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Q58.618
Q58
How many genes does the drug Ondansetron Hydrochloride target and what are they?
HTR3A is the only gene target of drug Ondansetron Hydrochloride.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ondansetron hydrochloride%" OR LOWER(tradeNames_...
[{'UUID': 'DrugGeneTargets_v2_4955', 'drugName': 'Ondansetron Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HTR3A (ENSG00000166736)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1991, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.1479
Q58
How many genes does the drug Insulin Lispro Protamine Recombinant target and what are they?
INSR is the only gene target of drug Insulin Lispro Protamine Recombinant.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%insulin lispro protamine recombinant%" OR LOWER(...
[{'UUID': 'DrugGeneTargets_v2_5121', 'drugName': 'Insulin Lispro Protamine Recombinant', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'INSR (ENSG00000171105)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1999, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.250
Q58
How many genes does the drug Aprotinin target and what are they?
There are 2 gene targets for the drug Aprotinin: PLG and KLKB1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%aprotinin%" OR LOWER(tradeNames_string) LIKE "%a...
[{'UUID': 'DrugGeneTargets_v2_4053', 'drugName': 'Aprotinin', 'drugMolecularType': 'Unknown', 'newLinkedTargets_string': 'PLG (ENSG00000122194), KLKB1 (ENSG00000164344)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1993, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_4054', 'drug...
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Genetic Target
Q58.734
Q58
How many genes does the drug Teriparatide target and what are they?
PTH1R is the only gene target of drug Teriparatide.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%teriparatide%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_3571', 'drugName': 'Teriparatide Acetate', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'PTH1R (ENSG00000160801)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1987, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_2407', 'drugName': 'Teri...
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Genetic Target
Q58.311
Q58
How many genes does the drug Mitapivat Sulfate target and what are they?
PKLR is the only gene target of drug Mitapivat Sulfate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%mitapivat sulfate%" OR LOWER(tradeNames_string) ...
[{'UUID': 'DrugGeneTargets_v2_2811', 'drugName': 'Mitapivat Sulfate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PKLR (ENSG00000143627)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2022, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.236
Q58
How many genes does the drug Diphemanil target and what are they?
There are 2 gene targets for the drug Diphemanil: CHRM3 and CHRM1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%diphemanil%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2135', 'drugName': 'Diphemanil', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CHRM3 (ENSG00000133019), CHRM1 (ENSG00000168539)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1982, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_21...
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Genetic Target
Q58.72
Q58
How many genes does the drug Isotretinoin target and what are they?
There are 3 gene targets for the drug Isotretinoin: RARG, RARB, and RARA.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%isotretinoin%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_3116', 'drugName': 'Isotretinoin', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'RARG (ENSG00000172819), RARB (ENSG00000077092), RARA (ENSG00000131759)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 1982, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.896
Q58
How many genes does the drug Bivalirudin target and what are they?
F2 is the only gene target of drug Bivalirudin.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%bivalirudin%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_4317', 'drugName': 'Bivalirudin', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'F2 (ENSG00000180210)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2000, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.1754
Q58
How many genes does the drug Avl-3288 target and what are they?
The drug Avl-3288 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene CHRNA7.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%avl-3288%" OR LOWER(tradeNames_string) LIKE "%av...
[{'UUID': 'DrugGeneTargets_v2_2542', 'drugName': 'Avl-3288', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CHRNA7 (ENSG00000175344)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drugIsApproved': False}]
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Q58.712
Q58
How many genes does the drug Epoetin Theta target and what are they?
EPOR is the only gene target of drug Epoetin Theta.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%epoetin theta%" OR LOWER(tradeNames_string) LIKE...
[{'UUID': 'DrugGeneTargets_v2_6035', 'drugName': 'Epoetin Theta', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'EPOR (ENSG00000187266)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.1383
Q58
How many genes does the drug Dexmethylphenidate Hydrochloride target and what are they?
There are 2 gene targets for the drug Dexmethylphenidate Hydrochloride: SLC6A2 and SLC6A3.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%dexmethylphenidate hydrochloride%" OR LOWER(trad...
[{'UUID': 'DrugGeneTargets_v2_5956', 'drugName': 'Dexmethylphenidate Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SLC6A2 (ENSG00000103546), SLC6A3 (ENSG00000142319)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2001, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID'...
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Q58.1329
Q58
How many genes does the drug Azacitidine target and what are they?
There are 2 gene targets for the drug Azacitidine: DNMT1 and DNMT3A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%azacitidine%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_4131', 'drugName': 'Azacitidine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'DNMT1 (ENSG00000130816), DNMT3A (ENSG00000119772)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2004, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_...
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Q58.624
Q58
How many genes does the drug Sevoflurane target and what are they?
There are 23 gene targets for the drug Sevoflurane: KCNK9, KCNK2, KCNK10, KCNK18, KCNK3, GABRA1, GABRB2, GABRG2, GABRB3, GABRA4, GABRG3, GABRQ, GABRA3, GABRP, GABRD, GABRG1, GABRB1, GABRE, GABRA2, GABRA5, GABRA6, GLRA1, and GLRB.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%sevoflurane%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_2923', 'drugName': 'Sevoflurane', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'KCNK9 (ENSG00000169427), KCNK2 (ENSG00000082482), KCNK10 (ENSG00000100433), KCNK18 (ENSG00000186795), KCNK3 (ENSG00000171303), GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (EN...
