Datasets:

uuid
stringlengths
4
8
template_uuid
stringclasses
40 values
question
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13
193
answer
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29
2.2k
benchmark_query
stringlengths
133
622
execution_results
stringlengths
2
1.14M
query_type
stringclasses
2 values
sql_category
stringclasses
26 values
bio_category
stringclasses
14 values
Q1.1055
Q1
Is PDE6C a druggable gene?
There are currently 2 approved drugs which target PDE6C, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%PDE6C %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6107', 'drugName': 'Dipyridamole', 'drugIsApproved': True, 'newLinkedTargets_string': 'PDE5A (ENSG00000138735), PDE4A (ENSG00000065989), PDE3A (ENSG00000172572), PDE6H (ENSG00000139053), PDE6G (ENSG00000185527), PDE2A (ENSG00000186642), PDE7A (ENSG00000205268), PDE1A (ENSG00000115252), PDE...
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Approval Status, Genetic Target
Q1.79
Q1
Is ASGR1 a druggable gene?
There are currently no approved drugs targeting ASGR1, but there are 2 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%ASGR1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2325', 'drugName': 'Vupanorsen', 'drugIsApproved': False, 'newLinkedTargets_string': 'ANGPTL3 (ENSG00000132855), ASGR1 (ENSG00000141505)', 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_2326', 'drugName': 'Vupanorsen', 'drugIsApproved': False, 'newLinkedTargets_string': 'ANGPTL3...
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Approval Status, Genetic Target
Q1.86
Q1
Is ATP1B3 a druggable gene?
There are currently 5 approved drugs which target ATP1B3, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%ATP1B3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2499', 'drugName': 'Digoxin', 'drugIsApproved': True, 'newLinkedTargets_string': 'ATP1A1 (ENSG00000163399), ATP1B2 (ENSG00000129244), ATP1B1 (ENSG00000143153), ATP1A2 (ENSG00000018625), ATP1B3 (ENSG00000069849), ATP1A3 (ENSG00000105409), ATP1A4 (ENSG00000132681), FXYD2 (ENSG00000137731)', ...
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Approval Status, Genetic Target
Q1.946
Q1
Is NDUFA7 a druggable gene?
There are currently 2 approved drugs which target NDUFA7, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%NDUFA7 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'drugIsApproved': True, 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (EN...
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Approval Status, Genetic Target
Q1.84
Q1
Is ATP1B1 a druggable gene?
There are currently 5 approved drugs which target ATP1B1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%ATP1B1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2499', 'drugName': 'Digoxin', 'drugIsApproved': True, 'newLinkedTargets_string': 'ATP1A1 (ENSG00000163399), ATP1B2 (ENSG00000129244), ATP1B1 (ENSG00000143153), ATP1A2 (ENSG00000018625), ATP1B3 (ENSG00000069849), ATP1A3 (ENSG00000105409), ATP1A4 (ENSG00000132681), FXYD2 (ENSG00000137731)', ...
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Approval Status, Genetic Target
Q1.459
Q1
Is FGA a druggable gene?
There is 1 drug, Fibrinolysin, Human, that targets FGA, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%FGA %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1199', 'drugName': 'Fibrinolysin, Human', 'drugIsApproved': True, 'newLinkedTargets_string': 'FGA (ENSG00000171560), FGB (ENSG00000171564), FGG (ENSG00000171557)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1397', 'drugName': 'Ancrod', 'drugIsApproved': False, 'newLinkedTarg...
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Approval Status, Genetic Target
Q1.947
Q1
Is NDUFA8 a druggable gene?
There are currently 2 approved drugs which target NDUFA8, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%NDUFA8 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'drugIsApproved': True, 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (EN...
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Approval Status, Genetic Target
Q1.681
Q1
Is IL18RAP a druggable gene?
There are currently no approved drugs targeting IL18RAP, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%IL18RAP %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2219', 'drugName': 'Iboctadekin', 'drugIsApproved': False, 'newLinkedTargets_string': 'IL18RAP (ENSG00000115607), IL18R1 (ENSG00000115604)', 'maxClinicalTrialPhase': 2}]
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Approval Status, Genetic Target
Q1.1532
Q1
Is WT1 a druggable gene?
There are currently no approved drugs targeting WT1, but there are 2 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%WT1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_240', 'drugName': 'Galinpepimut-S', 'drugIsApproved': False, 'newLinkedTargets_string': 'WT1 (ENSG00000184937)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_6067', 'drugName': 'Ombipepimut-S', 'drugIsApproved': False, 'newLinkedTargets_string': 'WT1 (ENSG00000184937)', 'maxCl...
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Approval Status, Genetic Target
Q1.1114
Q1
Is PPARD a druggable gene?
There is 1 drug, Bezafibrate, that targets PPARD, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%PPARD %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1564', 'drugName': 'Bezafibrate', 'drugIsApproved': True, 'newLinkedTargets_string': 'PPARG (ENSG00000132170), PPARA (ENSG00000186951), PPARD (ENSG00000112033)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1645', 'drugName': 'Lanifibranor', 'drugIsApproved': False, 'newLinked...
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Approval Status, Genetic Target
Q1.438
Q1
Is F2 a druggable gene?
There are currently 8 approved drugs which target F2, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%F2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1887', 'drugName': 'Metformin Hydrochloride', 'drugIsApproved': True, 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (EN...
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Approval Status, Genetic Target
Q1.775
Q1
Is KCNQ1 a druggable gene?
There are currently 6 approved drugs which target KCNQ1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%KCNQ1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2190', 'drugName': 'Guanidine', 'drugIsApproved': True, 'newLinkedTargets_string': 'KCNQ1 (ENSG00000053918), KCND3 (ENSG00000171385), KCNH2 (ENSG00000055118), KCNA2 (ENSG00000177301), KCNA1 (ENSG00000111262), KCNQ2 (ENSG00000075043), KCNQ3 (ENSG00000184156), KCNA7 (ENSG00000104848), KCNQ5 ...
