drugName': 'Carphenazine', 'newLinkedTargets_string': 'HTR2A (ENSG00000102468), HTR2C (ENSG00000147246), DRD2 (ENSG00000149295)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5097', 'drugName': 'Pimavanserin Tartrate', 'newLinkedTargets_string':...
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Q4.116
Q4
What drugs target the gene BLK?
The drug that targets BLK is Dasatinib.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%BLK %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4602', 'drugName': 'Dasatinib', 'newLinkedTargets_string': 'PDGFRB (ENSG00000113721), FYN (ENSG00000010810), SRC (ENSG00000197122), LCK (ENSG00000182866), YES1 (ENSG00000176105), BLK (ENSG00000136573), HCK (ENSG00000101336), LYN (ENSG00000254087), FRK (ENSG00000111816), FGR (ENSG0000000093...
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Q4.419
Q4
What drugs target the gene EPHB4?
The drug that targets EPHB4 is Vandetanib.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%EPHB4 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1936', 'drugName': 'Vandetanib', 'newLinkedTargets_string': 'TEK (ENSG00000120156), ERBB2 (ENSG00000141736), EGFR (ENSG00000146648), ERBB4 (ENSG00000178568), ERBB3 (ENSG00000065361), EPHA2 (ENSG00000142627), EPHB2 (ENSG00000133216), EPHA5 (ENSG00000145242), EPHA4 (ENSG00000116106), EPHA8 (...
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Q4.1464
Q4
What drugs target the gene TNNI3?
There are no approved drugs targeting TNNI3, but the drug Levosimendan, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TNNI3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2198', 'drugName': 'Levosimendan', 'newLinkedTargets_string': 'PDE3A (ENSG00000172572), PDE3B (ENSG00000152270), TNNC1 (ENSG00000114854), TNNI3 (ENSG00000129991), TNNT2 (ENSG00000118194)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_2199', 'drugName':...
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Q4.975
Q4
What drugs target the gene NDUFV1?
The drugs that target NDUFV1 are Metformin and Metformin Hydrochloride.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%NDUFV1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (ENSG00000165264), NDUFA4 (...
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Genetic Target
Q4.608
Q4
What drugs target the gene HSD3B2?
The drug that targets HSD3B2 is Trilostane.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%HSD3B2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2278', 'drugName': 'Trilostane', 'newLinkedTargets_string': 'HSD3B2 (ENSG00000203859)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}]
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Q4.1537
Q4
What drugs target the gene XPO1?
The drug that targets XPO1 is Selinexor.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%XPO1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_58', 'drugName': 'Selinexor', 'newLinkedTargets_string': 'XPO1 (ENSG00000082898)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}]
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Q4.91
Q4
What drugs target the gene ATP4B?
The drugs that target ATP4B are Dexlansoprazole, Pantoprazole Sodium, Esomeprazole, Esomeprazole Strontium, Lansoprazole, Omeprazole Magnesium, Rabeprazole, Esomeprazole Sodium, Esomeprazole Magnesium, Omeprazole, Pantoprazole, Rabeprazole Sodium, Vonoprazan, and Vonoprazan Fumarate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ATP4B %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5144', 'drugName': 'Rabeprazole Sodium', 'newLinkedTargets_string': 'ATP4A (ENSG00000105675), ATP4B (ENSG00000186009)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4835', 'drugName': 'Pantoprazole', 'newLinkedTargets_string': 'ATP4A (ENSG00000105675), ...
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Q4.853
Q4
What drugs target the gene MAP3K13?
There are no approved drugs targeting MAP3K13, but the drug Cep-1347, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%MAP3K13 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6091', 'drugName': 'Cep-1347', 'newLinkedTargets_string': 'MAP3K13 (ENSG00000073803), MAP3K12 (ENSG00000139625), MAP3K10 (ENSG00000130758), MAP3K9 (ENSG00000006432), MAP3K11 (ENSG00000173327)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_6088', 'drugN...
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Q4.1172
Q4
What drugs target the gene PSMC3?
The drugs that target PSMC3 are Bortezomib, Carfilzomib, Ixazomib, and Ixazomib Citrate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PSMC3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_559', 'drugName': 'Bortezomib', 'newLinkedTargets_string': 'PSMD1 (ENSG00000173692), PSMB2 (ENSG00000126067), PSMB1 (ENSG00000008018), PSMB5 (ENSG00000100804), PSMB8 (ENSG00000204264), PSMB9 (ENSG00000240065), PSMB6 (ENSG00000142507), PSMD14 (ENSG00000115233), PSMA1 (ENSG00000129084), PSMA...