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Q58.1464
Q58
How many genes does the drug Bromazepam target and what are they?
GABRA2 is the only gene target of drug Bromazepam.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%bromazepam%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2148', 'drugName': 'Bromazepam', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GABRA2 (ENSG00000151834)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.1556
Q58
How many genes does the drug Memantine target and what are they?
There are 7 gene targets for the drug Memantine: GRIN1, GRIN2A, GRIN2B, GRIN2D, GRIN3B, GRIN2C, and GRIN3A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%memantine%" OR LOWER(tradeNames_string) LIKE "%m...
[{'UUID': 'DrugGeneTargets_v2_2817', 'drugName': 'Memantine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GRIN1 (ENSG00000176884), GRIN2A (ENSG00000183454), GRIN2B (ENSG00000273079), GRIN2D (ENSG00000105464), GRIN3B (ENSG00000116032), GRIN2C (ENSG00000161509), GRIN3A (ENSG00000198785)', 'numberLi...
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Q58.708
Q58
How many genes does the drug Acrivastine target and what are they?
HRH1 is the only gene target of drug Acrivastine.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%acrivastine%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_2524', 'drugName': 'Acrivastine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HRH1 (ENSG00000196639)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1994, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.1928
Q58
How many genes does the drug Sodium Dichloroacetate target and what are they?
There are 4 gene targets for the drug Sodium Dichloroacetate: PDK2, PDK3, PDK4, and PDK1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%sodium dichloroacetate%" OR LOWER(tradeNames_str...
[{'UUID': 'DrugGeneTargets_v2_2764', 'drugName': 'Sodium Dichloroacetate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PDK2 (ENSG00000005882), PDK3 (ENSG00000067992), PDK4 (ENSG00000004799), PDK1 (ENSG00000152256)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, '...
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Q58.614
Q58
How many genes does the drug Alprazolam target and what are they?
There are 16 gene targets for the drug Alprazolam: GABRA1, GABRB2, GABRG2, GABRB3, GABRA4, GABRG3, GABRQ, GABRA3, GABRP, GABRD, GABRG1, GABRB1, GABRE, GABRA2, GABRA5, and GABRA6.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%alprazolam%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_4460', 'drugName': 'Alprazolam', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089), GABRA3 (E...
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Genetic Target
Q58.372
Q58
How many genes does the drug Duvoglustat target and what are they?
The drug Duvoglustat is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene GAA.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%duvoglustat%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_98', 'drugName': 'Duvoglustat', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GAA (ENSG00000171298)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}, {'UUID': 'DrugGeneTargets_v2_135', 'drugName': 'Duvoglustat H...
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Q58.1756
Q58
How many genes does the drug Bismuth Subgallate target and what are they?
F12 is the only gene target of drug Bismuth Subgallate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%bismuth subgallate%" OR LOWER(tradeNames_string)...
[{'UUID': 'DrugGeneTargets_v2_5123', 'drugName': 'Bismuth Subgallate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'F12 (ENSG00000131187)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.1669
Q58
How many genes does the drug Etalocib target and what are they?
The drug Etalocib is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 2 genes: PPARG and LTB4R.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%etalocib%" OR LOWER(tradeNames_string) LIKE "%et...
[{'UUID': 'DrugGeneTargets_v2_4852', 'drugName': 'Etalocib', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PPARG (ENSG00000132170), LTB4R (ENSG00000213903)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}, {'UUID': 'DrugGeneTargets_v2_4853',...
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Q58.533
Q58
How many genes does the drug Flecainide Acetate target and what are they?
SCN5A is the only gene target of drug Flecainide Acetate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%flecainide acetate%" OR LOWER(tradeNames_string)...
[{'UUID': 'DrugGeneTargets_v2_605', 'drugName': 'Flecainide Acetate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SCN5A (ENSG00000183873)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1985, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.1821
Q58
How many genes does the drug Clomipramine target and what are they?
SLC6A4 is the only gene target of drug Clomipramine.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%clomipramine%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_4905', 'drugName': 'Clomipramine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SLC6A4 (ENSG00000108576)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1989, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_1137', 'drugName': 'Clom...
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Q58.1442
Q58
How many genes does the drug Pasireotide target and what are they?
There are 4 gene targets for the drug Pasireotide: SSTR3, SSTR1, SSTR2, and SSTR5.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%pasireotide%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_1407', 'drugName': 'Pasireotide Diaspartate', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'SSTR3 (ENSG00000278195), SSTR2 (ENSG00000180616), SSTR1 (ENSG00000139874), SSTR5 (ENSG00000162009)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 2012, 'maxClinicalTrialPhase': 4, ...
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Q58.302
Q58
How many genes does the drug Protokylol Hydrochloride target and what are they?
ADRB2 is the only gene target of drug Protokylol Hydrochloride.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%protokylol hydrochloride%" OR LOWER(tradeNames_s...
[{'UUID': 'DrugGeneTargets_v2_5847', 'drugName': 'Protokylol Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRB2 (ENSG00000169252)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1982, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.1016
Q58
How many genes does the drug Teriflunomide target and what are they?
DHODH is the only gene target of drug Teriflunomide.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%teriflunomide%" OR LOWER(tradeNames_string) LIKE...
[{'UUID': 'DrugGeneTargets_v2_5674', 'drugName': 'Teriflunomide', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'DHODH (ENSG00000102967)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2012, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.1417
Q58
How many genes does the drug T84.66 target and what are they?
