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Q58.1571
Q58
How many genes does the drug Amg-820 target and what are they?
The drug Amg-820 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene CSF1R.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%amg-820%" OR LOWER(tradeNames_string) LIKE "%amg...
[{'UUID': 'DrugGeneTargets_v2_681', 'drugName': 'Amg-820', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'CSF1R (ENSG00000182578)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drugIsApproved': False}]
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Q58.1641
Q58
How many genes does the drug Moclobemide target and what are they?
MAOA is the only gene target of drug Moclobemide.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%moclobemide%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_6369', 'drugName': 'Moclobemide', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'MAOA (ENSG00000189221)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1565
Q58
How many genes does the drug Cangrelor Tetrasodium target and what are they?
P2RY12 is the only gene target of drug Cangrelor Tetrasodium.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%cangrelor tetrasodium%" OR LOWER(tradeNames_stri...
[{'UUID': 'DrugGeneTargets_v2_1075', 'drugName': 'Cangrelor Tetrasodium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'P2RY12 (ENSG00000169313)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2015, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.491
Q58
How many genes does the drug Azd-8055 target and what are they?
The drug Azd-8055 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene MTOR.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%azd-8055%" OR LOWER(tradeNames_string) LIKE "%az...
[{'UUID': 'DrugGeneTargets_v2_5914', 'drugName': 'Azd-8055', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'MTOR (ENSG00000198793)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drugIsApproved': False}]
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Genetic Target
Q58.1966
Q58
How many genes does the drug Modafinil target and what are they?
SLC6A3 is the only gene target of drug Modafinil.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%modafinil%" OR LOWER(tradeNames_string) LIKE "%m...
[{'UUID': 'DrugGeneTargets_v2_5145', 'drugName': 'Modafinil', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SLC6A3 (ENSG00000142319)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1998, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_2926', 'drugName': 'Armodaf...
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Q58.1800
Q58
How many genes does the drug Oxymorphone Hydrochloride target and what are they?
There are 3 gene targets for the drug Oxymorphone Hydrochloride: OPRK1, OPRD1, and OPRM1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%oxymorphone hydrochloride%" OR LOWER(tradeNames_...
[{'UUID': 'DrugGeneTargets_v2_4591', 'drugName': 'Oxymorphone Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'OPRK1 (ENSG00000082556), OPRD1 (ENSG00000116329), OPRM1 (ENSG00000112038)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 1959, 'maxClinicalTrialPhase': 4, 'drugIsApproved'...
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Genetic Target
Q58.1330
Q58
How many genes does the drug Midazolam Hydrochloride target and what are they?
There are 16 gene targets for the drug Midazolam Hydrochloride: GABRA1, GABRB2, GABRG2, GABRB3, GABRA4, GABRG3, GABRQ, GABRA3, GABRP, GABRD, GABRG1, GABRB1, GABRE, GABRA2, GABRA5, and GABRA6.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%midazolam hydrochloride%" OR LOWER(tradeNames_st...
[{'UUID': 'DrugGeneTargets_v2_4008', 'drugName': 'Midazolam Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG0000026808...
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Genetic Target
Q58.285
Q58
How many genes does the drug Tolterodine target and what are they?
There are 2 gene targets for the drug Tolterodine: CHRM2 and CHRM3.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tolterodine%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_1507', 'drugName': 'Tolterodine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CHRM2 (ENSG00000181072), CHRM3 (ENSG00000133019)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1998, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_1...
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Genetic Target
Q58.1375
Q58
How many genes does the drug Ranolazine target and what are they?
There are 2 gene targets for the drug Ranolazine: SCN4A and SCN5A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ranolazine%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_6340', 'drugName': 'Ranolazine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SCN4A (ENSG00000007314), SCN5A (ENSG00000183873)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2006, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_63...
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Genetic Target
Q58.221
Q58
How many genes does the drug Topiramate target and what are they?
There are 37 gene targets for the drug Topiramate: GRIK1, GRIK5, GRIK4, GRIK2, GRIK3, CA4, SCN1A, SCN5A, SCN4A, SCN7A, SCN2A, SCN9A, SCN3A, SCN11A, SCN8A, SCN10A, GABRA1, GABRB2, GABRG2, GABRB3, GABRA4, GABRG3, GABRQ, GABRA3, GABRP, GABRD, GABRG1, GABRB1, GABRE, GABRA2, GABRA5, GABRA6, CA2, GRIA4, GRIA3, GRIA2, and GRI...
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%topiramate%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1597', 'drugName': 'Topiramate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GRIK1 (ENSG00000171189), GRIK5 (ENSG00000105737), GRIK4 (ENSG00000149403), GRIK2 (ENSG00000164418), GRIK3 (ENSG00000163873), CA4 (ENSG00000167434), SCN1A (ENSG00000144285), SCN5A (ENSG000001...
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Q58.1931
Q58
How many genes does the drug Aripiprazole Lauroxil target and what are they?
There are 3 gene targets for the drug Aripiprazole Lauroxil: DRD2, HTR2A, and HTR1A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%aripiprazole lauroxil%" OR LOWER(tradeNames_stri...
[{'UUID': 'DrugGeneTargets_v2_4679', 'drugName': 'Aripiprazole Lauroxil', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'DRD2 (ENSG00000149295), HTR2A (ENSG00000102468), HTR1A (ENSG00000178394)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 2015, 'maxClinicalTrialPhase': 4, 'drugIsApproved': Tru...