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Approval Status, Genetic Target
Q1.648
Q1
Is IFNA4 a druggable gene?
There are currently no approved drugs targeting IFNA4, but there are 2 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%IFNA4 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5087', 'drugName': 'Sifalimumab', 'drugIsApproved': False, 'newLinkedTargets_string': 'IFNA6 (ENSG00000120235), IFNA8 (ENSG00000120242), IFNA5 (ENSG00000147873), IFNA10 (ENSG00000186803), IFNA2 (ENSG00000188379), IFNA1 (ENSG00000197919), IFNA13 (ENSG00000233816), IFNA7 (ENSG00000214042), I...
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Approval Status, Genetic Target
Q1.850
Q1
Is MAP3K10 a druggable gene?
There are currently no approved drugs targeting MAP3K10, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%MAP3K10 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6091', 'drugName': 'Cep-1347', 'drugIsApproved': False, 'newLinkedTargets_string': 'MAP3K13 (ENSG00000073803), MAP3K12 (ENSG00000139625), MAP3K10 (ENSG00000130758), MAP3K9 (ENSG00000006432), MAP3K11 (ENSG00000173327)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_6088', 'drugN...
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Approval Status, Genetic Target
Q1.1414
Q1
Is TACSTD2 a druggable gene?
There is 1 drug, Sacituzumab Govitecan, that targets TACSTD2, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%TACSTD2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4818', 'drugName': 'Sacituzumab Govitecan', 'drugIsApproved': True, 'newLinkedTargets_string': 'TACSTD2 (ENSG00000184292), TOP1 (ENSG00000198900)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4819', 'drugName': 'Sacituzumab Govitecan', 'drugIsApproved': True, 'newLinkedTarget...
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Approval Status, Genetic Target
Q1.1223
Q1
Is ROCK1 a druggable gene?
There are currently 4 approved drugs which target ROCK1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%ROCK1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4693', 'drugName': 'Netarsudil Dimesylate', 'drugIsApproved': True, 'newLinkedTargets_string': 'ROCK2 (ENSG00000134318), ROCK1 (ENSG00000067900)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4213', 'drugName': 'Belumosudil', 'drugIsApproved': True, 'newLinkedTargets_string': ...
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Approval Status, Genetic Target
Q1.406
Q1
Is EPCAM a druggable gene?
There is 1 drug, Catumaxomab, that targets EPCAM, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%EPCAM %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2537', 'drugName': 'Catumaxomab', 'drugIsApproved': True, 'newLinkedTargets_string': 'CD3E (ENSG00000198851), CD3G (ENSG00000160654), CD3D (ENSG00000167286), EPCAM (ENSG00000119888)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2538', 'drugName': 'Catumaxomab', 'drugIsApprove...
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Approval Status, Genetic Target
Q1.1336
Q1
Is SCN5A a druggable gene?
There are currently 85 approved drugs which target SCN5A, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%SCN5A %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_718', 'drugName': 'Vernakalant', 'drugIsApproved': True, 'newLinkedTargets_string': 'KCND3 (ENSG00000171385), KCNA5 (ENSG00000130037), KCNJ3 (ENSG00000162989), KCNJ5 (ENSG00000120457), KCNH2 (ENSG00000055118), SCN5A (ENSG00000183873)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets...
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Approval Status, Genetic Target
Q1.1110
Q1
Is POLR2A a druggable gene?
There are currently no approved drugs targeting POLR2A, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%POLR2A %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3830', 'drugName': 'Tas-106', 'drugIsApproved': False, 'newLinkedTargets_string': 'POLR1A (ENSG00000068654), POLR3A (ENSG00000148606), POLR2A (ENSG00000181222)', 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_3831', 'drugName': 'Tas-106', 'drugIsApproved': False, 'newLinkedTarge...
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Approval Status, Genetic Target
Q1.1429
Q1
Is THRA a druggable gene?
There are currently 6 approved drugs which target THRA, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%THRA %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_637', 'drugName': 'Levothyroxine', 'drugIsApproved': True, 'newLinkedTargets_string': 'THRA (ENSG00000126351), THRB (ENSG00000151090)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4914', 'drugName': 'Liothyronine Sodium', 'drugIsApproved': True, 'newLinkedTargets_string': 'TH...
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Approval Status, Genetic Target
Q1.106
Q1
Is BCL2L2 a druggable gene?
There are currently no approved drugs targeting BCL2L2, but there are 3 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%BCL2L2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2962', 'drugName': 'Obatoclax Mesylate', 'drugIsApproved': False, 'newLinkedTargets_string': 'BCL2 (ENSG00000171791), BCL2L1 (ENSG00000171552), MCL1 (ENSG00000143384), BCL2L2-PABPN1 (ENSG00000258643), BCL2L2 (ENSG00000129473), BCL2A1 (ENSG00000140379), BCL2L10 (ENSG00000137875)', 'maxClini...
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Approval Status, Genetic Target
Q1.613
Q1
Is HSPA8 a druggable gene?
There are currently no approved drugs targeting HSPA8, but there are 2 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%HSPA8 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1772', 'drugName': 'Forigerimod', 'drugIsApproved': False, 'newLinkedTargets_string': 'HSPA8 (ENSG00000109971)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_3527', 'drugName': 'Forigerimod Acetate', 'drugIsApproved': False, 'newLinkedTargets_string': 'HSPA8 (ENSG00000109971)'...
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Approval Status, Genetic Target
Q1.1338
Q1
Is SCN8A a druggable gene?
There are currently 78 approved drugs which target SCN8A, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%SCN8A %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1606', 'drugName': 'Chloroprocaine', 'drugIsApproved': True, 'newLinkedTargets_string': 'SCN1A (ENSG00000144285), SCN5A (ENSG00000183873), SCN4A (ENSG00000007314), SCN7A (ENSG00000136546), SCN2A (ENSG00000136531), SCN9A (ENSG00000169432), SCN3A (ENSG00000153253), SCN11A (ENSG00000168356), ...