The drug T84.66 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene CEACAM5.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%t84.66%" OR LOWER(tradeNames_string) LIKE "%t84....
[{'UUID': 'DrugGeneTargets_v2_2893', 'drugName': '90Y-Ct84.66', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'CEACAM5 (ENSG00000105388)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drugIsApproved': False}, {'UUID': 'DrugGeneTargets_v2_5856', 'drugName': 'T84.66', 'dr...
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Genetic Target
Q58.1567
Q58
How many genes does the drug Enlimomab target and what are they?
The drug Enlimomab is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene ICAM1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%enlimomab%" OR LOWER(tradeNames_string) LIKE "%e...
[{'UUID': 'DrugGeneTargets_v2_5504', 'drugName': 'Enlimomab Pegol', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'ICAM1 (ENSG00000090339)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}, {'UUID': 'DrugGeneTargets_v2_4244', 'drugName': 'Enlimomab'...
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Genetic Target
Q58.1311
Q58
How many genes does the drug Pioglitazone target and what are they?
PPARG is the only gene target of drug Pioglitazone.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%pioglitazone%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_878', 'drugName': 'Pioglitazone Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PPARG (ENSG00000132170)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1999, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_1041', 'drug...
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Genetic Target
Q58.862
Q58
How many genes does the drug Elagolix target and what are they?
GNRHR is the only gene target of drug Elagolix.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%elagolix%" OR LOWER(tradeNames_string) LIKE "%el...
[{'UUID': 'DrugGeneTargets_v2_5788', 'drugName': 'Elagolix', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GNRHR (ENSG00000109163)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2018, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_5526', 'drugName': 'Elagolix ...
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Genetic Target
Q58.591
Q58
How many genes does the drug Lfb-R603 target and what are they?
The drug Lfb-R603 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene MS4A1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%lfb-r603%" OR LOWER(tradeNames_string) LIKE "%lf...
[{'UUID': 'DrugGeneTargets_v2_3518', 'drugName': 'Lfb-R603', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'MS4A1 (ENSG00000156738)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drugIsApproved': False}]
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Genetic Target
Q58.485
Q58
How many genes does the drug Abatacept target and what are they?
There are 2 gene targets for the drug Abatacept: CD80 and CD86.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%abatacept%" OR LOWER(tradeNames_string) LIKE "%a...
[{'UUID': 'DrugGeneTargets_v2_3638', 'drugName': 'Abatacept', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'CD80 (ENSG00000121594), CD86 (ENSG00000114013)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2006, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_3639', 'drug...
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Genetic Target
Q58.1473
Q58
How many genes does the drug Tecadenoson target and what are they?
The drug Tecadenoson is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene ADORA1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tecadenoson%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_275', 'drugName': 'Tecadenoson', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADORA1 (ENSG00000163485)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1784
Q58
How many genes does the drug Vodobatinib target and what are they?
The drug Vodobatinib is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 2 genes: ABL1 and BCR.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%vodobatinib%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_5367', 'drugName': 'Vodobatinib', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ABL1 (ENSG00000097007), BCR (ENSG00000186716)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}, {'UUID': 'DrugGeneTargets_v2_5368',...
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Genetic Target
Q58.644
Q58
How many genes does the drug Abt-107 target and what are they?
The drug Abt-107 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene CHRNA7.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%abt-107%" OR LOWER(tradeNames_string) LIKE "%abt...
[{'UUID': 'DrugGeneTargets_v2_1344', 'drugName': 'Abt-107', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CHRNA7 (ENSG00000175344)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drugIsApproved': False}]
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Genetic Target
Q58.357
Q58
How many genes does the drug Olverembatinib target and what are they?
The drug Olverembatinib is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 2 genes: ABL1 and BCR.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%olverembatinib%" OR LOWER(tradeNames_string) LIK...
[{'UUID': 'DrugGeneTargets_v2_4219', 'drugName': 'Olverembatinib', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ABL1 (ENSG00000097007), BCR (ENSG00000186716)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.1128
Q58
How many genes does the drug Azelastine target and what are they?
HRH1 is the only gene target of drug Azelastine.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%azelastine%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_3567', 'drugName': 'Azelastine Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HRH1 (ENSG00000196639)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1996, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_2721', 'drugNa...
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Genetic Target
Q58.439
Q58
How many genes does the drug Avatrombopag Maleate target and what are they?
MPL is the only gene target of drug Avatrombopag Maleate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%avatrombopag maleate%" OR LOWER(tradeNames_strin...
[{'UUID': 'DrugGeneTargets_v2_6317', 'drugName': 'Avatrombopag Maleate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'MPL (ENSG00000117400)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2018, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1121
Q58
How many genes does the drug Mebanazine target and what are they?
There are 2 gene targets for the drug Mebanazine: MAOA and MAOB.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%mebanazine%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_401', 'drugName': 'Mebanazine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'MAOA (ENSG00000189221), MAOB (ENSG00000069535)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1103
Q58
How many genes does the drug Methylnaltrexone target and what are they?
OPRM1 is the only gene target of drug Methylnaltrexone.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%methylnaltrexone%" OR LOWER(tradeNames_string) L...
[{'UUID': 'DrugGeneTargets_v2_2413', 'drugName': 'Methylnaltrexone Bromide', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'OPRM1 (ENSG00000112038)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2008, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_1780', 'drugN...