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Genetic Target
Q58.888
Q58
How many genes does the drug Carmustine target and what are they?
GSR is the only gene target of drug Carmustine.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%carmustine%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_4261', 'drugName': 'Carmustine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GSR (ENSG00000104687)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1977, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1623
Q58
How many genes does the drug Granisetron target and what are they?
HTR3A is the only gene target of drug Granisetron.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%granisetron%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_520', 'drugName': 'Granisetron Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HTR3A (ENSG00000166736)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1993, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_2107', 'drugN...
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Q58.701
Q58
How many genes does the drug Idazoxan target and what are they?
The drug Idazoxan is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 3 genes: ADRA2A, ADRA2C, and ADRA2B.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%idazoxan%" OR LOWER(tradeNames_string) LIKE "%id...
[{'UUID': 'DrugGeneTargets_v2_4192', 'drugName': 'Idazoxan', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRA2A (ENSG00000150594), ADRA2C (ENSG00000184160), ADRA2B (ENSG00000274286)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Q58.61
Q58
How many genes does the drug Losartan target and what are they?
AGTR1 is the only gene target of drug Losartan.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%losartan%" OR LOWER(tradeNames_string) LIKE "%lo...
[{'UUID': 'DrugGeneTargets_v2_1912', 'drugName': 'Losartan Potassium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'AGTR1 (ENSG00000144891)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1995, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_6345', 'drugName': ...
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Q58.843
Q58
How many genes does the drug Hmpl-453 target and what are they?
The drug Hmpl-453 is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 3 genes: FGFR3, FGFR2, and FGFR1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%hmpl-453%" OR LOWER(tradeNames_string) LIKE "%hm...
[{'UUID': 'DrugGeneTargets_v2_4342', 'drugName': 'Hmpl-453', 'drugMolecularType': 'Unknown', 'newLinkedTargets_string': 'FGFR3 (ENSG00000068078), FGFR2 (ENSG00000066468), FGFR1 (ENSG00000077782)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}, {'UUID': 'DrugGen...
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Q58.1356
Q58
How many genes does the drug Selodenoson target and what are they?
The drug Selodenoson is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene ADORA1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%selodenoson%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_1822', 'drugName': 'Selodenoson', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADORA1 (ENSG00000163485)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Q58.76
Q58
How many genes does the drug Insulin Detemir target and what are they?
INSR is the only gene target of drug Insulin Detemir.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%insulin detemir%" OR LOWER(tradeNames_string) LI...
[{'UUID': 'DrugGeneTargets_v2_4168', 'drugName': 'Insulin Detemir', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'INSR (ENSG00000171105)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2005, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.165
Q58
How many genes does the drug Humax-Il15 target and what are they?
The drug Humax-Il15 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene CD38.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%humax-il15%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2244', 'drugName': 'Humax-Il15', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'CD38 (ENSG00000004468)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Q58.576
Q58
How many genes does the drug Phentolamine target and what are they?
There are 6 gene targets for the drug Phentolamine: ADRA1A, ADRA2A, ADRA2C, ADRA1D, ADRA1B, and ADRA2B.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%phentolamine%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_2547', 'drugName': 'Phentolamine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRA1A (ENSG00000120907), ADRA2A (ENSG00000150594), ADRA2C (ENSG00000184160), ADRA1D (ENSG00000171873), ADRA1B (ENSG00000170214), ADRA2B (ENSG00000274286)', 'numberLinkedTargets': 6, 'year...
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Q58.959
Q58
How many genes does the drug Moricizine target and what are they?
There are 10 gene targets for the drug Moricizine: SCN1A, SCN5A, SCN4A, SCN7A, SCN2A, SCN9A, SCN3A, SCN11A, SCN8A, and SCN10A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%moricizine%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_4424', 'drugName': 'Moricizine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SCN1A (ENSG00000144285), SCN5A (ENSG00000183873), SCN4A (ENSG00000007314), SCN7A (ENSG00000136546), SCN2A (ENSG00000136531), SCN9A (ENSG00000169432), SCN3A (ENSG00000153253), SCN11A (ENSG000...
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Q58.1540
Q58
How many genes does the drug Imatinib target and what are they?
There are 4 gene targets for the drug Imatinib: ABL1, PDGFRB, BCR, and KIT.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%imatinib%" OR LOWER(tradeNames_string) LIKE "%im...
[{'UUID': 'DrugGeneTargets_v2_3270', 'drugName': 'Imatinib Mesylate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ABL1 (ENSG00000097007), PDGFRB (ENSG00000113721), KIT (ENSG00000157404), BCR (ENSG00000186716)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 2001, 'maxClinicalTrialPhase': 4, 'dr...
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Q58.1046
Q58
How many genes does the drug Diclofenac Potassium target and what are they?
There are 2 gene targets for the drug Diclofenac Potassium: PTGS2 and PTGS1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%diclofenac potassium%" OR LOWER(tradeNames_strin...
[{'UUID': 'DrugGeneTargets_v2_5263', 'drugName': 'Diclofenac Potassium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PTGS2 (ENSG00000073756), PTGS1 (ENSG00000095303)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1993, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1706
Q58
How many genes does the drug Telotristat Etiprate target and what are they?
There are 2 gene targets for the drug Telotristat Etiprate: TPH2 and TPH1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%telotristat etiprate%" OR LOWER(tradeNames_strin...