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Approval Status, Genetic Target
Q1.693
Q1
Is IL2RA a druggable gene?
There are currently 4 approved drugs which target IL2RA, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%IL2RA %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5634', 'drugName': 'Denileukin Diftitox', 'drugIsApproved': True, 'newLinkedTargets_string': 'IL2RA (ENSG00000134460), IL2RG (ENSG00000147168), IL2RB (ENSG00000100385), EEF2 (ENSG00000167658)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5633', 'drugName': 'Denileukin Diftito...
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Approval Status, Genetic Target
Q1.1360
Q1
Is SLC10A2 a druggable gene?
There are currently 3 approved drugs which target SLC10A2, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%SLC10A2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5835', 'drugName': 'Maralixibat', 'drugIsApproved': True, 'newLinkedTargets_string': 'SLC10A2 (ENSG00000125255)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5944', 'drugName': 'Maralixibat Chloride', 'drugIsApproved': True, 'newLinkedTargets_string': 'SLC10A2 (ENSG0000012525...
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Approval Status, Genetic Target
Q1.1473
Q1
Is TPH1 a druggable gene?
There are currently 3 approved drugs which target TPH1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%TPH1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3468', 'drugName': 'Telotristat', 'drugIsApproved': True, 'newLinkedTargets_string': 'TPH2 (ENSG00000139287), TPH1 (ENSG00000129167)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1064', 'drugName': 'Telotristat Etiprate', 'drugIsApproved': True, 'newLinkedTargets_string': 'TP...
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Approval Status, Genetic Target
Q1.63
Q1
Is ANGPTL3 a druggable gene?
There is 1 drug, Evinacumab, that targets ANGPTL3, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%ANGPTL3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5281', 'drugName': 'Evinacumab', 'drugIsApproved': True, 'newLinkedTargets_string': 'ANGPTL3 (ENSG00000132855)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2325', 'drugName': 'Vupanorsen', 'drugIsApproved': False, 'newLinkedTargets_string': 'ANGPTL3 (ENSG00000132855), ASGR1 ...
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Approval Status, Genetic Target
Q1.283
Q1
Is CNR1 a druggable gene?
There are currently 4 approved drugs which target CNR1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CNR1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4055', 'drugName': 'Cannabidiol', 'drugIsApproved': True, 'newLinkedTargets_string': 'CNR1 (ENSG00000118432)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3038', 'drugName': 'Dronabinol', 'drugIsApproved': True, 'newLinkedTargets_string': 'CNR1 (ENSG00000118432)', 'maxClinica...
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Approval Status, Genetic Target
Q1.783
Q1
Is KCNV1 a druggable gene?
There are currently 5 approved drugs which target KCNV1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%KCNV1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5118', 'drugName': 'Guanidine Hydrochloride', 'drugIsApproved': True, 'newLinkedTargets_string': 'KCNQ1 (ENSG00000053918), KCND3 (ENSG00000171385), KCNH2 (ENSG00000055118), KCNA2 (ENSG00000177301), KCNA1 (ENSG00000111262), KCNQ2 (ENSG00000075043), KCNQ3 (ENSG00000184156), KCNA7 (ENSG000001...
general
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Approval Status, Genetic Target
Q1.1037
Q1
Is PARP3 a druggable gene?
There are currently 3 approved drugs which target PARP3, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%PARP3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3166', 'drugName': 'Rucaparib', 'drugIsApproved': True, 'newLinkedTargets_string': 'PARP1 (ENSG00000143799), PARP3 (ENSG00000041880), PARP2 (ENSG00000129484)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_279', 'drugName': 'Olaparib', 'drugIsApproved': True, 'newLinkedTargets_...
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Approval Status, Genetic Target
Q1.240
Q1
Is CDK19 a druggable gene?
There are currently no approved drugs targeting CDK19, but there are 4 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CDK19 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1429', 'drugName': 'Roniciclib', 'drugIsApproved': False, 'newLinkedTargets_string': 'CDK1 (ENSG00000170312), CDK4 (ENSG00000135446), CDK2 (ENSG00000123374), CDK5 (ENSG00000164885), CDK6 (ENSG00000105810), CDK7 (ENSG00000134058), CDK3 (ENSG00000250506), CDK16 (ENSG00000102225), CDK18 (ENSG...
general
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Approval Status, Genetic Target
Q1.225
Q1
Is CD80 a druggable gene?
There are currently 2 approved drugs which target CD80, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CD80 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4093', 'drugName': 'Belatacept', 'drugIsApproved': True, 'newLinkedTargets_string': 'CD80 (ENSG00000121594), CD86 (ENSG00000114013)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4094', 'drugName': 'Belatacept', 'drugIsApproved': True, 'newLinkedTargets_string': 'CD80 (ENSG000...
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Approval Status, Genetic Target
Q1.147
Q1
Is CACNA1F a druggable gene?
There are currently 35 approved drugs which target CACNA1F, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CACNA1F %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6292', 'drugName': 'Terodiline', 'drugIsApproved': True, 'newLinkedTargets_string': 'CHRM3 (ENSG00000133019), CHRM4 (ENSG00000180720), CHRM1 (ENSG00000168539), CHRM2 (ENSG00000181072), CHRM5 (ENSG00000184984), CACNA1H (ENSG00000196557), CACNA2D1 (ENSG00000153956), CACNA1C (ENSG00000151067)...
general
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Approval Status, Genetic Target
Q1.1434
Q1
Is TLR3 a druggable gene?
There are currently no approved drugs targeting TLR3, but there are 3 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%TLR3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4726', 'drugName': 'Bevasiranib', 'drugIsApproved': False, 'newLinkedTargets_string': 'TLR3 (ENSG00000164342)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_4727', 'drugName': 'Bevasiranib', 'drugIsApproved': False, 'newLinkedTargets_string': 'TLR3 (ENSG00000164342)', 'maxClin...
general
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Approval Status, Genetic Target
Q1.375
Q1
Is DRD3 a druggable gene?