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Q4.1469
Q4
What drugs target the gene TOP2A?
The drugs that target TOP2A are Idarubicin, Doxorubicin, Daunorubicin, Daunorubicin Citrate, Daunorubicin Hydrochloride, Mitoxantrone, Teniposide, Etoposide Phosphate, Amsacrine, Dexrazoxane, Doxorubicin Hydrochloride, Mitoxantrone Hydrochloride, Etoposide, Idarubicin Hydrochloride, and Valrubicin.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TOP2A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2612', 'drugName': 'Teniposide', 'newLinkedTargets_string': 'TOP2A (ENSG00000131747), TOP2B (ENSG00000077097)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4763', 'drugName': 'Etoposide', 'newLinkedTargets_string': 'TOP2A (ENSG00000131747), TOP2B (ENSG...
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Q4.758
Q4
What drugs target the gene KCNH4?
The drugs that target KCNH4 are Dalfampridine, Guanidine, Amifampridine Phosphate, Guanidine Hydrochloride, and Amifampridine.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%KCNH4 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5118', 'drugName': 'Guanidine Hydrochloride', 'newLinkedTargets_string': 'KCNQ1 (ENSG00000053918), KCND3 (ENSG00000171385), KCNH2 (ENSG00000055118), KCNA2 (ENSG00000177301), KCNA1 (ENSG00000111262), KCNQ2 (ENSG00000075043), KCNQ3 (ENSG00000184156), KCNA7 (ENSG00000104848), KCNQ5 (ENSG00000...
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Q4.501
Q4
What drugs target the gene GABRB3?
The drugs that target GABRB3 are Meprobamate, Acamprosate Calcium, Enflurane, Methohexital, Metharbital, Butabarbital, Flurazepam Hydrochloride, Pentobarbital Sodium, Acamprosate, Primidone, Temazepam, Flunitrazepam, Ganaxolone, Diazepam, Methyprylon, Thiopental, Clonazepam, Topiramate, Remimazolam Besylate, Brexanolon...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%GABRB3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2287', 'drugName': 'Clomethiazole', 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089), GABRA3 (ENSG00000011677), GABRP (ENSG00000094...
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Q4.12
Q4
What drugs target the gene ACHE?
The drugs that target ACHE are Ambenonium Chloride, Ambenonium, Rivastigmine, Pyridostigmine, Donepezil Hydrochloride, Galantamine Hydrobromide, Rivastigmine Tartrate, Neostigmine Methylsulfate, Isoflurophate, Tacrine, Echothiophate Iodide, Echothiophate, Demecarium, Distigmine, Physostigmine Salicylate, Galantamine, P...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ACHE %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1632', 'drugName': 'Galantamine Hydrobromide', 'newLinkedTargets_string': 'ACHE (ENSG00000087085)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_516', 'drugName': 'Pyridostigmine', 'newLinkedTargets_string': 'ACHE (ENSG00000087085)', 'drugIsApproved': T...
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Q4.398
Q4
What drugs target the gene ELANE?
The drug that targets ELANE is .Alpha.1-Proteinase Inhibitor Human.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ELANE %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2772', 'drugName': '.Alpha.1-Proteinase Inhibitor Human', 'newLinkedTargets_string': 'ELANE (ENSG00000197561)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3534', 'drugName': 'Sivelestat', 'newLinkedTargets_string': 'ELANE (ENSG00000197561)', 'drugIsAp...
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Q4.286
Q4
What drugs target the gene COL11A2?
The drugs that target COL11A2 are Collagenase Clostridium Histolyticum and Ocriplasmin.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%COL11A2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5818', 'drugName': 'Ocriplasmin', 'newLinkedTargets_string': 'FN1 (ENSG00000115414), COL1A2 (ENSG00000164692), COL1A1 (ENSG00000108821), COL2A1 (ENSG00000139219), COL3A1 (ENSG00000168542), COL4A1 (ENSG00000187498), COL5A1 (ENSG00000130635), COL6A1 (ENSG00000142156), COL11A1 (ENSG0000006071...
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Q4.1072
Q4
What drugs target the gene PGA5?