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Genetic Target
Q58.1348
Q58
How many genes does the drug Chlordiazepoxide target and what are they?
There are 16 gene targets for the drug Chlordiazepoxide: GABRA1, GABRB2, GABRG2, GABRB3, GABRA4, GABRG3, GABRQ, GABRA3, GABRP, GABRD, GABRG1, GABRB1, GABRE, GABRA2, GABRA5, and GABRA6.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%chlordiazepoxide%" OR LOWER(tradeNames_string) L...
[{'UUID': 'DrugGeneTargets_v2_4453', 'drugName': 'Chlordiazepoxide', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089), GAB...
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Genetic Target
Q58.597
Q58
How many genes does the drug Labetuzumab target and what are they?
The drug Labetuzumab is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene CEACAM5.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%labetuzumab%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_4444', 'drugName': 'Labetuzumab Govitecan', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'CEACAM5 (ENSG00000105388)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}, {'UUID': 'DrugGeneTargets_v2_4322', 'drugName': 'La...
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Genetic Target
Q58.1368
Q58
How many genes does the drug Lumasiran Sodium target and what are they?
HAO1 is the only gene target of drug Lumasiran Sodium.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%lumasiran sodium%" OR LOWER(tradeNames_string) L...
[{'UUID': 'DrugGeneTargets_v2_1071', 'drugName': 'Lumasiran Sodium', 'drugMolecularType': 'Oligonucleotide', 'newLinkedTargets_string': 'HAO1 (ENSG00000101323)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2020, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1401
Q58
How many genes does the drug Fentanyl target and what are they?
OPRM1 is the only gene target of drug Fentanyl.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%fentanyl%" OR LOWER(tradeNames_string) LIKE "%fe...
[{'UUID': 'DrugGeneTargets_v2_3916', 'drugName': 'Fentanyl Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'OPRM1 (ENSG00000112038)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2006, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_733', 'drugName...
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Genetic Target
Q58.753
Q58
How many genes does the drug Mdx-210 target and what are they?
The drug Mdx-210 is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 2 genes: ERBB2 and FCGR1A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%mdx-210%" OR LOWER(tradeNames_string) LIKE "%mdx...
[{'UUID': 'DrugGeneTargets_v2_2242', 'drugName': 'Mdx-210', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'ERBB2 (ENSG00000141736), FCGR1A (ENSG00000150337)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}, {'UUID': 'DrugGeneTargets_v2_2243', 'drug...
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Genetic Target
Q58.259
Q58
How many genes does the drug Ibodutant target and what are they?
The drug Ibodutant is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene TACR2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ibodutant%" OR LOWER(tradeNames_string) LIKE "%i...
[{'UUID': 'DrugGeneTargets_v2_1669', 'drugName': 'Ibodutant', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'TACR2 (ENSG00000075073)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.1687
Q58
How many genes does the drug Irampanel target and what are they?
The drug Irampanel is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 14 genes: GRIA4, GRIA3, GRIA2, GRIA1, SCN1A, SCN5A, SCN4A, SCN7A, SCN2A, SCN9A, SCN3A, SCN11A, SCN8A, and SCN10A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%irampanel%" OR LOWER(tradeNames_string) LIKE "%i...
[{'UUID': 'DrugGeneTargets_v2_782', 'drugName': 'Irampanel', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GRIA4 (ENSG00000152578), GRIA3 (ENSG00000125675), GRIA2 (ENSG00000120251), GRIA1 (ENSG00000155511), SCN1A (ENSG00000144285), SCN5A (ENSG00000183873), SCN4A (ENSG00000007314), SCN7A (ENSG000001...
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Genetic Target
Q58.1723
Q58
How many genes does the drug Adipiplon target and what are they?
The drug Adipiplon is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 16 genes: GABRA1, GABRB2, GABRG2, GABRB3, GABRA4, GABRG3, GABRQ, GABRA3, GABRP, GABRD, GABRG1, GABRB1, GABRE, GABRA2, GABRA5, and GABRA6.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%adipiplon%" OR LOWER(tradeNames_string) LIKE "%a...
[{'UUID': 'DrugGeneTargets_v2_1372', 'drugName': 'Adipiplon', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089), GABRA3 (EN...
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Genetic Target
Q58.544
Q58
How many genes does the drug Corifollitropin Alfa target and what are they?
FSHR is the only gene target of drug Corifollitropin Alfa.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%corifollitropin alfa%" OR LOWER(tradeNames_strin...
[{'UUID': 'DrugGeneTargets_v2_2306', 'drugName': 'Corifollitropin Alfa', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'FSHR (ENSG00000170820)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.792
Q58
How many genes does the drug Quavonlimab target and what are they?
The drug Quavonlimab is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene CTLA4.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%quavonlimab%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_4260', 'drugName': 'Quavonlimab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'CTLA4 (ENSG00000163599)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.1484
Q58
How many genes does the drug Alfuzosin target and what are they?
There are 3 gene targets for the drug Alfuzosin: ADRA1A, ADRA1D, and ADRA1B.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%alfuzosin%" OR LOWER(tradeNames_string) LIKE "%a...
[{'UUID': 'DrugGeneTargets_v2_1235', 'drugName': 'Alfuzosin Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRA1A (ENSG00000120907), ADRA1D (ENSG00000171873), ADRA1B (ENSG00000170214)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 2003, 'maxClinicalTrialPhase': 4, 'drugIsApproved...