There are currently 38 approved drugs which target DRD3, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%DRD3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4041', 'drugName': 'Loxapine', 'drugIsApproved': True, 'newLinkedTargets_string': 'HTR2A (ENSG00000102468), HTR2C (ENSG00000147246), DRD2 (ENSG00000149295), DRD3 (ENSG00000151577), DRD4 (ENSG00000069696)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1241', 'drugName': 'Caripr...
general
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Approval Status, Genetic Target
Q1.1271
Q1
Is RPL9 a druggable gene?
There is 1 drug, Ataluren, that targets RPL9, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%RPL9 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'drugIsApproved': True, 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.120
Q1
Is BRD2 a druggable gene?
There are currently no approved drugs targeting BRD2, but there are 6 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%BRD2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_866', 'drugName': 'Pelabresib', 'drugIsApproved': False, 'newLinkedTargets_string': 'BRD2 (ENSG00000204256), BRD4 (ENSG00000141867), BRDT (ENSG00000137948), BRD3 (ENSG00000169925)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_746', 'drugName': 'Apabetalone', 'drugIsApproved':...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1153
Q1
Is PSMA3 a druggable gene?
There are currently 4 approved drugs which target PSMA3, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%PSMA3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3334', 'drugName': 'Ixazomib', 'drugIsApproved': True, 'newLinkedTargets_string': 'PSMD1 (ENSG00000173692), PSMB2 (ENSG00000126067), PSMB1 (ENSG00000008018), PSMB5 (ENSG00000100804), PSMB8 (ENSG00000204264), PSMB9 (ENSG00000240065), PSMB6 (ENSG00000142507), PSMD14 (ENSG00000115233), PSMA1 ...
general
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Approval Status, Genetic Target
Q1.252
Q1
Is CETP a druggable gene?
There are currently no approved drugs targeting CETP, but there are 6 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CETP %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5790', 'drugName': 'Evacetrapib', 'drugIsApproved': False, 'newLinkedTargets_string': 'CETP (ENSG00000087237)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_2315', 'drugName': 'Obicetrapib', 'drugIsApproved': False, 'newLinkedTargets_string': 'CETP (ENSG00000087237)', 'maxClin...
general
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Approval Status, Genetic Target
Q1.1481
Q1
Is TRGV3 a druggable gene?
There are currently no approved drugs targeting TRGV3, but there are 3 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%TRGV3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1483', 'drugName': 'Medi-500', 'drugIsApproved': False, 'newLinkedTargets_string': 'TRAV29DV5 (ENSG00000211810), TRAC (ENSG00000277734), TRBV7-9 (ENSG00000278030), TRGV3 (ENSG00000211699)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_5971', 'drugName': 'Tol-101', 'drugIsAppro...
general
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Approval Status, Genetic Target
Q1.1239
Q1
Is RPL18A a druggable gene?
There is 1 drug, Ataluren, that targets RPL18A, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%RPL18A %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'drugIsApproved': True, 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.920
Q1
Is MUC16 a druggable gene?
There is 1 drug, Igovomab, that targets MUC16, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%MUC16 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_640', 'drugName': 'Igovomab', 'drugIsApproved': True, 'newLinkedTargets_string': 'MUC16 (ENSG00000181143)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3687', 'drugName': 'Oregovomab', 'drugIsApproved': False, 'newLinkedTargets_string': 'MUC16 (ENSG00000181143)', 'maxClinical...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.10
Q1
Is ACACB a druggable gene?
There are currently no approved drugs targeting ACACB, but there are 4 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%ACACB %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1425', 'drugName': 'Olumacostat Glasaretil', 'drugIsApproved': False, 'newLinkedTargets_string': 'ACACA (ENSG00000278540), ACACB (ENSG00000076555)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_2233', 'drugName': 'Clesacostat', 'drugIsApproved': False, 'newLinkedTargets_string...
general
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Approval Status, Genetic Target
Q1.451
Q1
Is FCGR1A a druggable gene?
There are currently no approved drugs targeting FCGR1A, but there are 2 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%FCGR1A %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4872', 'drugName': 'Mdx-447', 'drugIsApproved': False, 'newLinkedTargets_string': 'EGFR (ENSG00000146648), FCGR1A (ENSG00000150337)', 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_4871', 'drugName': 'Mdx-447', 'drugIsApproved': False, 'newLinkedTargets_string': 'EGFR (ENSG00000...
general
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Approval Status, Genetic Target
Q1.911
Q1
Is MT-ND4 a druggable gene?
There are currently 2 approved drugs which target MT-ND4, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%MT-ND4 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'drugIsApproved': True, 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (EN...
general
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Approval Status, Genetic Target
Q1.713
Q1
Is IRAK4 a druggable gene?
There are currently no approved drugs targeting IRAK4, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%IRAK4 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4254', 'drugName': 'Zimlovisertib', 'drugIsApproved': False, 'newLinkedTargets_string': 'IRAK4 (ENSG00000198001)', 'maxClinicalTrialPhase': 2}]
general
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Approval Status, Genetic Target
Q1.257
Q1
Is CHEK2 a druggable gene?
There are currently no approved drugs targeting CHEK2, but there are 2 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CHEK2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_562', 'drugName': 'Prexasertib', 'drugIsApproved': False, 'newLinkedTargets_string': 'CHEK1 (ENSG00000149554), CHEK2 (ENSG00000183765)', 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_563', 'drugName': 'Prexasertib', 'drugIsApproved': False, 'newLinkedTargets_string': 'CHEK1 (EN...
general
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Approval Status, Genetic Target
Q1.597
Q1
Is HMGCR a druggable gene?
There are currently 16 approved drugs which target HMGCR, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%HMGCR %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1184', 'drugName': 'Fluvastatin Sodium', 'drugIsApproved': True, 'newLinkedTargets_string': 'HMGCR (ENSG00000113161)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5208', 'drugName': 'Rosuvastatin Calcium', 'drugIsApproved': True, 'newLinkedTargets_string': 'HMGCR (ENSG0000011...
general
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Approval Status, Genetic Target
Q1.391
Q1
Is EFNB2 a druggable gene?