The drug that targets PGA5 is Sucralfate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PGA5 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4142', 'drugName': 'Sucralfate', 'newLinkedTargets_string': 'PGA5 (ENSG00000256713)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5872', 'drugName': 'Sucralfate', 'newLinkedTargets_string': 'PGA5 (ENSG00000256713)', 'drugIsApproved': True, 'maxClinical...
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Q4.695
Q4
What drugs target the gene IL2RG?
The drugs that target IL2RG are Basiliximab, Aldesleukin, Denileukin Diftitox, and Daclizumab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%IL2RG %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2628', 'drugName': 'Basiliximab', 'newLinkedTargets_string': 'IL2RA (ENSG00000134460), IL2RG (ENSG00000147168), IL2RB (ENSG00000100385)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5681', 'drugName': 'Daclizumab', 'newLinkedTargets_string': 'IL2RA (EN...
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Q4.1261
Q4
What drugs target the gene RPL37A?
The drug that targets RPL37A is Ataluren.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RPL37A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG00000083845), RPS7 (ENSG...
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Q4.1439
Q4
What drugs target the gene TLR9?
The drugs that target TLR9 are Hydroxychloroquine and Hydroxychloroquine Sulfate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TLR9 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3879', 'drugName': 'Hydroxychloroquine Sulfate', 'newLinkedTargets_string': 'TLR9 (ENSG00000239732), TLR7 (ENSG00000196664)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3878', 'drugName': 'Hydroxychloroquine Sulfate', 'newLinkedTargets_string': 'TLR9 ...
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Q4.694
Q4
What drugs target the gene IL2RB?
The drugs that target IL2RB are Basiliximab, Aldesleukin, Denileukin Diftitox, and Daclizumab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%IL2RB %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5633', 'drugName': 'Denileukin Diftitox', 'newLinkedTargets_string': 'IL2RA (ENSG00000134460), IL2RG (ENSG00000147168), IL2RB (ENSG00000100385), EEF2 (ENSG00000167658)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2628', 'drugName': 'Basiliximab', 'new...
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Q4.856
Q4
What drugs target the gene MAP3K9?
There are no approved drugs targeting MAP3K9, but the drug Cep-1347, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%MAP3K9 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6091', 'drugName': 'Cep-1347', 'newLinkedTargets_string': 'MAP3K13 (ENSG00000073803), MAP3K12 (ENSG00000139625), MAP3K10 (ENSG00000130758), MAP3K9 (ENSG00000006432), MAP3K11 (ENSG00000173327)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_6088', 'drugN...
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Q4.161
Q4
What drugs target the gene CACNG2?
The drugs that target CACNG2 are Gabapentin, Terodiline Hydrochloride, Phloroglucinol, Suloctidil, Pregabalin, Gabapentin Enacarbil, Bepridil Hydrochloride, Bepridil, and Terodiline.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CACNG2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_142', 'drugName': 'Gabapentin', 'newLinkedTargets_string': 'CACNA1H (ENSG00000196557), CACNA2D1 (ENSG00000153956), CACNA1C (ENSG00000151067), CACNA2D3 (ENSG00000157445), CACNA1S (ENSG00000081248), CACNA2D2 (ENSG00000007402), CACNA1D (ENSG00000157388), CACNA1A (ENSG00000141837), CACNA1B (EN...
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Q4.900
Q4
What drugs target the gene MMP8?
The drugs that target MMP8 are Doxycycline Anhydrous, Doxycycline Hyclate, Doxycycline, and Doxycycline Calcium.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%MMP8 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2398', 'drugName': 'Doxycycline Hyclate', 'newLinkedTargets_string': 'MMP13 (ENSG00000137745), MMP1 (ENSG00000196611), MMP7 (ENSG00000137673), MMP8 (ENSG00000118113)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3046', 'drugName': 'Doxycycline', 'newLi...
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Q4.1219
Q4
What drugs target the gene RHD?
There are no FDA approved drugs targeting the gene RHD. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Roledumab, Morolimumab, Atorolimumab, and Rozrolimupab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RHD %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3177', 'drugName': 'Roledumab', 'newLinkedTargets_string': 'RHD (ENSG00000187010)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_6033', 'drugName': 'Rozrolimupab', 'newLinkedTargets_string': 'RHD (ENSG00000187010)', 'drugIsApproved': False, 'maxClinica...
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Q4.259
Q4
What drugs target the gene CHRM1?