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Genetic Target
Q58.420
Q58
How many genes does the drug Rosiptor target and what are they?
The drug Rosiptor is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene INPP5D.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%rosiptor%" OR LOWER(tradeNames_string) LIKE "%ro...
[{'UUID': 'DrugGeneTargets_v2_2977', 'drugName': 'Rosiptor', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'INPP5D (ENSG00000168918)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.1849
Q58
How many genes does the drug Indecainide target and what are they?
There are 10 gene targets for the drug Indecainide: SCN1A, SCN5A, SCN4A, SCN7A, SCN2A, SCN9A, SCN3A, SCN11A, SCN8A, and SCN10A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%indecainide%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_112', 'drugName': 'Indecainide', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SCN1A (ENSG00000144285), SCN5A (ENSG00000183873), SCN4A (ENSG00000007314), SCN7A (ENSG00000136546), SCN2A (ENSG00000136531), SCN9A (ENSG00000169432), SCN3A (ENSG00000153253), SCN11A (ENSG000...
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Genetic Target
Q58.1920
Q58
How many genes does the drug Mestranol target and what are they?
ESR1 is the only gene target of drug Mestranol.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%mestranol%" OR LOWER(tradeNames_string) LIKE "%m...
[{'UUID': 'DrugGeneTargets_v2_1659', 'drugName': 'Mestranol', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ESR1 (ENSG00000091831)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1961, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1099
Q58
How many genes does the drug Formoterol Fumarate target and what are they?
ADRB2 is the only gene target of drug Formoterol Fumarate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%formoterol fumarate%" OR LOWER(tradeNames_string...
[{'UUID': 'DrugGeneTargets_v2_3747', 'drugName': 'Formoterol Fumarate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRB2 (ENSG00000169252)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2001, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.845
Q58
How many genes does the drug Varenicline Tartrate target and what are they?
There are 2 gene targets for the drug Varenicline Tartrate: CHRNB2 and CHRNA4.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%varenicline tartrate%" OR LOWER(tradeNames_strin...
[{'UUID': 'DrugGeneTargets_v2_259', 'drugName': 'Varenicline Tartrate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CHRNB2 (ENSG00000160716), CHRNA4 (ENSG00000101204)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2006, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.68
Q58
How many genes does the drug Mk-4280 target and what are they?
The drug Mk-4280 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene LAG3.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%mk-4280%" OR LOWER(tradeNames_string) LIKE "%mk-...
[{'UUID': 'DrugGeneTargets_v2_1383', 'drugName': 'Mk-4280', 'drugMolecularType': 'Unknown', 'newLinkedTargets_string': 'LAG3 (ENSG00000089692)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.1698
Q58
How many genes does the drug Potassium Oxybate target and what are they?
There are 2 gene targets for the drug Potassium Oxybate: GABBR1 and GABBR2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%potassium oxybate%" OR LOWER(tradeNames_string) ...
[{'UUID': 'DrugGeneTargets_v2_2573', 'drugName': 'Potassium Oxybate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GABBR1 (ENSG00000204681), GABBR2 (ENSG00000136928)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2020, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1733
Q58
How many genes does the drug Hydromorphone target and what are they?
OPRM1 is the only gene target of drug Hydromorphone.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%hydromorphone%" OR LOWER(tradeNames_string) LIKE...
[{'UUID': 'DrugGeneTargets_v2_245', 'drugName': 'Morphine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'OPRM1 (ENSG00000112038)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1984, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_3034', 'drugName': 'Hydromorph...
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Genetic Target
Q58.380
Q58
How many genes does the drug Osilodrostat Phosphate target and what are they?
CYP11B1 is the only gene target of drug Osilodrostat Phosphate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%osilodrostat phosphate%" OR LOWER(tradeNames_str...
[{'UUID': 'DrugGeneTargets_v2_5216', 'drugName': 'Osilodrostat Phosphate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CYP11B1 (ENSG00000160882)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2020, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.240
Q58
How many genes does the drug Thioguanine target and what are they?
There are 2 gene targets for the drug Thioguanine: IMPDH1 and IMPDH2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%thioguanine%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_5258', 'drugName': 'Thioguanine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'IMPDH1 (ENSG00000106348), IMPDH2 (ENSG00000178035)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1966, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.257
Q58
How many genes does the drug Abobotulinumtoxina target and what are they?
SNAP25 is the only gene target of drug Abobotulinumtoxina.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%abobotulinumtoxina%" OR LOWER(tradeNames_string)...
[{'UUID': 'DrugGeneTargets_v2_5684', 'drugName': 'Abobotulinumtoxina', 'drugMolecularType': 'Unknown', 'newLinkedTargets_string': 'SNAP25 (ENSG00000132639)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2009, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1032
Q58
How many genes does the drug Indacaterol Maleate target and what are they?
ADRB2 is the only gene target of drug Indacaterol Maleate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%indacaterol maleate%" OR LOWER(tradeNames_string...
[{'UUID': 'DrugGeneTargets_v2_3427', 'drugName': 'Indacaterol Maleate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRB2 (ENSG00000169252)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2011, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.30
Q58
How many genes does the drug Lixisenatide target and what are they?