There are currently no approved drugs targeting EFNB2, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%EFNB2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6169', 'drugName': 'Sephb4-Hsa', 'drugIsApproved': False, 'newLinkedTargets_string': 'EFNB2 (ENSG00000125266)', 'maxClinicalTrialPhase': 2}]
general
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Approval Status, Genetic Target
Q1.1321
Q1
Is RXRB a druggable gene?
There are currently 4 approved drugs which target RXRB, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%RXRB %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5080', 'drugName': 'Acitretin', 'drugIsApproved': True, 'newLinkedTargets_string': 'RXRB (ENSG00000204231), RARG (ENSG00000172819), RXRG (ENSG00000143171), RARB (ENSG00000077092), RARA (ENSG00000131759), RXRA (ENSG00000186350)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_701...
general
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Approval Status, Genetic Target
Q1.1231
Q1
Is RPL11 a druggable gene?
There is 1 drug, Ataluren, that targets RPL11, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%RPL11 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'drugIsApproved': True, 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG...
general
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Approval Status, Genetic Target
Q1.560
Q1
Is GSK3B a druggable gene?
There are currently 2 approved drugs which target GSK3B, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%GSK3B %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3119', 'drugName': 'Lithium Carbonate', 'drugIsApproved': True, 'newLinkedTargets_string': 'IMPA1 (ENSG00000133731), GSK3A (ENSG00000105723), GSK3B (ENSG00000082701)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5478', 'drugName': 'Lithium Citrate', 'drugIsApproved': True, 'n...
general
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Approval Status, Genetic Target
Q1.1320
Q1
Is RXRA a druggable gene?
There are currently 5 approved drugs which target RXRA, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%RXRA %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_701', 'drugName': 'Alitretinoin', 'drugIsApproved': True, 'newLinkedTargets_string': 'RXRB (ENSG00000204231), RARG (ENSG00000172819), RXRG (ENSG00000143171), RARB (ENSG00000077092), RARA (ENSG00000131759), RXRA (ENSG00000186350)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3...
general
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Approval Status, Genetic Target
Q1.867
Q1
Is MARCKS a druggable gene?
There are currently no approved drugs targeting MARCKS, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%MARCKS %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5771', 'drugName': 'Bio-11006', 'drugIsApproved': False, 'newLinkedTargets_string': 'MARCKS (ENSG00000277443)', 'maxClinicalTrialPhase': 2}]
general
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Approval Status, Genetic Target
Q1.462
Q1
Is FGF2 a druggable gene?
There are currently no approved drugs targeting FGF2, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%FGF2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5103', 'drugName': 'Muparfostat', 'drugIsApproved': False, 'newLinkedTargets_string': 'HPSE (ENSG00000173083), FGF1 (ENSG00000113578), FGF2 (ENSG00000138685), VEGFA (ENSG00000112715)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_5102', 'drugName': 'Muparfostat', 'drugIsApprov...
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Approval Status, Genetic Target
Q1.728
Q1
Is ITGB8 a druggable gene?
There are currently no approved drugs targeting ITGB8, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%ITGB8 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1968', 'drugName': 'Abituzumab', 'drugIsApproved': False, 'newLinkedTargets_string': 'ITGAV (ENSG00000138448), ITGB6 (ENSG00000115221), ITGB5 (ENSG00000082781), ITGB3 (ENSG00000259207), ITGB1 (ENSG00000150093), ITGB8 (ENSG00000105855)', 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTarget...
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Approval Status, Genetic Target
Q1.1417
Q1
Is TEC a druggable gene?
There are currently no approved drugs targeting TEC, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%TEC %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4380', 'drugName': 'Pf-06651600', 'drugIsApproved': False, 'newLinkedTargets_string': 'ITK (ENSG00000113263), BMX (ENSG00000102010), TEC (ENSG00000135605), TXK (ENSG00000074966), BTK (ENSG00000010671), JAK3 (ENSG00000105639)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_4381'...
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Approval Status, Genetic Target
Q1.146
Q1
Is CACNA1E a druggable gene?
There are currently 9 approved drugs which target CACNA1E, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CACNA1E %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_142', 'drugName': 'Gabapentin', 'drugIsApproved': True, 'newLinkedTargets_string': 'CACNA1H (ENSG00000196557), CACNA2D1 (ENSG00000153956), CACNA1C (ENSG00000151067), CACNA2D3 (ENSG00000157445), CACNA1S (ENSG00000081248), CACNA2D2 (ENSG00000007402), CACNA1D (ENSG00000157388), CACNA1A (ENSG0...
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Approval Status, Genetic Target
Q1.504
Q1
Is GABRG1 a druggable gene?
There are currently 66 approved drugs which target GABRG1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%GABRG1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1494', 'drugName': 'Thiopental', 'drugIsApproved': True, 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089), GABRA3 (ENSG00000011677)...
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Approval Status, Genetic Target
Q1.1175
Q1
Is PSMC6 a druggable gene?
There are currently 4 approved drugs which target PSMC6, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%PSMC6 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_559', 'drugName': 'Bortezomib', 'drugIsApproved': True, 'newLinkedTargets_string': 'PSMD1 (ENSG00000173692), PSMB2 (ENSG00000126067), PSMB1 (ENSG00000008018), PSMB5 (ENSG00000100804), PSMB8 (ENSG00000204264), PSMB9 (ENSG00000240065), PSMB6 (ENSG00000142507), PSMD14 (ENSG00000115233), PSMA1...
general
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Approval Status, Genetic Target
Q1.744
Q1
Is KCNC2 a druggable gene?
There are currently 5 approved drugs which target KCNC2, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%KCNC2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5118', 'drugName': 'Guanidine Hydrochloride', 'drugIsApproved': True, 'newLinkedTargets_string': 'KCNQ1 (ENSG00000053918), KCND3 (ENSG00000171385), KCNH2 (ENSG00000055118), KCNA2 (ENSG00000177301), KCNA1 (ENSG00000111262), KCNQ2 (ENSG00000075043), KCNQ3 (ENSG00000184156), KCNA7 (ENSG000001...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1420
Q1
Is TFPI a druggable gene?