[{'UUID': 'DrugGeneTargets_v2_1064', 'drugName': 'Telotristat Etiprate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'TPH2 (ENSG00000139287), TPH1 (ENSG00000129167)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2017, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.513
Q58
How many genes does the drug Diphemanil Methylsulfate target and what are they?
There are 2 gene targets for the drug Diphemanil Methylsulfate: CHRM3 and CHRM1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%diphemanil methylsulfate%" OR LOWER(tradeNames_s...
[{'UUID': 'DrugGeneTargets_v2_1327', 'drugName': 'Diphemanil Methylsulfate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CHRM3 (ENSG00000133019), CHRM1 (ENSG00000168539)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1982, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGen...
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Genetic Target
Q58.46
Q58
How many genes does the drug Tacrine target and what are they?
There are 2 gene targets for the drug Tacrine: BCHE and ACHE.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tacrine%" OR LOWER(tradeNames_string) LIKE "%tac...
[{'UUID': 'DrugGeneTargets_v2_2037', 'drugName': 'Tacrine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'BCHE (ENSG00000114200), ACHE (ENSG00000087085)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1993, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_6243', ...
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Genetic Target
Q58.946
Q58
How many genes does the drug As-703988 target and what are they?
The drug As-703988 is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 2 genes: MAP2K2 and MAP2K1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%as-703988%" OR LOWER(tradeNames_string) LIKE "%a...
[{'UUID': 'DrugGeneTargets_v2_2441', 'drugName': 'As-703988', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'MAP2K2 (ENSG00000126934), MAP2K1 (ENSG00000169032)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 1, 'drugIsApproved': False}, {'UUID': 'DrugGeneTargets_v2_244...
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Q58.366
Q58
How many genes does the drug Demecarium target and what are they?
ACHE is the only gene target of drug Demecarium.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%demecarium%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2522', 'drugName': 'Demecarium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ACHE (ENSG00000087085)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1959, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_4088', 'drugName': 'Demecari...
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Genetic Target
Q58.540
Q58
How many genes does the drug Sodelglitazar target and what are they?
The drug Sodelglitazar is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 3 genes: PPARG, PPARA, and PPARD.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%sodelglitazar%" OR LOWER(tradeNames_string) LIKE...
[{'UUID': 'DrugGeneTargets_v2_5445', 'drugName': 'Sodelglitazar', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PPARG (ENSG00000132170), PPARA (ENSG00000186951), PPARD (ENSG00000112033)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.79
Q58
How many genes does the drug Pyridostigmine target and what are they?
ACHE is the only gene target of drug Pyridostigmine.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%pyridostigmine%" OR LOWER(tradeNames_string) LIK...
[{'UUID': 'DrugGeneTargets_v2_516', 'drugName': 'Pyridostigmine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ACHE (ENSG00000087085)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1955, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_5554', 'drugName': 'Pyrid...
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Genetic Target
Q58.1917
Q58
How many genes does the drug Galcanezumab target and what are they?
There are 2 gene targets for the drug Galcanezumab: CALCA and CALCB.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%galcanezumab%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_1901', 'drugName': 'Galcanezumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'CALCA (ENSG00000110680), CALCB (ENSG00000175868)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2018, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1416
Q58
How many genes does the drug Osimertinib target and what are they?
EGFR is the only gene target of drug Osimertinib.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%osimertinib%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_5692', 'drugName': 'Osimertinib', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'EGFR (ENSG00000146648)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2015, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_649', 'drugName': 'Osimerti...
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Genetic Target
Q58.586
Q58
How many genes does the drug Angiotensin Ii target and what are they?
AGTR1 is the only gene target of drug Angiotensin Ii.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%angiotensin ii%" OR LOWER(tradeNames_string) LIK...
[{'UUID': 'DrugGeneTargets_v2_3311', 'drugName': 'Angiotensin Ii', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'AGTR1 (ENSG00000144891)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2017, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_3664', 'drugName': 'Angiotensi...
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Genetic Target
Q58.1795
Q58
How many genes does the drug Osi-632 target and what are they?
The drug Osi-632 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene KDR.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%osi-632%" OR LOWER(tradeNames_string) LIKE "%osi...
[{'UUID': 'DrugGeneTargets_v2_2437', 'drugName': 'Osi-632', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'KDR (ENSG00000128052)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.771
Q58
How many genes does the drug Bosentan target and what are they?
There are 2 gene targets for the drug Bosentan: EDNRB and EDNRA.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%bosentan%" OR LOWER(tradeNames_string) LIKE "%bo...
[{'UUID': 'DrugGeneTargets_v2_379', 'drugName': 'Bosentan', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'EDNRB (ENSG00000136160), EDNRA (ENSG00000151617)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2001, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.371
Q58
How many genes does the drug Tregalizumab target and what are they?
The drug Tregalizumab is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene CD4.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%tregalizumab%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_2022', 'drugName': 'Tregalizumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'CD4 (ENSG00000010610)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.809
Q58
How many genes does the drug Benzphetamine Hydrochloride target and what are they?
There are 2 gene targets for the drug Benzphetamine Hydrochloride: SLC6A2 and SLC18A2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%benzphetamine hydrochloride%" OR LOWER(tradeName...
[{'UUID': 'DrugGeneTargets_v2_167', 'drugName': 'Benzphetamine Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SLC6A2 (ENSG00000103546), SLC18A2 (ENSG00000165646)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1960, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'Dr...
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Genetic Target
Q58.31
Q58
How many genes does the drug Desipramine Hydrochloride target and what are they?