GLP1R is the only gene target of drug Lixisenatide.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%lixisenatide%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_5357', 'drugName': 'Lixisenatide', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'GLP1R (ENSG00000112164)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2016, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.293
Q58
How many genes does the drug Daridorexant Hydrochloride target and what are they?
There are 2 gene targets for the drug Daridorexant Hydrochloride: HCRTR2 and HCRTR1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%daridorexant hydrochloride%" OR LOWER(tradeNames...
[{'UUID': 'DrugGeneTargets_v2_5696', 'drugName': 'Daridorexant Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HCRTR2 (ENSG00000137252), HCRTR1 (ENSG00000121764)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2022, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'Dru...
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Genetic Target
Q58.1886
Q58
How many genes does the drug Cedelizumab target and what are they?
The drug Cedelizumab is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene CD4.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%cedelizumab%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_2501', 'drugName': 'Cedelizumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'CD4 (ENSG00000010610)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drugIsApproved': False}]
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Genetic Target
Q58.1823
Q58
How many genes does the drug Fremanezumab target and what are they?
There are 2 gene targets for the drug Fremanezumab: CALCA and CALCB.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%fremanezumab%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_5545', 'drugName': 'Fremanezumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'CALCA (ENSG00000110680), CALCB (ENSG00000175868)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2018, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.620
Q58
How many genes does the drug Flurazepam Hydrochloride target and what are they?
There are 16 gene targets for the drug Flurazepam Hydrochloride: GABRA1, GABRB2, GABRG2, GABRB3, GABRA4, GABRG3, GABRQ, GABRA3, GABRP, GABRD, GABRG1, GABRB1, GABRE, GABRA2, GABRA5, and GABRA6.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%flurazepam hydrochloride%" OR LOWER(tradeNames_s...
[{'UUID': 'DrugGeneTargets_v2_653', 'drugName': 'Flurazepam Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG0000026808...
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Genetic Target
Q58.1667
Q58
How many genes does the drug Retifanlimab target and what are they?
The drug Retifanlimab is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene PDCD1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%retifanlimab%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_178', 'drugName': 'Retifanlimab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'PDCD1 (ENSG00000188389)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.850
Q58
How many genes does the drug Esomeprazole Magnesium target and what are they?
There are 2 gene targets for the drug Esomeprazole Magnesium: ATP4A and ATP4B.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%esomeprazole magnesium%" OR LOWER(tradeNames_str...
[{'UUID': 'DrugGeneTargets_v2_4440', 'drugName': 'Esomeprazole Magnesium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ATP4A (ENSG00000105675), ATP4B (ENSG00000186009)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2001, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.215
Q58
How many genes does the drug Benzbromarone target and what are they?
SLC22A12 is the only gene target of drug Benzbromarone.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%benzbromarone%" OR LOWER(tradeNames_string) LIKE...
[{'UUID': 'DrugGeneTargets_v2_3284', 'drugName': 'Benzbromarone', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SLC22A12 (ENSG00000197891)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.524
Q58
How many genes does the drug Eluxadoline target and what are they?
OPRM1 is the only gene target of drug Eluxadoline.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%eluxadoline%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_6255', 'drugName': 'Eluxadoline', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'OPRM1 (ENSG00000112038)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2015, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.477
Q58
How many genes does the drug Tesamorelin Acetate target and what are they?
GHRHR is the only gene target of drug Tesamorelin Acetate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tesamorelin acetate%" OR LOWER(tradeNames_string...
[{'UUID': 'DrugGeneTargets_v2_4100', 'drugName': 'Tesamorelin Acetate', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'GHRHR (ENSG00000106128)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2010, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1327
Q58
How many genes does the drug Neostigmine target and what are they?
ACHE is the only gene target of drug Neostigmine.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%neostigmine%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_6228', 'drugName': 'Neostigmine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ACHE (ENSG00000087085)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2013, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_1766', 'drugName': 'Neostig...
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Genetic Target
Q58.1433
Q58
How many genes does the drug Oxandrolone target and what are they?
AR is the only gene target of drug Oxandrolone.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%oxandrolone%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_3386', 'drugName': 'Oxandrolone', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'AR (ENSG00000169083)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1964, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_2216', 'drugName': 'Methyltes...
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Genetic Target
Q58.123
Q58
How many genes does the drug Tamsulosin Hydrochloride target and what are they?
There are 3 gene targets for the drug Tamsulosin Hydrochloride: ADRA1A, ADRA1D, and ADRA1B.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tamsulosin hydrochloride%" OR LOWER(tradeNames_s...
[{'UUID': 'DrugGeneTargets_v2_5784', 'drugName': 'Tamsulosin Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRA1A (ENSG00000120907), ADRA1D (ENSG00000171873), ADRA1B (ENSG00000170214)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 1997, 'maxClinicalTrialPhase': 4, 'drugIsApprove...
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Genetic Target
Q58.1351
Q58
How many genes does the drug Cp-195543 target and what are they?
The drug Cp-195543 is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 2 genes: LTB4R2 and LTB4R.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%cp-195543%" OR LOWER(tradeNames_string) LIKE "%c...
[{'UUID': 'DrugGeneTargets_v2_193', 'drugName': 'Cp-195543', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'LTB4R2 (ENSG00000213906), LTB4R (ENSG00000213903)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1942
Q58
How many genes does the drug Gataparsen target and what are they?