There are currently no approved drugs targeting TFPI, but there are 4 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%TFPI %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6201', 'drugName': 'Marstacimab', 'drugIsApproved': False, 'newLinkedTargets_string': 'TFPI (ENSG00000003436)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_5154', 'drugName': 'Andexanet Alfa', 'drugIsApproved': False, 'newLinkedTargets_string': 'TFPI (ENSG00000003436)', 'maxC...
general
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Approval Status, Genetic Target
Q1.736
Q1
Is KCNA3 a druggable gene?
There are currently 5 approved drugs which target KCNA3, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%KCNA3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5118', 'drugName': 'Guanidine Hydrochloride', 'drugIsApproved': True, 'newLinkedTargets_string': 'KCNQ1 (ENSG00000053918), KCND3 (ENSG00000171385), KCNH2 (ENSG00000055118), KCNA2 (ENSG00000177301), KCNA1 (ENSG00000111262), KCNQ2 (ENSG00000075043), KCNQ3 (ENSG00000184156), KCNA7 (ENSG000001...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.542
Q1
Is GRIA4 a druggable gene?
There are currently 2 approved drugs which target GRIA4, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%GRIA4 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2165', 'drugName': 'Perampanel', 'drugIsApproved': True, 'newLinkedTargets_string': 'GRIA4 (ENSG00000152578), GRIA3 (ENSG00000125675), GRIA2 (ENSG00000120251), GRIA1 (ENSG00000155511)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1593', 'drugName': 'Topiramate', 'drugIsApprov...
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Approval Status, Genetic Target
Q1.179
Q1
Is CASP4 a druggable gene?
There are currently no approved drugs targeting CASP4, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CASP4 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_45', 'drugName': 'Emricasan', 'drugIsApproved': False, 'newLinkedTargets_string': 'CASP4 (ENSG00000196954), CASP9 (ENSG00000132906), CASP3 (ENSG00000164305), CASP5 (ENSG00000137757), CASP6 (ENSG00000138794), CASP7 (ENSG00000165806), CASP8 (ENSG00000064012), CASP1 (ENSG00000137752), CASP2 (...
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Approval Status, Genetic Target
Q1.1483
Q1
Is TRPA1 a druggable gene?
There are currently 3 approved drugs which target TRPA1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%TRPA1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5721', 'drugName': 'Menthol', 'drugIsApproved': True, 'newLinkedTargets_string': 'TRPA1 (ENSG00000104321), TRPM8 (ENSG00000144481)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5054', 'drugName': 'Butamben', 'drugIsApproved': True, 'newLinkedTargets_string': 'TRPA1 (ENSG00000...
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Approval Status, Genetic Target
Q1.702
Q1
Is IL5RA a druggable gene?
There is 1 drug, Benralizumab, that targets IL5RA, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%IL5RA %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5224', 'drugName': 'Benralizumab', 'drugIsApproved': True, 'newLinkedTargets_string': 'IL5RA (ENSG00000091181)', 'maxClinicalTrialPhase': 4}]
general
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Approval Status, Genetic Target
Q1.969
Q1
Is NDUFS3 a druggable gene?
There are currently 2 approved drugs which target NDUFS3, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%NDUFS3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'drugIsApproved': True, 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (EN...
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Approval Status, Genetic Target
Q1.1069
Q1
Is PDK3 a druggable gene?
There is 1 drug, Sodium Dichloroacetate, that targets PDK3, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%PDK3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2764', 'drugName': 'Sodium Dichloroacetate', 'drugIsApproved': True, 'newLinkedTargets_string': 'PDK2 (ENSG00000005882), PDK3 (ENSG00000067992), PDK4 (ENSG00000004799), PDK1 (ENSG00000152256)', 'maxClinicalTrialPhase': 4}]
general
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Approval Status, Genetic Target
Q1.903
Q1
Is MPO a druggable gene?
There are currently no approved drugs targeting MPO, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%MPO %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1006', 'drugName': 'Verdiperstat', 'drugIsApproved': False, 'newLinkedTargets_string': 'MPO (ENSG00000005381)', 'maxClinicalTrialPhase': 3}]
general
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Approval Status, Genetic Target
Q1.927
Q1
Is MYL4 a druggable gene?
There is 1 drug, Mavacamten, that targets MYL4, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%MYL4 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1036', 'drugName': 'Mavacamten', 'drugIsApproved': True, 'newLinkedTargets_string': 'MYH7 (ENSG00000092054), MYH6 (ENSG00000197616), MYH7B (ENSG00000078814), MYL3 (ENSG00000160808), MYL2 (ENSG00000111245), MYL7 (ENSG00000106631), MYL4 (ENSG00000198336)', 'maxClinicalTrialPhase': 4}, {'UUID...
general
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Approval Status, Genetic Target
Q1.1531
Q1
Is WEE1 a druggable gene?
There are currently no approved drugs targeting WEE1, but there are 2 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%WEE1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5552', 'drugName': 'Azenosertib', 'drugIsApproved': False, 'newLinkedTargets_string': 'WEE1 (ENSG00000166483)', 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_224', 'drugName': 'Adavosertib', 'drugIsApproved': False, 'newLinkedTargets_string': 'WEE1 (ENSG00000166483)', 'maxClini...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.8
Q1
Is ABL1 a druggable gene?
There are currently 13 approved drugs which target ABL1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%ABL1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_802', 'drugName': 'Regorafenib', 'drugIsApproved': True, 'newLinkedTargets_string': 'EPHA2 (ENSG00000142627), TEK (ENSG00000120156), MAPK11 (ENSG00000185386), RAF1 (ENSG00000132155), FRK (ENSG00000111816), PDGFRB (ENSG00000113721), PDGFRA (ENSG00000134853), KIT (ENSG00000157404), FGFR1 (EN...
general
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Approval Status, Genetic Target
Q1.908
Q1
Is MT-ND1 a druggable gene?