SLC6A2 is the only gene target of drug Desipramine Hydrochloride.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%desipramine hydrochloride%" OR LOWER(tradeNames_...
[{'UUID': 'DrugGeneTargets_v2_3926', 'drugName': 'Desipramine Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SLC6A2 (ENSG00000103546)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1964, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1960
Q58
How many genes does the drug Dibucaine target and what are they?
There are 2 gene targets for the drug Dibucaine: SCN5A and SCN10A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%dibucaine%" OR LOWER(tradeNames_string) LIKE "%d...
[{'UUID': 'DrugGeneTargets_v2_1657', 'drugName': 'Dibucaine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SCN5A (ENSG00000183873), SCN10A (ENSG00000185313)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1982, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_16...
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Genetic Target
Q58.1742
Q58
How many genes does the drug Ozanimod Hydrochloride target and what are they?
S1PR1 is the only gene target of drug Ozanimod Hydrochloride.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ozanimod hydrochloride%" OR LOWER(tradeNames_str...
[{'UUID': 'DrugGeneTargets_v2_5399', 'drugName': 'Ozanimod Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'S1PR1 (ENSG00000170989)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2020, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1577
Q58
How many genes does the drug Esflurbiprofen target and what are they?
The drug Esflurbiprofen is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 2 genes: PTGS2 and PTGS1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%esflurbiprofen%" OR LOWER(tradeNames_string) LIK...
[{'UUID': 'DrugGeneTargets_v2_5008', 'drugName': 'Esflurbiprofen', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PTGS2 (ENSG00000073756), PTGS1 (ENSG00000095303)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.794
Q58
How many genes does the drug Hydroxyamphetamine Hydrobromide target and what are they?
There are 9 gene targets for the drug Hydroxyamphetamine Hydrobromide: ADRA1A, ADRA2A, ADRB1, ADRB2, ADRA2C, ADRA1D, ADRA1B, ADRA2B, and ADRB3.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%hydroxyamphetamine hydrobromide%" OR LOWER(trade...
[{'UUID': 'DrugGeneTargets_v2_2950', 'drugName': 'Hydroxyamphetamine Hydrobromide', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRA1A (ENSG00000120907), ADRA2A (ENSG00000150594), ADRB1 (ENSG00000043591), ADRB2 (ENSG00000169252), ADRA2C (ENSG00000184160), ADRA1D (ENSG00000171873), ADRA1B (ENSG000...
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Genetic Target
Q58.1249
Q58
How many genes does the drug Levobupivacaine Hydrochloride target and what are they?
SCN4A is the only gene target of drug Levobupivacaine Hydrochloride.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%levobupivacaine hydrochloride%" OR LOWER(tradeNa...
[{'UUID': 'DrugGeneTargets_v2_4768', 'drugName': 'Levobupivacaine Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SCN4A (ENSG00000007314)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1999, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.501
Q58
How many genes does the drug Candesartan target and what are they?
The drug Candesartan is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene AGTR1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%candesartan%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_2579', 'drugName': 'Candesartan Cilexetil', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'AGTR1 (ENSG00000144891)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1998, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_3868', 'drugName...
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Genetic Target
Q58.1551
Q58
How many genes does the drug Probenecid target and what are they?
There are 3 gene targets for the drug Probenecid: SLC22A8, SLC22A6, and SLC22A11.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%probenecid%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_1876', 'drugName': 'Probenecid', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SLC22A8 (ENSG00000149452), SLC22A6 (ENSG00000197901), SLC22A11 (ENSG00000168065)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 1951, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True},...
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Genetic Target
Q58.1568
Q58
How many genes does the drug Methylnaltrexone Bromide target and what are they?
OPRM1 is the only gene target of drug Methylnaltrexone Bromide.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%methylnaltrexone bromide%" OR LOWER(tradeNames_s...
[{'UUID': 'DrugGeneTargets_v2_2413', 'drugName': 'Methylnaltrexone Bromide', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'OPRM1 (ENSG00000112038)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2008, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.991
Q58
How many genes does the drug Doxorubicin Hydrochloride target and what are they?
TOP2A is the only gene target of drug Doxorubicin Hydrochloride.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%doxorubicin hydrochloride%" OR LOWER(tradeNames_...
[{'UUID': 'DrugGeneTargets_v2_4222', 'drugName': 'Doxorubicin Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'TOP2A (ENSG00000131747)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1974, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1574
Q58
How many genes does the drug Sildenafil target and what are they?
PDE5A is the only gene target of drug Sildenafil.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%sildenafil%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_4134', 'drugName': 'Sildenafil Citrate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PDE5A (ENSG00000138735)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1998, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_5817', 'drugName': ...
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Genetic Target
Q58.45
Q58
How many genes does the drug Otamixaban target and what are they?
The drug Otamixaban is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene F10.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%otamixaban%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_3113', 'drugName': 'Otamixaban', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'F10 (ENSG00000126218)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.1608
Q58
How many genes does the drug Milveterol target and what are they?
The drug Milveterol is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene ADRB2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%milveterol%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2733', 'drugName': 'Milveterol', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRB2 (ENSG00000169252)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.171
Q58
How many genes does the drug Eplerenone target and what are they?
NR3C2 is the only gene target of drug Eplerenone.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%eplerenone%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_4937', 'drugName': 'Eplerenone', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'NR3C2 (ENSG00000151623)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2002, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.307
Q58
How many genes does the drug Nitroprusside target and what are they?