The drug Gataparsen is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene BIRC5.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%gataparsen%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_3583', 'drugName': 'Gataparsen', 'drugMolecularType': 'Oligonucleotide', 'newLinkedTargets_string': 'BIRC5 (ENSG00000089685)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1371
Q58
How many genes does the drug Lomitapide Mesylate target and what are they?
There are 2 gene targets for the drug Lomitapide Mesylate: MTTP and P4HB.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%lomitapide mesylate%" OR LOWER(tradeNames_string...
[{'UUID': 'DrugGeneTargets_v2_3058', 'drugName': 'Lomitapide Mesylate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'MTTP (ENSG00000138823), P4HB (ENSG00000185624)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2012, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1171
Q58
How many genes does the drug Safinamide target and what are they?
MAOB is the only gene target of drug Safinamide.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%safinamide%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_4183', 'drugName': 'Safinamide', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'MAOB (ENSG00000069535)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2017, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_1874', 'drugName': 'Safinami...
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Genetic Target
Q58.138
Q58
How many genes does the drug S-777469 target and what are they?
The drug S-777469 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene CNR2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%s-777469%" OR LOWER(tradeNames_string) LIKE "%s-...
[{'UUID': 'DrugGeneTargets_v2_678', 'drugName': 'S-777469', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CNR2 (ENSG00000188822)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1134
Q58
How many genes does the drug Sr-13668 target and what are they?
The drug Sr-13668 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene AKT1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%sr-13668%" OR LOWER(tradeNames_string) LIKE "%sr...
[{'UUID': 'DrugGeneTargets_v2_2050', 'drugName': 'Sr-13668', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'AKT1 (ENSG00000142208)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drugIsApproved': False}]
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Genetic Target
Q58.1874
Q58
How many genes does the drug Olanzapine Pamoate target and what are they?
There are 5 gene targets for the drug Olanzapine Pamoate: HTR2C, HTR2A, DRD2, DRD3, and DRD4.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%olanzapine pamoate%" OR LOWER(tradeNames_string)...
[{'UUID': 'DrugGeneTargets_v2_1529', 'drugName': 'Olanzapine Pamoate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HTR2C (ENSG00000147246), HTR2A (ENSG00000102468), DRD2 (ENSG00000149295), DRD3 (ENSG00000151577), DRD4 (ENSG00000069696)', 'numberLinkedTargets': 5, 'yearOfFirstApproval': 2009, 'max...
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Genetic Target
Q58.1241
Q58
How many genes does the drug Lofexidine Hydrochloride target and what are they?
There are 3 gene targets for the drug Lofexidine Hydrochloride: ADRA2A, ADRA2C, and ADRA2B.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%lofexidine hydrochloride%" OR LOWER(tradeNames_s...
[{'UUID': 'DrugGeneTargets_v2_3056', 'drugName': 'Lofexidine Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRA2A (ENSG00000150594), ADRA2C (ENSG00000184160), ADRA2B (ENSG00000274286)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 2018, 'maxClinicalTrialPhase': 4, 'drugIsApprove...
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Genetic Target
Q58.1338
Q58
How many genes does the drug Diclofenac Epolamine target and what are they?
There are 2 gene targets for the drug Diclofenac Epolamine: PTGS2 and PTGS1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%diclofenac epolamine%" OR LOWER(tradeNames_strin...
[{'UUID': 'DrugGeneTargets_v2_3087', 'drugName': 'Diclofenac Epolamine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PTGS2 (ENSG00000073756), PTGS1 (ENSG00000095303)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2007, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.958
Q58
How many genes does the drug Lapatinib Ditosylate target and what are they?
There are 2 gene targets for the drug Lapatinib Ditosylate: EGFR and ERBB2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%lapatinib ditosylate%" OR LOWER(tradeNames_strin...
[{'UUID': 'DrugGeneTargets_v2_2160', 'drugName': 'Lapatinib Ditosylate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'EGFR (ENSG00000146648), ERBB2 (ENSG00000141736)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2007, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTarg...
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Q58.929
Q58
How many genes does the drug Bretylium Tosylate target and what are they?
SLC6A2 is the only gene target of drug Bretylium Tosylate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%bretylium tosylate%" OR LOWER(tradeNames_string)...
[{'UUID': 'DrugGeneTargets_v2_904', 'drugName': 'Bretylium Tosylate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SLC6A2 (ENSG00000103546)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1986, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.112
Q58
How many genes does the drug Phenmetrazine Hydrochloride target and what are they?
There are 2 gene targets for the drug Phenmetrazine Hydrochloride: SLC6A3 and SLC6A2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%phenmetrazine hydrochloride%" OR LOWER(tradeName...
[{'UUID': 'DrugGeneTargets_v2_4238', 'drugName': 'Phenmetrazine Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SLC6A3 (ENSG00000142319), SLC6A2 (ENSG00000103546)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1982, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'Dr...
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Genetic Target
Q58.1240
Q58
How many genes does the drug Alosetron target and what are they?
HTR3A is the only gene target of drug Alosetron.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%alosetron%" OR LOWER(tradeNames_string) LIKE "%a...
[{'UUID': 'DrugGeneTargets_v2_4889', 'drugName': 'Alosetron', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HTR3A (ENSG00000166736)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2000, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_5986', 'drugName': 'Alosetro...
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Genetic Target
Q58.1921
Q58
How many genes does the drug Hydrocortisone target and what are they?