There are currently 2 approved drugs which target MT-ND1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%MT-ND1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'drugIsApproved': True, 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (EN...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.672
Q1
Is IL13RA1 a druggable gene?
There are currently no approved drugs targeting IL13RA1, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%IL13RA1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2466', 'drugName': 'Cintredekin Besudotox', 'drugIsApproved': False, 'newLinkedTargets_string': 'IL4R (ENSG00000077238), IL13RA1 (ENSG00000131724), IL13RA2 (ENSG00000123496)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_2467', 'drugName': 'Cintredekin Besudotox', 'drugIsAppro...
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Approval Status, Genetic Target
Q1.1436
Q1
Is TLR5 a druggable gene?
There are currently no approved drugs targeting TLR5, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%TLR5 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3738', 'drugName': 'Entolimod', 'drugIsApproved': False, 'newLinkedTargets_string': 'TLR5 (ENSG00000187554)', 'maxClinicalTrialPhase': 2}]
general
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Approval Status, Genetic Target
Q1.359
Q1
Is DHCR24 a druggable gene?
There is 1 drug, Triparanol, that targets DHCR24, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%DHCR24 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3812', 'drugName': 'Triparanol', 'drugIsApproved': True, 'newLinkedTargets_string': 'DHCR24 (ENSG00000116133)', 'maxClinicalTrialPhase': 4}]
general
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Approval Status, Genetic Target
Q1.788
Q1
Is KIF11 a druggable gene?
There are currently no approved drugs targeting KIF11, but there are 4 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%KIF11 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5386', 'drugName': 'Litronesib', 'drugIsApproved': False, 'newLinkedTargets_string': 'KIF11 (ENSG00000138160)', 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_3893', 'drugName': 'Ispinesib', 'drugIsApproved': False, 'newLinkedTargets_string': 'KIF11 (ENSG00000138160)', 'maxClini...
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Approval Status, Genetic Target
Q1.740
Q1
Is KCNA7 a druggable gene?
There are currently 5 approved drugs which target KCNA7, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%KCNA7 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5118', 'drugName': 'Guanidine Hydrochloride', 'drugIsApproved': True, 'newLinkedTargets_string': 'KCNQ1 (ENSG00000053918), KCND3 (ENSG00000171385), KCNH2 (ENSG00000055118), KCNA2 (ENSG00000177301), KCNA1 (ENSG00000111262), KCNQ2 (ENSG00000075043), KCNQ3 (ENSG00000184156), KCNA7 (ENSG000001...
general
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Approval Status, Genetic Target
Q1.331
Q1
Is CTSC a druggable gene?
There are currently no approved drugs targeting CTSC, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CTSC %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1902', 'drugName': 'Brensocatib', 'drugIsApproved': False, 'newLinkedTargets_string': 'CTSC (ENSG00000109861)', 'maxClinicalTrialPhase': 3}]
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Approval Status, Genetic Target
Q1.1230
Q1
Is RPL10A a druggable gene?
There is 1 drug, Ataluren, that targets RPL10A, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%RPL10A %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'drugIsApproved': True, 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG...
general
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Approval Status, Genetic Target
Q1.1176
Q1
Is PSMD1 a druggable gene?
There are currently 4 approved drugs which target PSMD1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%PSMD1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_559', 'drugName': 'Bortezomib', 'drugIsApproved': True, 'newLinkedTargets_string': 'PSMD1 (ENSG00000173692), PSMB2 (ENSG00000126067), PSMB1 (ENSG00000008018), PSMB5 (ENSG00000100804), PSMB8 (ENSG00000204264), PSMB9 (ENSG00000240065), PSMB6 (ENSG00000142507), PSMD14 (ENSG00000115233), PSMA1...
general
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Approval Status, Genetic Target
Q1.1270
Q1
Is RPL8 a druggable gene?
There is 1 drug, Ataluren, that targets RPL8, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%RPL8 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'drugIsApproved': True, 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG...
general
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Approval Status, Genetic Target
Q1.260
Q1
Is CHRM2 a druggable gene?
There are currently 21 approved drugs which target CHRM2, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CHRM2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3301', 'drugName': 'Tolterodine Tartrate', 'drugIsApproved': True, 'newLinkedTargets_string': 'CHRM3 (ENSG00000133019), CHRM2 (ENSG00000181072)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_871', 'drugName': 'Oxybutynin Chloride', 'drugIsApproved': True, 'newLinkedTargets_str...
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Approval Status, Genetic Target
Q1.1255
Q1
Is RPL34 a druggable gene?
There is 1 drug, Ataluren, that targets RPL34, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%RPL34 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'drugIsApproved': True, 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG...
general
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Approval Status, Genetic Target
Q1.374
Q1
Is DRD2 a druggable gene?
There are currently 98 approved drugs which target DRD2, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%DRD2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5204', 'drugName': 'Metoclopramide Hydrochloride', 'drugIsApproved': True, 'newLinkedTargets_string': 'HTR4 (ENSG00000164270), HTR3A (ENSG00000166736), DRD2 (ENSG00000149295)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_426', 'drugName': 'Prochlorperazine', 'drugIsApproved':...
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Approval Status, Genetic Target
Q1.1128
Q1
Is PRKACA a druggable gene?
There are currently no approved drugs targeting PRKACA, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%PRKACA %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1835', 'drugName': 'Gsk-690693', 'drugIsApproved': False, 'newLinkedTargets_string': 'PRKACB (ENSG00000142875), PRKACA (ENSG00000072062), PRKACG (ENSG00000165059), AKT2 (ENSG00000105221), AKT3 (ENSG00000117020), AKT1 (ENSG00000142208), PRKD3 (ENSG00000115825), PRKCI (ENSG00000163558), PRKC...
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Approval Status, Genetic Target
Q1.954
Q1
Is NDUFB1 a druggable gene?
There are currently 2 approved drugs which target NDUFB1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%NDUFB1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'drugIsApproved': True, 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (EN...