There are 4 gene targets for the drug Nitroprusside: GUCY1B1, GUCY1B2, GUCY1A2, and GUCY1A1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%nitroprusside%" OR LOWER(tradeNames_string) LIKE...
[{'UUID': 'DrugGeneTargets_v2_1208', 'drugName': 'Nitroprusside', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GUCY1B1 (ENSG00000061918), GUCY1B2 (ENSG00000123201), GUCY1A2 (ENSG00000152402), GUCY1A1 (ENSG00000164116)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 1981, 'maxClinicalTrialPhase'...
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Genetic Target
Q58.1957
Q58
How many genes does the drug Ticlopidine target and what are they?
P2RY12 is the only gene target of drug Ticlopidine.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ticlopidine%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_3795', 'drugName': 'Ticlopidine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'P2RY12 (ENSG00000169313)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1991, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_1201', 'drugName': 'Ticlo...
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Genetic Target
Q58.1105
Q58
How many genes does the drug Metolazone target and what are they?
SLC12A3 is the only gene target of drug Metolazone.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%metolazone%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_4829', 'drugName': 'Metolazone', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SLC12A3 (ENSG00000070915)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1973, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1925
Q58
How many genes does the drug Cocaine Hydrochloride target and what are they?
There are 10 gene targets for the drug Cocaine Hydrochloride: SCN1A, SCN5A, SCN4A, SCN7A, SCN2A, SCN9A, SCN3A, SCN11A, SCN8A, and SCN10A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%cocaine hydrochloride%" OR LOWER(tradeNames_stri...
[{'UUID': 'DrugGeneTargets_v2_3417', 'drugName': 'Cocaine Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SCN1A (ENSG00000144285), SCN5A (ENSG00000183873), SCN4A (ENSG00000007314), SCN7A (ENSG00000136546), SCN2A (ENSG00000136531), SCN9A (ENSG00000169432), SCN3A (ENSG00000153253), SCN1...
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Genetic Target
Q58.1038
Q58
How many genes does the drug Moxonidine target and what are they?
NISCH is the only gene target of drug Moxonidine.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%moxonidine%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2347', 'drugName': 'Moxonidine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'NISCH (ENSG00000010322)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.658
Q58
How many genes does the drug Torcetrapib target and what are they?
The drug Torcetrapib is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene CETP.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%torcetrapib%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_1801', 'drugName': 'Torcetrapib', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CETP (ENSG00000087237)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.373
Q58
How many genes does the drug Apazone target and what are they?
There are 2 gene targets for the drug Apazone: PTGS2 and PTGS1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%apazone%" OR LOWER(tradeNames_string) LIKE "%apa...
[{'UUID': 'DrugGeneTargets_v2_3917', 'drugName': 'Apazone', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PTGS2 (ENSG00000073756), PTGS1 (ENSG00000095303)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1661
Q58
How many genes does the drug Bunazosin target and what are they?
The drug Bunazosin is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 3 genes: ADRA1A, ADRA1D, and ADRA1B.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%bunazosin%" OR LOWER(tradeNames_string) LIKE "%b...
[{'UUID': 'DrugGeneTargets_v2_4492', 'drugName': 'Bunazosin', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRA1A (ENSG00000120907), ADRA1D (ENSG00000171873), ADRA1B (ENSG00000170214)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.1513
Q58
How many genes does the drug Deucravacitinib target and what are they?
TYK2 is the only gene target of drug Deucravacitinib.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%deucravacitinib%" OR LOWER(tradeNames_string) LI...
[{'UUID': 'DrugGeneTargets_v2_1979', 'drugName': 'Deucravacitinib', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'TYK2 (ENSG00000105397)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2022, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_6268', 'drugName': 'Deu...
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Genetic Target
Q58.778
Q58
How many genes does the drug Mazindol target and what are they?
There are 3 gene targets for the drug Mazindol: SLC6A4, SLC6A3, and SLC6A2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%mazindol%" OR LOWER(tradeNames_string) LIKE "%ma...
[{'UUID': 'DrugGeneTargets_v2_5589', 'drugName': 'Mazindol', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SLC6A4 (ENSG00000108576), SLC6A3 (ENSG00000142319), SLC6A2 (ENSG00000103546)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 1973, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.328
Q58
How many genes does the drug Alogliptin Benzoate target and what are they?
DPP4 is the only gene target of drug Alogliptin Benzoate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%alogliptin benzoate%" OR LOWER(tradeNames_string...
[{'UUID': 'DrugGeneTargets_v2_2469', 'drugName': 'Alogliptin Benzoate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'DPP4 (ENSG00000197635)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2013, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1988
Q58
How many genes does the drug Sodium Nitroprusside target and what are they?
There are 4 gene targets for the drug Sodium Nitroprusside: GUCY1B1, GUCY1B2, GUCY1A2, and GUCY1A1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%sodium nitroprusside%" OR LOWER(tradeNames_strin...
[{'UUID': 'DrugGeneTargets_v2_3464', 'drugName': 'Sodium Nitroprusside', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GUCY1B1 (ENSG00000061918), GUCY1B2 (ENSG00000123201), GUCY1A2 (ENSG00000152402), GUCY1A1 (ENSG00000164116)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 1981, 'maxClinicalTria...
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Genetic Target
Q58.1924
Q58
How many genes does the drug Prednisolone Acetate target and what are they?
NR3C1 is the only gene target of drug Prednisolone Acetate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%prednisolone acetate%" OR LOWER(tradeNames_strin...