The drugs that target CHRM1 are Clidinium Bromide, Terodiline Hydrochloride, Benztropine Mesylate, Methixene Hydrochloride, Oxyphencyclimine, Glycopyrrolate, Oxyphenonium Bromide, Methixene, Diphemanil Methylsulfate, Biperiden, Diphenidol Hydrochloride, Biperiden Hydrochloride, Oxyphenonium, Mepenzolate Bromide, Methsc...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CHRM1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2995', 'drugName': 'Glycopyrronium', 'newLinkedTargets_string': 'CHRM3 (ENSG00000133019), CHRM1 (ENSG00000168539)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_6050', 'drugName': 'Trihexyphenidyl Hydrochloride', 'newLinkedTargets_string': 'CHRM1 (ENSG0...
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Q4.337
Q4
What drugs target the gene CXCL12?
There are no approved drugs targeting CXCL12, but the drug Olaptesed Pegol, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CXCL12 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3593', 'drugName': 'Olaptesed Pegol', 'newLinkedTargets_string': 'CXCL12 (ENSG00000107562)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}]
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Q4.1443
Q4
What drugs target the gene TNFRSF10A?
There are no FDA approved drugs targeting the gene TNFRSF10A. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Dulanermin and Mapatumumab.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%TNFRSF10A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5538', 'drugName': 'Mapatumumab', 'newLinkedTargets_string': 'TNFRSF10A (ENSG00000104689)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_638', 'drugName': 'Dulanermin', 'newLinkedTargets_string': 'TNFRSF10A (ENSG00000104689), TNFRSF10B (ENSG00000120889...
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Q4.1045
Q4
What drugs target the gene PDE2A?
The drugs that target PDE2A are Pentoxifylline and Dipyridamole.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PDE2A %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6107', 'drugName': 'Dipyridamole', 'newLinkedTargets_string': 'PDE5A (ENSG00000138735), PDE4A (ENSG00000065989), PDE3A (ENSG00000172572), PDE6H (ENSG00000139053), PDE6G (ENSG00000185527), PDE2A (ENSG00000186642), PDE7A (ENSG00000205268), PDE1A (ENSG00000115252), PDE9A (ENSG00000160191), PD...
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Q4.518
Q4
What drugs target the gene GHRHR?
The drugs that target GHRHR are Tesamorelin, Tesamorelin Acetate, and Sermorelin Acetate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%GHRHR %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2825', 'drugName': 'Tesamorelin', 'newLinkedTargets_string': 'GHRHR (ENSG00000106128)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5465', 'drugName': 'Sermorelin Acetate', 'newLinkedTargets_string': 'GHRHR (ENSG00000106128)', 'drugIsApproved': True, '...
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Q4.1021
Q4
What drugs target the gene OPRM1?
The drugs that target OPRM1 are Morphine, Diphenoxylate, Naloxegol Oxalate, Propoxyphene Napsylate, Codeine Polistirex, Meperidine Hydrochloride, Benzhydrocodone, Remifentanil Hydrochloride, Difenoxin, Nalmefene Hydrochloride, Fentanyl Citrate, Butorphanol, Oxycodone Terephthalate, Alfentanil Hydrochloride, Naldemedine...
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%OPRM1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1750', 'drugName': 'Methadone', 'newLinkedTargets_string': 'OPRM1 (ENSG00000112038)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3858', 'drugName': 'Diacetylmorphine', 'newLinkedTargets_string': 'OPRM1 (ENSG00000112038)', 'drugIsApproved': True, 'maxC...
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Q4.773
Q4
What drugs target the gene KCNMA1?
There are no FDA approved drugs targeting the gene KCNMA1. However, the following drugs, which potentially target this gene, are currently in various clinical trial stages: Flindokalner, Bms-223131, and Andolast.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%KCNMA1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2864', 'drugName': 'Flindokalner', 'newLinkedTargets_string': 'KCNMA1 (ENSG00000156113), KCNQ2 (ENSG00000075043), KCNQ3 (ENSG00000184156), KCNQ4 (ENSG00000117013), KCNQ5 (ENSG00000185760)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_2869', 'drugName'...
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Q4.1349
Q4
What drugs target the gene SEM1?
The drugs that target SEM1 are Bortezomib, Carfilzomib, Ixazomib, and Ixazomib Citrate.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%SEM1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_559', 'drugName': 'Bortezomib', 'newLinkedTargets_string': 'PSMD1 (ENSG00000173692), PSMB2 (ENSG00000126067), PSMB1 (ENSG00000008018), PSMB5 (ENSG00000100804), PSMB8 (ENSG00000204264), PSMB9 (ENSG00000240065), PSMB6 (ENSG00000142507), PSMD14 (ENSG00000115233), PSMA1 (ENSG00000129084), PSMA...