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Q1.144
Q1
Is CACNA1C a druggable gene?
There are currently 35 approved drugs which target CACNA1C, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CACNA1C %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6292', 'drugName': 'Terodiline', 'drugIsApproved': True, 'newLinkedTargets_string': 'CHRM3 (ENSG00000133019), CHRM4 (ENSG00000180720), CHRM1 (ENSG00000168539), CHRM2 (ENSG00000181072), CHRM5 (ENSG00000184984), CACNA1H (ENSG00000196557), CACNA2D1 (ENSG00000153956), CACNA1C (ENSG00000151067)...
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Q1.528
Q1
Is GNRHR a druggable gene?
There are currently 25 approved drugs which target GNRHR, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%GNRHR %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4802', 'drugName': 'Leuprolide Acetate', 'drugIsApproved': True, 'newLinkedTargets_string': 'GNRHR (ENSG00000109163)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2259', 'drugName': 'Goserelin', 'drugIsApproved': True, 'newLinkedTargets_string': 'GNRHR (ENSG00000109163)', 'ma...
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Q1.1164
Q1
Is PSMB4 a druggable gene?
There are currently 4 approved drugs which target PSMB4, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%PSMB4 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3334', 'drugName': 'Ixazomib', 'drugIsApproved': True, 'newLinkedTargets_string': 'PSMD1 (ENSG00000173692), PSMB2 (ENSG00000126067), PSMB1 (ENSG00000008018), PSMB5 (ENSG00000100804), PSMB8 (ENSG00000204264), PSMB9 (ENSG00000240065), PSMB6 (ENSG00000142507), PSMD14 (ENSG00000115233), PSMA1 ...
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Q1.234
Q1
Is CDK13 a druggable gene?
There are currently no approved drugs targeting CDK13, but there are 4 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CDK13 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1429', 'drugName': 'Roniciclib', 'drugIsApproved': False, 'newLinkedTargets_string': 'CDK1 (ENSG00000170312), CDK4 (ENSG00000135446), CDK2 (ENSG00000123374), CDK5 (ENSG00000164885), CDK6 (ENSG00000105810), CDK7 (ENSG00000134058), CDK3 (ENSG00000250506), CDK16 (ENSG00000102225), CDK18 (ENSG...
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Q1.1212
Q1
Is RARB a druggable gene?
There are currently 7 approved drugs which target RARB, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%RARB %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5080', 'drugName': 'Acitretin', 'drugIsApproved': True, 'newLinkedTargets_string': 'RXRB (ENSG00000204231), RARG (ENSG00000172819), RXRG (ENSG00000143171), RARB (ENSG00000077092), RARA (ENSG00000131759), RXRA (ENSG00000186350)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_701...
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Q1.1459
Q1
Is TNKS a druggable gene?
There are currently no approved drugs targeting TNKS, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%TNKS %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1419', 'drugName': '2X-121', 'drugIsApproved': False, 'newLinkedTargets_string': 'TNKS2 (ENSG00000107854), TNKS (ENSG00000173273), PARP1 (ENSG00000143799), PARP2 (ENSG00000129484)', 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_1420', 'drugName': '2X-121', 'drugIsApproved': Fal...
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Q1.442
Q1
Is F5 a druggable gene?
There is 1 drug, Drotrecogin Alfa (Activated), that targets F5, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%F5 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2502', 'drugName': 'Drotrecogin Alfa (Activated)', 'drugIsApproved': True, 'newLinkedTargets_string': 'F8 (ENSG00000185010), F5 (ENSG00000198734)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2503', 'drugName': 'Drotrecogin Alfa (Activated)', 'drugIsApproved': True, 'newLinke...
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Q1.534
Q1
Is GPNMB a druggable gene?
There are currently no approved drugs targeting GPNMB, but there are 2 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%GPNMB %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6315', 'drugName': 'Glembatumumab Vedotin', 'drugIsApproved': False, 'newLinkedTargets_string': 'GPNMB (ENSG00000136235), TUBB4B (ENSG00000188229), TUBB1 (ENSG00000101162), TUBA3C (ENSG00000198033), TUBA4A (ENSG00000127824), TUBB3 (ENSG00000258947), TUBA1A (ENSG00000167552), TUBB4A (ENSG00...
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Q1.1232
Q1
Is RPL12 a druggable gene?
There is 1 drug, Ataluren, that targets RPL12, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%RPL12 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'drugIsApproved': True, 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG...
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Q1.228
Q1
Is CDC7 a druggable gene?
There are currently no approved drugs targeting CDC7, but there are 4 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CDC7 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1097', 'drugName': 'Bms-863233', 'drugIsApproved': False, 'newLinkedTargets_string': 'CDC7 (ENSG00000097046)', 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_5195', 'drugName': 'Simurosertib', 'drugIsApproved': False, 'newLinkedTargets_string': 'CDC7 (ENSG00000097046)', 'maxClin...
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Q1.1056
Q1
Is PDE6D a druggable gene?
There are currently 2 approved drugs which target PDE6D, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%PDE6D %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6107', 'drugName': 'Dipyridamole', 'drugIsApproved': True, 'newLinkedTargets_string': 'PDE5A (ENSG00000138735), PDE4A (ENSG00000065989), PDE3A (ENSG00000172572), PDE6H (ENSG00000139053), PDE6G (ENSG00000185527), PDE2A (ENSG00000186642), PDE7A (ENSG00000205268), PDE1A (ENSG00000115252), PDE...
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Q1.230
Q1
Is CDK1 a druggable gene?
There are currently no approved drugs targeting CDK1, but there are 13 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CDK1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5622', 'drugName': 'Alvocidib', 'drugIsApproved': False, 'newLinkedTargets_string': 'CDK1 (ENSG00000170312), CDK7 (ENSG00000134058), CDK9 (ENSG00000136807), CDK6 (ENSG00000105810), CDK2 (ENSG00000123374), CDK4 (ENSG00000135446)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_49...
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