[{'UUID': 'DrugGeneTargets_v2_5344', 'drugName': 'Prednisolone Acetate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'NR3C1 (ENSG00000113580)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1955, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_675', 'drugName':...
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Genetic Target
Q58.931
Q58
How many genes does the drug Bromodiphenhydramine target and what are they?
HRH1 is the only gene target of drug Bromodiphenhydramine.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%bromodiphenhydramine%" OR LOWER(tradeNames_strin...
[{'UUID': 'DrugGeneTargets_v2_4863', 'drugName': 'Bromodiphenhydramine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HRH1 (ENSG00000196639)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1954, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_1015', 'drugName':...
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Genetic Target
Q58.188
Q58
How many genes does the drug Ralimetinib target and what are they?
The drug Ralimetinib is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene MAPK14.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ralimetinib%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_5096', 'drugName': 'Ralimetinib', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'MAPK14 (ENSG00000112062)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1595
Q58
How many genes does the drug Apilimod Mesylate target and what are they?
The drug Apilimod Mesylate is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene PIKFYVE.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%apilimod mesylate%" OR LOWER(tradeNames_string) ...
[{'UUID': 'DrugGeneTargets_v2_1384', 'drugName': 'Apilimod Mesylate', 'drugMolecularType': 'Unknown', 'newLinkedTargets_string': 'PIKFYVE (ENSG00000115020)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.772
Q58
How many genes does the drug Prasugrel target and what are they?
P2RY12 is the only gene target of drug Prasugrel.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%prasugrel%" OR LOWER(tradeNames_string) LIKE "%p...
[{'UUID': 'DrugGeneTargets_v2_2823', 'drugName': 'Prasugrel Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'P2RY12 (ENSG00000169313)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2009, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_3169', 'drugN...
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Genetic Target
Q58.1203
Q58
How many genes does the drug Bexarotene target and what are they?
There are 3 gene targets for the drug Bexarotene: RXRB, RXRG, and RXRA.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%bexarotene%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_3322', 'drugName': 'Bexarotene', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'RXRB (ENSG00000204231), RXRG (ENSG00000143171), RXRA (ENSG00000186350)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 1999, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.500
Q58
How many genes does the drug Reproterol target and what are they?
ADRB2 is the only gene target of drug Reproterol.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%reproterol%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_487', 'drugName': 'Reproterol', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRB2 (ENSG00000169252)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1064
Q58
How many genes does the drug Duloxetine Hydrochloride target and what are they?
There are 2 gene targets for the drug Duloxetine Hydrochloride: SLC6A4 and SLC6A2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%duloxetine hydrochloride%" OR LOWER(tradeNames_s...
[{'UUID': 'DrugGeneTargets_v2_5702', 'drugName': 'Duloxetine Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SLC6A4 (ENSG00000108576), SLC6A2 (ENSG00000103546)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2004, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugG...
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Genetic Target
Q58.1111
Q58
How many genes does the drug Methylprednisolone target and what are they?
NR3C1 is the only gene target of drug Methylprednisolone.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%methylprednisolone%" OR LOWER(tradeNames_string)...
[{'UUID': 'DrugGeneTargets_v2_5705', 'drugName': 'Methylprednisolone Sodium Succinate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'NR3C1 (ENSG00000113580)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1959, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_47...
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Genetic Target
Q58.536
Q58
How many genes does the drug Mk-2461 target and what are they?
The drug Mk-2461 is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene MET.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%mk-2461%" OR LOWER(tradeNames_string) LIKE "%mk-...
[{'UUID': 'DrugGeneTargets_v2_1238', 'drugName': 'Mk-2461', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'MET (ENSG00000105976)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}]
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Genetic Target
Q58.1601
Q58
How many genes does the drug Perindopril Erbumine target and what are they?
ACE is the only gene target of drug Perindopril Erbumine.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%perindopril erbumine%" OR LOWER(tradeNames_strin...
[{'UUID': 'DrugGeneTargets_v2_1718', 'drugName': 'Perindopril Erbumine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ACE (ENSG00000159640)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1993, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.752
Q58
How many genes does the drug Fosphenytoin target and what are they?
There are 10 gene targets for the drug Fosphenytoin: SCN1A, SCN5A, SCN4A, SCN7A, SCN2A, SCN9A, SCN3A, SCN11A, SCN8A, and SCN10A.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%fosphenytoin%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_993', 'drugName': 'Fosphenytoin', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SCN1A (ENSG00000144285), SCN5A (ENSG00000183873), SCN4A (ENSG00000007314), SCN7A (ENSG00000136546), SCN2A (ENSG00000136531), SCN9A (ENSG00000169432), SCN3A (ENSG00000153253), SCN11A (ENSG00...
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Genetic Target
Q58.1933
Q58
How many genes does the drug Cabozantinib target and what are they?
There are 2 gene targets for the drug Cabozantinib: MET and KDR.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%cabozantinib%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_3580', 'drugName': 'Cabozantinib S-Malate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'MET (ENSG00000105976), KDR (ENSG00000128052)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 2012, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTarget...
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Genetic Target
Q58.1367
Q58
How many genes does the drug Itepekimab target and what are they?
The drug Itepekimab is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene IL33.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%itepekimab%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_2908', 'drugName': 'Itepekimab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'IL33 (ENSG00000137033)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.1444
Q58
How many genes does the drug Donepezil target and what are they?
ACHE is the only gene target of drug Donepezil.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%donepezil%" OR LOWER(tradeNames_string) LIKE "%d...