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Q4.766
Q4
What drugs target the gene KCNJ5?
The drug that targets KCNJ5 is Vernakalant.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%KCNJ5 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_716', 'drugName': 'Vernakalant', 'newLinkedTargets_string': 'KCND3 (ENSG00000171385), KCNA5 (ENSG00000130037), KCNJ3 (ENSG00000162989), KCNJ5 (ENSG00000120457), KCNH2 (ENSG00000055118), SCN5A (ENSG00000183873)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets...
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Q4.1127
Q4
What drugs target the gene PRKAB2?
There are no approved drugs targeting PRKAB2, but the drug Acadesine, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%PRKAB2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5888', 'drugName': 'Acadesine', 'newLinkedTargets_string': 'PRKAA2 (ENSG00000162409), PRKAB2 (ENSG00000131791), PRKAG1 (ENSG00000181929), PRKAG2 (ENSG00000106617), PRKAB1 (ENSG00000111725), PRKAA1 (ENSG00000132356), PRKAG3 (ENSG00000115592)', 'drugIsApproved': False, 'maxClinicalTrialPhase...
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Q4.524
Q4
What drugs target the gene GLRA1?
The drugs that target GLRA1 are Enflurane, Methoxyflurane, Sevoflurane, Desflurane, Halothane, and Isoflurane.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%GLRA1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5597', 'drugName': 'Isoflurane', 'newLinkedTargets_string': 'KCNK10 (ENSG00000100433), KCNK9 (ENSG00000169427), GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089...
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Q4.23
Q4
What drugs target the gene ADH4?
The drug that targets ADH4 is Nitrefazole.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%ADH4 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6344', 'drugName': 'Nitrefazole', 'newLinkedTargets_string': 'ADH1A (ENSG00000187758), ADH4 (ENSG00000198099), ADH1B (ENSG00000196616), ADH1C (ENSG00000248144), ADH7 (ENSG00000196344), ADH5 (ENSG00000197894), ADH6 (ENSG00000172955)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}]
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Q4.358
Q4
What drugs target the gene DGAT1?
There are no approved drugs targeting DGAT1, but the drug Pradigastat, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%DGAT1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3433', 'drugName': 'Pradigastat', 'newLinkedTargets_string': 'DGAT1 (ENSG00000185000)', 'drugIsApproved': False, 'maxClinicalTrialPhase': 3}]
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Q4.1304
Q4
What drugs target the gene RPS6KA3?
There are no approved drugs targeting RPS6KA3, but the drug Tas0612, which potentially targets this gene, is currently undergoing clinical trials.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%RPS6KA3 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3347', 'drugName': 'Tas0612', 'newLinkedTargets_string': 'RPS6KB2 (ENSG00000175634), RPS6KB1 (ENSG00000108443), AKT2 (ENSG00000105221), AKT3 (ENSG00000117020), AKT1 (ENSG00000142208), RPS6KA3 (ENSG00000177189), RPS6KA2 (ENSG00000071242), RPS6KA6 (ENSG00000072133), RPS6KA1 (ENSG00000117676)...
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Q4.342
Q4
What drugs target the gene CYP11A1?
The drugs that target CYP11A1 are Aminoglutethimide, Levoketoconazole, and Mitotane.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%CYP11A1 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3930', 'drugName': 'Levoketoconazole', 'newLinkedTargets_string': 'CYP11B1 (ENSG00000160882), CYP11B2 (ENSG00000179142), CYP17A1 (ENSG00000148795), CYP11A1 (ENSG00000140459)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3932', 'drugName': 'Levoketocona...
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Q4.433
Q4
What drugs target the gene EZH2?
The drugs that target EZH2 are Tazemetostat and Tazemetostat Hydrobromide.
SELECT DISTINCT UUID, drugName, newLinkedTargets_string, drugIsApproved, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE '%EZH2 %' ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4960', 'drugName': 'Tazemetostat Hydrobromide', 'newLinkedTargets_string': 'EZH2 (ENSG00000106462)', 'drugIsApproved': True, 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1211', 'drugName': 'Tazemetostat', 'newLinkedTargets_string': 'EZH2 (ENSG00000106462)', 'drugIsApproved': T...
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