NR3C1 is the only gene target of drug Hydrocortisone.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%hydrocortisone%" OR LOWER(tradeNames_string) LIK...
[{'UUID': 'DrugGeneTargets_v2_2255', 'drugName': 'Prednisone', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'NR3C1 (ENSG00000113580)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1955, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_5998', 'drugName': 'Hydroco...
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Genetic Target
Q58.1963
Q58
How many genes does the drug Propranolol Hydrochloride target and what are they?
There are 2 gene targets for the drug Propranolol Hydrochloride: ADRB2 and ADRB1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%propranolol hydrochloride%" OR LOWER(tradeNames_...
[{'UUID': 'DrugGeneTargets_v2_4718', 'drugName': 'Propranolol Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRB2 (ENSG00000169252), ADRB1 (ENSG00000043591)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1967, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGe...
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Genetic Target
Q58.214
Q58
How many genes does the drug Levocabastine Hydrochloride target and what are they?
HRH1 is the only gene target of drug Levocabastine Hydrochloride.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%levocabastine hydrochloride%" OR LOWER(tradeName...
[{'UUID': 'DrugGeneTargets_v2_674', 'drugName': 'Levocabastine Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HRH1 (ENSG00000196639)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1993, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.999
Q58
How many genes does the drug Rilonacept target and what are they?
IL1B is the only gene target of drug Rilonacept.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%rilonacept%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_3681', 'drugName': 'Rilonacept', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'IL1B (ENSG00000125538)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2008, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1269
Q58
How many genes does the drug Carbetapentane Citrate target and what are they?
SIGMAR1 is the only gene target of drug Carbetapentane Citrate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%carbetapentane citrate%" OR LOWER(tradeNames_str...
[{'UUID': 'DrugGeneTargets_v2_5379', 'drugName': 'Carbetapentane Citrate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SIGMAR1 (ENSG00000147955)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.592
Q58
How many genes does the drug Ziprasidone Mesylate target and what are they?
There are 3 gene targets for the drug Ziprasidone Mesylate: HTR2A, DRD2, and HTR2C.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ziprasidone mesylate%" OR LOWER(tradeNames_strin...
[{'UUID': 'DrugGeneTargets_v2_4286', 'drugName': 'Ziprasidone Mesylate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HTR2A (ENSG00000102468), DRD2 (ENSG00000149295), HTR2C (ENSG00000147246)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 2002, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True...
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Genetic Target
Q58.1391
Q58
How many genes does the drug Thalidomide target and what are they?
There are 4 gene targets for the drug Thalidomide: CRBN, DDB1, CUL4A, and RBX1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%thalidomide%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_64', 'drugName': 'Thalidomide', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CRBN (ENSG00000113851), DDB1 (ENSG00000167986), CUL4A (ENSG00000139842), RBX1 (ENSG00000100387)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 1998, 'maxClinicalTrialPhase': 4, 'drugIsApp...
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Genetic Target
Q58.1450
Q58
How many genes does the drug Vinorelbine Tartrate target and what are they?
There are 15 gene targets for the drug Vinorelbine Tartrate: TUBB4B, TUBB1, TUBA3C, TUBA4A, TUBB3, TUBA1A, TUBB4A, TUBB8, TUBB, TUBA1B, TUBA1C, TUBA3E, TUBB2A, TUBB2B, and TUBB6.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%vinorelbine tartrate%" OR LOWER(tradeNames_strin...
[{'UUID': 'DrugGeneTargets_v2_6364', 'drugName': 'Vinorelbine Tartrate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'TUBB4B (ENSG00000188229), TUBB1 (ENSG00000101162), TUBA3C (ENSG00000198033), TUBA4A (ENSG00000127824), TUBB3 (ENSG00000258947), TUBA1A (ENSG00000167552), TUBB4A (ENSG00000104833), ...
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Genetic Target
Q58.279
Q58
How many genes does the drug Temsirolimus target and what are they?
FKBP1A is the only gene target of drug Temsirolimus.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%temsirolimus%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_5750', 'drugName': 'Temsirolimus', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'FKBP1A (ENSG00000088832)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2007, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1507
Q58
How many genes does the drug Agomelatine target and what are they?
There are 3 gene targets for the drug Agomelatine: MTNR1A, MTNR1B, and HTR2C.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%agomelatine%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_4045', 'drugName': 'Agomelatine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'MTNR1A (ENSG00000168412), MTNR1B (ENSG00000134640), HTR2C (ENSG00000147246)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID...
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Genetic Target
Q58.1328
Q58
How many genes does the drug Rg-7600 target and what are they?
The drug Rg-7600 is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 16 genes: TUBB4B, TUBB1, TUBA3C, TUBA4A, TUBB3, TUBA1A, TUBB4A, TUBB8, TUBB, TUBA1B, TUBA1C, TUBA3E, TUBB2A, TUBB2B, TUBB6, and MSLN.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%rg-7600%" OR LOWER(tradeNames_string) LIKE "%rg-...
[{'UUID': 'DrugGeneTargets_v2_641', 'drugName': 'Rg-7600', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'TUBB4B (ENSG00000188229), TUBB1 (ENSG00000101162), TUBA3C (ENSG00000198033), TUBA4A (ENSG00000127824), TUBB3 (ENSG00000258947), TUBA1A (ENSG00000167552), TUBB4A (ENSG00000104833), TUBB8 (ENSG000002614...
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