[{'UUID': 'DrugGeneTargets_v2_795', 'drugName': 'Donepezil Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ACHE (ENSG00000087085)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1996, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_4037', 'drugName...
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Genetic Target
Q58.178
Q58
How many genes does the drug Nialamide target and what are they?
There are 2 gene targets for the drug Nialamide: MAOA and MAOB.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%nialamide%" OR LOWER(tradeNames_string) LIKE "%n...
[{'UUID': 'DrugGeneTargets_v2_3121', 'drugName': 'Nialamide', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'MAOA (ENSG00000189221), MAOB (ENSG00000069535)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.470
Q58
How many genes does the drug Dantrolene target and what are they?
There are 2 gene targets for the drug Dantrolene: RYR3 and RYR1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%dantrolene%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_4505', 'drugName': 'Dantrolene Sodium', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'RYR3 (ENSG00000198838), RYR1 (ENSG00000196218)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1974, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_...
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Genetic Target
Q58.1337
Q58
How many genes does the drug Carphenazine target and what are they?
There are 3 gene targets for the drug Carphenazine: HTR2A, HTR2C, and DRD2.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%carphenazine%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_4893', 'drugName': 'Carphenazine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HTR2A (ENSG00000102468), HTR2C (ENSG00000147246), DRD2 (ENSG00000149295)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 1982, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUI...
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Genetic Target
Q58.1611
Q58
How many genes does the drug Meprobamate target and what are they?
There are 16 gene targets for the drug Meprobamate: GABRA1, GABRB2, GABRG2, GABRB3, GABRA4, GABRG3, GABRQ, GABRA3, GABRP, GABRD, GABRG1, GABRB1, GABRE, GABRA2, GABRA5, and GABRA6.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%meprobamate%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_143', 'drugName': 'Meprobamate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089), GABRA3 (E...
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Genetic Target
Q58.126
Q58
How many genes does the drug Orp-101 target and what are they?
The drug Orp-101 is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 2 genes: OPRK1 and OPRM1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%orp-101%" OR LOWER(tradeNames_string) LIKE "%orp...
[{'UUID': 'DrugGeneTargets_v2_1458', 'drugName': 'Orp-101', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'OPRK1 (ENSG00000082556), OPRM1 (ENSG00000112038)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved': False}, {'UUID': 'DrugGeneTargets_v2_1459', ...
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Genetic Target
Q58.355
Q58
How many genes does the drug Ibuprofen target and what are they?
There are 2 gene targets for the drug Ibuprofen: PTGS2 and PTGS1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%ibuprofen%" OR LOWER(tradeNames_string) LIKE "%i...
[{'UUID': 'DrugGeneTargets_v2_3209', 'drugName': 'Ibuprofen', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PTGS2 (ENSG00000073756), PTGS1 (ENSG00000095303)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1974, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_144...
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Genetic Target
Q58.388
Q58
How many genes does the drug Levoketoconazole target and what are they?
There are 4 gene targets for the drug Levoketoconazole: CYP11B1, CYP11B2, CYP17A1, and CYP11A1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%levoketoconazole%" OR LOWER(tradeNames_string) L...
[{'UUID': 'DrugGeneTargets_v2_3930', 'drugName': 'Levoketoconazole', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'CYP11B1 (ENSG00000160882), CYP11B2 (ENSG00000179142), CYP17A1 (ENSG00000148795), CYP11A1 (ENSG00000140459)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 2021, 'maxClinicalTrialPha...
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Q58.1435
Q58
How many genes does the drug Secretin Synthetic Porcine target and what are they?
SCTR is the only gene target of drug Secretin Synthetic Porcine.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%secretin synthetic porcine%" OR LOWER(tradeNames...
[{'UUID': 'DrugGeneTargets_v2_462', 'drugName': 'Secretin Synthetic Porcine', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'SCTR (ENSG00000080293)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2002, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.1007
Q58
How many genes does the drug Almorexant target and what are they?
The drug Almorexant is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 2 genes: HCRTR2 and HCRTR1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%almorexant%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_4454', 'drugName': 'Almorexant', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HCRTR2 (ENSG00000137252), HCRTR1 (ENSG00000121764)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Q58.894
Q58
How many genes does the drug Dapoxetine target and what are they?
SLC6A4 is the only gene target of drug Dapoxetine.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%dapoxetine%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_3188', 'drugName': 'Dapoxetine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'SLC6A4 (ENSG00000108576)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.1495
Q58
How many genes does the drug Brimonidine Tartrate target and what are they?
There are 3 gene targets for the drug Brimonidine Tartrate: ADRA2A, ADRA2C, and ADRA2B.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%brimonidine tartrate%" OR LOWER(tradeNames_strin...
[{'UUID': 'DrugGeneTargets_v2_4923', 'drugName': 'Brimonidine Tartrate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRA2A (ENSG00000150594), ADRA2C (ENSG00000184160), ADRA2B (ENSG00000274286)', 'numberLinkedTargets': 3, 'yearOfFirstApproval': 1996, 'maxClinicalTrialPhase': 4, 'drugIsApproved': ...
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Genetic Target
Q58.335
Q58
How many genes does the drug Nesiritide target and what are they?
NPR1 is the only gene target of drug Nesiritide.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%nesiritide%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_3389', 'drugName': 'Nesiritide', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'NPR1 (ENSG00000169418)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 2001, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.975
Q58
How many genes does the drug Odronextamab target and what are they?
The drug Odronextamab is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 4 genes: CD3E, CD3G, CD3D, and MS4A1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%odronextamab%" OR LOWER(tradeNames_string) LIKE ...
[{'UUID': 'DrugGeneTargets_v2_1602', 'drugName': 'Odronextamab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'CD3E (ENSG00000198851), CD3G (ENSG00000160654), CD3D (ENSG00000167286), MS4A1 (ENSG00000156738)', 'numberLinkedTargets': 4, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 2, 'drugIsApproved'...
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Q58.197
Q58
How many genes does the drug Phenoxybenzamine target and what are they?
There are 6 gene targets for the drug Phenoxybenzamine: ADRA1A, ADRA2A, ADRA2C, ADRA1D, ADRA1B, and ADRA2B.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%phenoxybenzamine%" OR LOWER(tradeNames_string) L...
[{'UUID': 'DrugGeneTargets_v2_5463', 'drugName': 'Phenoxybenzamine', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'ADRA1A (ENSG00000120907), ADRA2A (ENSG00000150594), ADRA2C (ENSG00000184160), ADRA1D (ENSG00000171873), ADRA1B (ENSG00000170214), ADRA2B (ENSG00000274286)', 'numberLinkedTargets': 6, '...
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Genetic Target
Q58.520
Q58
How many genes does the drug Codeine Phosphate target and what are they?
There are 3 gene targets for the drug Codeine Phosphate: OPRK1, OPRD1, and OPRM1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%codeine phosphate%" OR LOWER(tradeNames_string) ...
[{'UUID': 'DrugGeneTargets_v2_4198', 'drugName': 'Dihydrocodeine Bitartrate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'OPRM1 (ENSG00000112038)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1983, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_1990', 'drug...
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Genetic Target
Q58.459
Q58
How many genes does the drug Rilotumumab target and what are they?
The drug Rilotumumab is not approved by the FDA. However, it is currently undergoing clinical trials and indecated to target the gene HGF.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%rilotumumab%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_1237', 'drugName': 'Rilotumumab', 'drugMolecularType': 'Antibody', 'newLinkedTargets_string': 'HGF (ENSG00000019991)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 3, 'drugIsApproved': False}]
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Genetic Target
Q58.1714
Q58
How many genes does the drug Cosyntropin target and what are they?
MC2R is the only gene target of drug Cosyntropin.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%cosyntropin%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_4137', 'drugName': 'Cosyntropin', 'drugMolecularType': 'Protein', 'newLinkedTargets_string': 'MC2R (ENSG00000185231)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1970, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.326
Q58
How many genes does the drug Pravastatin target and what are they?
HMGCR is the only gene target of drug Pravastatin.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%pravastatin%" OR LOWER(tradeNames_string) LIKE "...
[{'UUID': 'DrugGeneTargets_v2_5677', 'drugName': 'Pravastatin', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'HMGCR (ENSG00000113161)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1991, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}, {'UUID': 'DrugGeneTargets_v2_1605', 'drugName': 'Pravas...
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Genetic Target
Q58.1323
Q58
How many genes does the drug Lorediplon target and what are they?
The drug Lorediplon is not approved by the FDA. However, it is currently undergoing clinical trials and indicated to target 16 genes: GABRA1, GABRB2, GABRG2, GABRB3, GABRA4, GABRG3, GABRQ, GABRA3, GABRP, GABRD, GABRG1, GABRB1, GABRE, GABRA2, GABRA5, and GABRA6.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%lorediplon%" OR LOWER(tradeNames_string) LIKE "%...
[{'UUID': 'DrugGeneTargets_v2_5767', 'drugName': 'Lorediplon', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089), GABRA3 (E...
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Genetic Target
Q58.269
Q58
How many genes does the drug Pargyline Hydrochloride target and what are they?
There are 2 gene targets for the drug Pargyline Hydrochloride: MAOA and MAOB.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%pargyline hydrochloride%" OR LOWER(tradeNames_st...
[{'UUID': 'DrugGeneTargets_v2_1196', 'drugName': 'Pargyline Hydrochloride', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'MAOA (ENSG00000189221), MAOB (ENSG00000069535)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 1982, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Genetic Target
Q58.799
Q58
How many genes does the drug Isoxicam target and what are they?
There are 2 gene targets for the drug Isoxicam: PTGS2 and PTGS1.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%isoxicam%" OR LOWER(tradeNames_string) LIKE "%is...
[{'UUID': 'DrugGeneTargets_v2_1802', 'drugName': 'Isoxicam', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PTGS2 (ENSG00000073756), PTGS1 (ENSG00000095303)', 'numberLinkedTargets': 2, 'yearOfFirstApproval': 0, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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Q58.1432
Q58
How many genes does the drug Milrinone Lactate target and what are they?
PDE3A is the only gene target of drug Milrinone Lactate.
SELECT DISTINCT UUID, drugName, drugMolecularType, newLinkedTargets_string, numberLinkedTargets, yearOfFirstApproval, maxClinicalTrialPhase, drugIsApproved FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE (LOWER(drugName) LIKE "%milrinone lactate%" OR LOWER(tradeNames_string) ...
[{'UUID': 'DrugGeneTargets_v2_3912', 'drugName': 'Milrinone Lactate', 'drugMolecularType': 'Small molecule', 'newLinkedTargets_string': 'PDE3A (ENSG00000172572)', 'numberLinkedTargets': 1, 'yearOfFirstApproval': 1987, 'maxClinicalTrialPhase': 4, 'drugIsApproved': True}]
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